Synthesis and anticonvulsant activity of the (+)- and (-)-enantiomers of 1,2,3,4-tetrahydro-5-(2-phosphonoethyl)-3-isoquinolinecarboxylic acid, a competitive NMDA antagonist (Unbekannt)
- Neue Suche nach: Bigge, C. F.
- Neue Suche nach: Wu, J.-P.
- Neue Suche nach: Malone, T. C.
- Neue Suche nach: Taylor, C. P.
- Neue Suche nach: Bigge, C. F.
- Neue Suche nach: Wu, J.-P.
- Neue Suche nach: Malone, T. C.
- Neue Suche nach: Taylor, C. P.
In:
BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS
;
3
, 1
;
39
;
1993
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ISSN:
- Aufsatz (Zeitschrift) / Print
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Titel:Synthesis and anticonvulsant activity of the (+)- and (-)-enantiomers of 1,2,3,4-tetrahydro-5-(2-phosphonoethyl)-3-isoquinolinecarboxylic acid, a competitive NMDA antagonist
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Beteiligte:Bigge, C. F. ( Autor:in ) / Wu, J.-P. ( Autor:in ) / Malone, T. C. ( Autor:in ) / Taylor, C. P. ( Autor:in )
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Erschienen in:BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS ; 3, 1 ; 39
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Verlag:
- Neue Suche nach: PERGAMON PRESS
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Erscheinungsdatum:01.01.1993
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Format / Umfang:39 pages
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ISSN:
-
Medientyp:Aufsatz (Zeitschrift)
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Format:Print
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Sprache:Unbekannt
- Neue Suche nach: 572.5
- Weitere Informationen zu Dewey Decimal Classification
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Klassifikation:
DDC: 572.5 -
Datenquelle:
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- 1
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Contributors to this issue| 1993
- 3
-
Graphical abstracts| 1993
- 9
-
Foreword| 1993
- 9
-
Excitatory amino acid related agentsJohnson, Graham et al. | 1993
- 15
-
Synthesis of L-2-(2,3-dicarboxyclopropyl)glycines. Novel conformationally restricted glutamate analogues.Ohfune, Yasufumi / Shimamoto, Keiko / Ishida, Michiko / Shinozaki, Haruhiko et al. | 1993
- 15
-
Synthesis of L-2-(2,3-dicarboxycyclopropyl)glycines. Novel conformationally restricted glutamate analoguesOhfune, Y. / Shimamoto, K. / Ishida, M. / Shinozaki, H. et al. | 1993
- 15
-
Synthesis of L-2-(2,3-dicarboxvcydopropyl)glycines. Novel conformationally restricted glutamate analoguesOhfune, Y. et al. | 1993
- 19
-
Competitive NMDA receptor antagonists: synthesis of β-ketophosphonate-substituted piperidine carboxylic acid derivativesWhitten, Jeffrey P. / Cube, Rowena V. / Baron, Bruce M. / McDonald, Ian A. et al. | 1993
- 19
-
Competitive NMDA receptor antagonists: synthesis of b-ketophosphonatesubstituted piperidine carboxylic acid derivativesWhitten, J.P. et al. | 1993
- 23
-
Competitive NMDA receptor antagonists; (R)-4-Oxo-5-phosphononorvaline structure-activity relationshipsWhitten, Jeffrey P. / Baron, Bruce M. / McDonald, Ian A. et al. | 1993
- 27
-
Enzymatic asymmetric synthesis of (2R, 4R, 5S)-2-amino-4,5-(1,2-cyclohexyl)-7-phosphonoheptanoic acid, a potent, selective and competitive NMDA antagonistHamilton, G.S. / Huang, Z. / Patch, R.J. / Narayanan, B.A. / Ferkany, J.W. et al. | 1993
- 27
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Enzymatic asymmetric synthesis of (2R,4R,5S)-2-amino-4,5-(1,2-cyclohexyl)-7-phosphonohetanoic acid, a potent, selective and competitive NMDA antagonistHamilton, G.S. et al. | 1993
- 33
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Pharmacology of (2R, 4R, 5S)-2-amino-4,5-(1,2-cyclohexyl)-7-phosphonoheptanoic acid (NPC 17742); a selective, systemically active, competitive NMDA antagonistFerkany, J.W. / Willetts, J.S.A. / Borosky, D.B. / Clissold, E.W. / Karbon / Hamilton, G.S. et al. | 1993
- 33
-
Pharmacology of (2R,4R,5S)-2-amino-4,5-(1,2-cyclohexyl)-7-phosphonoheptanoic acid (NPC 17742) a selective,systemlcally active, competitive NMDA antagonistFerkany, J.W. et al. | 1993
- 39
-
Synthesis and anticonvulsant activity of the (+)- and (−)-enantiomers of 1,2,3,4-tetrahydro-5-(2-phosphonoethyl)-3-isoquinolinecarboxylic acid, a competitive NMDA antagonistBigge, Christopher F. / Wu, Jiang-Ping / Malone, Thomas C. / Taylor, Charles P. / Vartanian, Mark G. et al. | 1993
- 39
-
Synthesis and anticonvulsant activity of the (+)- and (-)-enantiomers of 1,2,3,4-tetrahydro-5-(2-phosphonoethyl)-3-isoqulnolinecarboxylic acid, a competitive NMDA antagonistBiqge, C.F. et al. | 1993
- 43
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Tetrazole amino acids as competitive NMDA antagonistsOrnstein, Paul L. / Arnold, M.Brian / Evrard, Debbie / Leander, J.David / Lodge, David / Schoepp, Darryle D. et al. | 1993
- 49
-
Synthesis and biological activity of conformationally constrained 4a-phenanthreneamine derivatives as noncompetitive NMDA antagonistsMalone, Thomas C. / Ortwine, Daniel F. / Johnson, Graham / Probert, Albert W. Jr. et al. | 1993
- 55
-
Synthesis and activity of spiroisoindolines as novel noncompetitive NMDA antagonistsBare, Thomas M. / Draper, Clyde W. / McLaren, Charles D. / Pullan, Linda M. / Patel, Jitendra / Patel, Jitendra B. et al. | 1993
- 61
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Anticonvulsant activity of glycine-site NMDA antagonists--I. 2-Carboxyl prodrugs of 5,7-dichlorokynurenic acidMoore, K.W. et al. | 1993
- 61
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Anticonvulsant activity of glycine-site NMDA antagonists. 1. 2-carboxyl prodrugs of 5,7-dichlorokynurenic acidMoore, Kevin W. / Leeson, Paul D. / Carling, Robert W. / Ticklebank, Mark D. / Singh, Lakhbir et al. | 1993
- 65
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Anticonvulsant activity of glycine-site NMDA antagonists. 2. trans 2-carboxy-4-substituted tetrahydroquinolines.Carling, Robert W. / Leeson, Paul D. / Moseley, Angela M. / Smith, Julian D. / Saywell, Kay / Tricklebank, Mark D. / Kemp, John A. / Marshall, George R. / Foster, Alan C. / Grimwood, Sarah et al. | 1993
- 65
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Anticonvulsant activity of glycine-site NMDA antagonists--II. trans 2-Carboxy-4-substituted tetrahydroquinolinesCarlinq, R.W. et al. | 1993
- 71
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Derivatives of 1-hydroxy-3-aminopyrrolidin-2-one (HA-966). Partial agonists at the glycine site of the NMDA receptorLeeson, Paul D. / Williams, Brian J. / Rowley, Michael / Moore, Kevin W. / Baker, Raymond / Kemp, John A. / Priestley, Tony / Foster, Alan C. / Donald, Angus E. et al. | 1993
- 77
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N-sulfonyl derivatives of 6,7-dichloro 3,4-dihydro-3-oxo-quinoxalinecarboxylate as glycine-site NMDA and AMPA antagonistsHays, Sheryl J. / Boxer, Peter A. / Taylor, Charles P. / Vartanian, Mark G. / Robichaud, Lillian J. / Nielsen, Elsebet Ø. et al. | 1993
- 81
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Structure-activity relationships of a series of glycine antagonists related to 5,7-dichlorokynurenic acid and 3-(2-carboxy-6-chloroindol-3-yl)acetic acidSmith, Edward C.R. / McQuaid, Loretta A. / Calligaro, David O. / O'Malley, Patrick J. et al. | 1993
- 85
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Interaction of rigid polyamine analogues with the NMDA receptor complex from rat brainReynolds, Ian J. / Rothermund, Kristi D. / Rajdev, Sunita et al. | 1993
- 85
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Interaction of rigid polyamine analogues with the NMDA receptor complex from rat bralnReynolds, I.J. et al. | 1993
- 91
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Oxindole N-Methyl-D-Aspartate (NMDA) antagonistsChenard, B.L. / Butler, T.W. / Shalaby, I.A. / Prochniak, M.A. / Koe, B.K. / Fox, C.B. et al. | 1993
- 95
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Synthesis and pharmacological characterization of l-trans-4-tetrazolylproline (ly300020): A novel systemically-active ampa receptor agonistMonn, James A. / Valli, Matthew J. / True, Rebecca A. / Schoepp, Darryl D. / Leander, J.David / Lodge, David et al. | 1993
- 99
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Structure-activity relationships of 2,3-benzodiazepine compounds with glutamate antagonistic actionTarnawa, István / Berzsenyi, Pál / Andrási, Ferenc / Botka, Péter / Hámori, Tamás / Ling, István / Körösi, Jenö et al. | 1993
- 105
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Isatin oximes - A novel series of bioavailable non-NMDA antagonistsWätjen, Frank / Nielsen, Elsebet Ø. / Drejer, Jørgen / Jensen, Leif H. et al. | 1993
- 107
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Enzymatic resolution of AMPA by use of α-chymotrypsinNielsen, Birgitte / Fisker, Herdis / Ebert, Bjarke / Madsen, Ulf / Curtis, David R. / Krogsgaard-Larsen, Povl / Hansen, Jan J. et al. | 1993
- 107
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Enzymatic resolution of AMPA by use of a-chymotrypsinNielsen, B. et al. | 1993
- 115
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Conformationally restricted inhibitors of the high affinity -glutamate transporterBridges, Richard J. / Lovering, Frank E. / Humphrey, John M. / Stanley, Mark S. / Blakely, Tracy N. / Cristofaro, Michael F. / Chamberlin, A.Richard et al. | 1993