Antipsoriatic Anthrones with Modulated Redox Properties. 3. 10-Thio-Substituted 1,8-Dihydroxy-9(10H)-anthracenones as Inhibitors of Keratinocyte Growth, 5-Lipoxygenase, and the Formation of 12(S)-HETE in Mouse Epidermis1 (Englisch)

In: Journal of Medicinal Chemistry   ;  39 ,  16  ;  3132-3138  ;  1996

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Inhaltsverzeichnis – Band 39, Ausgabe 16

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3035
Identification of a Retinoic Acid Receptor α Subtype Specific Agonist
Teng, Min / Duong, Tien T. / Klein, Elliott S. / Pino, Mary E. / Chandraratna, Roshantha A. S. | 1996
3035
Identification of a Retinoic Acid Receptor a Subtype Specific Agonist
Teng, Min / Duong, Tien T. / Klein, Elliott S. / Pino, Mary E. / Chandraratna, Roshantha A.S. | 1996
3039
Potent Thrombin Inhibitors That the S~1^' Subsite: Tripeptide Transition State Analogues Based on a Heterocycle-Activated Carbonyl Group
Costanzo, M. J. / Maryanoff, B. E. / Hecker, L. R. / Schott, M. R. / Yabut, S. C. / Zhang, H.-C. / Andrade-Gordon, P. / Kauffman, J. A. / Lewis, J. M. / Krishnan, R. | 1996
3039
Potent Thrombin Inhibitors That Probe the S1‘ Subsite:  Tripeptide Transition State Analogues Based on a Heterocycle-Activated Carbonyl Group1
Costanzo, Michael J. / Maryanoff, Bruce E. / Hecker, Leonard R. / Schott, Mary R. / Yabut, Stephen C. / Zhang, Han-Cheng / Andrade-Gordon, Patricia / Kauffman, Jack A. / Lewis, Joan M. / Krishnan, Raman et al. | 1996
3039
Potent Thrombin Inhibitors That Probe the S1' Subsite: Tripeptide Transition State Analogues Based on a Heterocycle-Activated Carbonyl Group
Costanzo, Michael J. / Maryanoff, Bruce E. / Hecker, Leonard R. / Schott, Mary R. / Yabut, Stephen C. / Zhang, Han-Cheng / Andrade-Gordon, Patricia / Kauffman, Jack A. / Lewis, Joan M. / Krishnan, Raman et al. | 1996
3044
Potent Inhibition of Tumor Necrosis Factor-� Production by Tetraflourothalidomide and Tetraflourophthalimides
Niwayama, S. / Turk, B. E. / Liu, J. O. | 1996
3044
Potent Inhibition of Tumor Necrosis Factor-a Production by Tetrafluorothalidomide and Tetrafluorophthalimides
Niwayama, Satomi / Turk, Benjamin E. / Liu, Jun O. | 1996
3044
Potent Inhibition of Tumor Necrosis Factor-α Production by Tetrafluorothalidomide and Tetrafluorophthalimides
Niwayama, Satomi / Turk, Benjamin E. / Liu, Jun O. | 1996
3046
Mechanism-Based Inhibition ofl-Pipecolate Oxidase by 4,5-Dehydro-l-Pipecolic Acid
Zabriskie, T. Mark | 1996
3049
Neighborhood Behavior:  A Useful Concept for Validation of “Molecular Diversity” Descriptors
Patterson, David E. / Cramer, Richard D. / Ferguson, Allan M. / Clark, Robert D. / Weinberger, Laurence E. | 1996
3060
Bioisosterism as a Molecular Diversity Descriptor:  Steric Fields of Single “Topomeric” Conformers
Cramer, Richard D. / Clark, Robert D. / Patterson, David E. / Ferguson, Allan M. | 1996
3070
Synthesis and Structure−Activity Relationships of 2-Pyridones:  A Novel Series of Potent DNA Gyrase Inhibitors as Antibacterial Agents
Li, Qun / Chu, Daniel T. W. / Claiborne, Akiyo / Cooper, Curt S. / Lee, Cheuk M. / Raye, Kathleen / Berst, Kristine B. / Donner, Pamela / Wang, Weibo / Hasvold, Lisa et al. | 1996
3089
Synthesis of 2-Amido-2,3-dihydro-1H-phenalene Derivatives as New Conformationally Restricted Ligands for Melatonin Receptors
Mathé-Allainmat, Monique / Gaudy, Florence / Sicsic, Sames / Dangy-Caye, Anne-Laure / Shen, Shuren / Brémont, Béatrice / Benatalah, Zohra / Langlois, Michel / Renard, Pierre / Delagrange, Philippe | 1996
3096
Evaluation of the Stability and Animal Biodistribution of Gadolinium(III) Benzylamine-Derivatized Diethylenetriaminepentaacetic Acid
Deal, Kim A. / Motekaitis, Ramunas J. / Martell, Arthur E. / Welch, Michael J. | 1996
3107
De Novo Antimicrobial Peptides with Low Mammalian Cell Toxicity
Javadpour, Maryam M. / Juban, Martha M. / Lo, Wai-Chun J. / Bishop, Steven M. / Alberty, J. Brannon / Cowell, Scott M. / Becker, Calvin L. / McLaughlin, Mark L. | 1996
3114
Peptidyl Anthraquinones as Potential Antineoplastic Drugs:  Synthesis, DNA Binding, Redox Cycling, and Biological Activity
Gatto, Barbara / Zagotto, Giuseppe / Sissi, Claudia / Cera, Cinzia / Uriarte, Eugenio / Palù, Giorgio / Capranico, Giovanni / Palumbo, Manlio | 1996
3123
Synthesis and Evaluation of Phorboid 20-Homovanillates:  Discovery of a Class of Ligands Binding to the Vanilloid (Capsaicin) Receptor with Different Degrees of Cooperativity
Appendino, Giovanni / Cravotto, Giancarlo / Palmisano, Giovanni / Annunziata, Rita / Szallasi, Arpad | 1996
3132
Antipsoriatic Anthrones with Modulated Redox Properties. 3. 10-Thio-Substituted 1,8-Dihydroxy-9(10H)-anthracenones as Inhibitors of Keratinocyte Growth, 5-Lipoxygenase, and the Formation of 12(S)-HETE in Mouse Epidermis
Müller, Klaus / Huang, Hsu-Shan / Wiegrebe, Wolfgang | 1996
3132
Antipsoriatic Anthrones with Modulated Redox Properties. 3. 10-Thio-Substituted 1,8-Dihydroxy-9(10H)-anthracenones as Inhibitors of Keratinocyte Growth, 5-Lipoxygenase, and the Formation of 12(S)-HETE in Mouse Epidermis1
Müller, Klaus / Huang, Hsu-Shan / Wiegrebe, Wolfgang | 1996
3139
Orally Active Fibrinogen Receptor Antagonists. 2. Amidoximes as Prodrugs of Amidines
Weller, Thomas / Alig, Leo / Beresini, Maureen / Blackburn, Brent / Bunting, Stuart / Hadváry, Paul / Hürzeler Müller, Marianne / Knopp, Dietmar / Levet-Trafit, Bernard / Lipari, M. Terry et al. | 1996
3148
Structure−Activity Relationships of (E)-3-(1,4-Benzoquinonyl)-2-[(3-pyridyl)- alkyl]-2-propenoic Acid Derivatives That Inhibit Both 5-Lipoxygenase and Thromboxane A2Synthetase
Hibi, Shigeki / Okamoto, Yasushi / Tagami, Katsuya / Numata, Hirotoshi / Kobayashi, Naoki / Shinoda, Masanobu / Kawahara, Tetsuya / Harada, Koukichi / Miyamoto, Kaname / Yamatsu, Isao | 1996
3158
Mercaptoacyl Dipeptides as Orally Active Dual Inhibitors of Angiotensin-Converting Enzyme and Neutral Endopeptidase
Fink, Cynthia A. / Carlson, J. Eric / McTaggart, Patricia A. / Qiao, Ying / Webb, Randy / Chatelain, Ricardo / Jeng, Arco Y. / Trapani, Angelo J. | 1996
3169
Synthesis and Characterization of Pseudopeptide Bradykinin B2 Receptor Antagonists Containing the 1,3,8-Triazaspiro[4.5]decan-4-one Ring System
Mavunkel, Babu J. / Lu, Zhijian / Goehring, R. Richard / Lu, Songfeng / Chakravarty, Sarvajit / Perumattam, John / Novotny, Elizabeth A. / Connolly, Maureen / Valentine, Heather / Kyle, Donald J. | 1996
3174
Synthesis and Biological Activity of NK-1 Selective, N-Backbone Cyclic Analogs of the C-Terminal Hexapeptide of Substance P
Byk, Gerardo / Halle, David / Zeltser, Irena / Bitan, Gal / Selinger, Zvi / Gilon, Chaim | 1996
3179
Aryl 1-But-3-ynyl-4-phenyl-1,2,3,6-tetrahydropyridines as Potential Antipsychotic Agents:  Synthesis and Structure−Activity Relationships
Glase, Shelly A. / Akunne, Hyacinth C. / Heffner, Thomas G. / Jaen, Juan C. / MacKenzie, Robert G. / Meltzer, Leonard T. / Pugsley, Thomas A. / Smith, Sarah J. / Wise, Lawrence D. | 1996
3188
A New Highly Selective Metabotropic Excitatory Amino Acid Agonist:  2-Amino-4-(3-hydroxy-5-methylisoxazol-4-yl)butyric Acid
Bräuner-Osborne, Hans / Sløk, Frank A. / Skjærbæk, Niels / Ebert, Bjarke / Sekiyama, Naohiro / Nakanishi, Shigetada / Krogsgaard-Larsen, Povl | 1996
3195
1-Aryl-4-((1-tetralinyl)alkyl)piperazines: Alkylamido and Alkylamino Derivatives. Synthesis, 5-HT1A Receptor Affinity, and Selectivity. 3
Perrone, Roberto / Berardi, Francesco / Leopoldo, Marcello / Tortorella, Vincenzo / Fornaretto, Maria Gioia / Caccia, Carla / McArthur, Robert A. | 1996
3195
1-Aryl-4-[(1-tetralinyl)alkyl]piperazines:  Alkylamido and Alkylamino Derivatives. Synthesis, 5-HT1AReceptor Affinity, and Selectivity. 31
Perrone, Roberto / Berardi, Francesco / Leopoldo, Marcello / Tortorella, Vincenzo / Fornaretto, Maria Gioia / Caccia, Carla / McArthur, Robert A. | 1996
3203
Aza-Peptide Analogs as Potent Human Immunodeficiency Virus Type-1 Protease Inhibitors with Oral Bioavailability
Fässler, Alexander / Bold, Guido / Capraro, Hans-Georg / Cozens, Robert / Mestan, Jürgen / Poncioni, Bernard / Rösel, Johannes / Tintelnot-Blomley, Marina / Lang, Marc | 1996
3217
Synthesis and Biological Evaluation of Certain Alkenyldiarylmethanes as Anti-HIV-1 Agents Which Act as Non-Nucleoside Reverse Transcriptase Inhibitors
Cushman, Mark / Golebiewski, W. Marek / Graham, Lisa / Turpin, Jim A. / Rice, William G. / Fliakas-Boltz, Valerie / Buckheit, Robert W. | 1996
3228
2,4-Diamino-5-deaza-6-Substituted Pyrido[2,3-d]pyrimidine Antifolates as Potent and Selective Nonclassical Inhibitors of Dihydrofolate Reductases
Gangjee, Aleem / Vasudevan, Anil / Queener, Sherry F. / Kisliuk, Roy L. | 1996