Synthesis and Calcium Channel Antagonist Activity of New 1,4-Dihydropyridine Derivatives Containing Dichloroimidazolyl Substituents (English)
- New search for: Amini, M.
- New search for: Golabchifar, A. A.
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- New search for: Shafiee, A.
- New search for: Amini, M.
- New search for: Golabchifar, A. A.
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In:
ARZNEIMITTEL FORSCHUNG
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52
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21-26
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2002
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ISSN:
- Article (Journal) / Print
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Title:Synthesis and Calcium Channel Antagonist Activity of New 1,4-Dihydropyridine Derivatives Containing Dichloroimidazolyl Substituents
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Contributors:Amini, M. ( author ) / Golabchifar, A. A. ( author ) / Dehpour, A. R. ( author ) / Pirali, H. M. ( author ) / Shafiee, A. ( author )
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Published in:ARZNEIMITTEL FORSCHUNG ; 52 ; 21-26
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Publisher:
- New search for: EDITIO CANTOR GMBH
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Publication date:2002-01-01
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Size:6 pages
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ISSN:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 610.7
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Classification:
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Table of contents – Volume 52
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1
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Cholesterol-lowering Properties and Safety of ChitosanYlitalo, Ritva / Lehtinen, Saara / Wuolijoki, Erkki / Ylitalo, Pauli / Lehtimäki, Terho et al. | 2002
- 8
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Microbiological and Pharmaco-toxicological Profile of Nifuratel and its Favourable Risk/Benefit Ratio for the Treatment of Vulvo-vaginal Infections. A reviewMendling, Werner / Mailland, Federico et al. | 2002
- 14
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General Pharmacological Profile of the Novel Muscarinic Receptor Agonist SNI-2011, a Drug for Xerostomia in Sjögren’s Syndrome. 1st Communication: Effects on general behavior and central nervous systemArisawa, Hirohiko / Imai, Eiichi / Fujise, Nobuaki / Fukui, Kenji / Masunaga, Hiroaki et al. | 2002
- 14
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General Pharmacological Profile of the Novel Muscarinic Receptor Agonist SNI-2011, a Drug for Xerostomia in Sjogren's Syndrome / 1st Communication: Effects on general behaviour and central nervous systemArisawa, H. / Imai, E. / Fujise, N. / Fukui, K. / Masunaga, H. et al. | 2002
- 21
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Synthesis and Calcium Channel Antagonist Activity of New 1,4-Dihydropyridine Derivatives Containing Dichloroimidazolyl SubstituentsAmini, Mohsen / Golabchifar, Ali A. / Dehpour, Ahmad R. / Pirali, Hamedani M. / Abbas, Shafieea et al. | 2002
- 27
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Synthesis, Enantioseparation and Pharmacological Activity of 4-Aryl-7,7-dimethyl-5-oxo-1,2,3,4,5,6,7,8-octahydroquinazoline-2-thionesYarim, Mine / Saraç, Selma / Ertan, Mevlüt / Kiliç, F. Sultan / Erol, Kevser et al. | 2002
- 34
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Effect of Troglitazone on Endothelial Function in Type 2 Diabetic PatientsTakase, Hiroyuki / Hakamata, Mutsumi / Toriyama, Takayuki / Hayashi, Kunihiko / Gotoa, Takatoshi / Sato, Koichi / Ueda, Ryuzo / Dohi, Yasuaki et al. | 2002
- 39
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Synthesis of Some New Diaryl and Triaryl Hydrazone Derivatives as Possible Estrogen Receptor ModulatorsPandey, Jaya / Pal, Rekha / Dwivedi, Anila / Hajela, Kanchan et al. | 2002
- 45
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Effects on Mycobacterium avium Replication in Normal Human Macrophages by Deferiprone (L1) and Other Iron Chelators. Possible implications on toxicityDouvas, George S. / May, Mary H. / Kolnagou, Annita / Kontoghiorghes, George J. et al. | 2002
- 53
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The Pharma Market as Reflected by Patents. Information for Marketing and Scientific WorkHabernickel, Valentin J. et al. | 2002
- 53
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The Pharma Market as Reflected by Patents / Agents for the treatment of cancer and tumors / Agents for the treatment of glaucoma and elevated intraocular pressureHabernickel, V. J. et al. | 2002
- 57
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Book Reviews| 2002
- 60
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Lekteplase — a Secreted Tissue Plasminogen Activator Derivative from Escherichia coliManosroi, Jiradey / Tayapiwatana, Chatchai / Manosroi, Aranya / Beer, Jürgen / Bergemann, Klaus / Werner, Rolf Günter et al. | 2002
- 67
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Detection of Isolated Mistletoe Lectin Chains in Plant ExtractsTonevitsky, Alexander G. / Marx, Uwe / Agapov, Igor / Moisenovich, Mikhail et al. | 2002
- 73
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Comparing beta-Blockers and their Relevance in the Pharmacotherapy of Cardiovascular DiseasesWehling, M. et al. | 2002
- 73
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β-Blocker und ihre Bedeutung für die Pharmakotherapie kardiovaskulärer Erkrankungen im VergleichWehling, Martin et al. | 2002
- 81
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General Pharmacological Profile of the Novel Muscarinic Receptor Agonist SNI-2011, a Drug for Xerostomia in Sjögren’s Syndrome. 2nd Communication: Effects on somatic nervous system and on autonomic nervous system and smooth muscle1)Arisawa, Hirohiko / Fukui, Kenji / Fujise, Nobuaki / Masunaga, Hiroaki et al. | 2002
- 81
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General Pharmacological Profile of the Novel Muscarinic Receptor Agonist SNI-2011, a Drug for Xerostomia in Sjogren's Syndrome / 2nd Communication: Effects on somatic nervous system and on autonomic nervous system and smooth muscleArisawa, H. / Fukui, K. / Fujise, N. / Masunaga, H. et al. | 2002
- 89
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Quantification of Procyanidins in Oral Herbal Medicinal Products Containing Extracts of Crataegus SpeciesWittig, Jörg / Leipolz, Ingrid / Graefe, Eva Ulrike / Jaki, Birgit / Treutter, Dieter / Veit, Markus et al. | 2002
- 97
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Effects of Antihistamines on Leukotriene and Cytokine Release from Dispersed Nasal Polyp CellsKüsters, Sabine / Schuligoi, Rufina / Hüttenbrink, Karl-Bernd / Rudert, Jutta / Wachs, Angela / Szelenyi, Istvan / Peskar, Bernhard A. et al. | 2002
- 103
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Synthesis and Antitumour Evaluation of 4-Bromophenyl SemicarbazonesPandeya, Surendra N. / Yogeeswari, Perumal / Sausville, Edward A. / Mauger, Anthony B. / Narayanan, Ven L. et al. | 2002
- 109
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Effects of Sub-minimum Inhibitory Concentrations of Gatifloxacin on the Inhibition Staphylococcus aureus and Escherichia coli AdherenceBraga, P. C. / Dal Sasso, M. et al. | 2002
- 109
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Effects of Sub-minimum Inhibitory Concentrations of Gatifloxacin on the Inhibition of Staphylococcus aureus and Escherichia coli AdherenceBraga, Pier Carlo / Sasso, Monica Dal et al. | 2002
- 113
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Anti-Mycobacterium tuberculosis Agents Derived from Quinoxaline-2-carbonitrile and Quinoxaline-2-carbonitrile 1,4-di-N-oxideOrtega, Miguel AÁngel / Sainz, Yolanda / Montoya, Marŕıa Elena / Jaso, Andreés / Zarranz, Beleén / Aldana, Ignacio / Monge, Antonio et al. | 2002
- 120
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Synthetic Derivatives of Curcumin and their Activity against Leishmania amazonensisGomes, Denise de C. F. / Alegrio, Leila Vilela / Lim, Marco Edilson Freire de / Leon, Leonor L. / Araújo, Catarina A. C. et al. | 2002
- 125
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From the Manual Method of Topliss to a Modified Quantitative MethodYunesa, Rosendo A. / Heinzena, Vilma E. Fonseca / Filhob, Valdir Cechinel / Lazzarottoa, Marcelo et al. | 2002
- 133
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The Pharma Market as Reflected by Patents / Agents for the treatment of anxiety and depression / Agents for the treatment of e.g. cognitive disorders / Compounds having antibacterial activity / Agents for the treatment of thromboembolic disordersHabernickel, V. J. et al. | 2002
- 140
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BioRegioN – Biotechnology in Lower Saxony| 2002
- 145
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Physiologische und therapeutische Bedeutung von Serotonin und des serotoninergen SystemsMolderings, Gerhard J. et al. | 2002
- 145
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Physiological and Therapeutic Relevance of Serotonin and the Serotonergic SystemMolderings, G. J. et al. | 2002
- 155
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Interaction Potential of Lercanidipine, a New Vasoselective Dihydropyridine Calcium AntagonistKlotz, Ulrich et al. | 2002
- 162
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General Pharmacological Profile of the Novel Muscarinic Receptor Agonist SNI-2011, a Drug for Xerostomia in Sjogren's Syndrome / 3rd Communication: Effects on respiratory and cardiovascular systemsArisawa, H. / Fukui, K. / Masunaga, H. et al. | 2002
- 162
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General Pharmacological Profile of the Novel Muscarinic Receptor Agonist SNI-2011, a Drug for Xerostomia in Sjögren’s Syndrome. 3rd Communication: Effects on respiratory and cardiovascular systems1)Arisawa, Hirohiko / Fukui, Kenji / Masunaga, Hiroaki et al. | 2002
- 168
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Neuroprotective Activity of a Nanoparticulate Formulation of the GlycineB Site Antagonist MRZ 2/576 in Transient Focal Ischaemia in RatsSopala, Monika / Schweizer, Steffen / Schäfer, Nicole / Nürnberg, Eberhard / Kreuter, Jörg / Seiller, Erhard / Danysz, Wojciech et al. | 2002
- 175
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Study of the Novel Non-xanthine Heterocyclic Compound GU285 as a Potent Non-selective Adenosine Receptor Antagonist in the RatHarden, Fiona A. / Brown, Lindsay / Quinn, Ronald J. / Harrison, Glenn J. / Headrick, John P. / Rose’Meyer, Roselyn B. / Willis, Roger J. et al. | 2002
- 182
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Evaluation of the Bioequivalence and Pharmacokinetics of Two Tablet Formulations of Isosorbide-5-mononitrate after Single Oral Administration in Healthy VolunteersNiopas, Ioannis / Daftsios, Athanasios C. / Nikolaidis, Nicolaos et al. | 2002
- 187
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Pharmacokinetic Behaviour of Antithrombin III Following Intravenous Infusion in Healthy VolunteersMarzo, Antonio / Ceppi-Monti, Nunzia / Giusti, Andrea / Abbiati, Gianalfredo / Maddalena, Parenti et al. | 2002
- 194
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Local Anaesthetic Properties of Ambroxol Hydrochloride Lozenges in View of Sore Throat. Clinical proof of conceptSchutz, Alexander / Gund, Hans-Jürgen / Pschorn, Uwe / Aicher, Bernhard / Peil, Hubertus / Müller, Achim / Mey, Christian de / Gillissen, Adrian et al. | 2002
- 200
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Randomised Crossover Studies of the Bioequivalence of Two Fenofibrate Formulations after Administration of a Single Oral Dose in Healthy VolunteersSonet, Bernard / Vanderbist, Francis / Streel, Bruno / Houin, Georges et al. | 2002
- 205
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Nitric Oxide Release from Coumarin 4-Carboxamidoximes in the Presence of ThiolsKontogiorgis, Christos A. / Hadjipavlou-Litina, Dimitra J. et al. | 2002
- 211
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Erfassung von Arzneimittel-assoziierten Schädigungen an der Schleimhaut des oberen Intestinaltraktes. Zum Problem einer Charakterisierung des Gesundheitsstatus gesunder ProbandenWildgrube, Hans Jörg / Kierschke, Gerd / Weigmann, Ingo / Terhaag, Bernd et al. | 2002
- 211
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Registration of Drug-associated Lesions at the Mucosa of the Upper Gastrointestinal Tract / The problem of the characterisation of the health status of healthy volunteersWildgrube, H. J. / Kierschke, G. / Weigmann, I. / Terhaag, B. et al. | 2002
- 219
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The Pharma Market as Reflected by Patents / Cardiac agents / Antimalarial agents / AnalgesicsHabernickel, V. J. et al. | 2002
- 225
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General Pharmacological Profile of the Novel Muscarinic Receptor Agonist SNI-2011, a Drug for Xerostomia in Sjogren's Syndrome / 4th Communication: Effects on gastrointestinal, urinary and reproductive systems and other effectsArisawa, H. / Fukui, K. / Imai, E. / Fujise, N. / Masunaga, H. et al. | 2002
- 225
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General Pharmacological Profile of the Novel Muscarinic Receptor Agonist SNI-2011, a Drug for Xerostomia in Sjögren’s Syndrome. 4th Communication: Effects on gastrointestinal, urinary and reproductive systems and other effects1)Arisawa, Hirohiko / Fukui, Kenji / Imai, Eiichi / Fujise, Nobuaki / Masunaga, Hiroaki et al. | 2002
- 233
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Pharmacokinetic and Pharmacodynamic Comparative Study of Zofenopril and Enalapril in Healthy VolunteersMarzo, Antonio / Bo, Lorenzo Dal / Mazzucchelli, Paolo / Monti, Nunzia Ceppi / Crivelli, Fabrizio / Ismaili, Shevqet / Giusti, Andrea / Uhr, Mario Richard et al. | 2002
- 243
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Efficacy and Safety of a Butcher’s Broom Preparation (Ruscus aculeatus L. Extract) Compared to Placebo in Patients Suffering from Chronic Venous InsufficiencyVanscheidt, Wolfgang / Jost, Volker / Wolna, Peter / Lücker, Peter W. / Müller, Alfred / Theurer, Christoph / Patz, Brigitte / Grützner, Karen I. et al. | 2002
- 251
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Clinical Efficacy of Pitavastatin, a New 3-Hydroxy-3-methylglutaryl Coenzyme A Reductase Inhibitor, in Patients with Hyperlipidemia. Dose-finding study using the double-blind, three-group parallel comparisonSaito, Yasushi / Yamada, Nobuhiro / Teramoto, Tamio / Itakura, Hiroshige / Hata, Yoshiya / Nakaya, Noriaki / Mabuchi, Hiroshi / Tushima, Motoo / Sasaki, Jun / Goto, Yuichiro et al. | 2002
- 256
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Efficacy and Tolerability of Ambroxol Hydrochloride Lozenges in Sore Throat. Randomised, double-blind, placebo-controlled trials regarding the local anaesthetic propertiesFischer, Jürgen / Pschorn, Uwe / Vix, Jean-Michel / Peil, Hubertus / Aicher, Bernhard / Müller, Achim / Mey, Christian de et al. | 2002
- 264
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Application of Quantifying Scoring Systems for the Determination of Changes of the Mucosa of the Upper Gastrointestinal Tract / A comparative study of a diclofenac effervescent tablet with conventional diclofenac preparations and acetylsalicyclic acid after repeated administrationWildgrube, H. J. / Kierschke, G. / Nowak, H. / Weigmann, I. / Terhaag, B. et al. | 2002
- 264
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Einsatz quantifizierender Scoring-Systeme zur Ermittlung von Schleimhautveränderungen des oberen Gastrointestinaltraktes. Vergleichende Untersuchung einer Diclofenac-Brausetablette, konventioneller Diclofenac-Zubereitungen sowie von Acetylsalicylsäure nach wiederholter AnwendungWildgrube, Hans Jörg / Kierschke, Gerd / Nowak, Horst / Weigmann, Ingo / Terhaag, Bernd et al. | 2002
- 273
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Synthesis, Biological Activity and Molecular Modeling Studies of 1,2,3,4-Tetrahydroiso-quinoline Derivatives as Conformationally Constrained Analogues of KN62, a Potent Antagonist of the P2X7-Receptor Containing a Tyrosine MoietyBaraldi, Pier Giovanni / Makaeva, Rimma / Pavani, Maria Giovanna / Nuñez, Maria del Carmen / Spalluto, Giampiero / Moro, Stefano / Falzoni, Simonetta / Virgilio, Francesco Di / Romagnoli, Romeo et al. | 2002
- 286
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Syntheses, Antibacterial, Cytotoxic and Antifungal Effects of New 3-Carboxy-1-phenacylpyridinium SaltsKhan, Khalid Mohammed / Saify, Zafar Saeed / Shah, Syed Tasadaque Ali / Ahmed, Mansoor / Saeed, Muhammad / Hayat, Safdar / Abbas, Muhammad / Voelter, Wolfgang et al. | 2002
- 294
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Effect of Combined Chemotherapy and Anti-inflammatory Drugs on Murine SchistosomiasisMahmoud, Madiha R. / Zoheiry, Mona M. K. / Nosseir, Mona M. F. et al. | 2002
- 302
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The Pharma Market as Reflected by Patents / Cytostatics / Agents for the Treatment of Prostatic HyperplasiaHabernickel, V. J. et al. | 2002
- 353
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Influence of Inhibition of Adenosine Uptake on the gamma-Aminobutyric Acid Level of the Ischemic Rat BrainSeif-El-Nasr, M. / Khattab, M. et al. | 2002
- 353
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Influence of Inhibition of Adenosine Uptake on the γ-Aminobutyric Acid Level of the Ischemic Rat BrainSeif-El-Nasr, Mona / Khattab, Mahmoud et al. | 2002
- 358
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Inhibitory Effects of Alprostadil (Prostaglandin E1) Incorporated in Lipid Microspheres of Soybean Oil on Intimal Hyperplasia Following Balloon Injury in RabbitsKunihara, Mineo / Tsuchida, Katsuharu / Kaneko, Katsuyoshi / Suga, Hiroyuki / Hasegawa, Tomohiko / Mochizuki, Saeri / Kawai, Keiko / Shiga, Atsushi / Yamaguchi, Tatsuya et al. | 2002
- 365
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The Effects of Calcium Channel Antagonists on Coronary Nitrite Outflow in Isolated Rat HeartDjuric, Dragan / Mitrovic, Veselin / Jakovljevic, Vladimir et al. | 2002
- 371
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In vitro and in vivo Equivalence of Two Oral Atenolol Tablet FormulationsCuadrado, Antonio / Gascón, Alicia Rodríguez / Hernández, Rosa María / Castilla, Ana María / Maza, Ane de la / Ocáriz, Alici López de / Calvo, Begoña / Pedraz, José Luis et al. | 2002
- 379
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Prospective Controlled Trial of Two Nifedipine Extended Release Formulations in the Treatment of Essential HypertensionPivac, Nediljko / Naranća, Mario / Vujic-Podlipec, Dunja / Bagatin, Jugoslav / Rumboldt, Zvonko et al. | 2002
- 385
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Studies of Piroxicam Absorption by Oral MucosaDiez-Ortego, Irene / Cruz, Margarida / Largo, Raquel / Navarro, Antonio / Palacios, Itziar / Solans, Ana / Sanchez-Pernaute, Olga / Egido, Jesús / Herrero-Beaumont, Gabriel et al. | 2002
- 388
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Synthesis and Evaluation of Anticancer Activity of Some Imidazothiazolyl, Imidazobenzothiazolyl and Dihydroimidazothiazolyl CoumarinsSrimanth, Kagne / Rao, Vedula Rajeswar / Krishna, Devarakonda R. et al. | 2002
- 393
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In vitro Antiviral Activity of Aphidicolin and its Derivates. Synergistic effects of aphidicolin with other antiviral drugsMichaelis, Martin / Langer, Klaus / Vogel, Jens-Uwe / Kreuter, Jörg / Rabenau, Holger / Doerr, Hans-Wilhelm / Cinatl, Jindrich et al. | 2002
- 400
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Effect of Chloroquine on Glucose MetabolismGaafar, Khadiga M. / Khedr, Mona I. / Bashandy, Samir A. / Sharaf, Olaa A. / El-Zayat, Salwa R. et al. | 2002
- 407
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Bioequivalence Evaluation of a Fixed Combination of Chloroquine and Proguanil in a Capsule Formulation versus a Standard MedicationChaulet, Jean Franćois / Nony, Patrice / Bévalot, Fabien / Girard, Pascal / Chabaud, Sylvie / Mounier, Cyril / Clair, Pascal / Boissel, Jean Pierre / Grelaud, Gilles et al. | 2002
- 413
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The Pharma Market as Reflected by Patents / Antidiabetic Agents / AntidepressantsHabernickel, V. J. et al. | 2002
- 423
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From Toxic Precursors to Safe Drugs. Mechanisms and relevance of idiosyncratic drug reactionsPetersen, Karl-Uwe et al. | 2002
- 430
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Pharmacokinetics of Pipamperone from Three Different Tablet FormulationsPotgieter, Gerbrecht E. / Groenewoud, Gerhard / Jordaan, Pierre J. / Hundt, Hans K. L. / Schall, Robert / Kummer, Michael / Sewarte-Ross, Günter et al. | 2002
- 435
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Effects on the Reactive Oxygen Species of Erdosteine and its Metabolite in vitroHosoe, Hisashi / Kaise, Toshihiko / Ohmori, Kenji et al. | 2002
- 441
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Mechanism of the Antitussive Effect of Azelastine in Guinea PigsIto, Nobuaki / Shioya, Takanobu / Watanabe, Akiko / Sano, Masaaki / Sasaki, Masahiro / Miura, Mamoru et al. | 2002
- 448
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Synthesis and Activity of Phenyl Derivatives Containing 5,6-Dimethylthieno[2,3-d]pyrimidin-4(1H)-one or 4H-Pyrimido [5,4-b] indol-4-one Heterocyclic System as Potential Non-steroidal Anti-inflammatory DrugsSantagati, Andrea / Granata, Giuseppe / Santagati, Maria / Cutuli, Vincenza / Mangano, Nunzio Guido / Caruso, Antonina et al. | 2002
- 455
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Studies on New Cyclic Imides Obtained from Aminophenazone with Analgesic Properties / Potent effects of a 3,4-dichlormaleimide derivativede Campos, F. / Correa, R. / de Souza, M. M. / Yunes, R. A. / Nunes, R. J. / Cechinel-Filho, V. et al. | 2002
- 455
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Studies on New Cyclic Imides Obtained from Aminophenazone with Analgesic Properties. Potent effects of a 3,4-dichloromaleimide derivativeCampos, Fátima de / Corrêa, Rogério / Souza, Márcia Maria de / Yunes, Rosendo Augusto / Nunes, Ricardo José / Cechinel-Filho, Valdir et al. | 2002
- 462
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Evaluation of the Analgesic and Anti-inflammatory Activities of Some Thiazolo[4,5-d]pyrimidinesBalkan, Ayla / Gören, Zafer / Urgun, Hüsne / Çalιş, Ünsal / Çakar, A. Nur / Atilla, Pergin / Uzbay, Tayfun et al. | 2002
- 468
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Effects of Gold-Chloroquine Complexes on Respiratory Burst of Polymorphonuclear LeukocytesNavarro, Maribel / Vásquez, Flor / Velásquez, Mait / Medina, Rafael / Reggio, Ronald / Fraile, German et al. | 2002
- 475
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Synthesis and Antitumour Activity of a Series of Cyclic Amidines of 2,3-Dihydro-1H-1,5-benzodiazepinesJančienė, Regina / Kosychova, Lidija / Bukelskienė, Virginija / Domkus, Vigintas / Stumbrevičiūtė, Zita / Ragalevičienè, Vida / Puodžiūnaitè, Benedikta D. et al. | 2002
- 482
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Synthesis and Antimalarial Activity of Substituted Pyrazole DerivativesDomínguez, José N. / Charris, Jaime E. / Caparelli, Mario / Riggione, Flavia et al. | 2002
- 489
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Effects of Amidine Derivatives on Parasite-Macrophage Interaction and Evaluation of ToxicityTemporal, Rosane M. / Cysne-Finkelstein, Léa / Echevarria, Aurea / Souza, Marco A. S. de / Sertã, Mônica / Silva-Gonçalves, Antônio J. da / Pirmez, Claude / Leon, Lenor L. et al. | 2002
- 494
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The Pharma Market as Reflected by Patents / Antitumor Agents / Neuroprotective AgentsHabernickel, V. J. et al. | 2002
- 500
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Comparison between the Mechanisms of Action of Plant Toxins Ricin and Viscumin on the Stage of Intracellular DissociationTonevitsky, Alexander / Agapov, Igor / Chelnokova, Olga / Moisenovich, Mikhail / Marx, Uwe et al. | 2002
- 507
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Meta-analysis of Flecainide Safety in Patients with Supraventricular ArrhythmiasWehling, Martin et al. | 2002
- 515
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Local Treatment of Hemorrhoidal Disease and Perianal Eczema. Meta-analysis of the efficacy and safety of an Escherichia coli culture suspension alone or in combination with hydrocortisoneWienert, Volker / Heusinger, Jörg H. et al. | 2002
- 524
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Reproductive Toxicity of γ-Ethyl-γ-phenyl-butyrolactone, a New Anticonvulsant and Hypnotic Drug, in Mice. Fertility and peri- and post-natal studiesChamorro, Germán / Vega, Fernando / Madrigal, Eduardo / Salazar, María et al. | 2002
- 529
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A Randomised, Placebo-controlled Study Comparing Two Formulations of Dimenhydrinate with Respect to Efficacy in Motion Sickness and SedationSeibel, Klaus / Schaffler, Klaus / Reitmeir, Peter et al. | 2002
- 537
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Synthesis and Calcium Channel Antagonist Activity of 1,4-Dihydropyridine Derivatives Containing 4-Nitroimidazolyl SubstituentsShaflee, Abbas / Rastkary, Noushin / Jorjani, Masoumeh et al. | 2002
- 543
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Studies on the Cardiotoxicity of Noradrenaline in Isolated Rabbit HeartsRump, Alexis F. E. / Schierholz, Jörg / Klaus, Wolfgang et al. | 2002
- 552
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Haemodynamic and Metabolic Effects of Low Daily Dose Sulphonylureas in Diabetic Dog HeartsPósa, Ildikó / Kocsis, Erzsébet / Nieszner, Éva / Pogátsa, Gábor / Koltai, Mária Zsófia et al. | 2002
- 560
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HPLC Method for the Determination of Rosiglitazone in Human Plasma and its Application in a Clinical Pharmacokinetic StudyMamidi, Rao N. V. S. / Chaluvadi, Madhusudana R. / Benjamin, Biju / Ramesh, Mullangi / Katneni, Kasiram / Babu, Aravinda P. / Bhanduri, Jaydip / Rao, Naidu M. U. / Rajagopalan, Ramanujam et al. | 2002
- 565
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Synthesis and Antituberculosis Activity of Cycloalkylidenehydrazide and 4-Aza-1-thiaspiro [4.5] decan-3-one Derivatives of Imidazo [2][1-b]thiazoleUlusoy, Nuray et al. | 2002
- 572
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Synthesis and Antifungal and Antioxidant Properties of some New 5-Substituted-4-amino(or aryl)-3-mercapto-4(H)-1,2,4-triazolesMarakos, Panagiotis / Papakonstantinou-Garoufalias, Spyroula / Tani, Ekaterini / Kourounakis, Panos N. / Athanasiou, George / Chytyroglou-Lada, Aikaterini et al. | 2002
- 583
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Mode of Action of Gabapentin in Chronic Neuropathic Pain Syndromes. A short review about its cellular mechanisms in nociceptive neurotransmissionSurges, Rainer / Feuerstein, Thomas J. et al. | 2002
- 587
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Disposition of TAK-044, a New Endothelin Antagonist, in Rats and DogsMaeshiba, Yoshihiro / Takeuchi, Toshiyuki / Kondo, Takahiro / Yamashita, Kenji / Tsukuda, Ryoichi / Yoshimura, Yoshinobu et al. | 2002
- 593
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Preformulation Approaches to Improve the Oral Bioavailability of Two Novel Piperidine Renin Inhibitors in DogBittner, Beate / Chou, Ruby / Schleimer, Michael / Morgenroth, Brita / Zell, Manfred / Lavé, Thierry et al. | 2002
- 600
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Effects of Anti-ulcer Agents on Ethanol-induced Gastric Mucosal Lesions in D-Galactosamine-induced Hepatitis RatsTaniguchi, Hiroyuki / Yomota, Eiji / Nogi, Koji / Onoda, Yuichi et al. | 2002
- 605
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Study of the Insulinotropic Effect of the Novel Antihyperglycemic Agent KAD-1229 Using HIT T15 Cells, a Hamster’s Insulinoma Cell LineIchikawa, Kiyoshi / Yamato, Tokuhisa / Tsuji, Atsutoshi / Ojima, Kazuma / Kusama, Hiroshi / Kojima, Masami et al. | 2002
- 610
-
Effects of the Lipoprotein Lipase Activator NO-1886 as a Suppressor Agent of Atherosclerosis in Aorta of Mild Diabetic RabbitsYin, Weidong / Tsutsumi, Kazuhiko / Yuan, Zhonghua / Yang, Baotang et al. | 2002
- 615
-
Vergleichende Pharmakokinetik von Progesteron-Kapseln und einem Progesteron-Gel nach vaginaler AnwendungKleinstein, Jürgen / Schlegelmilch, Ronald / Mazur, Dago / Vens-Cappell, Bernd et al. | 2002
- 622
-
Verminderung der Rezidivhäufigkeit bei Patienten mit chronisch rezidivierender hypertrophischer Sinusitis unter Behandlung mit einem bakteriellen Immunstimulans (Enterococcus faecalis-Bakterien humaner Herkunft)Habermann, Werner / Zimmermann, Kurt / Skarabis, Horst / Kunze, Rudolf / Rusch, Volker et al. | 2002
- 628
-
Syntheses and Stability Studies of Some Mannich Bases of Acetophenones and Evaluation of their Cytotoxicity against Jurkat CellsGul, Halise Inci / Gul, Mustafa / Erciyas, Ercin et al. | 2002
- 636
-
Effect of Fluconazole on the Fertility of Male RabbitsEl-Medany, Azza H. / Hagar, Hanan H. et al. | 2002
- 649
-
Principles of a Topical Chemosensory Receptor Intervention. The basis for a chemosensory CNS medicineLiedtke, Rainer K. et al. | 2002
- 654
-
Synthesis and β1-, β2-Adrenergic Receptor Binding Studies of 4-Acylaminosubstituted Phenoxypropanolamine and 5-Acylamino-substituted Naphthyloxypropanolamine DerivativesJindal, Dharam Paul / Coumar, Mohane S. / Bruni, Giancarlo / Massarelli, Paola et al. | 2002
- 664
-
Pharmacokinetic Interaction between TAK-044, a New Endothelin Antagonist, and Ciclosporin in RatsMaeshiba, Yoshihiro / Yamashita, Kenji / Tsukuda, Ryoichi / Yoshimura, Yoshinobu et al. | 2002
- 669
-
Human Neutrophil Oxidative Bursts and their in vitro Modulation by Different N-Acetylcysteine ConcentrationsAllegra, Luigi / Sasso, Monica Dal / Bovio, Cinzia / Massoni, Carola / Fonti, Elena / Braga, Pier Carlo et al. | 2002
- 677
-
Volume Independent Stimulation of Renin Secretion by a Single Dose of Amiloride in ManEndemann, Dierk / Marienhagen, Jörg / Stubanus, Mike / Luger, Rainer J. / Fischereder, Michael / Riegger, Günter A. J. / Krämer, Bernhard K. et al. | 2002
- 684
-
Improvement of the Bioavailability of Colchicine in Rats by Co-administration of D-α-Tocopherol Polyethylene Glycol 1000 Succinate and a Polyethoxylated Derivative of 12-Hydroxy-Stearic AcidBittner, Beate / Guenzi, Alberto / Fullhardt, Pascal / Zuercher, Gerhard / González, Roberto Carlos Bravo / Mountfield, Richard Jolyon et al. | 2002
- 689
-
Effects of Lerisetron, a New 5-HT3 Receptor Antagonist, on Ipecacuanha- induced Emesis in Healthy VolunteersCooper, Mark / Sologuren, Ander / Valiente, Roman / Smith, Jeffery et al. | 2002
- 695
-
Total Synthesis and Anti-leishmanial Activity of Some Curcumin AnaloguesGomes, Denise de Castro Ferreira / Alegrioa, Leila Vilela / Leon, Leonor L. / Limaa, Marco Edilson Freire de et al. | 2002
- 699
-
Antimicrobial Activity of Dequalinium Chloride against Leading Germs of Vaginal InfectionsCasa, Vera Della / Noll, Harald / Gonser, Susanne / Grob, Philipp / Graf, Federico / Pohlig, Gabriele et al. | 2002
- 706
-
Local Treatment of Vaginal Infections of Varying Etiology with Dequalinium Chloride or Povidone Iodine. A randomised, double-blind, active-controlled, multicentric clinical studyPetersen, Eiko E. / Weissenbacher, Ernst R. / Hengst, Peter / Spitzbart, Heinz / Wolfgang, Weise / Wolff, Friedrich / Dreher, Ekkehard / Ernst, Uwe / Casa, Vera Della / Pohlig, Gabriele et al. | 2002
- 716
-
Studies of Interferences of Apomorphine and its Metabolites or Decomposition Products with Immunochemical Screening Tests for Legal and Illicit Drugs after Therapeutic Doses of ApomorphineSchütz, Harald / Erdmann, Freidoon / Riße, Manfred / Weiler, Günter et al. | 2002
- 725
-
Clinical Effects of Nifuratel in Vulvovaginal Infections. A meta-analysis of metronidazole-controlled trialsMendling, Werner / Poli, Aldo / Magnani, Paola et al. | 2002
- 731
-
Structure-Activity Relationships Investigation in a Mixed Series of Cannabinoids. An electronic-topological approachKandemirli, Fatma et al. | 2002
- 740
-
Cerebral Blood Perfusion after Treatment with Zolpidem and Flumazenil in the BaboonClauss, Ralf P. / Dormehl, Irene C. / Kilian, Elmaré / Louw, Werner K.A. / Nel, Wally H. / Oliver, Douglas W. et al. | 2002
- 745
-
Metabolic Fate of Pitavastatin (NK-104), a New Inhibitor of 3-Hydroxy-3-methylglutaryl Coenzyme A Reductase / Effects on drug-metabolizing systems in rats and humansFujino, H. / Yamada, I. / Shimada, S. / Nagao, T. / Yoneda, M. et al. | 2002
- 745
-
Metabolic Fate of Pitavastatin (NK-104), a New Inhibitor of 3-Hydroxy-3-methyllutaryl Coenzyme A Reductase. Effects on drug-metabolizing systems in rats and humansFujino, Hideki / Yamada, Iwao / Shimada, Syunsuke / Nagao, Takeshi / Yoneda, Michiaki et al. | 2002
- 754
-
High-Performance Liquid Chromatographic Determination of Oxatomide and its Metabolite and its Application to Pharmacokinetic Study in Rat PlasmaKikuchi, Kazuo / Ohishi, Takayoshi / Masuike, Taketoshi / Ohmori, Kenji / Sakai, Kenichi et al. | 2002
- 764
-
Study on the Usefulness of Seratrodast in the Treatment of Chronic Pulmonary EmphysemaHoriguchi, Takahiko / Tachikawa, Soichi / Kondo, Rieko / Shiga, Mamoru / Hirose, Masahiro / Fukumoto, Koji et al. | 2002
- 769
-
Paracetamol Metabolism in Indian PopulationPabba, Santosh K. / Bolla, Sambamurthy / Kandhagatla, Rajnarayana / Chaluvadi, Madhusudana R. / Krishna, Devarakonda R. et al. | 2002
- 773
-
Antimicrobial Evaluation of Some Mannich Bases of Acetophenones and Representative Quaternary DerivativesGul, Halise Inci / Denizci, A. Akin / Erciyas, Ercin et al. | 2002
- 778
-
Synthesis and Antimicrobial Activity Evaluation of Some New Adamantane DerivativesÜnsal, Çalısş / Yarıma, Mine / Köksala, Mericç / Özalpb, Meral et al. | 2002
- 782
-
The Pharma Market as Reflected by Patents / Fungicides / Agents for the treatment of diabetes / Agents for the treatment of asthma and related diseases / AnalgesicsHabernickel, V. J. et al. | 2002
- 787
-
Synthesis and Anticonvulsant Activity of 1-Acetyl-5-arylidenyl-3-(2’-oxo/thio-barbiturinyl) -2-pyrazolinesno surname, Archana / Srivastava, Virendra Kishor / Kumar, Ashok et al. | 2002
- 792
-
Synthesis and a~1-Adrenoceptor Antagonistic Activity of Some 4-Amino-5,7-dimethyl-2-(substituted) aminopyrido(2,3-d)pyrimidinesChhabria, M. T. / Srinivas, S. / Rajan, K. S. / Ravikumar, T. / Rathnam, S. et al. | 2002
- 792
-
Synthesis and α1-Adrenoceptor Antagonistic Activity of Some 4-Amino-5,7-dimethyl-2-(substituted) aminopyrido(2,3-d) pyrimidinesChhabria, Mahesh T. / Srinivas, Sreeramaiah / Rajan, Kombu S. / Ravikumar, Tadiparthy / Rathnam, Shivprakash et al. | 2002
- 797
-
Blood Pressure Lowering Effect of an Olive Leaf Extract (Olea europaea) in L-NAME Induced Hypertension in RatsKhayyal, M. T. / El-Ghazaly, M. A. / Abdallah, D. M. / Nassar, N. N. / Okpanyi, S. N. / Kreuter, M.-H. et al. | 2002
- 797
-
Blood Pressure Lowering Effect of an Olive Leaf Extract {Olea europaed) in L-NAME Induced Hypertension in RatsKhayyal, Mohamed T. / El-Ghazaly, Mona A. / Abdallah, Dalai M. / Nassar, Noha N. / Okpanyi, Samuel N. / Kreuter, Matthias-Heinrich et al. | 2002
- 803
-
Effects of Direct and Indirect Activation of G Protein of Adenylyl Cyclase on the Subsequent Response to ß-Adrenergic Receptor Agonists in Human TrachealisSudo, Yukio / Kume, Hiroaki / Ito, Satoru / Ito, Yasushi / Yamaki, Kenichi / Takagi, Kenzo et al. | 2002
- 803
-
Effects of Direct and Indirect Activation of G Protein of Adenylyl Cyclase on the Subsequent Response to beta-Adrenergic Receptor Agonists in Human TrachealisSudo, Y. / Kume, H. / Ito, S. / Ito, Y. / Yamaki, K. / Takagi, K. et al. | 2002
- 813
-
Evaluation of the Combined Effect of Pranlukast during High-dose Steroid InhalationHoriguchi, Takahiko / Tachikawa, Soichi / Kondo, Rieko / Miyazaki, Junichi / Sasaki, Yasushi / Banno, Kengo / Handa, Misuzu et al. | 2002
- 817
-
Synthesis, Spectral Studies and Antiinflammatory Activity of Glycolamide Esters of Niflumic Acid as Potential ProdrugsGadad, Andanappa K. / Bhat, Shailija / Tegeli, Varsha S. / Redasani, Vivek V. et al. | 2002
- 822
-
Tissue Absorption and Distribution of Ketoprofen after Patch Application in Subjects Undergoing Knee Arthroscopy or Endoscopic Carpal Ligament ReleaseOsterwalder, Andreas / Reiner, Valentina / Reiner, Giorgio / Lualdi, Paolo et al. | 2002
- 828
-
Effects of the Anti-ulcer Agents Ecabet Sodium, Cimetidine and Sucralfate on Acetylsalicylic Acid-induced Gastric Mucosal Damage Deteriorated by Renal Failure in RatsNogi, Koji / Taniguchi, Hiroyuki / Onoda, Yuichi et al. | 2002
- 833
-
Synthesis and Evaluation of Anti-HIV-1 and Anti-HSV-1 Activities of 4H-[1,2,4]-Triazolo [1,5-a]pyrimidin-5-one DerivativesAbdel-Hafez, Atef A. / Elsherief, Hosny A. H. / Jo, Michiko / Kurokawa, Masahiko / Shiraki, Kimiyasu / Kawahata, Takuya / Otake, Toru / Nakamura, Norio / Hattori, Masao et al. | 2002
- 840
-
Cytotoxic Activities of Some Mono and Bis Mannich Bases Derived from Acetophenone in Brine Shrimp BioassayGul, Halise Inci / Gul, Mustafa / Hänninen, Osmo et al. | 2002
- 844
-
Mediation of the Schistosomicidal Effect of Praziquantel through Nitric OxideAmmar, Elsayed M. / Said, Shehta A. / Eissa, Laila A. et al. | 2002
- 849
-
Agents for the treatment of viral infections / Agents for the treatment of tumor and cancer / Agents for the treatment of sexual dysfunction / Agents for the treatment of thromboembolic disordersHabernickel, V. J. et al. | 2002
- 857
-
Effects of Interleukin-11 on the Hematopoietic Action of Granulocyte Colony-stimulating FactorMomose, Kazuhiro / Taguchi, Katsunari / Saitoh, Minori / Yasuda, Shuhei / Miyata, Keiji et al. | 2002
- 863
-
Synthesis and Evaluation of Anticonvulsant Activities of Some Bis Mannich Bases and Corresponding PiperidinolsGul, Halise Inci / Calis, Unsal / Vepsalainen, Jouko et al. | 2002
- 870
-
Sufentanil-related Respiratory Depression and Antinociception in the Dog. Mediation by different receptor typesLatasch, Leo / Freye, Enno et al. | 2002
- 877
-
Topical Treatment of Rhinosinusitis with Fusafungine Nasal Spray. A double-blind, placebo-controlled, parallel-group study in 20 patientsMösges, Ralph / Spaeth, Joachim / Berger, Kristine / Dubois, Frederic et al. | 2002
- 884
-
1-Ethyl and 1-Propylazacycloalkan-2-one Ester Prodrugs of Ketoprofen. Synthesis, chemical stability, enzymatic hydrolysis, anti-inflammatory activity, and gastrointestinal toxicityBonina, Francesco Paolo / Puglia, Carmelo / Ventura, Dario / Santagati, Natale Alfredo / Saija, Antonella / Trombetta, Domenico et al. | 2002
- 890
-
Effect of Tolterodine on the Anticoagulant Actions and Pharmacokinetics of Single-dose Warfarin in Healthy VolunteersRahimy, Mohamad / Hallén, Bengt / Narang, Prem et al. | 2002
- 896
-
Transport of Anionic Drugs across the Basolateral Membrane of Proximal S2 Segments of the Rabbit Kidney. Inverse relationship between the affinity to the p-aminohippurate transport system and the transport ratePerst, Volker / Haßler, Martin / Greven, Joachim et al. | 2002
- 903
-
Synthesis, Antibacterial Activity, and Toxicity of 7-(Isoindolin-5-yl)-4-oxoquinoline-3-carboxylic Acids. Discovery of the novel Des-F(6)-quinolone antibacterial agent garenoxacin (T-3811 or BMS-284756)Hayashi, Kazuya / Takahata, Masahiro / Kawamura, Yasuhito / Todo, Yozo et al. | 2002
- 914
-
The Pharma Market as Reflected by Patents / Antidiarrhoeal agents / Compounds useful as antiallergic and antiinflammatory agents / Agents for the treatment of arteriosclerosis and related diseases / Agents for treating heart failureHabernickel, V. J. et al. | 2002
- 918
-
Announcements| 2002
- 922
-
Symposium of the Paul Martini Foundation on "Pharmacogenomics: Promises and Expectations for Drug Therapy and Drug Development" on 7 September 2002 in Halle/Saale (Germany)| 2002
- 922
-
Pharmacogenomics: Promises and Expectations for Drug Therapy and Drug Development| 2002
- 928
-
Kombinationstherapie der chronischen Virushepatitis CZeuzem, S. et al. | 2002
- 930
-
Aktuelle Therapie der chronischen Virus-hepatitis BManns, M. P. et al. | 2002
- 931
-
Medikamentose Therapie bei Aszites und hepatorenalem SyndromGerbes, A. L. et al. | 2002
- 933
-
Rolle von nuklearen Rezeptoren beim hepatischen und intestinalen Medikamenten-transportKullak-Ublick, G. A. et al. | 2002
- 933
-
Enterohepatic Circulation of Bile Acids in Lipid TherapyKramer, W. et al. | 2002
- 935
-
Zelltherapie in der Hepatologievon Weizsacker, F. et al. | 2002
- 936
-
Immunsuppression bei chronisch entzundlichen DarmerkrankungenStange, E. F. et al. | 2002
- 938
-
Strategien gegen Tumor-Nekrose-FaktorSchreiber, S. et al. | 2002
- 939
-
Anti-Interleukin-18-Strategien zur Therapie der Colitis im TiermodellSiegmund, B. et al. | 2002
- 941
-
Probiotika und chronisch entzundliche DarmerkrankungenFolwaczny, C. et al. | 2002
- 943
-
Gastroosophageale Refluxkrankheit und H. pylori-Infektion: Rolle neuer Protonenpum-peninhibitorenMalfertheiner, P. et al. | 2002
- 944
-
Atiologie, Definition und Therapie des ReizdarmsyndromsMuller-Lissner, S. et al. | 2002
- 945
-
Botulinum-Toxin: Wirkgrundlage und Stellenwert in der TherapieAllescher, H. D. et al. | 2002
- 946
-
Signaltransduktion des Pankreaskarzinoms: Ansatzpunkte fur die TherapieSchmid, R. M. et al. | 2002
- 947
-
Neue Zytostatika in der Therapie des kolorektalen KarzinomsGalle, P. R. et al. | 2002
- 948
-
5-ASA-Praparate zur Pravention des KolonkarzinomsReinacher-Schick, A. et al. | 2002
- 950
-
Dendritische Zellen und CpG-Oligonukleotide in der Immuntherapie experimenteller gastrointestinaler TumoreEndres, S. et al. | 2002
- 953
-
Therapie der neuroendokrinen Tumoren des gastroenteropankreatischen Systems (GEP)Wiedenmann, B. et al. | 2002
- 954
-
Medikamentose Therapie und Pravention des hepatozellularen KarzinomsBlum, H. E. et al. | 2002
- 958
-
Tyrosinkinase-Inhibition mit Imatinib bei chronisch-myeloischer Leukamie und gastrointestinalen StromatotumorenWolf, H. et al. | 2002
- E524
-
Reproductive Toxicity of gamma-Ethyl-gamma-phenyl-butyrolactone, a New Anticonvulsant and Hypnotic Drug, in Mice / Fertility and peri- and post-natal studiesChamorro, G. / Vega, F. / Madrigal, E. / Salazar, M. et al. | 2002
- E654
-
Synthesis and beta~1-, beta~2-Adrenergic Receptor Binding Studies of 4-Acylamino-substituted Phenoxypropanolamine and 5-Acylamino-substituted Naphthyloxypropanolamine DerivativesJindal, D. P. / Coumar, M. S. / Bruni, G. / Massarelli, P. et al. | 2002
- E684
-
Improvement of the Bioavailability of Colchicine in Rats by Co-administration of D-a-Tocopherol Polyethylene Glycol 1000 Succinate and a Polyethoxylated Derivative of 12-Hydroxy-Stearic AcidBittner, B. / Guenzi, A. / Fullhardt, P. / Zuercher, G. / Gonzalez, R. C. B. / Mountfield, R. J. et al. | 2002
- G615
-
Comparative Pharmacokinetics of a Progesterone Capsule and a Progesterone Gel Following Vaginal AdministrationKleinstein, J. / Schlegelmilch, R. / Mazur, D. / Vens-Cappell, B. et al. | 2002
-
Reduction of Acute Relapses in Patients with Chronic Recurrent Hypertrophic Sinusitis during Treatment with a Bacterial Immunostimulant (Enterococcus faecalis Bacteriae of Human Origin)Habermann, W. / Zimmermann, K. / Skarabis, H. / Kunze, R. / Rusch, V. et al. | 2002