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Molecular Diversity in Drug Design [2002]

1
Issues in Molecular Diversity and the Role of Ligand Binding Sites
23
Molecular Diversity in Drug Design. Application to High-speed Synthesis and High-Throughput Screening
43
Background Theory of Molecular Diversity
67
Absolute vs Relative Similarity and Diversity
93
Diversity in Very Large Libraries
115
Subset-Selection Methods For Chemical Databases
141
Molecular Diversity in Site-focused Libraries
175
Managing Combinatorial Chemistry Information
197
Design of Small Libraries for Lead Exploration
221
The Design of Small- and Medium-sized Focused Combinatorial Libraries
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