BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS
Die Inhaltsverzeichnisse werden automatisch erzeugt und basieren auf den im Index des TIB-Portals verfügbaren Einzelnachweisen der enthaltenen Beiträge. Die Anzeige der Inhaltsverzeichnisse kann daher unvollständig oder lückenhaft sein.
Inhaltsverzeichnis
- 1
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Graphical contents list| 2008
- 17
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Identification of a small molecule β-secretase inhibitor that binds without catalytic aspartate engagementSteele, Thomas G. / Hills, Ivory D. / Nomland, Ashley A. et al. | 2008
- 17
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Identification of a small molecule b-secretase inhibitor that binds without catalytic aspartate engagementSteele, T. G. / Hills, I. D. / Nomland, A. A. et al. | 2009
- 21
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Synthesis and stereochemical effects of pyrrolidinyl-acetylenic thieno[3,2-d]pyrimidines as EGFR and ErbB-2 inhibitorsStevens, Kirk L. / Alligood, Krystal J. / Alberti, Jennifer G. Badiang et al. | 2008
- 27
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Discovery of potent, selective sulfonylfuran urea endothelial lipase inhibitorsGoodman, Krista B. / Bury, Michael J. / Cheung, Mui et al. | 2008
- 31
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Discovery of α-amidosulfones as potent and selective agonists of CB2: Synthesis, SAR, and pharmacokinetic propertiesMarx, Isaac E. / DiMauro, Erin F. / Cheng, Alan et al. | 2008
- 31
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Discovery of a-amidosulfones as potent and selective agonists of CB2: Synthesis, SAR, and pharmacokinetic propertiesMarx, I. E. / DiMauro, E. F. / Cheng, A. et al. | 2009
- 36
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PEG-immobilization of cardol and soluble polymer-supported synthesis of some cardol–coumarin derivatives: Preliminary evaluation of their inhibitory activity on mushroom tyrosinaseTocco, Graziella / Fais, Antonella / Meli, Gabriele et al. | 2008
- 40
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Identification and synthesis of 2,7-diamino-thiazolo[5,4-d]pyrimidine derivatives as TRPV1 antagonistsLebsack, Alec D. / Branstetter, Bryan J. / Hack, Michael D. et al. | 2008
- 47
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Calculation of binding free energies for non-zinc chelating pyrimidine dicarboxamide inhibitors with MMP-13Carrascal, Noel / Rizzo, Robert C. et al. | 2008
- 51
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Synthesis and neuropharmacological evaluation of esters of R(−)-N-alkyl-11-hydroxy-2-methoxynoraporphinesSi, Yu-Gui / Choi, Yong-Kee / Gardner, Matthew P. et al. | 2008
- 54
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Discovery of novel spirocyclopropyl hydroxamate and carboxylate compounds as TACE inhibitorsGuo, Zhuyan / Orth, Peter / Wong, Shing-Chun et al. | 2008
- 58
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1-Naphthyl and 4-indolyl arylalkylamines as selective monoamine reuptake inhibitorsManning, James R. / Sexton, Tammy / Childers, Steven R. et al. | 2008
- 62
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Lead identification to generate 3-cyanoquinoline inhibitors of insulin-like growth factor receptor (IGF-1R) for potential use in cancer treatmentMiller, Lori M. / Mayer, Scott C. / Berger, Dan M. et al. | 2008
- 67
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Modification of the N-terminal sulfonyl residue in 3-amidinophenylalanine-based matriptase inhibitorsSteinmetzer, Torsten / Dönnecke, Daniel / Korsonewski, Martin et al. | 2008
- 74
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Synthesis of biflavones having a 6-O-7’’ linkage and effects on cyclooxygenase-2 and inducible nitric oxide synthaseChe, Haiyan / Park, Byung Kyu / Lim, Hyun et al. | 2008
- 77
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Multifidone: A novel cytotoxic lathyrane-type diterpene having an unusual six-membered A ring from Jatropha multifidaDas, Biswanath / Reddy, Kongara Ravinder / Ravikanth, Bommena et al. | 2008
- 80
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Synthesis and evaluation of novel photoreactive α-amino acid analog carrying acidic and cleavable functionsBongo, Nlandu B. / Tomohiro, Takenori / Hatanaka, Yasumaru et al. | 2008
- 80
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Synthesis and evaluation of novel photoreactive a-amino acid analog carrying acidic and cleavable functionsBongo, N. B. / Tomohiro, T. / Hatanaka, Y. et al. | 2009
- 83
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Novel fluorinated pseudopeptides as proteasome inhibitorsFormicola, Lucia / Maréchal, Xavier / Basse, Nicolas et al. | 2008
- 87
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Carbamoylcholine analogs as nicotinic acetylcholine receptor agonists—Structural modifications of 3-(dimethylamino)butyl dimethylcarbamate (DMABC)Hansen, Camilla P. / Jensen, Anders A. / Balle, Thomas et al. | 2008
- 92
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Design, synthesis, and biological evaluation of biotin-labeled (−)-ternatin, a potent fat-accumulation inhibitor against 3T3-L1 adipocytesShimokawa, Kenichiro / Yamada, Kaoru / Ohno, Osamu et al. | 2008
- 96
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Urea based CCR3 antagonists employing a tetrahydro-1,3-oxazin-2-one spacerDhar, T.G. Murali / Yang, Guchen / Davies, Paul et al. | 2008
- 100
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Efficient nucleic acid transduction with lipoplexes containing novel piperazine- and polyamine-conjugated cholesterol derivativesIslam, Rafique Ul / Hean, Justin / van Otterlo, Willem A.L. et al. | 2008
- 104
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11-Phenyl-[b,e]-dibenzazepine compounds: Novel antitumor agentsAl-Qawasmeh, Raed A. / Lee, Yoon / Cao, Ming-Yu et al. | 2008
- 108
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Analogs of methyl-piperidinopyrazole (MPP): Antiestrogens with estrogen receptor α selective activityZhou, Hai-Bing / Carlson, Kathryn E. / Stossi, Fabio et al. | 2008
- 108
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Analogs of methyl-piperidinopyrazole (MPP): Antiestrogens with estrogen receptor a selective activityZhou, H. B. / Carlson, K. E. / Stossi, F. et al. | 2009
- 111
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Synthesis of a fluorescent 2′3′-dideoxycytosine analog, tCddPorterfield, William / Tahmassebi, Deborah C. et al. | 2008
- 111
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Synthesis of a fluorescent 2prime3prime-dideoxycytosine analog, tCddPorterfield, W. / Tahmassebi, D. C. et al. | 2009
- 114
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Camphor sulfonamide derivatives as novel, potent and selective CXCR3 antagonistsWang, Yonghui / Busch-Petersen, Jakob / Wang, Feng et al. | 2008
- 119
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Sulfonamido-aryl ethers as bradykinin B1 receptor antagonistsCole, Andrew G. / Metzger, Axel / Brescia, Marc-Raleigh et al. | 2008
- 123
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3,4-Disubstituted indole acylsulfonamides: A novel series of potent and selective human EP3 receptor antagonistsZhou, Nian / Zeller, Wayne / Krohn, Michael et al. | 2008
- 127
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3D-QSAR and QSSR studies of 3,8-diazabicyclo[4.2.0]octane derivatives as neuronal nicotinic acetylcholine receptors by comparative molecular field analysis (CoMFA)Ye, Mao / Dawson, Marcia I. et al. | 2008
- 132
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Design, synthesis, and biological evaluation of a scaffold for iGluR ligands based on the structure of (−)-kaitocephalinVaswani, Rishi G. / Limon, Agenor / Reyes-Ruiz, Jorge Mauricio et al. | 2008
- 136
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One-pot synthesis of 5-phenylimino, 5-thieno or 5-oxo-1,2,3-dithiazoles and evaluation of their antimicrobial and antitumor activityKonstantinova, Lidia S. / Bol’shakov, Oleg I. / Obruchnikova, Natalia V. et al. | 2008
- 142
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Diarylimidazolyl oxadiazole and thiadiazole derivatives as cannabinoid CB1 receptor antagonistsKim, Jong Yup / Seo, Hee Jeong / Lee, Sung-Han et al. | 2008
- 146
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Synthesis and antifungal activity of 1H-pyrrolo[3,2-g]quinoline-4,9-diones and 4,9-dioxo-4,9-dihydro-1H-benzo[f]indolesRyu, Chung-Kyu / Lee, Jung Yoon / Jeong, Seong Hee et al. | 2008
- 149
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A model ternary heparin conjugate by direct covalent bond strategy applied to drug delivery systemWang, Ying / Xin, Dingcheng / Hu, Jiawen et al. | 2008
- 153
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Synthesis and biological evaluation of new glutamic acid-based inhibitors of MurD ligaseTomašić, Tihomir / Zidar, Nace / Rupnik, Veronika et al. | 2008
- 158
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Aryl aminopyrazole benzamides as oral non-steroidal selective glucocorticoid receptor agonistsBarnett, Heather A. / Coe, Diane M. / Cooper, Tony W.J. et al. | 2008
- 163
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Inhibition of purple acid phosphatase with α-alkoxynaphthylmethylphosphonic acidsMcGeary, Ross P. / Vella, Peter / Mak, Jeffrey Y.W. et al. | 2008
- 163
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Inhibition of purple acid phosphatase with a-alkoxynaphthylmethylphosphonic acidsMcGeary, R. P. / Vella, P. / Mak, J. Y. et al. | 2009
- 167
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Synthesis and biological evaluation of a series of tangeretin-derived chalconesQuintin, Jérôme / Desrivot, Julie / Thoret, Sylviane et al. | 2008
- 170
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Pleuromutilin derivatives having a purine ring. Part 2: Influence of the central spacer on the antibacterial activity against Gram-positive pathogensHirokawa, Yoshimi / Kinoshita, Hironori / Tanaka, Tomoyuki et al. | 2008
- 175
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Pleuromutilin derivatives having a purine ring. Part 3: Synthesis and antibacterial activity of novel compounds possessing a piperazine ring spacerHirokawa, Yoshimi / Kinoshita, Hironori / Tanaka, Tomoyuki et al. | 2008
- 180
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Potent inhibitors of HCV-NS3 protease derived from boronic acidsVenkatraman, Srikanth / Wu, Wanli / Prongay, Andrew et al. | 2008
- 184
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Design, synthesis, and pharmacological and pharmacokinetic evaluation of 3-phenyl-5-pyridyl-1,2,4-triazole derivatives as xanthine oxidoreductase inhibitorsSato, Takahiro / Ashizawa, Naoki / Iwanaga, Takashi et al. | 2008
- 188
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Synthesis of tyrosinase inhibitory (4-oxo-4H-pyran-2-yl)acrylic acid ester derivativesKang, Soo Sung / Kim, Hyoung Ja / Jin, Changbae et al. | 2008
- 192
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Two new cytotoxic diterpenes from the rhizomes of Hedychium spicatumReddy, P. Prabhakar / Rao, R. Ranga / Rekha, K. et al. | 2008
- 196
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N,N-Dichloroaminosulfonic acids as novel topical antimicrobial agentsLow, Eddy / Nair, Satheesh / Shiau, Timothy et al. | 2008
- 199
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Synthesis and structure–activity relationships of oxamyl dipeptide caspase inhibitors developed for the treatment of liver diseaseUeno, Hirokazu / Kawai, Makoto / Shimokawa, Hirohisa et al. | 2008
- 203
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Syntheses and opioid receptor binding properties of carboxamido-substituted opioidsWentland, Mark P. / Lou, Rongliang / Lu, Qun et al. | 2008
- 209
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Discovery of a potent, selective and orally bioavailable 3,9-diazaspiro[5.5]undeca-2-one CCR5 antagonistYang, Hanbiao / Lin, Xiao-Fa / Padilla, Fernando et al. | 2008
- 214
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The discovery of highly potent CGRP receptor antagonistsStump, Craig A. / Bell, Ian M. / Bednar, Rodney A. et al. | 2008
- 218
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Biologically relevant chemical properties of peroxymonophosphate (O3POOH)LaButti, Jason N. / Gates, Kent S. et al. | 2008
- 222
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Design and synthesis of pyrazole derivatives as potent and selective inhibitors of tissue-nonspecific alkaline phosphatase (TNAP)Sidique, Shyama / Ardecky, Robert / Su, Ying et al. | 2008
- 226
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Beyond the MEK-pocket: Can current MEK kinase inhibitors be utilized to synthesize novel type III NCKIs? Does the MEK-pocket exist in kinases other than MEK?Tecle, Haile / Shao, Jianxing / Li, Yanhong et al. | 2008
- 230
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Tetrahydroisoquinoline amide substituted phenyl pyrazoles as selective Bcl-2 inhibitorsPorter, John / Payne, Andrew / de Candole, Ben et al. | 2008
- 234
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TRAIL-enhancing activity of Erythrinan alkaloids from Erythrina velutinaOzawa, Masaaki / Etoh, Tadahiro / Hayashi, Masahiko et al. | 2008
- 237
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Alcohol dehydrogenase-catalyzed in vitro oxidation of anandamide to N-arachidonoyl glycine, a lipid mediator: Synthesis of N-acyl glycinalsAneetha, Halikhedkar / O’Dell, David K. / Tan, Bo et al. | 2008
- 242
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2,6,9-Trisubstituted purine derivatives as protein A mimetics for the treatment of autoimmune diseasesZacharie, Boulos / Fortin, Daniel / Wilb, Nicole et al. | 2008
- 247
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Oxadiazolone bioisosteres of pregabalin and gabapentinWustrow, David J. / Belliotti, Thomas R. / Capiris, Thomas et al. | 2008
- 251
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Molecular modeling of the α9α10 nicotinic acetylcholine receptor subtypePérez, Edwin G. / Cassels, Bruce K. / Zapata-Torres, Gerald et al. | 2008
- 251
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Molecular modeling of the a9a10 nicotinic acetylcholine receptor subtypePerez, E. G. / Cassels, B. K. / Zapata-Torres, G. et al. | 2009
- 255
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Synthesis and antiinflammatory activity of some new 1,3,5-trisubstituted pyrazolines bearing benzene sulfonamideRathish, I.G. / Javed, Kalim / Ahmad, Shamim et al. | 2008
- 259
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Pyridine-3-carboxamides as novel CB2 agonists for analgesiaMitchell, William L. / Giblin, Gerard M.P. / Naylor, Alan et al. | 2008
- 264
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Molecular modeling, synthesis, and activity studies of novel biaryl and fused-ring BACE1 inhibitorsChirapu, Srinivas Reddy / Pachaiyappan, Boobalan / Nural, Hikmet F. et al. | 2008
- 275
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Synthesis and biological evaluation of novel 2,4,5-substituted pyrimidine derivatives for anticancer activityXie, Fuchun / Zhao, Hongbing / Zhao, Lizhi et al. | 2008
- 279
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Fragment-based discovery of JAK-2 inhibitorsAntonysamy, Stephen / Hirst, Gavin / Park, Frances et al. | 2008
- 283
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Corrigendum to “Synthesis of a 200-member library of squaric acid N-hydroxylamide amides” [Bioorg. Med. Chem. Lett. 18 (2008) 4968–4971]Charton, Julie / Leroux, Florence / Delaroche, Sylvain et al. | 2008
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Corrigendum to “Structural modifications of N-arylamide oxadiazoles: Identification of N-arylpiperidine oxadiazoles as potent and selective agonists of CB2” [Bioorg. Med. Chem. Lett. 18 (2008) 4267–4274]DiMauro, Erin F. / Buchanan, John L. / Chen, Alan et al. | 2008
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Instructions to contributors| 2008
- IFC
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Editorial board| 2008