BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS
Die Inhaltsverzeichnisse werden automatisch erzeugt und basieren auf den im Index des TIB-Portals verfügbaren Einzelnachweisen der enthaltenen Beiträge. Die Anzeige der Inhaltsverzeichnisse kann daher unvollständig oder lückenhaft sein.
Inhaltsverzeichnis
- 753
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Graphical contents list| 2005
- 771
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Concise and efficient asymmetric synthesis of (S)-2-ethylphenylpropanoic acid derivatives: Dual agonists for human peroxisome proliferator-activated receptor #945 and #948Kasuga, Jun-ichi et al. | 2006
- 771
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Concise and efficient asymmetric synthesis of (S)-2-ethylphenylpropanoic acid derivatives: Dual agonists for human peroxisome proliferator-activated receptor α and δKasuga, Jun-ichi / Hashimoto, Yuichi / Miyachi, Hiroyuki et al. | 2005
- 775
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The synthesis and aqueous superoxide anion scavenging of water-dispersible lutein estersNadolski, Geoff / Cardounel, Arturo J. / Zweier, Jay L. et al. | 2005
- 782
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Two methylene groups in phospholipids distinguish between apoptosis and necrosis for tumor cellsNagami, Hideaki / Nakano, Koji / Ichihara, Hideaki et al. | 2005
- 786
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Isolation, synthesis, and anti-tumor activities of a novel class of podocarpic diterpenesXiong, Yi / Wang, Kuiwu / Pan, Yuanjiang et al. | 2005
- 790
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Microbial transformation of silybin by Trichoderma koningiiKim, Hyun Jung / Park, Hae-Suk / Lee, Ik-Soo et al. | 2005
- 794
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Design, synthesis, and biological evaluation of BODIPY(R)#8211erythromycin probes for bacterial ribosomesLi, Jing et al. | 2006
- 794
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Design, synthesis, and biological evaluation of BODIPY®–erythromycin probes for bacterial ribosomesLi, Jing / Kim, In Ho / Roche, Eric D. et al. | 2005
- 798
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Structure#8211activity relationship study of 1,4-dihydropyridine derivatives blocking N-type calcium channelsYamamoto, Takashi et al. | 2006
- 798
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Structure–activity relationship study of 1,4-dihydropyridine derivatives blocking N-type calcium channelsYamamoto, Takashi / Niwa, Seiji / Ohno, Seiji et al. | 2005
- 803
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Hydrolysis of plasmid DNA and RNA by amino alkyl naphthalimide as metal-free artificial nucleaseYang, Qing / Xu, Jianqiang / Sun, Yuanshe et al. | 2005
- 807
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Enhancing the synthetic utility of aldolase antibody 38C2Mondal, Kalyani / Ramesh, Namakkal G. / Roy, Ipsita et al. | 2005
- 811
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Synthesis and structure–activity relationships of 8-azabicyclo[3.2.1]octane benzylamine NK1 antagonistsThomson, Christopher G. / Carlson, Emma / Chicchi, Gary G. et al. | 2005
- 811
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Synthesis and structure#8211activity relationships of 8-azabicyclo(3.2.1)octane benzylamine NK1 antagonistsThomson, Christopher G. et al. | 2006
- 815
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Synthesis and antiprotozoal activity of some new synthetic substituted quinoxalinesHui, Xu / Desrivot, Julie / Bories, Christian et al. | 2005
- 821
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Structure-guided synthesis of tamoxifen analogs with improved selectivity for the orphan ERR#947Chao, Esther Y.H. et al. | 2006
- 821
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Structure-guided synthesis of tamoxifen analogs with improved selectivity for the orphan ERRγChao, Esther Y.H. / Collins, Jon L. / Gaillard, Stéphanie et al. | 2005
- 825
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Synthesis and pharmacochemical study of novel polyfunctional molecules combining anti-inflammatory, antioxidant, and hypocholesterolemic propertiesDoulgkeris, Christos M. / Galanakis, Dimitrios / Kourounakis, Angeliki P. et al. | 2005
- 830
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From genome to drug lead: Identification of a small-molecule inhibitor of the SARS virusDooley, Andrea J. / Shindo, Nice / Taggart, Barbara et al. | 2005
- 834
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Androstenediol analogs as ER-β-selective SERMsBlizzard, Timothy A. / Gude, Candido / Morgan, Jerry D. II et al. | 2005
- 834
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Androstenediol analogs as ER-#946-selective SERMsBlizzard, Timothy A. et al. | 2006
- 839
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Convergent, parallel synthesis of a series of β-substituted 1,2,4-oxadiazole butanoic acids as potent and selective αvβ3 receptor antagonistsBoys, Mark L. / Schretzman, Lori A. / Chandrakumar, Nizal S. et al. | 2005
- 839
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Convergent, parallel synthesis of a series of #946-substituted 1,2,4-oxadiazole butanoic acids as potent and selective #945v#9463 receptor antagonistsBoys, Mark L. et al. | 2006
- 845
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Synthesis of 2,5-thiazole butanoic acids as potent and selective αvβ3 integrin receptor antagonists with improved oral pharmacokinetic propertiesWendt, John A. / Wu, Hongwei / Stenmark, Heather G. et al. | 2005
- 845
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Synthesis of 2,5-thiazole butanoic acids as potent and selective #945v#9463 integrin receptor antagonists with improved oral pharmacokinetic propertiesWendt, John A. et al. | 2006
- 850
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Conformation stability and organization of mefloquine molecules in different environmentsSkórska, Agnieszka / Śliwiński, Jan / Oleksyn, Barbara J. et al. | 2005
- 854
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Substituted 4-hydroxyphenyl sulfonamides as pathway-selective estrogen receptor ligandsSabatucci, Joseph P. / Ashwell, Mark A. / Trybulski, Eugene et al. | 2005
- 859
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Design, synthesis, and biological evaluation of monopyrrolinone-based HIV-1 protease inhibitors possessing augmented P2′ side chainsSmith, Amos B. III / Charnley, Adam K. / Harada, Hironori et al. | 2005
- 859
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Design, synthesis, and biological evaluation of monopyrrolinone-based HIV-1 protease inhibitors possessing augmented P2#8242 side chainsSmith, Amos B. et al. | 2006
- 864
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Synthesis and structure–activity relationships of a new series of 2α-substituted trans-4,5-dimethyl-4-(3-hydroxyphenyl)piperidine as μ-selective opioid antagonistsLe Bourdonnec, Bertrand / Goodman, Allan J. / Michaut, Mathieu et al. | 2005
- 864
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Synthesis and structure#8211activity relationships of a new series of 2#945-substituted trans-4,5-dimethyl-4-(3-hydroxyphenyl)piperidine as #956-selective opioid antagonistsLe Bourdonnec, Bertrand et al. | 2006
- 869
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Synthesis and reactivity with β-lactamases of a monobactam bearing a retro-amide side chainAdediran, S.A. / Lohier, J.-F. / Cabaret, D. et al. | 2005
- 869
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Synthesis and reactivity with #946-lactamases of a monobactam bearing a retro-amide side chainAdediran, S.A. et al. | 2006
- 872
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Pharmacokinetics and metabolism studies on (3-tert-butyl-7-(5-methylisoxazol-3-yl)-2-(1-methyl-1H-1,2,4-triazo- l-5-ylmethoxy) pyrazolo(1,5-d)(1,2,4)triazine, a functionally selective GABAA #9455 inverse agonist for cognitive dysfunctionJones, Philip et al. | 2006
- 872
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Pharmacokinetics and metabolism studies on (3-tert-butyl-7-(5-methylisoxazol-3-yl)-2-(1-methyl-1H-1,2,4-triazol-5-ylmethoxy) pyrazolo[1,5-d][1,2,4]triazine, a functionally selective GABAA α5 inverse agonist for cognitive dysfunctionJones, Philip / Atack, John R. / Braun, Matthew P. et al. | 2005
- 876
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Synthesis and in vitro antitubercular activity of some 1-[(4-sub)phenyl]-3-(4-{1-[(pyridine-4-carbonyl)hydrazono]ethyl}phenyl)thioureaSriram, Dharmarajan / Yogeeswari, Perumal / Madhu, Kasinathan et al. | 2005
- 879
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Discovery of a potent phenolic N1-benzylidene–pyridinecarboxamidrazone selective against Gram-positive bacteriaRathbone, Daniel L. / Parker, Katy J. / Coleman, Michael D. et al. | 2005
- 879
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Discovery of a potent phenolic N 1-benzylidene#8211pyridinecarboxamidrazone selective against Gram-positive bacteriaRathbone, Daniel L. et al. | 2006
- 884
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Thyroid receptor ligands. Part 4: 4′-amido bioisosteric ligands selective for the thyroid hormone receptor betaLi, Yi-Lin / Litten, Chris / Koehler, Konrad F. et al. | 2005
- 884
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Thyroid receptor ligands. Part 4: 4#8242-amido bioisosteric ligands selective for the thyroid hormone receptor betaLi, Yi-Lin et al. | 2006
- 887
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Partial structures of ketoconazole as modulators of the large conductance calcium-activated potassium channel (BKCa)Power, Eoin C. / Ganellin, C. Robin / Benton, David C.H. et al. | 2005
- 891
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Novel non-nucleobase inhibitors of Staphylococcus aureus DNA polymerase IIICRose, Yannick / Ciblat, Stéphane / Reddy, Ranga et al. | 2005
- 897
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Aplysamine-1 and related analogs as histamine H3 receptor antagonistsSwanson, Devin M. / Wilson, Sandy J. / Boggs, Jamin D. et al. | 2005
- 901
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Design and total synthesis of a fluorescent phorboxazole a analog for cellular studiesChen, Jiehao / Ying, Lu / Hansen, T. Matthew et al. | 2005
- 905
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Highly potent and selective zwitterionic agonists of the #948-opioid receptor. Part 1Middleton, Donald S. et al. | 2006
- 905
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Highly potent and selective zwitterionic agonists of the δ-opioid receptor. Part 1Middleton, Donald S. / Maw, Graham N. / Challenger, Clare et al. | 2005
- 911
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Synthesis of 1-(3′,4′,5′-trimethoxy) phenyl naphtho[2,1b]furan as a novel anticancer agentSrivastava, Vandana / Negi, Arvind S. / Kumar, J.K. et al. | 2005
- 911
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Synthesis of 1-(3#8242,4#8242,5#8242-trimethoxy) phenyl naphtho(2,1b)furan as a novel anticancer agentSrivastava, Vandana et al. | 2006
- 915
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Design, synthesis, and evaluation of 2-alkoxydihydrocinnamates as PPAR agonistsLu, Ying / Guo, Zongru / Guo, Yanshen et al. | 2005
- 920
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Novel endoperoxides: Synthesis and activity against Candida speciesMacreadie, Peter / Avery, Thomas / Greatrex, Ben et al. | 2005
- 923
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Inhibition of DNA helicases with DNA-competitive inhibitorsDubaele, Sandy / Jahnke, Wolfang / Schoepfer, Joseph et al. | 2005
- 928
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Synthesis of complex-type glycans derived from parasitic helminthsNakano, Jun / Ohta, Hiromichi / Ito, Yukishige et al. | 2005
- 934
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Synthesis and evaluation of 2-anilino-3-phenylsulfonyl-6-methylpyridines as corticotropin-releasing factor1 receptor ligandsHartz, Richard A. / Arvanitis, Argyrios G. / Arnold, Charles et al. | 2005
- 938
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Synthesis and structure#8211activity relationships of novel poly(ADP-ribose) polymerase-1 inhibitorsTao, Ming et al. | 2006
- 938
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Synthesis and structure–activity relationships of novel poly(ADP-ribose) polymerase-1 inhibitorsTao, Ming / Park, Chung Ho / Bihovsky, Ron et al. | 2005
- 943
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Novel fluorescent labelled affinity probes for diadenosine-5′,5‴-P1,P4-tetraphosphate (Ap4A)-binding studiesWright, Michael / Miller, Andrew D. et al. | 2005
- 943
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Novel fluorescent labelled affinity probes for diadenosine-5#8242,5#8244-P 1,P 4-tetraphosphate (Ap4A)-binding studiesWright, Michael et al. | 2006
- 949
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Isolation, structure elucidation, antioxidative and immunomodulatory properties of two novel dihydrocoumarins from Aloe veraZhang, Xiu-feng / Wang, Hong-mei / Song, Yuan-li et al. | 2005
- 954
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Pyridobenzodiazepines: A novel class of orally active, vasopressin V2 receptor selective agonistsFailli, Amedeo A. / Shumsky, Jay S. / Steffan, Robert J. et al. | 2005
- 960
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Hit-to-Lead studies: The discovery of potent, orally bioavailable thiazolopyrimidine CXCR2 receptor antagonistsBaxter, Andrew / Cooper, Anne / Kinchin, Elizabeth et al. | 2005
- 964
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The discovery of a potent and selective lethal factor inhibitor for adjunct therapy of anthrax infectionXiong, Yusheng / Wiltsie, Judyann / Woods, Andrea et al. | 2005
- 969
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Analysis of anti-PDE3 activity of 2-morpholinochromone derivatives reveals multiple mechanisms of anti-platelet activityAbbott, Belinda M. / Thompson, Philip E. et al. | 2005
- 974
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Syntheses and evaluation of novel fatty acid-second-generation taxoid conjugates as promising anticancer agentsKuznetsova, Larissa / Chen, Jin / Sun, Liang et al. | 2005
- 978
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Semicarbazone-based inhibitors of cathepsin K, are they prodrugs for aldehyde inhibitors?Adkison, Kim K. / Barrett, David G. / Deaton, David N. et al. | 2005
- 984
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Enhanced FTase activity achieved via piperazine interaction with catalytic zincNjoroge, F. George / Vibulbhan, Bancha / Pinto, Patrick et al. | 2005
- 989
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Reduction of CYP450 inhibition in the 4-[(1H-imidazol-4-yl)methyl]piperidine series of histamine H3 receptor antagonistsBerlin, Michael / Ting, Pauline C. / Vaccaro, Wayne D. et al. | 2005
- 995
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#9514-Pyrone iron(0)carbonyl complexes as effective CO-releasing molecules (CO-RMs)Fairlamb, Ian J.S. et al. | 2006
- 995
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η4-Pyrone iron(0)carbonyl complexes as effective CO-releasing molecules (CO-RMs)Fairlamb, Ian J.S. / Duhme-Klair, Anne-Kathrin / Lynam, Jason M. et al. | 2005
- 999
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Microwave-assisted synthesis of N-alkylated benzotriazole derivatives: Antimicrobial studiesNanjunda Swamy, S. / Basappa / Sarala, G. et al. | 2005
- 1005
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Intermolecular interactions in the crystal structures of potential HIV-1 integrase inhibitorsMajerz-Maniecka, Katarzyna / Musiol, Robert / Nitek, Wojciech et al. | 2005
- 1010
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Synthesis and anti-HSV-1 activity of quinolonic acyclovir analoguesLucero, Bianca d’A. / Gomes, Claudia Regina B. / Frugulhetti, Izabel Christina de P.P. et al. | 2005
- 1014
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3D-QSAR studies on antitubercular thymidine monophosphate kinase inhibitors based on different alignment methodsAparna, V. / Jeevan, J. / Ravi, M. et al. | 2005
- 1021
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Kinetic investigation on aqueous decomposition of 2-chloroethylnitrososulfamideSeridi, Achour / Kadri, Mekki / Abdaoui, Mohamed et al. | 2005
- 1028
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Conversion of potent MMP inhibitors into selective TACE inhibitorsCherney, Robert J. / King, Bryan W. / Gilmore, John L. et al. | 2005
- 1032
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Phenolic P2/P3 core motif as thrombin inhibitors—Design, synthesis, and X-ray co-crystal structureHanessian, Stephen / Therrien, Eric / van Otterlo, Willem A.L. et al. | 2005
- 1032
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Phenolic P2-P3 core motif as thrombin inhibitors#8212Design, synthesis, and X-ray co-crystal structureHanessian, Stephen et al. | 2006
- 1037
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A neural network based classification scheme for cytotoxicity predictions:Validation on 30,000 compoundsMolnár, László / Keserű, György M. / Papp, Ákos et al. | 2005
- 1040
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Phthalazinones 2: Optimisation and synthesis of novel potent inhibitors of poly(ADP-ribose)polymeraseCockcroft, Xiao-ling / Dillon, Krystyna J. / Dixon, Lesley et al. | 2005
- 1045
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Piperazinyl oxime ethers as NK-1 receptor antagonistsvan den Hoogenband, Adri / van Maarseveen, Jan H. / McCreary, Andrew C. et al. | 2005
- 1049
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A novel nicotinic acetylcholine receptor antagonist radioligand for PET studiesDing, Yu-Shin / Kil, Kun-eek / Lin, Kuo-Shyan et al. | 2005
- 1054
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Synthesis and antibacterial activity of 3-O-acyl-6-O-carbamoyl erythromycin A derivativesZhu, Bin / Marinelli, Brett A. / Abbanat, Darren et al. | 2005
- 1060
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The discovery of fluoropyridine-based inhibitors of the factor VIIa/TF complex—Part 2Kohrt, Jeffrey T. / Filipski, Kevin J. / Cody, Wayne L. et al. | 2005
- 1060
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The discovery of fluoropyridine-based inhibitors of the factor VIIa-TF complex#8212Part 2Kohrt, Jeffrey T. et al. | 2006
- 1065
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Cyclic urea derivatives as potent NK1 selective antagonists. Part II: Effects of fluoro and benzylic methyl substitutionsShue, Ho-Jane / Chen, Xiao / Schwerdt, John H. et al. | 2005
- 1070
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6-Acylamino-2-amino-4-methylquinolines as potent melanin-concentrating hormone 1 receptor antagonists: Structure–activity exploration of eastern and western partsUlven, Trond / Little, Paul Brian / Receveur, Jean-Marie et al. | 2005
- 1070
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6-Acylamino-2-amino-4-methylquinolines as potent melanin-concentrating hormone 1 receptor antagonists: Structure#8211activity exploration of eastern and western partsUlven, Trond et al. | 2006
- 1076
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Inhibiting protein–amyloid interactions with small molecules: A surface chemistry approachInbar, Petra / Yang, Jerry et al. | 2005
- 1076
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Inhibiting protein#8211amyloid interactions with small molecules: A surface chemistry approachInbar, Petra et al. | 2006
- 1080
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Pyridazines part 41: Synthesis, antiplatelet activity and SAR of 2,4,6-substituted 5-(3-oxo-3-phenylprop-1-en-1-yl)- or 5-(3-phenylprop-2-enoyl)pyridazin-3(2H)-onesCrespo, Abel / Meyers, Caroline / Coelho, Alberto et al. | 2005
- 1084
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3-Amino-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazoles: A new class of CDK2 inhibitorsPevarello, Paolo / Fancelli, Daniele / Vulpetti, Anna et al. | 2005
- CO2
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Editorial Board| 2005
- I
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Instructions to contributors| 2005