BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS
Die Inhaltsverzeichnisse werden automatisch erzeugt und basieren auf den im Index des TIB-Portals verfügbaren Einzelnachweisen der enthaltenen Beiträge. Die Anzeige der Inhaltsverzeichnisse kann daher unvollständig oder lückenhaft sein.
Inhaltsverzeichnis
- 4727
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Graphical contents list| 2013
- 4741
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A medicinal chemists’ guide to the unique difficulties of lead optimization for tuberculosisDartois, Véronique / Barry, Clifton E. 3rd et al. | 2013
- 4751
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Peripherally restricted CB1 receptor blockersChorvat, Robert J. et al. | 2013
- 4761
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Selective orexin receptor antagonistsLebold, Terry P. / Bonaventure, Pascal / Shireman, Brock T. et al. | 2013
- 4770
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Increase of anti-HIV activity of C-peptide fusion inhibitors using a bivalent drug design approachLing, Yanbo / Xue, Huifang / Jiang, Xifeng et al. | 2013
- 4774
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Peroxisome proliferator-activated receptor delta antagonists inhibit hepatitis C virus RNA replicationBan, Shintaro / Ueda, Youki / Ohashi, Masao et al. | 2013
- 4779
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Antithrombotic effects of LB30870, a potent, orally active, selective and direct thrombin inhibitor, and pharmacokinetics of its prodrugPark, Hee Dong / Lee, Sung-Hack / Kim, Tae Hoon et al. | 2013
- 4785
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Design, synthesis, and anti-tumor activities of novel triphenylethylene–coumarin hybrids, and their interactions with Ct-DNAChen, Hua / Li, Shuai / Yao, Yuchao et al. | 2013
- 4790
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Identification of novel HDAC inhibitors through cell based screening and their evaluation as potential anticancer agentsWang, Tong / Sepulveda, Mario / Gonzales, Paul et al. | 2013
- 4794
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Design and synthesis of bicyclic heterocycles as potent γ-secretase modulatorsOehlrich, Daniel / Rombouts, Frederik J.R. / Berthelot, Didier et al. | 2013
- 4794
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Design and synthesis of bicyclic heterocycles as potent @c-secretase modulatorsOehlrich, D. / Rombouts, F. J. R. / Berthelot, D. et al. | 2013
- 4801
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Promotion effect of constituents from the root of Polygonum multiflorum on hair growthSun, Ya Nan / Cui, Long / Li, Wei et al. | 2013
- 4806
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Semisynthesis and quantitative structure–activity relationship (QSAR) study of some cholesterol-based hydrazone derivatives as insecticidal agentsYang, Chun / Shao, Yonghua / Zhi, Xiaoyan et al. | 2013
- 4813
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Adipogenetic effects of retrofractamide A derivatives in 3T3-L1 cellsMourad, Ahmed Aboul-Fotouh / Nakamura, Seikou / Ueno, Tsubasa et al. | 2013
- 4817
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Investigation into the functional impact of the vancomycin C-ring aryl chloridePinchman, Joseph R. / Boger, Dale L. et al. | 2013
- 4820
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A convenient synthesis of lubeluzole and its enantiomer: Evaluation as chemosensitizing agents on human ovarian adenocarcinoma and lung carcinoma cellsCavalluzzi, Maria Maddalena / Viale, Maurizio / Bruno, Claudio et al. | 2013
- 4824
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3,4-Dihydroxy- and 3,4-methylenedioxy- phenanthrene-type alkaloids with high selectivity for D2 dopamine receptorMoreno, Laura / Cabedo, Nuria / Ivorra, María Dolores et al. | 2013
- 4828
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Synthesis and antifungal activities of miltefosine analogsRavu, Ranga Rao / Chen, Ying-Lien / Jacob, Melissa R. et al. | 2013
- 4832
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Novel selective inhibitors of aminopeptidases that generate antigenic peptidesPapakyriakou, Athanasios / Zervoudi, Efthalia / Theodorakis, Emmanuel A. et al. | 2013
- 4837
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Synthesis of quaternary α-amino acid-based arginase inhibitors via the Ugi reactionGolebiowski, Adam / Whitehouse, Darren / Beckett, R. Paul et al. | 2013
- 4837
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Synthesis of quaternary @a-amino acid-based arginase inhibitors via the Ugi reactionGolebiowski, A. / Whitehouse, D. / Beckett, R. P. et al. | 2013
- 4842
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QM-polarized ligand docking accurately predicts the trend in binding affinity of a series of arylmethylene quinuclidine-like derivatives at the @a4@b2 and @a3@b4 nicotinic acetylcholine receptors (nAChRs)Kombo, D. C. / Grinevich, V. P. / Hauser, T. A. et al. | 2013
- 4842
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QM-polarized ligand docking accurately predicts the trend in binding affinity of a series of arylmethylene quinuclidine-like derivatives at the α4β2 and α3β4 nicotinic acetylcholine receptors (nAChRs)Kombo, David C. / Grinevich, Vladimir P. / Hauser, Terry A. et al. | 2013
- 4848
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A FRET-based assay for the discovery of West Nile Virus NS2B-NS3 protease inhibitorsAdamek, Rebecca N. / Maniquis, Roxanne V. / Khakoo, Sabaha et al. | 2013
- 4851
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Selective activity of 2,4-diaryl-1,2,3,4-tetrahydroquinolines on Trypanosoma cruzi epimastigotes and amastigotes expressing β-galactosidaseFonseca-Berzal, Cristina / Merchán Arenas, Diego R. / Romero Bohórquez, Arnold R. et al. | 2013
- 4851
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Selective activity of 2,4-diaryl-1,2,3,4-tetrahydroquinolines on Trypanosoma cruzi epimastigotes and amastigotes expressing @b-galactosidaseFonseca-Berzal, C. / Merchan Arenas, D. R. / Romero Bohorquez, A. R. et al. | 2013
- 4857
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Synthesis and SAR of 4-aminocyclopentapyrrolidines as orally active N-type calcium channel inhibitors for inflammatory and neuropathic painBeebe, Xenia / Yeung, Clinton M. / Darczak, Daria et al. | 2013
- 4862
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Psammaplysin F: A unique inhibitor of bacterial chromosomal partitioningRamsey, Deborah M. / Amirul Islam, Md. / Turnbull, Lynne et al. | 2013
- 4867
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Neuroactive diol and acyloin metabolites from cone snail-associated bacteriaLin, Zhenjian / Marett, Lenny / Hughen, Ronald W. et al. | 2013
- 4870
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Access to 7@b-analogs of codeine with mixed @m/@d agonist activity via 6,7-@a-epoxide openingMagnus, P. / Ghavimi, B. / Coe, J. W. et al. | 2013
- 4870
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Access to 7β-analogs of codeine with mixed μ/δ agonist activity via 6,7-α-epoxide openingMagnus, Philip / Ghavimi, Bahman / Coe, Jotham W. et al. | 2013
- 4875
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Identification of 2,3-dihydro-1H-pyrrolo[3,4-c]pyridine-derived ureas as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT)Dragovich, Peter S. / Bair, Kenneth W. / Baumeister, Timm et al. | 2013
- 4886
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Anticonvulsant properties of histamine H3 receptor ligands belonging to N-substituted carbamates of imidazopropanolSadek, Bassem / Shehab, Safa / Więcek, Małgorzata et al. | 2013
- 4892
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De novo design and synthesis of a @m-conotoxin KIIIA peptidomimeticBrady, R. M. / Zhang, M. / Gable, R. et al. | 2013
- 4892
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De novo design and synthesis of a μ-conotoxin KIIIA peptidomimeticBrady, Ryan M. / Zhang, Minmin / Gable, Robert et al. | 2013
- 4896
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Synthesis and binary QSAR study of antitubercular quinolylhydrazidesManvar, Atul / Khedkar, Vijay / Patel, Jignesh et al. | 2013
- 4903
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A novel necroptosis inhibitor—necrostatin-21 and its SAR studyWu, Zhijie / Li, Ying / Cai, Yu et al. | 2013
- 4907
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Search for a novel SIRT1 activator: Structural modification of SRT1720 and biological evaluationMatsuya, Yuji / Kobayashi, Yuta / Uchida, Sayumi et al. | 2013
- 4911
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Discovery of 7-azaindole based anaplastic lymphoma kinase (ALK) inhibitors: Wild type and mutant (L1196M) active compounds with unique binding modeGummadi, Venkateshwar Rao / Rajagopalan, Sujatha / Looi, Chung-Yeng et al. | 2013
- 4919
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Synthesis and structure–activity relationships evaluation of benzothiazinone derivatives as potential anti-tubercular agentsGao, Chao / Ye, Ting-Hong / Wang, Ning-Yu et al. | 2013
- 4923
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Structure–cytotoxic activity relationship of sesquilignan, morinol AYamauchi, Satoshi / Kawahara, Saya / Wukirsari, Tuti et al. | 2013
- 4931
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Synthesis and biological evaluation of amino analogs of Ludartin: Potent and selective cytotoxic agentsLone, Shabir H. / Bhat, Khursheed A. / Shakeel-u-Rehman et al. | 2013
- 4935
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Syntheses of procyanidin B2 and B3 gallate derivatives using equimolar condensation mediated by Yb(OTf)3 and their antitumor activitiesSuda, Manato / Katoh, Miyuki / Toda, Kazuya et al. | 2013
- 4940
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A monosaccharide-modified peptide phage library for screening of ligands to carbohydrate-binding proteinsArai, Kanako / Tsutsumi, Hiroshi / Mihara, Hisakazu et al. | 2013
- 4944
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Exploration of the 5-bromopyrimidin-4(3H)-ones as potent inhibitors of PDE5Gong, Xudong / Wang, Guan / Ren, Jing et al. | 2013
- 4948
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Novel β-dicarbonyl derivatives as inhibitors of aminopeptidase N (APN)Ma, Chunhua / Li, Xiaoguang / liang, Xuewu et al. | 2013
- 4948
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Novel @b-dicarbonyl derivatives as inhibitors of aminopeptidase N (APN)Ma, C. / Li, X. / liang, X. et al. | 2013
- 4953
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Identification of GNE-293, a potent and selective PI3Kδ inhibitor: Navigating in vitro genotoxicity while improving potency and selectivitySafina, Brian S. / Sweeney, Zachary K. / Li, Jun et al. | 2013
- 4953
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Identification of GNE-293, a potent and selective PI3K@d inhibitor: Navigating in vitro genotoxicity while improving potency and selectivitySafina, B. S. / Sweeney, Z. K. / Li, J. et al. | 2013
- 4960
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Design, synthesis and biological evaluation of novel triaryl (Z)-olefins as tamoxifen analoguesAbdellatif, Khaled R.A. / Belal, Amany / Omar, Hany A. et al. | 2013
- 4964
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Preparation and antitrypanosomal activity of secochiliolide acid derivativesSiless, Gastón E. / Lozano, Esteban / Sánchez, Marianela et al. | 2013
- 4968
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Antibacterial activity of quinoxalines, quinazolines, and 1,5-naphthyridinesParhi, Ajit K. / Zhang, Yongzheng / Saionz, Kurt W. et al. | 2013
- 4975
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Truncation of the peptide sequence in bifunctional ligands with mu and delta opioid receptor agonist and neurokinin 1 receptor antagonist activitiesNair, Padma / Yamamoto, Takashi / Largent-Milnes, Tally M. et al. | 2013
- 4979
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The discovery of potent blockers of the canonical transient receptor channels, TRPC3 and TRPC6, based on an anilino-thiazole pharmacophoreWashburn, David G. / Holt, Dennis A. / Dodson, Jason et al. | 2013
- 4985
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Selected furanochalcones as inhibitors of monoamine oxidaseRobinson, Sarel J. / Petzer, Jacobus P. / Petzer, Anél et al. | 2013
- 4990
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Synthesis and cytotoxic activity evaluation of 2,3-thiazolidin-4-one derivatives on human breast cancer cell linesSala, Marina / Chimento, Adele / Saturnino, Carmela et al. | 2013
- 4996
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Synthesis and structure activity relationship of imidazo[1,2-a]pyridine-8-carboxamides as a novel antimycobacterial lead seriesRamachandran, Sreekanth / Panda, Manoranjan / Mukherjee, Kakoli et al. | 2013
- 5002
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Regioselective synthesis of 6-aryl-benzo[h][1,2,4]-triazolo[5,1-b]quinazoline-7,8-diones as potent antitumoral agentswu, Liqiang / Zhang, Chong / Li, Weilin et al. | 2013
- 5006
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Convenient synthesis of heterobifunctional poly(ethylene glycol) suitable for the functionalization of iron oxide nanoparticles for biomedical applicationsPassemard, Solène / Staedler, Davide / Učňová, Lucia et al. | 2013
- 5011
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Structure activity relationship study of benzo[d]thiazol-2(3H)one based σ receptor ligandsBhat, Rohit / Fishback, James A. / Matsumoto, Rae R. et al. | 2013
- 5011
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Structure activity relationship study of benzo[d]thiazol-2(3H)one based @s receptor ligandsBhat, R. / Fishback, J. A. / Matsumoto, R. R. et al. | 2013
- 5014
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2-Amino-[1,2,4]triazolo[1,5-a]pyridines as JAK2 inhibitorsSiu, Michael / Pastor, Richard / Liu, Wendy et al. | 2013
- 5022
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Corrigendum to “The design and synthesis of indazole and pyrazolopyridine based glucokinase activators for the treatment of Type 2 diabetes mellitus” [Bioorg. Med. Chem. Lett. 22 (2012) 7100–7105]Pfefferkorn, Jeffrey A. / Tu, Meihua / Filipski, Kevin J. et al. | 2013
- IFC
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Editorial board| 2013