BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS
Die Inhaltsverzeichnisse werden automatisch erzeugt und basieren auf den im Index des TIB-Portals verfügbaren Einzelnachweisen der enthaltenen Beiträge. Die Anzeige der Inhaltsverzeichnisse kann daher unvollständig oder lückenhaft sein.
Inhaltsverzeichnis
- 6017
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Graphical contents list| 2008
- 6033
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Highly potent and selective chiral inhibitors of PDE5: An illustration of Pfeiffer’s ruleBunnage, Mark E. / Mathias, John P. / Wood, Anthony et al. | 2008
- 6037
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Rotational deviation of 3-acetyl group from cyclic tetrapyrrole p-plane in synthetic bacteriochlorophyll-a analogs by 20-substitutionTamiaki, H. / Kotegawa, Y. / Mizutani, K. et al. | 2008
- 6037
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Rotational deviation of 3-acetyl group from cyclic tetrapyrrole π-plane in synthetic bacteriochlorophyll-a analogs by 20-substitutionTamiaki, Hitoshi / Kotegawa, Yuki / Mizutani, Keisuke et al. | 2008
- 6041
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Development of novel 2-[4-(aminoalkoxy)phenyl]-4(3H)-quinazolinone derivatives as potent and selective histamine H3 receptor inverse agonistsMizutani, Takashi / Nagase, Tsuyoshi / Ito, Sayaka et al. | 2008
- 6046
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Pterocarpans and flavanones from Sophora flavescens displaying potent neuraminidase inhibitionRyu, Young Bae / Curtis-Long, Marcus J. / Kim, Jin Hyo et al. | 2008
- 6050
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Pyrrospirones A and B, apoptosis inducers in HL-60 cells, from an endophytic fungus, Neonectria ramulariae Wollenw KS-246Shiono, Yoshihito / Shimanuki, Keiko / Hiramatsu, Fuminori et al. | 2008
- 6054
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Synthesis and preliminary pharmacological evaluation of N-2-(4-(4-(2-substitutedthiazol-4-yl) piperazin-1-yl)-2-oxoethyl)acetamides as novel atypical antipsychotic agentsSekhar, K.V.G. Chandra / Rao, V.S. / Vyas, Devambatla Ravi Kumar et al. | 2008
- 6058
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Synthesis and characterization of novel natural product-Gd(III) MRI contrast agent conjugatesEfthimiadou, Eleni K. / Katsarou, Maria E. / Fardis, Michael et al. | 2008
- 6062
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Novel 3,3-disubstituted pyrrolidines as selective triple serotonin/norepinephrine/dopamine reuptake inhibitorsBannwart, Linda M. / Carter, David S. / Cai, Hai-Ying et al. | 2008
- 6067
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Synthesis and activity of novel 1- or 3-(3-amino-1-phenyl propyl)-1,3-dihydro-2H-benzimidazol-2-ones as selective norepinephrine reuptake inhibitorsZhang, Puwen / Terefenko, Eugene A. / McComas, Casey C. et al. | 2008
- 6071
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Trifluoromethylpyrimidine-based inhibitors of proline-rich tyrosine kinase 2 (PYK2): Structure–activity relationships and strategies for the elimination of reactive metabolite formationWalker, Daniel P. / Christopher Bi, F. / Kalgutkar, Amit S. et al. | 2008
- 6078
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Studies of the metabolic stability in cells of 5-(trifluoroacetyl)thiophene-2-carboxamides and identification of more stable class II histone deacetylase (HDAC) inhibitorsScarpelli, Rita / Di Marco, Annalise / Ferrigno, Federica et al. | 2008
- 6083
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2-Trifluoroacetylthiophene oxadiazoles as potent and selective class II human histone deacetylase inhibitorsMuraglia, Ester / Altamura, Sergio / Branca, Danila et al. | 2008
- 6088
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Quantitative structure–activity relationship of phenoxyphenyl-methanamine compounds with 5HT2A, SERT, and hERG activitiesMente, Scot / Gallaschun, Randall / Schmidt, Anne et al. | 2008
- 6093
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Identification of KD5170: A novel mercaptoketone-based histone deacetylase inhibitorPayne, Joseph E. / Bonnefous, Céline / Hassig, Christian A. et al. | 2008
- 6097
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The first X-ray crystal structure of the glucocorticoid receptor bound to a non-steroidal agonistMadauss, Kevin P. / Bledsoe, Randy K. / Mclay, Iain et al. | 2008
- 6100
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Exploring 8-benzyl pteridine-6,7-diones as inhibitors of glutamate racemase (MurI) in Gram-positive bacteriaBreault, Gloria A. / Comita-Prevoir, Janelle / Eyermann, Charles J. et al. | 2008
- 6104
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SAR profiles of spirocyclic nicotinamide derived selective HDAC1/HDAC2 inhibitors (SHI-1:2)Methot, Joey L. / Hamblett, Christopher L. / Mampreian, Dawn M. et al. | 2008
- 6110
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Non-nucleoside inhibitors of the hepatitis C virus NS5B RNA-dependant RNA polymerase: 2-Aryl-3-heteroaryl-1,3-thiazolidin-4-one derivativesRawal, Ravindra K. / Katti, S.B. / Kaushik-Basu, Neerja et al. | 2008
- 6115
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Interaction of ladder-shaped polyethers with transmembrane α-helix of glycophorin A as evidenced by saturation transfer difference NMR and surface plasmon resonanceUjihara, Satoru / Oishi, Tohru / Torikai, Kohei et al. | 2008
- 6115
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Interaction of ladder-shaped polyethers with transmembrane a-helix of glycophorin A as evidenced by saturation transfer difference NMR and surface plasmon resonanceUjihara, S. / Oishi, T. / Torikai, K. et al. | 2008
- 6119
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In situ blood–brain barrier permeability of a C-10 paclitaxel carbamateBallatore, Carlo / Zhang, Bin / Trojanowski, John Q. et al. | 2008
- 6122
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Potent benzimidazolone-based CGRP receptor antagonistsTheberge, Cory R. / Bednar, Rodney A. / Bell, Ian M. et al. | 2008
- 6126
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Radiolytic one-electron reduction characteristics of tyrosine derivative caged by 2-oxopropyl groupTanabe, Kazuhito / Ebihara, Masahiko / Hirata, Nao et al. | 2008
- 6130
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Cathepsin B inhibitory activities of three new phthalate derivatives isolated from seahorse, Hippocampus Kuda BleelerLi, Yong / Qian, Zhong-Ji / Kim, Se-Kwon et al. | 2008
- 6135
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Gold nanoparticles functionalised by Gd-complex of DTPA-bis(amide) conjugate of glutathione as an MRI contrast agentPark, Ji-Ae / Reddy, Pattubala A.N. / Kim, Hee-Kyung et al. | 2008
- 6138
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Synthesis of celecoxib analogs that possess a N-hydroxypyrid-2(1H)one 5-lipoxygenase pharmacophore: Biological evaluation as dual inhibitors of cyclooxygenases and 5-lipoxygenase with anti-inflammatory activityChowdhury, Morshed Alam / Abdellatif, Khaled R.A. / Dong, Ying et al. | 2008
- 6142
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Pyrrolo-pyrimidones: A novel class of MK2 inhibitors with potent cellular activitySchlapbach, Achim / Feifel, Roland / Hawtin, Stuart et al. | 2008
- 6147
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Synthesis of 3,6-diazabicyclo[3.1.1]heptanes as novel ligands for neuronal nicotinic acetylcholine receptorsMurineddu, Gabriele / Murruzzu, Caterina / Curzu, Maria M. et al. | 2008
- 6151
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Synthesis and structure–activity relationships of selective norepinephrine reuptake inhibitors (sNRI) with improved pharmaceutical characteristicsPontillo, Joseph / Wu, Dongpei / Ching, Brett et al. | 2008
- 6156
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Comparisons of the influenza virus A M2 channel binding affinities, anti-influenza virus potencies and NMDA antagonistic activities of 2-alkyl-2-aminoadamantanes and analoguesKolocouris, Antonios / Spearpoint, Philip / Martin, Stephen R. et al. | 2008
- 6161
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Peptides based on CcdB protein as novel inhibitors of bacterial topoisomerasesTrovatti, Eliane / Cotrim, Camila A. / Garrido, Saulo S. et al. | 2008
- 6165
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Synthesis, tubulin assembly, and antiproliferative activity against MCF7 and NCI/ADR-RES cancer cells of 10-O-acetyl-5prime-hydroxybutitaxelGe, H. / Wang, J. / Kayser, M. M. et al. | 2008
- 6165
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Synthesis, tubulin assembly, and antiproliferative activity against MCF7 and NCI/ADR-RES cancer cells of 10-O-acetyl-5′-hydroxybutitaxelGe, Haibo / Wang, Jianmei / Kayser, Margaret M. et al. | 2008
- 6168
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New synthesis and evaluation of enantiomers of 7-methyl-2-exo-(3′-iodo-5′-pyridinyl)-7-azabicyclo[2.2.1]heptane as stereoselective ligands for PET imaging of nicotinic acetylcholine receptorsGao, Yongjun / Horti, Andrew G. / Kuwabara, Hiroto et al. | 2008
- 6168
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New synthesis and evaluation of enantiomers of 7-methyl-2-exo-(3prime-iodo-5prime-pyridinyl)-7-azabicyclo[2.2.1]heptane as stereoselective ligands for PET imaging of nicotinic acetylcholine receptorsGao, Y. / Horti, A. G. / Kuwabara, H. et al. | 2008
- 6171
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2-Alkylamino- and alkoxy-substituted 2-amino-1,3,4-oxadiazoles—O-Alkyl benzohydroxamate esters replacements retain the desired inhibition and selectivity against MEK (MAP ERK kinase)Warmus, Joseph S. / Flamme, Cathlin / Zhang, Lu Yan et al. | 2008
- 6175
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Design at the atomic level: Design of biaryloxazolidinones as potent orally active antibioticsZhou, Jiacheng / Bhattacharjee, Ashoke / Chen, Shili et al. | 2008
- 6179
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Design at the atomic level: Generation of novel hybrid biaryloxazolidinones as promising new antibioticsZhou, Jiacheng / Bhattacharjee, Ashoke / Chen, Shili et al. | 2008
- 6184
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A bulge binding agent with novel wedge-shape topology for stimulation of DNA triplet repeat strand slippage synthesisLiu, Liangliang / Li, Heyang / Yi, Long et al. | 2008
- 6189
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Discovery of novel, potent and bioavailable proline-urea based macrocyclic HCV NS3/4A protease inhibitorsVendeville, Sandrine / Nilsson, Magnus / Kock, Herman de et al. | 2008
- 6194
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Carbonic anhydrase activators: Activation of the archaeal β-class (Cab) and γ-class (Cam) carbonic anhydrases with amino acids and aminesInnocenti, Alessio / Zimmerman, Sabrina A. / Scozzafava, Andrea et al. | 2008
- 6194
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Carbonic anhydrase activators: Activation of the archaeal b-class (Cab) and g-class (Cam) carbonic anhydrases with amino acids and aminesInnocenti, A. / Zimmerman, S. A. / Scozzafava, A. et al. | 2008
- 6199
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New cyclic somatostatin analogues containing a pyrazinone ring: Importance of Tyr for antiproliferative activityMiyazaki, Anna / Tsuda, Yuko / Fukushima, Shoji et al. | 2008
- 6202
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Possible involvement of radical intermediates in the inhibition of cysteine proteases by allenyl esters and amidesTakeuchi, Yoshio / Fujiwara, Tomoya / Shimone, Yoshihito et al. | 2008
- 6206
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The design, synthesis and biological evaluation of 7-alkoxy-4-heteroarylamino-3-cyanoquinolines as dual inhibitors of c-Src and iNOSCao, Xin / You, Qi-Dong / Li, Zhi-Yu et al. | 2008
- 6210
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Naphthalimide intercalators with chiral amino side chains: Effects of chirality on DNA binding, photodamage and antitumor cytotoxicityYang, Qing / Yang, Peng / Qian, Xuhong et al. | 2008
- 6214
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Imidazo[5,1-f][1,2,4]triazin-2-amines as novel inhibitors of polo-like kinase 1Cheung, M. / Kuntz, K.W. / Pobanz, M. et al. | 2008
- 6218
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2-Aminobenzimidazoles as potent ITK antagonists: trans-stilbene-like moieties targeting the kinase specificity pocketLo, Ho Yin / Bentzien, Jörg / Fleck, Roman W. et al. | 2008
- 6222
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Tetrahydro-4-quinolinamines identified as novel P2Y1 receptor antagonistsMorales-Ramos, Ángel I. / Mecom, John S. / Kiesow, Terry J. et al. | 2008
- 6227
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Synthetic chalcones as efficient inhibitors of Mycobacterium tuberculosis protein tyrosine phosphatase PtpAChiaradia, Louise Domeneghini / Mascarello, Alessandra / Purificação, Marcela et al. | 2008
- 6231
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Discovery and SAR of novel 4-thiazolyl-2-phenylaminopyrimidines as potent inhibitors of spleen tyrosine kinase (SYK)Farmer, Luc J. / Bemis, Guy / Britt, Shawn D. et al. | 2008
- 6236
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Modifications of the isonipecotic acid fragment of SNS-032: Analogs with improved permeability and lower efflux ratioFan, Junfa / Fahr, Bruce / Stockett, David et al. | 2008
- 6240
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Synthesis of new sulfonate and phosphonate derivatives for cation-independent mannose 6-phosphate receptor targetingJeanjean, Audrey / Gary-Bobo, Magali / Nirdé, Philippe et al. | 2008
- 6244
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Clubbed [1,2,3] triazoles by fluorine benzimidazole: A novel approach to H37Rv inhibitors as a potential treatment for tuberculosisGill, Charansingh / Jadhav, Ganesh / Shaikh, Mohammad et al. | 2008
- 6248
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Synthesis and Ribonucleotide reductase inhibitory activity of thiosemicarbazonesKrishnan, Kesavan / Prathiba, Kumari / Jayaprakash, Venkatesan et al. | 2008
- 6251
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The discovery of equipotent PPARa/g dual activatorsMartres, P. / Faucher, N. / Laroze, A. et al. | 2008
- 6251
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The discovery of equipotent PPARα/γ dual activatorsMartres, Paul / Faucher, Nicolas / Laroze, Alain et al. | 2008
- 6255
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RNA bandages for photoregulating in vitro protein synthesisRichards, Julia L. / Tang, XinJing / Turetsky, Anna et al. | 2008
- 6259
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Discovery of 1-benzoyl-3-cyanopyrrolo[1,2-a]quinolines as a new series of apoptosis inducers using a cell- and caspase-based high-throughput screening assay. Part 1: Structure–activity relationships of the 1- and 3-positionsKemnitzer, William / Kuemmerle, Jared / Jiang, Songchun et al. | 2008
- 6265
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Synthesis of Arabino glycosyl triazoles as potential inhibitors of mycobacterial cell wall biosynthesisWilkinson, Brendan L. / Long, Hilary / Sim, Edith et al. | 2008
- 6268
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Total synthesis and biological evaluation of potent analogues of dictyostatin: Modification of the C2–C6 dienoate regionPaterson, Ian / Gardner, Nicola M. / Guzmán, Esther et al. | 2008
- 6273
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Dihydroxylphenyl amides as inhibitors of the Hsp90 molecular chaperoneKung, Pei-Pei / Funk, Lee / Meng, Jerry et al. | 2008
- 6279
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Quinazolines as potent and highly selective PDE5 inhibitors as potential therapeutics for male erectile dysfunctionKim, Young Hoon / Choi, Hojin / Lee, Jaekwang et al. | 2008
- 6283
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3D QSAR CoMFA/CoMSIA, molecular docking and molecular dynamics studies of fullerene-based HIV-1 PR inhibitorsDurdagi, Serdar / Mavromoustakos, Thomas / Papadopoulos, Manthos G. et al. | 2008
- 6290
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Validation of high-affinity binding sites for succinic acid through distinguishable binding of gamma-hydroxybutyric acid receptor-specific NCS 382 antipodesMolnár, Tünde / Visy, Júlia / Simon, Ágnes et al. | 2008
- 6293
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Bacterial translation inhibitors, 1-acylindazol-3-ols as anthranilic acid mimicsStiff, Cory / Graber, David R. / Thorarensen, Atli et al. | 2007
- I
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Instructions to contributors| 2008
- IFC
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Editorial board| 2008