Organic Process Research & Development
Die Inhaltsverzeichnisse werden automatisch erzeugt und basieren auf den im Index des TIB-Portals verfügbaren Einzelnachweisen der enthaltenen Beiträge. Die Anzeige der Inhaltsverzeichnisse kann daher unvollständig oder lückenhaft sein.
Inhaltsverzeichnis
- 417
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Process Chemi-Stories in Japan| 2019
- 418
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The Spirit of the Japanese Society for Process ChemistrySajiki, Hironao et al. | 2019
- 419
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Efficient Azacycle Formations Developed in Japanese Pharmaceutical Industries: Elegancy, Logistics, and Training (ELT) “Sandwich” for Process ChemistsMizufune, Hideya et al. | 2019
- 443
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Catalytic Deprotonative α‑Formylation of Heteroarenes by an Amide Base Generated in Situ from Tetramethylammonium Fluoride and Tris(trimethylsilyl)amineShigeno, Masanori / Fujii, Yuki / Kajima, Akihisa et al. | 2019
- 452
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Development of Asymmetric Transfer Hydrogenation with a Bifunctional Oxo-Tethered Ruthenium Catalyst in Flow for the Synthesis of a Ceramide (d-erythro-CER[NDS])Touge, Taichiro / Kuwana, Masahiro / Komatsuki, Yasuhiro et al. | 2019
- 462
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Application of Thiol-Modified Dual-Pore Silica Beads as a Practical Scavenger of Leached Palladium Catalyst in C–C Coupling ReactionsYamada, Tsuyoshi / Matsuo, Tomohiro / Ogawa, Aya et al. | 2019
- 470
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Development of a Synthetic Process for K‑8986, an H1-Receptor AntagonistFukuda, Tomoaki / Hara, Takeaki / Ina, Shinji et al. | 2019
- 477
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Stereoselective Acetalization for the Synthesis of Liquid-Crystal Compounds Possessing a trans-2,5-Disubstituted 1,3-Dioxane Ring with Saturated Aqueous Solutions of Inorganic SaltsMaebayashi, Haruki / Fuchigami, Tsugumichi / Gotoh, Yasuyuki et al. | 2019
- 484
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Practical Preparation of a 1,3,5-Trisubstituted Pyridazin-4(1H)‑one Using Selective C1 Unit Insertion and CyclizationSuzuki, Akihiro / Fukuda, Naohiro / Kajiwara, Takeshi et al. | 2019
- 493
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Self-Assembled Polymeric Pyridine Copper Catalysts for Huisgen Cycloaddition with Alkynes and Acetylene Gas: Application in Synthesis of TazobactamHu, Hao / Ohno, Aya / Sato, Takuma et al. | 2019
- 499
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Process Development of an Efficient and Cost-Effective Telescoping Route to a Key Synthetic Precursor for the Preparation of a Renin InhibitorNonoyama, Akihito / Nakai, Yoshio / Lee, Shoukou et al. | 2019
- 512
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Improved Manufacturing Route and Polymorphic Control of a Potent and Selective Anaplastic Lymphoma Kinase (ALK) Inhibitor ASP3026Takahama, Yuji / Obitsu, Kazuyoshi / Takeguchi, Kazuhiro et al. | 2019
- 524
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Development of an Efficient Manufacturing Process for a Key Intermediate in the Synthesis of EdoxabanMichida, Makoto / Ishikawa, Hideaki / Kaneda, Takeshi et al. | 2019
- 535
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Construction of a (3aR,4R,9bR)‑Hexahydropyrroloquinoline by Stereoselective Hydrogen-Mediated Domino CyclizationYamada, Masatoshi / Usutani, Hirotsugu / Ito, Tatsuya et al. | 2019
- 548
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Synthesis of Tofogliflozin as an SGLT2 Inhibitor via Construction of Dihydroisobenzofuran by Intramolecular [4 + 2] CycloadditionMurakata, Masatoshi / Kawase, Akira / Kimura, Nobuaki et al. | 2019
- 558
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Practical and Scalable Synthetic Method for Preparation of Dolutegravir Sodium: Improvement of a Synthetic Route for Large-Scale SynthesisAoyama, Yasunori / Hakogi, Toshikazu / Fukui, Yuki et al. | 2019
- 565
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Practical Synthetic Method for the Preparation of Pyrone Diesters: An Efficient Synthetic Route for the Synthesis of Dolutegravir SodiumYasukata, Tatsuro / Masui, Moriyasu / Ikarashi, Fumiya et al. | 2019
- 571
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Safe and Scalable Aerobic Oxidation by 2‑Azaadamantan-2-ol (AZADOL)/NO x Catalysis: Large-Scale Preparation of Shi’s CatalystSasano, Yusuke / Sato, Hikaru / Tadokoro, Shinsuke et al. | 2019
- 578
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Scalable Process Design for a PDE10A Inhibitor Consisting of Pyrazolopyrimidine and Quinoxaline as Key UnitsYamagami, Takafumi / Kobayashi, Ryo / Moriyama, Noriaki et al. | 2019
- 588
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Ammonium Salt-Accelerated Hydrazinolysis of Unactivated Amides: Mechanistic Investigation and Application to a Microwave Flow ProcessNoshita, Megumi / Shimizu, Yuhei / Morimoto, Hiroyuki et al. | 2019
- 595
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Practical Synthesis of Polymethylated Flavones: Nobiletin and Its Desmethyl DerivativesAsakawa, Tomohiro / Sagara, Hiroto / Kanakogi, Masaki et al. | 2019
- 603
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Development of an Efficient Manufacturing Process for E2212 toward Rapid Clinical IntroductionIsomura, Minetaka / Nakamura, Taiju / Kamada, Atsushi et al. | 2019
- 614
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Regioselective Formylation of Pyrrole-2-Carboxylate: Crystalline Vilsmeier Reagent vs Dichloromethyl Alkyl EtherWarashina, Takuya / Matsuura, Daisuke / Sengoku, Tetsuya et al. | 2019
- 619
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Large Scale Synthesis of Chiral (3Z,5Z)‑2,7-Dihydro‑1H‑azepine-Derived Hamari Ligand for General Asymmetric Synthesis of Tailor-Made Amino AcidsTakahashi, Motohiro / Moriwaki, Hiroki / Miwa, Toshio et al. | 2019
- 629
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Expedient Asymmetric Synthesis of (S)‑2-Amino-4,4,4-trifluorobutanoic Acid via Alkylation of Chiral Nucleophilic Glycine EquivalentMei, Haibo / Hiramatsu, Takahiro / Takeda, Ryosuke et al. | 2019
- 635
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Molecular Weight Distribution of Polymers Produced by Anionic Polymerization Enables Mixability EvaluationEndo, Yuta / Furusawa, Mai / Shimazaki, Toshiya et al. | 2019
- 641
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Modeling and Design of a Flow-Microreactor-Based Process for Synthesizing Ionic LiquidsNakahara, Yuichi / Metten, Bert / Tonomura, Osamu et al. | 2019
- 648
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H–D Exchange Deuteration of Arenes at Room TemperatureSawama, Yoshinari / Nakano, Akihiro / Matsuda, Takumi et al. | 2019
- 654
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Efficient and Practical Deacylation Reaction System in a Continuous Packed-Bed ReactorYasukouchi, Hiroaki / Machida, Koji / Nishiyama, Akira et al. | 2019
- 660
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Enantioselective Synthesis of α‑Substituted Serine Derivatives via Cu-Catalyzed Oxidative Desymmetrization of 2‑Amino-1,3-diolsYamamoto, Kosuke / Ishimaru, Shota / Oyama, Tatsuya et al. | 2019
- 667
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Improved Synthesis of Unsymmetrical Carbonate Derivatives Using Calcium SaltsHamada, Tomohito / Okada, Michiaki / Yamauchi, Akiyoshi et al. | 2019
- 674
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Some Items of Interest to Process R&D Chemists and EngineersZhao, Wenyi / Guizzetti, Sylvain / Schwindeman, James A. et al. | 2019