BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS
Die Inhaltsverzeichnisse werden automatisch erzeugt und basieren auf den im Index des TIB-Portals verfügbaren Einzelnachweisen der enthaltenen Beiträge. Die Anzeige der Inhaltsverzeichnisse kann daher unvollständig oder lückenhaft sein.
Inhaltsverzeichnis
- 1
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Instructions to Contributors| 1993
- 477
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Contributors to this issue| 1993
- 481
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Graphical abstracts| 1993
- 497
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Design of C-terminal peptide antagonists of endothelin: structure-activity relationships of ET-[16–21, D-His16]Doherty, A.M. / Cody, W.L. / He, J.X. et al. | 1992
- 497
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Design of C-terminal peptide antagonists of endothelin: structure-activity relationships of ET-1(16-21,D-His16)Doherty, A.M. et al. | 1993
- 503
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Novel dimeric penicillin derived inhibitors of HIV-1 proteinase: interaction with the catalytic aspartatesHolmes, Duncan S. / Clemens, Ian R. / Cobley, Kevin N. et al. | 1992
- 509
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Synthesis and pharmacological properties of BW315C and other inotropic 2-arylimidazo(1 2-alpyrazinesBarraclough, P. et al. | 1993
- 509
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Synthesis and pharmacological properties of BW315c and other inotropic 2-arylimidazo[1,2-a]pyrazinesBarraclough, Paul / Black, James W. / Cambridge, David et al. | 1992
- 515
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Biological activity of 3-aminopropyl (methyl) phosphinic acid, a potent and selective GABAB agonist with CNS activityHowson, William / Mistry, Jaystree / Broekman, marianne et al. | 1993
- 519
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Endothelin receptor ligands. replacement net approach to SAR determination of potent hexapeptidesSpellmeyer, David C. / Brown, Suzy / Stauber, Gregory B. et al. | 1992
- 525
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Janus compounds: dual inhibitors of proteinasesAngelastro, Michael R. / Bey, Philippe / Mehdi, Shujaath et al. | 1992
- 531
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Carbon-carbon bond formation mediated by papain chemically modified by thiazolium saltsSuckling, Colin J. / Zhu, Li-Min et al. | 1992
- 535
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Synthesis of 1,3-diamino-2-hydroxypropane derivatives as pseudosymmetric HIV protease inhibitorsYu, Kuo-Long / Harte, William E. / Spinazze, Patrick et al. | 1992
- 539
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Selective incorporation of D-amino acid esters into peptides catalyzed by alcalase in t-butanolChen, Shui-Tein / Tu, Chen-Chen / Wang, Kung-Tsung et al. | 1992
- 543
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Synthesis of 1-(2-aminopropyl)benzimidazoles, structurally related to the TIBO derivative R82150, with activity against human immunodeficiency virusSwayze, Eric E. / Peiris, Sithumini M. / Kucera, Louis S. et al. | 1992
- 547
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Synthesis and anticonvulsant activity of 3-arylamino-4-aryl-5-(N-4-chlorophenylthiocarbamido)-1,2,4-thiadiazolesSrivastava, Kamna / Pandeya, S.N. et al. | 1992
- 553
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Benzopyran sulfoxide derivatives as New potassium channel activatorYoo, Sung-eun / Kim, Sun-Joo / Shin, Hwa-sup et al. | 1992
- 555
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4-alkylamino-3-bromo-N-alkyl-1,8-naphthalimides: new photochemically activatable antiviral compoundsChang, Shao-Chieh / Archer, Bradley J. / Utecht, Ronald E. et al. | 1992
- 557
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The synthesis of [3H]-losartan, [3H]-L-158,641 and [3H]-L-158,809Rivero, R.A. / Chakravarty, P.K. / Chen, R. et al. | 1992
- 561
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Preparation and in vitro biological evaluation of the enantiomers of the dihydropyridine BMY 20014, a combination calcium and ~1-adrenoreceptor antagonistLawson, J. E. / Poindexter, G. S. / Owens, D. A. et al. | 1993
- 561
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Preparation and in vitro biological evaluation of the enantiomers of the dihydropyridine BMY 20014, a combination calcium and a1-adrenoreceptor antagonistLawson, J.E. et al. | 1993
- 561
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Preparation and in vitro biological evaluation of the enantiomers of the diydropyridine BMY 20014, a combination calcium and α1-adrenoreceptor antagonistLawson, John E. / Poindexter, Graham S. / Owens, Donald A. et al. | 1992
- 565
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“Combretatropones”—hybrids of combretastatin and colchicine. Synthesis and biochemical evaluationAndres, C.J. / Bernardo, J.E. / Yan, Q. et al. | 1992
- 571
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N-oleoyl-1,2,3,4-tetrahydroisoquinolines as conformationally restricted inhibitors of acyl-CoA:cholesterol acyl transferase (ACAT)Dugar, Sundeep / Clader, John W. / Burrier, Robert E. et al. | 1992
- 577
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Synthesis of ingenol analogs with affinity for protein kinase CWinkler, J.D. et al. | 1993
- 577
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Synthesis of ingenol analogs wth affinity for protein kinase CWinkler, Jeffrey D. / Hong, Bor-Cherng / Bahador, Afshin et al. | 1993
- 581
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Centaureidin, a cytotoxic flavone from Polymnia fruticosa, inhibits tubulin polymerizationBeutler, John A. / Cardellina, John H. II / Lin, Chii M. et al. | 1992
- 585
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Regioselective enzyme-catalyzed deacetylation of benzyl phenyl ketone peracetates in organic solventsParmar, Virinder S. / Prasad, Ashok K. / Sharma, Nawal K. et al. | 1992
- 589
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Benzofuran based angiotensin II antagonists related to GR117289: enhancement of potency in vitro and oral activityMiddlemiss, D. / Watson, S.P. / Ross, B.C. et al. | 1992
- 595
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Aromatic isosteres as conformational probes for an isoprenyl subunit: application to inhibitors of squalene synthaseBiller, Scott A. / Abt, Jeffrey W. / Pudzianowski, Andrew T. et al. | 1992
- 601
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Synthesis of 5 glycosylamino pyrimidines. A new class of compounds with potential anb-AIDS activityNogueras, M. et al. | 1993
- 601
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Synthesis of 5-glycosylamino pyrimidines. A new class of compounds with potential anti-aids activityNogueras, Manuel / Sánchez, Adolfo / Melguizo, Manuel et al. | 1992
- 607
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Biselectrostatic interaction with DNA as potential anti-tumor agents: novel 2,11 -diamino-5,8-dithiaundecane derivativesOng, C.W. et al. | 1993
- 607
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Biselectrostatic interaction with DNA as potential anti-turmor agents: novel 2,11-diamino-5,8-dithiaundecane derivativesOng, Chi Wi / Yen, Feng Wen / Chou, Yi Meen et al. | 1992
- 611
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Preparation and evaluation of the antiaggregating and vasodilating activities of the novel 3-nitro-4(3H)-quinazolinone derivativesIto, Shigeru / Ando, Syuzo / Yamaguchi, Kentaro et al. | 1992
- 615
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Nucleosides & nucleotides. 118. Synthesis of oligonucleotides containing a novel 2′-deoxyuridine analogue that carries an aminoalkyl tether at 1′-position; stabilization of duplex formation by an intercalatin group accommodated in the minor grooveDan, Akihito / Yoshimura, Yuichi / Ono, Akira et al. | 1992
- 615
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Nucleosides and nucleotides--CXVIII. Synthesis of oligonucleotides containing a novel 2'-deoxyuridine analogue that carries an aminoalkyl tether at 1'-position; stabilization of duplex formation by an intercalating group accommodated in the minor grooveDan, A. et al. | 1993
- 619
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Chemoselective thioacylation of amino acids. Preparation of the four monothiothymopentin analogs and their biological activityZacharie, Boulos / Martel, Rene / Sauve, Gilles et al. | 1992
- 625
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Design of potent K+ channel openers by pharmacophore modelKoga, Hiroshi / Ohta, Masateru / Sato, Haruhiko et al. | 1992
- 633
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Quaternised renzapride as a potent and selective 5-HT4 receptor agonistBaxter, G.S. / Boyland, P. / Gaster, L.M. et al. | 1992
- 635
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Boric acid effect ont he hydrolysis of 4-nitrophenyl 2,3-dihydroxybenzoate: mimic of borate inhibition of serine proteasesYatsimirsky, Anatoly K. / Bezsoudnova, Katherine Yu. / Sakodinskaya, Inna K. et al. | 1992
- 639
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Synthesis and pharmacological evaluation of the enantiomers of the dopamine autoreceptor agonist PD 135385Jaén, Juan C. / Caprathe, Bradley W. / Wise, Lawrence D. et al. | 1992
- 639
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Synthesis and pharmacological evaluation of the enantiomers of the dopamine autoreceptor agomst PD 135385Jaen, J.C. et al. | 1993
- 645
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The use of neural networks for variable selection in QSARWikel, James H. / Dow, Ernst R. et al. | 1992
- 653
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Demonstration of Baeyer-Villiger oxidation and the course of cyclization in bisfuran ring formation during aflatoxin B1 biosynthesisMcGuire, Sean M. / Townsend, Craig A. et al. | 1993
- 657
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Novel derivatives at the C21 position of the FK-506 macrocycleOrgan, Helen M. / Holmes, Mark A. / Pisano, Judith M. et al. | 1992
- 663
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(±)-7-deazaaristeromycin lacking the hydroxymethyl substituentSiddiqi, Suhaib M. / Raissian, Manijeh / Schneller, Stewart W. et al. | 1992
- 667
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Diastereoselective synthesis of cyclopropyl phenylalanines and their incorporation into dipeptidesCampbell, Malcolm M. / Horwell, David C. / Mahon, Mary F. et al. | 1992
- 671
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U-87947E, a protein quinolone antibacterial agent incorporating a bicyclo[1.1.1]pent-1-yl (BCP) subunitBarbachyn, Michael R. / Hutchinson, Douglas K. / Toops, Dana S. et al. | 1992
- 671
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U-87947E, A potent quinolone antibacterial agent incorporating a bicyclo(1.1.1)pent-1-yl (BCP) subunitBarbachyn, M.R. et al. | 1993
- 677
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The synthesis of novel, rigid and water soluble analogues of coleonol (forskolinChauhan, P.M.S. / Varma, Neeraj / Tandon, J.S. et al. | 1992
- 681
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Enantioselective acetylation of primary amines by Cylindrocarpon radicicolaMouna, A. / Ouazzani, J. / Lenfant, M. et al. | 1992
- 685
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Synthesis of the 4,5 diphosphonate analog of D,L-myo-inositol 4,5-diphosphateLyssikatos, Joseph P. / Bednarski, Mark D. et al. | 1992
- 689
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8-amino(2-aminoethyl)-2′-deoxyadenosine incorporation into DNA by solid phase synthesisParkash, T.P. / Ganesh, K.N. et al. | 1992
- 693
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Synthesis, anti-human immunodeficiency virus, and anti-hepatitis B virus activity of pyrimidine oxathiolane nucleosidesChoi, Woo-Baeng / Yeola, Suresh / Liotta, Dennis C. et al. | 1992
- 697
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Synthesis of the complete glycotetrapeptide core of structurally variant glycopeptidolipidGurjar, M.K. / Saha, U.K. et al. | 1992
- 703
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Synthesis of a biotin conjugate of darglitazone, a new antidiabetic agent. A general protocol for the reversible biotinylation of ketonesHulin, B. / Lau, C.L. / Gibbs, E.M. et al. | 1993
- 707
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Synthesis of Nα-Fmoc-Nε-Nvoc-Lysine and use in the preparation of selectively functionalized peptidesRusiecki, Victoria K. / Warne, Susan A. et al. | 1993
- 707
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Synthesis of Na-Fmoc-Ne-Nvoc-lysine and use in the preparation of selectively functionalized peptidesRusiecki, V.K. et al. | 1993
- 711
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Antiinflammatory β-benzeneethanamines. IIIWilkerson, W.W. / DeLucca, I. / Galbraith, W. et al. | 1993
- 711
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Anti-inflammatory b-benzeneethanamines--IIIWilkerson, W.W. et al. | 1993
- 717
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Total synthesis of D-myo-inositol 3,4,5-trisphosphate and 1,3,4 5-tetrakisphosphateFalck, J.R. et al. | 1993
- 717
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Total synthesis of D-myo-inositole 3,4,5-trisphosphate and 1,3,4,5-tetrakisphosphateFalck, J.R. / Abdali, Abdelkrim et al. | 1993
- 721
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Preliminary structural analysis of the mutations selected by non-nucleoside inhibitors of HIV-1 reverse transcriptaseTong, Liang / Cardozo, Mario / Jones, Paul-James et al. | 1992
- 727
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Probing the S-1′ subsite selectivity of an industrial alkaline protease in anhydrous t-butanolChen, Shui-Tein / Chen, Shiah-Yun / Chen, Hsiu-Jen et al. | 1992
- 735
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Spiroepoxycyclohexadienone dimers: cytotoxic bisalkylating agentsGesson, J.-P. / Mondon, M. et al. | 1992
- 739
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Synthesis of homologs of cysteine suitable for peptide and protein crosslinkingLutgring, Ray / Sujatha, K. / Chmielewski, Jean et al. | 1992
- 743
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Synthesis and antimicrobial activity of 5-thioabbeymycin: limitations of the iminothioether approach to carbinolamine-containing pyrrolobenzodiazepinesKamal, Ahmed / Praveen Reddy, B.S. / Thurston, David E. et al. | 1992
- 747
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Synthesis of methyl α-sialosides N-substituted with large alkanoyl groups, and investigation of their inhibition of agglutination of erythrocytes by influenza A virusSchmid, Walther / Avila, Luis Z. / Williams, Kevin W. et al. | 1993
- 747
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Synthesis of methyl a-sialosides N-substituted with large alkanoyl groups, and investigation of their inhibition of agglutination of erythrocytes by influenza A virusSchmid, W. et al. | 1993
- 753
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A convergent synthesis of 4-(2-benzothiazoyl)piperidines with antihistaminic activityMaynard, G.D. et al. | 1993
- 753
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A convergent synthesis of 4-(2-benzothiazoyl)piperidines with antihistamic activityMaynard, George D. / Cheng, Hsien C. / Kane, John M. et al. | 1993
- 757
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3-hydroxy-3-cyclobutene-1,2-dione: Application of novel carboxylic acid bioisostere to an in-vivo active non-tetrazole angiotensin-II antagonistSoll, R.M. / Kinney, W.A. / Primeau, J. et al. | 1993
- 757
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3-Hydroxy-3-cyclobutene-1,2-dione: application of a novel carboxylic acid bioisostere to an in vivo active non-tetrazole angiotensin II antagonistSoll, R.M. et al. | 1993
- 761
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Synthesis of oligodeoxynucleoside methylphosphonothioatesPadmapriya, A.A. / Agrawal, Sudhir et al. | 1993
- 765
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A systematic evaluation of the inhibition of HIV-1 protease by its C- and N-terminal peptidesFranciskovich, Jeff / Houseman, Kathryn / Mueller, Richard et al. | 1993
- 769
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Cooperative binding of potassium ions to trans-isohumulone in the presence of divalent and trivalent cationsSimpson, William J. / Hughes, Paul S. et al. | 1993
- 773
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elastase inhibitors containing conformationally restricted lactams as P3-P2 dipeptide replacementsSkiles, Jerry W. / Sorcek, Ronald / Jacober, Stephen et al. | 1993
- 779
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Synthesis of myristic acid analogs with anti-HIV activity that may be resistant to metabolic processing by β-oxidationDevadas, Balekudru / Kishore, Nandini S. / Adams, Steven P. et al. | 1992
- 779
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Synthesis of myristic acid analogs with anti-HIV activity that may be resistant to metabolic processing by b-oxidationDevadas, B. et al. | 1993
- 785
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Additions and corrections| 1993
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Announcements| 1993