BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS
Die Inhaltsverzeichnisse werden automatisch erzeugt und basieren auf den im Index des TIB-Portals verfügbaren Einzelnachweisen der enthaltenen Beiträge. Die Anzeige der Inhaltsverzeichnisse kann daher unvollständig oder lückenhaft sein.
Inhaltsverzeichnis
- 1131
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Graphical contents list| 2007
- 1149
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Synthesis of O-prenylated and O-geranylated derivatives of 5-benzylidene2,4-thiazolidinediones and evaluation of their free radical scavenging activity as well as effect on some phase II antioxidant/detoxifying enzymesHossain, Sk. Ugir / Bhattacharya, Sudin et al. | 2006
- 1155
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Synthesis and structure evaluation of a novel cantharimide and its cytotoxicity on SK-Hep-1 hepatoma cellsKok, Stanton Hon Lung / Chui, Chung Hin / Lam, Wing Sze et al. | 2006
- 1160
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Opioids and efflux transporters. Part 1: P-Glycoprotein substrate activity of N-substituted analogs of meperidineMercer, Susan L. / Hassan, Hazem E. / Cunningham, Christopher W. et al. | 2006
- 1163
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Synthesis of new xanthone analogues and their biological activity test—Cytotoxicity, topoisomerase II inhibition, and DNA cross-linking studyWoo, Sangwook / Jung, Ji / Lee, Chongsoon et al. | 2006
- 1167
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Discovery of thienopyridines as Src-family selective Lck inhibitorsAbbott, Lily / Betschmann, Patrick / Burchat, Andrew et al. | 2006
- 1172
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A new visual screening assay for catalytic antibodies with retro-aldol retro-Michael activityShamis, Marina / Barbas, Carlos F. III / Shabat, Doron et al. | 2006
- 1176
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Chiral tetrahydroquinoline derivatives as potent anti-hyperalgesic agents in animal models of sustained inflammation and chronic neuropathic painDi Fabio, Romano / Alvaro, Giuseppe / Bertani, Barbara et al. | 2006
- 1181
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Synthesis and antibacterial evaluation of a novel series of rifabutin-like spirorifamycinsKim, In Ho / Combrink, Keith D. / Ma, Zhenkun et al. | 2006
- 1185
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Synthesis and evaluation of aryl thioxothiazolidinone inhibitors of ADAMTS-5 (Aggrecanase-2)Bursavich, Matthew G. / Gilbert, Adam M. / Lombardi, Sabrina et al. | 2006
- 1189
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5-((1H-Pyrazol-4-yl)methylene)-2-thioxothiazolidin-4-one inhibitors of ADAMTS-5Gilbert, Adam M. / Bursavich, Matthew G. / Lombardi, Sabrina et al. | 2006
- 1193
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Novel pyridinyl and pyrimidinylcarbazole sulfonamides as antiproliferative agentsHu, Laixing / Li, Zhuo-rong / Wang, Yue-ming et al. | 2006
- 1197
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Hydrolytic cleavage of DNA by quercetin zinc(II) complexJun, Tan / Bochu, Wang / Liancai, Zhu et al. | 2006
- 1200
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Discovery of novel, non-acidic 1,5-biaryl pyrrole EP1 receptor antagonistsHall, Adrian / Atkinson, Stephen / Brown, Susan H. et al. | 2006
- 1206
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Synthesis and SAR of 3,5-diamino-piperidine derivatives: Novel antibacterial translation inhibitors as aminoglycoside mimeticsZhou, Yuefen / Gregor, Vlad E. / Ayida, Benjamin K. et al. | 2006
- 1211
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Discovery and preliminary evaluation of 5-(4-phenylbenzyl)oxazole-4-carboxamides as prostacyclin receptor antagonistsBrescia, Marc-Raleigh / Rokosz, Laura L. / Cole, Andrew G. et al. | 2006
- 1216
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In vitro selection of RNA aptamer against Escherichia coli release factor 1Sando, Shinsuke / Ogawa, Atsushi / Nishi, Teruyuki et al. | 2006
- 1221
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Discovery of uracil-based histone deacetylase inhibitors able to reduce acquired antifungal resistance and trailing growth in Candida albicansMai, Antonello / Rotili, Dante / Massa, Silvio et al. | 2006
- 1226
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Simple criterion for selection of flavonoid compounds with anti-HIV activityVeljkovic, Veljko / Mouscadet, Jean-François / Veljkovic, Nevena et al. | 2006
- 1233
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Synthesis and biological evaluation of 4-amino derivatives of benzimidazoquinoxaline, benzimidazoquinoline, and benzopyrazoloquinazoline as potent IKK inhibitorsBeaulieu, Francis / Ouellet, Carl / Ruediger, Edward H. et al. | 2006
- 1238
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Synthesis, characterization, antibacterial activity, and interaction with DNA of the vanadyl-enrofloxacin complexEfthimiadou, Eleni K. / Katsaros, Nikos / Karaliota, Alexandra et al. | 2006
- 1243
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Synthesis of 3-(1H-benzimidazol-2-yl)-5-isoquinolin-4-ylpyrazolo[1,2-b]pyridine, a potent cyclin dependent kinase 1 (CDK1) inhibitorHuang, Shenlin / Lin, Ronghui / Yu, Yang et al. | 2006
- 1246
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Thienopyridine urea inhibitors of KDR kinaseHeyman, H. Robin / Frey, Robin R. / Bousquet, Peter F. et al. | 2006
- 1250
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Development of new pyrrolopyrimidine-based inhibitors of Janus kinase 3 (JAK3)Clark, Michael P. / George, Kelly M. / Bookland, Roger G. et al. | 2006
- 1254
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Bicyclic carbamates as inhibitors of papain-like cathepsin proteasesEpple, Robert / Urbina, Hugo D. / Russo, Ross et al. | 2006
- 1260
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Weak base dispiro-1,2,4-trioxolanes: Potent antimalarial ozonidesTang, Yuanqing / Dong, Yuxiang / Wittlin, Sergio et al. | 2006
- 1266
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A novel diketo phosphonic acid that exhibits specific, strand-transfer inhibition of HIV integrase and anti-HIV activityChi, Guochen / Nair, Vasu / Semenova, Elena et al. | 2006
- 1270
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Identification of arylsulfonamides as Aquaporin 4 inhibitorsHuber, Vincent J. / Tsujita, Mika / Yamazaki, Maya et al. | 2006
- 1274
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3-[2-((2S)-2-Cyano-pyrrolidin-1-yl)-2-oxo-ethylamino]-3-methyl-butyramide analogues as selective DPP-IV inhibitors for the treatment of type-II diabetesCoumar, Mohane Selvaraj / Chang, Chung-Nien / Chen, Chiung-Tong et al. | 2006
- 1280
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High-throughput screening affords novel and selective trypanothione reductase inhibitors with anti-trypanosomal activityMartyn, Derek C. / Jones, Deuan C. / Fairlamb, Alan H. et al. | 2006
- 1284
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3-Hydroxychromones as cyclin-dependent kinase inhibitors: Synthesis and biological evaluationLee, Jinho / Park, Taesik / Jeong, Shinwu et al. | 2006
- 1288
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Synthesis, structural revision, and antioxidant activities of antimutagenic homoisoflavonoids from Hoffmanosseggia intricataSiddaiah, Vidavalur / Maheswara, Muchchintala / Venkata Rao, Chunduri et al. | 2006
- 1291
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3-Substituted-(5-arylfuran-2-ylcarbonyl)guanidines as NHE-1 inhibitorsLee, Sunkyung / Kim, Taemi / Lee, Byung Ho et al. | 2006
- 1296
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N-(3-Cyano-4,5,6,7-tetrahydro-1-benzothien-2-yl)amides as potent, selective, inhibitors of JNK2 and JNK3Angell, Richard M. / Atkinson, Francis L. / Brown, Murray J. et al. | 2006
- 1302
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Rational design, synthesis, and structure–activity relationship of benzoxazolones: New potent mglu5 receptor antagonists based on the fenobam structureCeccarelli, Simona M. / Jaeschke, Georg / Buettelmann, Bernd et al. | 2006
- 1307
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Synthesis and biological evaluation of fenobam analogs as mGlu5 receptor antagonistsJaeschke, Georg / Porter, Richard / Büttelmann, Bernd et al. | 2006
- 1312
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Structure–activity relationships of 3-aminoquinazolinediones, a new class of bacterial type-2 topoisomerase (DNA gyrase and topo IV) inhibitorsTran, Tuan P. / Ellsworth, Edmund L. / Sanchez, Joseph P. et al. | 2006
- 1321
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Diastereoselective synthesis of glycosylated prolines as a-glucosidase inhibitors and organocatalyst in asymmetric aldol reactionPandey, J. / Dwivedi, N. / Singh, N. et al. | 2007
- 1321
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Diastereoselective synthesis of glycosylated prolines as α-glucosidase inhibitors and organocatalyst in asymmetric aldol reactionPandey, Jyoti / Dwivedi, Namrata / Singh, Nimisha et al. | 2006
- 1326
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Amino acid-based enantiomerically pure 3-substituted 1,4-benzodiazepin-2-ones: A new class of anti-ischemic agentsMishra, Jitendra Kumar / Garg, Puja / Dohare, Preeti et al. | 2006
- 1332
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Novel antiproliferative analogs of the Taq DNA polymerase inhibitor catalpolPungitore, Carlos R. / León, Leticia G. / García, Celina et al. | 2006
- 1336
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Carbonic anhydrase activators: An activation study of the human mitochondrial isoforms VA and VB with amino acids and aminesVullo, Daniela / Nishimori, Isao / Innocenti, Alessio et al. | 2006
- 1341
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Synthesis and biological evaluation of new conformationally biased integrin ligands based on a tetrahydroazoninone scaffoldBanfi, Luca / Basso, Andrea / Damonte, Gianluca et al. | 2006
- 1346
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Synthesis and antitubercular activity of quaternized promazine and promethazine derivativesBate, Aaron B. / Kalin, Jay H. / Fooksman, Eric M. et al. | 2006
- 1349
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3-Mercaptopropionic acids as efficacious inhibitors of activated thrombin activatable fibrinolysis inhibitor (TAFIa)Islam, Imadul / Bryant, Judi / May, Karen et al. | 2006
- 1355
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Anti-mycobacterial activity of a bis-sulfonamideWilkinson, Brendan L. / Bornaghi, Laurent F. / Wright, Anthony D. et al. | 2006
- 1358
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Inhibition of Src kinase activity by 7-ethynyl-4-phenylamino-3-quinolinecarbonitriles: Identification of SKS-927Boschelli, Diane H. / Barrios Sosa, Ana Carolina / Golas, Jennifer M. et al. | 2006
- 1362
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Synthesis and HIV-1 integrase inhibitory activity of spiroundecane(ene) derivativesShults, Elvira E. / Semenova, Elena A. / Johnson, Allison A. et al. | 2006
- 1369
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ortho-Substituted azoles as selective and dual inhibitors of VEGF receptors 1 and 2Kiselyov, Alexander S. / Piatnitski, Evgueni L. / Samet, Alexander V. et al. | 2006
- 1376
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Potent, selective, and orally active adenosine A2A receptor antagonists: Arylpiperazine derivatives of pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidinesNeustadt, Bernard R. / Hao, Jinsong / Lindo, Neil et al. | 2006
- 1381
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Structural simplification of bioactive natural products with multicomponent synthesis: Dihydropyridopyrazole analogues of podophyllotoxinMagedov, Igor V. / Manpadi, Madhuri / Rozhkova, Elena et al. | 2006
- 1386
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Challenges in the development of mGluR5 positive allosteric modulators: The discovery of CPPHAZhao, Zhijian / Wisnoski, David D. / O’Brien, Julie A. et al. | 2006
- 1392
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A potent and orally active HIV-1 integrase inhibitorEgbertson, Melissa S. / Moritz, H. Marie / Melamed, Jeffrey Y. et al. | 2006
- 1399
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Dopamine/serotonin receptor ligands. Part 15: Oxygenation of the benz-indolo-azecine LE 300 leads to novel subnanomolar dopamine D1/D5 antagonistsEnzensperger, Christoph / Kilian, Susann / Ackermann, Marit et al. | 2006
- 1403
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Quinazoline and benzimidazole MCH-1R antagonistsArienzo, Rosa / Cramp, Sue / Dyke, Hazel J. et al. | 2006
- 1408
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A molecular modeling analysis of novel non-hydroxamate inhibitors of TACESheppeck, James E. II / Tebben, Andrew / Gilmore, John L. et al. | 2006
- 1413
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Discovery of novel hydantoins as selective non-hydroxamate inhibitors of tumor necrosis factor-a converting enzyme (TACE)Sheppeck, J. E. / Gilmore, J. L. / Yang, A. et al. | 2007
- 1413
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Discovery of novel hydantoins as selective non-hydroxamate inhibitors of tumor necrosis factor-α converting enzyme (TACE)Sheppeck, James E. II / Gilmore, John L. / Yang, Anle et al. | 2006
- 1418
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Synthesis and evaluation of novel chromogenic aminopeptidase substrates for microorganism detection and identificationJames, Arthur L. / Perry, John D. / Rigby, Annette et al. | 2006
- 1422
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Discovery of 2-iminobenzimidazoles as a new class of trypanothione reductase inhibitor by high-throughput screeningHolloway, Georgina A. / Baell, Jonathan B. / Fairlamb, Alan H. et al. | 2006
- 1428
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Ac2-DPD, the bis-(O)-acetylated derivative of 4,5-dihydroxy-2,3-pentanedione (DPD) is a convenient stable precursor of bacterial quorum sensing autoinducer AI-2Frezza, Marine / Soulère, Laurent / Balestrino, Damien et al. | 2006
- 1432
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Pyrazole-based factor Xa inhibitors containing N-arylpiperidinyl P4 residuesQiao, Jennifer X. / Cheng, Xuhong / Smallheer, Joanne M. et al. | 2006
- 1438
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Synthesis and structure–activity relationship of N-acyl-Gly-, N-acyl-Sar- and N-blocked-boroPro inhibitors of FAP, DPP4, and POPTran, Thuy / Quan, Clifford / Edosada, Conrad Yap et al. | 2006
- 1443
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4-[6-(2-Aminoethyl)naphthalen-2-yl]benzonitriles are potent histamine H3 receptor antagonists with high CNS penetrationBlack, Lawrence A. / Nersesian, Diana L. / Sharma, Padam et al. | 2006
- 1447
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N-Alkyl-N-alkyloxycarbonylaminomethyl (NANAOCAM) prodrugs of carboxylic acid containing drugsMajumdar, Susruta / Sloan, Kenneth B. et al. | 2006
- 1451
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Novel membrane-localizing TEMPO derivatives for measurement of cellular oxidative stress at the cell membraneBan, Shizuka / Nakagawa, Hidehiko / Suzuki, Takayoshi et al. | 2006
- 1455
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Structure–activity relationship analysis of a novel necroptosis inhibitor, Necrostatin-5Wang, Ke / Li, Jinfeng / Degterev, Alexei et al. | 2006
- 1466
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Bis-styrylpyridine and bis-styrylbenzene derivatives as inhibitors for Ab fibril formationByeon, S. R. / Lee, J. H. / Sohn, J. H. et al. | 2007
- 1466
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Bis-styrylpyridine and bis-styrylbenzene derivatives as inhibitors for Aβ fibril formationByeon, Seong Rim / Lee, Ji Hoon / Sohn, Ji-Hoon et al. | 2006
- 1471
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Discovery of novel phosphorus-containing steroids as selective glucocorticoid receptor antagonistJiang, Weiqin / Fiordeliso, James J. / Allan, George et al. | 2006
- 1475
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Synthesis and cytotoxic activity of 17-carboxylic acid modified 23-hydroxy betulinic acid ester derivativesBi, Yi / Xu, Jinyi / Wu, Xiaoming et al. | 2006
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Editorial board| 2007
- I
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Instructions to contributors| 2007