A chiral template-driven synthesis of a 3′-deoxy-3′-18F-fluorothymidine precursor (Unbekannt)
- Neue Suche nach: Dey, Papiya
- Neue Suche nach: Ajish Kumar, K.S.
- Neue Suche nach: Sharma, Anubha
- Neue Suche nach: Chattopadhyay, Subrata
- Neue Suche nach: Dey, Papiya
- Neue Suche nach: Ajish Kumar, K.S.
- Neue Suche nach: Sharma, Anubha
- Neue Suche nach: Chattopadhyay, Subrata
In:
European journal of medicinal chemistry
;
143
;
1457-1462
;
2018
-
ISSN:
- Aufsatz (Zeitschrift) / Print
-
Titel:A chiral template-driven synthesis of a 3′-deoxy-3′-18F-fluorothymidine precursor
-
Beteiligte:Dey, Papiya ( Autor:in ) / Ajish Kumar, K.S. ( Autor:in ) / Sharma, Anubha ( Autor:in ) / Chattopadhyay, Subrata ( Autor:in )
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Erschienen in:European journal of medicinal chemistry ; 143 ; 1457-1462
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Verlag:
- Neue Suche nach: Elsevier Science B.V., Amsterdam.
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Erscheinungsdatum:01.01.2018
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Format / Umfang:6 pages
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ISSN:
-
Medientyp:Aufsatz (Zeitschrift)
-
Format:Print
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Sprache:Unbekannt
- Neue Suche nach: 615.1
- Weitere Informationen zu Dewey Decimal Classification
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Klassifikation:
DDC: 615.1 -
Datenquelle:
© Metadata Copyright the British Library Board and other contributors. All rights reserved.
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Discovery of naphtho[1,2-d]oxazole derivatives as potential anti-HCV agents through inducing heme oxygenase-1 expressionTseng, Chih-Hua / Lin, Chun-Kuang / Chen, Yeh-Long / Tseng, Chin-Kai / Lee, Jar-Yu / Lee, Jin-Ching et al. | 2018
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Bioactive products from singlet oxygen photooxygenation of cannabinoidsGalal Osman, Ahmed / Elokely, Khaled M. / Yadav, Vivek K. / Carvalho, Paulo / Radwan, Mohamed / Slade, Desmond / Gul, Waseem / Khan, Shabana / Dale, Olivia R. / Husni, Afeef S. et al. | 2018
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Peptides having antimicrobial activity and their complexes with transition metal ionsJeżowska-Bojczuk, Małgorzata / Stokowa-Sołtys, Kamila et al. | 2018
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Hetero-Diels-Alder reactions of novel 3-triazolyl-nitrosoalkenes as an approach to functionalized 1,2,3-triazoles with antibacterial profileLopes, Susana M.M. / Novais, Juliana S. / Costa, Dora C.S. / Castro, Helena C. / Figueiredo, Agnes Marie S. / Ferreira, Vitor F. / Pinho e Melo, Teresa M.V.D. / da Silva, Fernando de Carvalho et al. | 2018
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Structure-based identification of a NEDD8-activating enzyme inhibitor via drug repurposingWu, Ke-Jia / Zhong, Hai-Jing / Li, Guodong / Liu, Chenfu / Wang, Hui-Min David / Ma, Dik-Lung / Leung, Chung-Hang et al. | 2018
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Design and synthesis of novel quinacrine-[1, 3]-thiazinan-4-one hybrids for their anti-breast cancer activitySolomon, V. Raja / Pundir, Sheetal / Le, Hoang-Thanh / Lee, Hoyun et al. | 2018
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Homo- and heteroleptic Pt(II) complexes of ONN donor hydrazone and 4-picoline: A synthetic, structural and detailed mechanistic anticancer investigationRahman, Faiz-Ur / Bhatti, Muhammad Zeeshan / Ali, Amjad / Duong, Hong-Quan / Zhang, Yao / Yang, Bo / Koppireddi, Satish / Lin, Yuejian / Wang, Hui / Li, Zhan-Ting et al. | 2018
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Discovery and evolution of aloperine derivatives as a new family of HCV inhibitors with novel mechanismZhang, Xin / Lv, Xiao–Qin / Tang, Sheng / Mei, Lin / Li, Ying–Hong / Zhang, Jing–Pu / Jiang, Jian–Dong / Peng, Zong–Gen / Song, Dan–Qing et al. | 2018
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Development of novel bis-pyrazole derivatives as antitumor agents with potent apoptosis induction effects and DNA damageDai, Hong / Ge, Shushan / Guo, Jing / Chen, Shi / Huang, Meiling / Yang, Jiaying / Sun, Siyu / Ling, Yong / Shi, Yujun et al. | 2018
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Natural product inspired library synthesis - Identification of 2,3-diarylbenzofuran and 2,3-dihydrobenzofuran based inhibitors of Chlamydia trachomatisSaleeb, Michael / Mojica, Sergio / Eriksson, Anna U. / Andersson, C. David / Gylfe, Åsa / Elofsson, Mikael et al. | 2018
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Organic arsenicals target thioredoxin reductase followed by oxidative stress and mitochondrial dysfunction resulting in apoptosisFan, Xiao-Yang / Liu, Yu-Jiao / Chen, Kai / Jiang, Feng-Lei / Hu, Yan-Jun / Liu, Dan / Liu, Yi / Ge, Yu-Shu et al. | 2018
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Recent advances in the discovery of small molecule c-Met Kinase inhibitorsParikh, Palak K. / Ghate, Manjunath D. et al. | 2018
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Structure-activity analysis of CJ-15,801 analogues that interact with Plasmodium falciparum pantothenate kinase and inhibit parasite proliferationSpry, Christina / Sewell, Alan L. / Hering, Yuliya / Villa, Mathew V.J. / Weber, Jonas / Hobson, Stephen J. / Harnor, Suzannah J. / Gul, Sheraz / Marquez, Rodolfo / Saliba, Kevin J. et al. | 2018
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Structural optimization and structure-activity relationship studies of N-phenyl-7,8-dihydro-6H-pyrimido[5,4-b][1,4]oxazin-4-amine derivatives as a new class of inhibitors of RET and its drug resistance mutantsYang, Jiao / Chen, Kai / Zhang, Guo / Yang, Qiu-Yuan / Li, Yue-Shan / Huang, Shen-Zhen / Wang, Yan-Lin / Yang, Wei / Jiang, Xiao-Juan / Yan, Heng-Xiu et al. | 2018
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Design, synthesis, and evaluation of NDGA analogues as potential anti-ischemic stroke agentsHuang, Lili / Wang, Jiabing / Chen, Liping / Zhu, Min / Wu, Shoubiao / Chu, Shenghui / Zheng, Yuantie / Fan, Ziliang / Zhang, Jiafeng / Li, Wulan et al. | 2018
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A routinely used protein staining dye acts as an inhibitor of wild type and mutant alpha-synuclein aggregation and modulator of neurotoxicityAhsan, Nuzhat / Siddique, Ibrar Ahmed / Gupta, Sarika / Surolia, Avadhesha et al. | 2018
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Allicin-inspired pyridyl disulfides as antimicrobial agents for multidrug-resistant Staphylococcus aureusSheppard, Jordan G. / McAleer, Jeremy P. / Saralkar, Pushkar / Geldenhuys, Werner J. / Long, Timothy E. et al. | 2018
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Anti-amyloidogenic and anti-apoptotic effect of α-bisabolol against Aβ induced neurotoxicity in PC12 cellsShanmuganathan, Balakrishnan / Suryanarayanan, Venkatesan / Sathya, Sethuraman / Narenkumar, Muralidharan / Singh, Sanjeev Kumar / Ruckmani, Kandasamy / Pandima Devi, Kasi et al. | 2018
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Amphiphilic glycoconjugates as potential anti-cancer chemotherapeuticsGovindarajan, Mugunthan et al. | 2018
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Design, synthesis and evaluation of novel dihydrostilbene derivatives as potential anti-melanogenic skin-protecting agentsZhu, Yu / Pan, Wen-Hui / Ku, Chuen Fai / Zhang, Hong-Jie / Tsang, Siu Wai et al. | 2018
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Design and synthesis of small molecule agonists of EphA2 receptorPetty, Aaron / Idippily, Nethrie / Bobba, Viharika / Geldenhuys, Werner J. / Zhong, Bo / Su, Bin / Wang, Bingcheng et al. | 2018
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Dual or multi-targeting inhibitors: The next generation anticancer agentsRaghavendra, Nulgumnalli Manjunathaiah / Pingili, Divya / Kadasi, Sundeep / Mettu, Akhila / Prasad, S.V.U.M. et al. | 2018
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2-Arylbenzofurans from Artocarpus lakoocha and methyl ether analogs with potent cholinesterase inhibitory activityNamdaung, Umalee / Athipornchai, Anan / Khammee, Thongchai / Kuno, Mayuso / Suksamrarn, Sunit et al. | 2018
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Design, synthesis and evaluation of amino-substituted 1H-phenalen-1-ones as anti-leishmanial agentsFreijo, Mónica Blanco / López-Arencibia, Atteneri / Piñero, José E. / McNaughton-Smith, Grant / Abad-Grillo, Teresa et al. | 2018
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Exploring the tetrahydroisoquinoline thiohydantoin scaffold blockade the androgen receptor as potent anti-prostate cancer agentsXu, Xi / Ge, Raoling / Li, Lei / Wang, Jubo / Lu, Xiaoyu / Xue, Siqi / Chen, Xijing / Li, Zhiyu / Bian, Jinlei et al. | 2018
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Novel indole and triazole based hybrid molecules exhibit potent anti-adipogenic and antidyslipidemic activity by activating Wnt3a/β-catenin pathwayRajan, Sujith / Puri, Surendra / Kumar, Durgesh / Babu, Madala Hari / Shankar, Kripa / Varshney, Salil / Srivastava, Ankita / Gupta, Abhishek / Reddy, M. Sridhar / Gaikwad, Anil N. et al. | 2018
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1, 4-Naphthoquinones potently inhibiting P2X7 receptor activityFaria, R.X. / Oliveira, F.H. / Salles, J.P. / Oliveira, A.S. / von Ranke, N.L. / Bello, M.L. / Rodrigues, C.R. / Castro, H.C. / Louvis, A.R. / Martins, D.L. et al. | 2018
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Synthesis, monoamine oxidase inhibition activity and molecular docking studies of novel 4-hydroxy-N′-[benzylidene or 1-phenylethylidene]-2-H/methyl/benzyl-1,2-benzothiazine-3-carbohydrazide 1,1-dioxidesSaddique, Furqan Ahmad / Zaib, Sumera / Jalil, Saquib / Aslam, Sana / Ahmad, Matloob / Sultan, Sadia / Naz, Humera / Iqbal, Mazhar / Iqbal, Jamshed et al. | 2018
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Synthesis and in vitro biological evaluation of three 4′-(4-methoxyphenyl)-2,2′:6′,2″-terpyridine iridium(III) complexes as new telomerase inhibitorsQin, Qi-Pin / Meng, Ting / Tan, Ming-Xiong / Liu, Yan-Cheng / Luo, Xu-Jian / Zou, Bi-Qun / Liang, Hong et al. | 2018
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Synthesis and preliminary antiproliferative activity of new pteridin-7(8H)-one derivativesLi, Zhong-Hua / Zhao, Tao-Qian / Liu, Xue-Qi / Zhao, Bing / Wang, Chao / Geng, Peng-Fei / Cao, Ya-Quan / Fu, Dong-Jun / Jiang, Li-Ping / Yu, Bin et al. | 2018
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Recent advances in the discovery of potent and selective HDAC6 inhibitorsWang, Xiu-Xiu / Wan, Ren-Zhong / Liu, Zhao-Peng et al. | 2018
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Discovery of new potent molecular entities able to inhibit mPGES-1Di Micco, Simone / Terracciano, Stefania / Cantone, Vincenza / Fischer, Katrin / Koeberle, Andreas / Foglia, Antonio / Riccio, Raffaele / Werz, Oliver / Bruno, Ines / Bifulco, Giuseppe et al. | 2018
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Development of noviomimetics that modulate molecular chaperones and manifest neuroprotective effectsForsberg, Leah K. / Anyika, Mercy / You, Zhenyuan / Emery, Sean / McMullen, Mason / Dobrowsky, Rick T. / Blagg, Brian S.J. et al. | 2018
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Optimization of pharmacokinetic properties by modification of a carbazole-based cannabinoid receptor subtype 2 (CB2) ligandHeimann, Dominik / Börgel, Frederik / de Vries, Henk / Bachmann, Kim / Rose, Victoria E. / Frehland, Bastian / Schepmann, Dirk / Heitman, Laura H. / Wünsch, Bernhard et al. | 2018
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Biphenylthiazole antibiotics with an oxadiazole linker: An approach to improve physicochemical properties and oral bioavailabilityHagras, Mohamed / Hegazy, Youssef A. / Elkabbany, Amr H. / Mohammad, Haroon / Ghiaty, Adel / Abdelghany, Tamer M. / Seleem, Mohamed N. / Mayhoub, Abdelrahman S. et al. | 2018
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A chiral template-driven synthesis of a 3′-deoxy-3′-18F-fluorothymidine precursorDey, Papiya / Ajish Kumar, K.S. / Sharma, Anubha / Chattopadhyay, Subrata et al. | 2018
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Quinoline derivatives bearing pyrazole moiety: Synthesis and biological evaluation as possible antibacterial and antifungal agentsEl Shehry, Mohamed F. / Ghorab, Mostafa M. / Abbas, Samir Y. / Fayed, Eman A. / Shedid, Said A. / Ammar, Yousry A. et al. | 2018
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Design, synthesis and biological evaluation of novel aryldiketo acids with enhanced antibacterial activity against multidrug resistant bacterial strainsCvijetić, Ilija N. / Verbić, Tatjana Ž. / Ernesto de Resende, Pedro / Stapleton, Paul / Gibbons, Simon / Juranić, Ivan O. / Drakulić, Branko J. / Zloh, Mire et al. | 2018
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Synthesis and bioactivities study of new antibacterial peptide mimics: The dialkyl cationic amphiphilesZhang, En / Bai, Peng-Yan / Cui, De-Yun / Chu, Wen-Chao / Hua, Yong-Gang / Liu, Qin / Yin, Hai-Yang / Zhang, Yong-Jie / Qin, Shangshang / Liu, Hong-Min et al. | 2018
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Discovery of simplified sampangine derivatives as novel fungal biofilm inhibitorsLiu, Na / Zhong, Hua / Tu, Jie / Jiang, Zhigan / Jiang, Yanjuan / Jiang, Yan / Jiang, Yuanying / Li, Jian / Zhang, Wannian / Wang, Yan et al. | 2018
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Synthesis, antibacterial properties and 2D-QSAR studies of quinolone-triazole conjugatesFaidallah, Hassan M. / Girgis, Adel S. / Tiwari, Anand D. / Honkanadavar, Hitesh H. / Thomas, Sean J. / Samir, Ahmed / Kalmouch, Atef / Alamry, Khalid A. / Khan, Khalid A. / Ibrahim, Tarek S. et al. | 2018
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Exploration of 1, 2, 3-triazole-pyrimidine hybrids as potent reversal agents against ABCB1-mediated multidrug resistanceWang, Bo / Zhao, Bing / Chen, Zhe-Sheng / Pang, Lu-Ping / Zhao, Yuan-Di / Guo, Qian / Zhang, Xin-Hui / Liu, Ying / Liu, Guang-Yao / Zhang, Xin-Yuan et al. | 2018
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Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agentsCarradori, Simone / Ortuso, Francesco / Petzer, Anél / Bagetta, Donatella / De Monte, Celeste / Secci, Daniela / De Vita, Daniela / Guglielmi, Paolo / Zengin, Gokhan / Aktumsek, Abdurrahman et al. | 2018
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Aminomethylation of heliomycin: Preparation and anticancer characterization of the first series of semi-synthetic derivativesNadysev, Georgy Y. / Tikhomirov, Alexander S. / Lin, Ming-Hung / Yang, Ya-Ting / Dezhenkova, Lyubov G. / Chen, Huei-Yu / Kaluzhny, Dmitry N. / Schols, Dominique / Shtil, Alexander A. / Shchekotikhin, Andrey E. et al. | 2018
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Design, synthesis and biological evaluation of new β-carboline-bisindole compounds as DNA binding, photocleavage agents and topoisomerase I inhibitorsKovvuri, Jeshma / Nagaraju, Burri / Nayak, V. Lakshma / Akunuri, Ravikumar / Rao, M.P. Narasimha / Ajitha, Ayyappan / Nagesh, Narayan / Kamal, Ahmed et al. | 2018
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Discovery of a head-to-tail cyclic peptide as the Keap1-Nrf2 protein-protein interaction inhibitor with high cell potencyLu, Meng-Chen / Jiao, Qiong / Liu, Tian / Tan, Shi-Jie / Zhou, Hai-Shan / You, Qi-Dong / Jiang, Zheng-Yu et al. | 2018
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Indole and Benzimidazole Bichalcophenes: Synthesis, DNA Binding and Antiparasitic ActivityFarahat, Abdelbasset A. / Ismail, Mohamed A. / Kumar, Arvind / Wenzler, Tanja / Brun, Reto / Paul, Ananya / Wilson, W. David / Boykin, David W. et al. | 2018
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Synthesis, crystal structure and biological evaluation of a new dasatinib copper(II) complex as telomerase inhibitorQin, Qi-Pin / Meng, Ting / Tan, Ming-Xiong / Liu, Yan-Cheng / Luo, Xu-Jian / Zou, Bi-Qun / Liang, Hong et al. | 2018
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Synthesis, molecular docking, and QSAR study of sulfonamide-based indoles as aromatase inhibitorsPingaew, Ratchanok / Mandi, Prasit / Prachayasittikul, Veda / Prachayasittikul, Supaluk / Ruchirawat, Somsak / Prachayasittikul, Virapong et al. | 2018
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Design, synthesis and biological evaluation of novel benzimidazole amidines as potent multi-target inhibitors for the treatment of non-small cell lung cancerBistrović, Andrea / Krstulović, Luka / Harej, Anja / Grbčić, Petra / Sedić, Mirela / Koštrun, Sanja / Pavelić, Sandra Kraljević / Bajić, Miroslav / Raić-Malić, Silvana et al. | 2018