ARTICLES - N-(2-Benzoylphenyl)-L-tyrosine PPARg Agonists. 3. Structure-Activity Relationship and Optimization of the N-Aryl Substituent (Englisch)
- Neue Suche nach: Cobb, Jeff E.
- Neue Suche nach: Cobb, Jeff E.
- Neue Suche nach: Blanchard, Steven G.
- Neue Suche nach: Boswell, Evan G.
- Neue Suche nach: Brown, Kathleen K.
- Neue Suche nach: Charifson, Paul S.
- Neue Suche nach: Cooper, Joel P.
- Neue Suche nach: Collins, Jon L.
- Neue Suche nach: Dezube, Milana
- Neue Suche nach: Henke, Brad R.
- Neue Suche nach: Hull-Ryde, Emily A.
- Neue Suche nach: Lake, Debra H.
- Neue Suche nach: Lenhard, James M.
- Neue Suche nach: Oliver Jr, William
- Neue Suche nach: Oplinger, Jeffery
- Neue Suche nach: Pentti, Mila
- Neue Suche nach: Parks, Derek J.
- Neue Suche nach: Plunket, Kelli D.
- Neue Suche nach: Tong, Wei-Qin
In:
Journal of medicinal chemistry
;
41
, 25
; 5055-5069
;
1998
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ISSN:
- Aufsatz (Zeitschrift) / Print
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Titel:ARTICLES - N-(2-Benzoylphenyl)-L-tyrosine PPARg Agonists. 3. Structure-Activity Relationship and Optimization of the N-Aryl Substituent
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Beteiligte:
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Erschienen in:Journal of medicinal chemistry ; 41, 25 ; 5055-5069
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Verlag:
- Neue Suche nach: American Chemical Society
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Erscheinungsort:Easton, Pa.
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Erscheinungsdatum:1998
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ISSN:
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ZDBID:
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Medientyp:Aufsatz (Zeitschrift)
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Format:Print
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Sprache:Englisch
- Neue Suche nach: 770/4230
- Neue Suche nach: 44.42 / 44.42
- Weitere Informationen zu Basisklassifikation
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Schlagwörter:
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Klassifikation:
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Datenquelle:
Inhaltsverzeichnis – Band 41, Ausgabe 25
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Die Inhaltsverzeichnisse werden automatisch erzeugt und basieren auf den im Index des TIB-Portals verfügbaren Einzelnachweisen der enthaltenen Beiträge. Die Anzeige der Inhaltsverzeichnisse kann daher unvollständig oder lückenhaft sein.
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Mutational Evidence for a Common κ Antagonist Binding Pocket in the Wild-Type κ and Mutant μ[K303E] Opioid Receptors †Jones, Robert M. / Hjorth, Siv A. / Schwartz, Thue W. / Portoghese, Philip S. et al. | 1998
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Mutational Evidence for a Common kappa Antagonist Binding Pocket in the Wild-Type kappa and Mutant [K303E] Opioid ReceptorsJones, R. M. / Hjorth, S. A. / Schwartz, T. W. / Portoghese, P. S. et al. | 1998
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COMMUNICATIONS TO THE EDITOR - Mutational Evidence for a Common K Antagonist Binding Pocket in the Wild-Type k and Mutant m(K303E) Opioid ReceptorsJones, Robert M. et al. | 1998
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COMMUNICATIONS TO THE EDITOR - Dual D2-Receptor and b2-Adrenoceptor Agonists for the Treatment of Airway Diseases. 1. Discovery and Biological Evaluation of Some 7-(2-Aminoethyl)-4-hydroxybenzothiazol-2(3H)-one AnaloguesBonnert, Roger V. et al. | 1998
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Dual D2-Receptor and β2-Adrenoceptor Agonists for the Treatment of Airway Diseases. 1. Discovery and Biological Evaluation of Some 7-(2-Aminoethyl)- 4-hydroxybenzothiazol-2(3H)-one AnaloguesBonnert, Roger V. / Brown, Roger C. / Chapman, David / Cheshire, David R. / Dixon, John / Ince, Francis / Kinchin, Elizabeth C. / Lyons, Amanda J. / Davis, Andrew M. / Hallam, Catherine et al. | 1998
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Structure−Activity Relationships for Antiplasmodial Activity among 7-Substituted 4-AminoquinolinesDe, Dibyendu / Krogstad, Frances M. / Byers, Larry D. / Krogstad, Donald J. et al. | 1998
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ARTICLES - Polyanion Inhibitors of HIV and Other Viruses. 7. Polyanionic Compounds and Polyzwitterionic Compounds Derived from Cyclodextrins as Inhibitors of HIV TransmissionLeydet, Alain et al. | 1998
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ARTICLES - N-n-Propyl-Substituted 3-(Dimethylphenyl)piperidines Display Novel Discriminative Properties between Dopamine Receptor Subtypes: Synthesis and Receptor Binding StudiesCervetto, Luigi et al. | 1998
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N-n-Propyl-Substituted 3-(Dimethylphenyl)piperidines Display Novel Discriminative Properties between Dopamine Receptor Subtypes: Synthesis and Receptor Binding StudiesCervetto, Luigi / Demontis, Gian Carlo / Giannaccini, Gino / Longoni, Biancamaria / Macchia, Bruno / Macchia, Marco / Martinelli, Adriano / Orlandini, Elisabetta et al. | 1998
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Correlation of Human Jejunal Permeability (in Vivo) of Drugs with Experimentally and Theoretically Derived Parameters. A Multivariate Data Analysis ApproachWiniwarter, Susanne / Bonham, Nicholas M. / Ax, Fredrik / Hallberg, Anders / Lennernäs, Hans / Karlén, Anders et al. | 1998
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ARTICLES - Characterization of Novel N,N'-Disubstituted Piperazines as s Receptor LigandsZhang, Ying et al. | 1998
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Characterization of Novel N,N‘-Disubstituted Piperazines as σ Receptor LigandsZhang, Ying / Williams, Wanda / Torrence-Campbell, Cheryl / Bowen, Wayne D. / Rice, Kenner C. et al. | 1998
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ARTICLES - Antiviral Oligo- and Polyribonucleotides Containing Selected Triazolo(2,3-a)purinesTutonda, Mayoka G. et al. | 1998
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Antiviral Oligo- and Polyribonucleotides Containing Selected Triazolo[2,3-a]purines ‖Tutonda, Mayoka G. / Buckheit,, Robert W. / Agrawal, Vijai K. / Broom, Arthur D. et al. | 1998
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Antiviral Oligo- and Polyribonucleotides Containing Selected Triazolo[2,3-]purinesTutonda, M. G. / Buckheit, R. W. / Agrawal, V. K. / Broom, A. D. et al. | 1998
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Methoxy-Substituted 3-Formyl-2-phenylindoles Inhibit Tubulin PolymerizationGastpar, Robert / Goldbrunner, Michael / Marko, Doris / von Angerer, Erwin et al. | 1998
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ARTICLES - Methoxy-Substituted 3-Formyl-2-phenylindoles Inhibit Tubulin PolymerizationGastpar, Robert et al. | 1998
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Synthesis and Biological Properties of New 2β-Alkyl- and 2β-Aryl-3-(substituted phenyl)tropane Derivatives: Stereochemical Effect of C-3 on Affinity and Selectivity for Neuronal Dopamine and Serotonin TransportersKozikowski, Alan P. / Araldi, Gian Luca / Prakash, K. R. C. / Zhang, Mei / Johnson, Kenneth M. et al. | 1998
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ARTICLES - Synthesis and Biological Properties of New 2b-Alkyl- and 2b-Aryl-3-(substituted phenyl)tropane Derivatives: Stereochemical Effect of C-3 on Affinity and Selectivity for Neuronal Dopamine and Serotonin TransportersKozikowski, Alan P. et al. | 1998
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ARTICLES - Tetrahydro-isoquinoline-Based Factor Xa InhibitorsKucznierz, Ralf et al. | 1998
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Tetrahydro-isoquinoline-Based Factor Xa InhibitorsKucznierz, Ralf / Grams, Frank / Leinert, Herbert / Marzenell, Klaus / Engh, Richard A. / von der Saal, Wolfgang et al. | 1998
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Synthesis and Serotonin Receptor Affinities of a Series of trans-2-(Indol-3-yl)cyclopropylamine DerivativesVangveravong, Suwanna / Kanthasamy, Arthi / Lucaites, Virginia L. / Nelson, David L. / Nichols, David E. et al. | 1998
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ARTICLES - Synthesis and Serotonin Receptor Affinities of a Series of trans-2-(Indol-3-yl)cyclopropylamine DerivativesVangveravong, Suwanna et al. | 1998
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Constrained Corticotropin-Releasing Factor (CRF) Agonists and Antagonists with i−(i+3) Glu-Xaa-dXbb-Lys Bridges †Koerber, Steven C. / Gulyas, Jozsef / Lahrichi, Sabine L. / Corrigan, Anne / Craig, A. Grey / Rivier, Catherine / Vale, Wylie / Rivier, Jean et al. | 1998
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ARTICLES - Constrained Corticotropin-Releasing Factor (CRF) Agonists and Antagonists with i-(i+3) Glu-Xaa-DXbb-Lys BridgesKoerber, Steven C. et al. | 1998
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Astressin Analogues (Corticotropin-Releasing Factor Antagonists) with Extended Duration of Action in the Rat ‖Rivier, Jean / Gulyas, Jozsef / Corrigan, Anne / Martinez, Vicente / Craig, A. Grey / Taché, Yvette / Vale, Wylie / Rivier, Catherine et al. | 1998
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ARTICLES - Astressin Analogues (Corticotropin-Releasing Factor Antagonists) with Extended Duration of Action in the RatRivier, Jean et al. | 1998
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N-(2-Benzoylphenyl)-l-tyrosine PPARγ Agonists. 1. Discovery of a Novel Series of Potent Antihyperglycemic and Antihyperlipidemic AgentsHenke, Brad R. / Blanchard, Steven G. / Brackeen, Marcus F. / Brown, Kathleen K. / Cobb, Jeff E. / Collins, Jon L. / Harrington,, W. Wallace / Hashim, Mir A. / Hull-Ryde, Emily A. / Kaldor, Istvan et al. | 1998
- 5020
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ARTICLES - N-(2-Benzoylphenyl)-L-tyrosine PPARg Agonists. 1. Discovery of a Novel Series of Potent Antihyperglycemic and Antihyperlipidemic AgentsHenke, Brad R. et al. | 1998
- 5037
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ARTICLES - N-(2-Benzoylphenyl)-L-tyrosine PPARg Agonists. 2. Structure-Activity Relationship and Optimization of the Phenyl Alkyl Ether MoietyCollins, Jon L. et al. | 1998
- 5037
-
N-(2-Benzoylphenyl)-l-tyrosine PPARγ Agonists. 2. Structure−Activity Relationship and Optimization of the Phenyl Alkyl Ether MoietyCollins, Jon L. / Blanchard, Steven G. / Boswell, G. Evan / Charifson, Paul S. / Cobb, Jeff E. / Henke, Brad R. / Hull-Ryde, Emily A. / Kazmierski, Wieslaw M. / Lake, Debra H. / Leesnitzer, Lisa M. et al. | 1998
- 5055
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N-(2-Benzoylphenyl)-l-tyrosine PPARγ Agonists. 3. Structure−Activity Relationship and Optimization of the N-Aryl SubstituentCobb, Jeff E. / Blanchard, Steven G. / Boswell, Evan G. / Brown, Kathleen K. / Charifson, Paul S. / Cooper, Joel P. / Collins, Jon L. / Dezube, Milana / Henke, Brad R. / Hull-Ryde, Emily A. et al. | 1998
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ARTICLES - N-(2-Benzoylphenyl)-L-tyrosine PPARg Agonists. 3. Structure-Activity Relationship and Optimization of the N-Aryl SubstituentCobb, Jeff E. et al. | 1998
- 5070
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Design and Synthesis of a Series of 6-Substituted-2-pyridinylmethylamine Derivatives as Novel, High-Affinity, Selective Agonists at 5-HT1A ReceptorsVacher, Bernard / Bonnaud, Bernard / Funes, Philippe / Jubault, Nathalie / Koek, Wouter / Assié, Marie-Bernadette / Cosi, Cristina et al. | 1998
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ARTICLES - Design and Synthesis of a Series of 6-Substituted-2-pyridinylmethylamine Derivatives as Novel, High-Affinity, Selective Agonists at 5-HT1A ReceptorsVacher, Bernard et al. | 1998
- 5084
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ARTICLES - Spiperone: Influence of Spiro Ring Substituents on 5-HT2A Serotonin Receptor BindingMetwally, Kamel A. et al. | 1998
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Nucleosides and Nucleotides. 180. Synthesis and Antitumor Activity of Nucleosides That Have a Hydroxylamino Group Instead of a Hydroxyl Group at the 2‘- or 3‘-Position of the Sugar MoietyOgawa, Akira / Tanaka, Motohiro / Sasaki, Takuma / Matsuda, Akira et al. | 1998
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ARTICLES - Nucleosides and Nucleotides. 180. Synthesis and Antitumor Activity of Nucleosides That Have a Hydroxylamino Group Instead of a Hydroxyl Group at the 2'- or 3'-Position of the Sugar MoietyOgawa, Akira et al. | 1998
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Synthesis of Imidazo[1,2-a]pyridines as Antiviral AgentsGueiffier, Alain / Mavel, Sylvie / Lhassani, Mohammed / Elhakmaoui, Ahmed / Snoeck, Robert / Andrei, Graciela / Chavignon, Olivier / Teulade, Jean-Claude / Witvrouw, Myriam / Balzarini, Jan et al. | 1998
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NOTES - Synthesis of Imidazo(1,2-a)pyridines as Antiviral AgentsGueiffier, Alain et al. | 1998
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Stereoisomers of Cyclic Urea HIV-1 Protease Inhibitors: Synthesis and Binding AffinitiesKaltenbach, Robert F. / Nugiel, David A. / Lam, Patrick Y. S. / Klabe, Ronald M. / Seitz, Steven P. et al. | 1998
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NOTES - Stereoisomers of Cyclic Urea HIV-1 Protease Inhibitors: Synthesis and Binding AffinitiesKaltenbach III, Robert F. et al. | 1998
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-
BOOK REVIEWS - The Molecular and Supramolecular Chemistry of CarbohydratesLevy, Daniel E. et al. | 1998
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The Molecular and Supramolecular Chemistry of CarbohydratesLevy, D. E. et al. | 1998
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The Molecular and Supramolecular Chemistry of Carbohydrates By Serge David. Oxford University Press, New York. 1998. vii + 320 pp. 15.5 × 23 cm. ISBN 0-19-850046-7. $45.00.Levy, Daniel E. et al. | 1998