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Synonyme wurden verwendet für: BACE1
Suche ohne Synonyme: keywords:(BACE1)
Verwendete Synonyme:
- asp2
- b site of app cleaving enzyme
- bace
- beta secretase 1
- beta sekretase
- beta site alzheimer's amyloid precursor protein cleaving enzyme 1
- beta site app cleaving enzyme 1
- cas 158736 49 3
- ec 3 4 23 46
- flj90568
- hspc104
- kiaa1149
- memapsin 2
- membrane associated aspartic protease 2
-
BACE1 Inhibitor Peptides: Can an Infinitely Small k cat Value Turn the Substrate of an Enzyme into Its Inhibitor?
American Chemical Society | 2012|Schlagwörter: BACE1, BACE1 inhibitor -
Screening Platform Based on Inductively Coupled Plasma Mass Spectrometry for β‑Site Amyloid Protein Cleaving Enzyme 1 (BACE1) Inhibitors
American Chemical Society | 2021|Schlagwörter: BACE1 inhibitor, BACE1 -
Increased Secondary Nucleation Underlies Accelerated Aggregation of the Four-Residue N‑Terminally Truncated Aβ42 Species Aβ5–42
American Chemical Society | 2019|Schlagwörter: BACE -
Lilly, AstraZeneca drop BACE inhibitor
American Chemical Society | 2018Schlagwörter: BACE inhibitors -
miR-29a/b1 Regulates BACE1 in Aluminum-Induced Aβ Deposition in Vitro
American Chemical Society | 2021|Schlagwörter: BACE1 -
Targeting the BACE1 Active Site Flap Leads to a Potent Inhibitor That Elicits Robust Brain Aβ Reduction in Rodents
American Chemical Society | 2016|Schlagwörter: BACE1 -
Thiazolyl-thiadiazines as Beta Site Amyloid Precursor Protein Cleaving Enzyme‑1 (BACE-1) Inhibitors and Anti-inflammatory Agents: Multitarget-Directed Ligands for the Efficient Management of Alzheimer’s Disease
American Chemical Society | 2018|Schlagwörter: BACE-1 -
Discovery of an Orally Available, Brain Penetrant BACE1 Inhibitor That Affords Robust CNS Aβ Reduction
American Chemical Society | 2012|Schlagwörter: BACE1 -
Synthesis, Optimization, and Large-Scale Preparation of the Low-Dose Central Nervous System-Penetrant BACE1 Inhibitor LY3202626 via a [3 + 2] Nitrone Cycloaddition
American Chemical Society | 2020|Schlagwörter: BACE inhibitor -
Structure-Based Survey of the Binding Modes of BACE1 Inhibitors
American Chemical Society | 2019|Schlagwörter: BACE1 -
Scope of β‑Secretase (BACE1)-Targeted Therapy in Alzheimer’s Disease: Emphasizing the Flavonoid Based Natural Scaffold for BACE1 Inhibition
American Chemical Society | 2020|Schlagwörter: BACE1 -
Process Development of a Second Generation β‑Amyloid-Cleaving Enzyme InhibitorImproving the Robustness of a Halogen-Metal Exchange Using Continuous Stirred-Tank Reactors
American Chemical Society | 2021|Schlagwörter: BACE1 -
Improved Process for a Copper-Catalyzed C–N Coupling in the Synthesis of Verubecestat
American Chemical Society | 2019|Schlagwörter: BACE1 inhibitor -
A Brain-Penetrant and Bioavailable Pyrazolopiperazine BACE1 Inhibitor Elicits Sustained Reduction of Amyloid β In Vivo
American Chemical Society | 2022|Schlagwörter: BACE inhibitor -
Polyrhachis vicina Roger Alleviates Memory Impairment in a Rat Model of Alzheimer’s Disease Through the EGR1/BACE1/APP Axis
American Chemical Society | 2022|Schlagwörter: BACE1 -
Discovery of Multitarget-Directed Ligands from Piperidine Alkaloid Piperine as a Cap Group for the Management of Alzheimer’s Disease
American Chemical Society | 2023|Schlagwörter: BACE1 -
Evaluation of a Series of β‑Secretase 1 Inhibitors Containing Novel Heteroaryl-Fused-Piperazine Amidine Warheads
American Chemical Society | 2019|Schlagwörter: BACE inhibitor -
Determining Structural Changes for Ligand Recognition between Human and Rat Phosphorylated BACE1 in Silico and Its Phosphorylation by GSK3β at Thr252 by in Vitro Studies
American Chemical Society | 2024|Schlagwörter: BACE1
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