Erscheinungsjahr
Medientyp
Format
Lizenz
Sprache
Synonyme wurden verwendet für: Chemistry
Suche ohne Synonyme: journal:(Journal of Medicinal Chemistry)
Verwendete Synonyme:
- allgemeine chemie
- chemie
-
Identification of MRTX1133, a Noncovalent, Potent, and Selective KRASG12D Inhibitor
Freier ZugriffAmerican Chemical Society | 2022| -
Discovery of S‑217622, a Noncovalent Oral SARS-CoV‑2 3CL Protease Inhibitor Clinical Candidate for Treating COVID-19
Freier ZugriffAmerican Chemical Society | 2022| -
Thiazoles, Their Benzofused Systems, and Thiazolidinone Derivatives: Versatile and Promising Tools to Combat Antibiotic Resistance
Freier ZugriffAmerican Chemical Society | 2020| -
Movement to the Clinic of Soluble Epoxide Hydrolase Inhibitor EC5026 as an Analgesic for Neuropathic Pain and for Use as a Nonaddictive Opioid Alternative
Freier ZugriffAmerican Chemical Society | 2021| -
The Medicinal Chemistry in the Era of Machines and Automation: Recent Advances in Continuous Flow Technology
Freier ZugriffAmerican Chemical Society | 2020| -
Small Molecule Kinase Inhibitor Drugs (1995–2021): Medical Indication, Pharmacology, and Synthesis
Freier ZugriffAmerican Chemical Society | 2022| -
Understanding the Metabolism of Proteolysis Targeting Chimeras (PROTACs): The Next Step toward Pharmaceutical Applications
Freier ZugriffAmerican Chemical Society | 2020| -
Nonclassical Phenyl Bioisosteres as Effective Replacements in a Series of Novel Open-Source Antimalarials
Freier ZugriffAmerican Chemical Society | 2020| -
Sustainable Drug Discovery of Multi-Target-Directed Ligands for Alzheimer’s Disease
Freier ZugriffAmerican Chemical Society | 2021| -
Sulfonamide Inhibitors of Human Carbonic Anhydrases Designed through a Three-Tails Approach: Improving Ligand/Isoform Matching and Selectivity of Action
Freier ZugriffAmerican Chemical Society | 2020| -
Glycogen Synthase Kinase 3β: A New Gold Rush in Anti-Alzheimer’s Disease Multitarget Drug Discovery?
Freier ZugriffMiniperspectiveAmerican Chemical Society | 2021| -
Direct Observation of Protonation State Modulation in SARS-CoV‑2 Main Protease upon Inhibitor Binding with Neutron Crystallography
Freier ZugriffAmerican Chemical Society | 2021| -
Discovery of TAK-981, a First-in-Class Inhibitor of SUMO-Activating Enzyme for the Treatment of Cancer
Freier ZugriffAmerican Chemical Society | 2021| -
Pyrrolo[2′,3′:3,4]cyclohepta[1,2‑d][1,2]oxazoles, a New Class of Antimitotic Agents Active against Multiple Malignant Cell Types
Freier ZugriffAmerican Chemical Society | 2020| -
The Alpha Keto Amide Moiety as a Privileged Motif in Medicinal Chemistry: Current Insights and Emerging Opportunities
Freier ZugriffAmerican Chemical Society | 2021| -
Discovery and Mechanism of SARS-CoV‑2 Main Protease Inhibitors
Freier ZugriffAmerican Chemical Society | 2022| -
Molecular Engineering of Insulin Icodec, the First Acylated Insulin Analog for Once-Weekly Administration in Humans
Freier ZugriffAmerican Chemical Society | 2021| -
Fragment-to-Lead Medicinal Chemistry Publications in 2020
Freier ZugriffAmerican Chemical Society | 2022| -
Amide-to-Ester Substitution as a Strategy for Optimizing PROTAC Permeability and Cellular Activity
Freier ZugriffAmerican Chemical Society | 2021| -
Fragment-Based Discovery of MRTX1719, a Synthetic Lethal Inhibitor of the PRMT5•MTA Complex for the Treatment of MTAP-Deleted Cancers
Freier ZugriffAmerican Chemical Society | 2022| -
Potent Anti-SARS-CoV‑2 Activity by the Natural Product Gallinamide A and Analogues via Inhibition of Cathepsin L
Freier ZugriffAmerican Chemical Society | 2022| -
Drug Research Meets Network Science: Where Are We?
Freier ZugriffAmerican Chemical Society | 2020| -
Potent Inhibition of Nicotinamide N‑Methyltransferase by Alkene-Linked Bisubstrate Mimics Bearing Electron Deficient Aromatics
Freier ZugriffAmerican Chemical Society | 2021| -
Discovery of AG-270, a First-in-Class Oral MAT2A Inhibitor for the Treatment of Tumors with Homozygous MTAP Deletion
Freier ZugriffAmerican Chemical Society | 2021| -
Discovery of Aficamten (CK-274), a Next-Generation Cardiac Myosin Inhibitor for the Treatment of Hypertrophic Cardiomyopathy
Freier ZugriffAmerican Chemical Society | 2021| -
Garcinoic Acid Is a Natural and Selective Agonist of Pregnane X Receptor
Freier ZugriffAmerican Chemical Society | 2020| -
Development of HDAC Inhibitors Exhibiting Therapeutic Potential in T‑Cell Prolymphocytic Leukemia
Freier ZugriffAmerican Chemical Society | 2021| -
Terphenyl-Based Small-Molecule Inhibitors of Programmed Cell Death-1/Programmed Death-Ligand 1 Protein–Protein Interaction
Freier ZugriffAmerican Chemical Society | 2021| -
Identification of Novel Carbocyclic Pyrimidine Cyclic Dinucleotide STING Agonists for Antitumor Immunotherapy Using Systemic Intravenous Route
Freier ZugriffAmerican Chemical Society | 2021| -
Discovery of GLPG1972/S201086, a Potent, Selective, and Orally Bioavailable ADAMTS‑5 Inhibitor for the Treatment of Osteoarthritis
Freier ZugriffAmerican Chemical Society | 2021| -
Monohydrazone Based G‑Quadruplex Selective Ligands Induce DNA Damage and Genome Instability in Human Cancer Cells
Freier ZugriffAmerican Chemical Society | 2020| -
Structure–Activity Relationships of Triple-Action Platinum(IV) Prodrugs with Albumin-Binding Properties and Immunomodulating Ligands
Freier ZugriffAmerican Chemical Society | 2021| -
Development of Cagrilintide, a Long-Acting Amylin Analogue
Freier ZugriffAmerican Chemical Society | 2021| -
Azidothymidine “Clicked” into 1,2,3-Triazoles: First Report on Carbonic Anhydrase–Telomerase Dual-Hybrid Inhibitors
Freier ZugriffAmerican Chemical Society | 2020| -
Rings in Clinical Trials and Drugs: Present and Future
Freier ZugriffAmerican Chemical Society | 2022| -
A Novel Mitragynine Analog with Low-Efficacy Mu Opioid Receptor Agonism Displays Antinociception with Attenuated Adverse Effects
Freier ZugriffAmerican Chemical Society | 2021| -
Disentangling the Structure–Activity Relationships of Naphthalene Diimides as Anticancer G‑Quadruplex-Targeting Drugs
Freier ZugriffAmerican Chemical Society | 2021| -
Development of BromoTag: A “Bump-and-Hole”–PROTAC System to Induce Potent, Rapid, and Selective Degradation of Tagged Target Proteins
Freier ZugriffAmerican Chemical Society | 2021| -
ACS medicinal chemistry letters
Freier ZugriffGWLB - Gottfried Wilhelm Leibniz Bibliothek | 1.2010 - -
Identification of Potent, Selective, and Orally Bioavailable Small-Molecule GSPT1/2 Degraders from a Focused Library of Cereblon Modulators
Freier ZugriffAmerican Chemical Society | 2021| -
Preclinical Lead Optimization of a 1,2,4-Triazole Based Tankyrase Inhibitor
Freier ZugriffAmerican Chemical Society | 2020| -
Computational Design of Potent D‑Peptide Inhibitors of SARS-CoV‑2
Freier ZugriffAmerican Chemical Society | 2021| -
Designing Chimeric Molecules for Drug Discovery by Leveraging Chemical Biology
Freier ZugriffAmerican Chemical Society | 2020| -
Discovery of Soticlestat, a Potent and Selective Inhibitor for Cholesterol 24-Hydroxylase (CH24H)
Freier ZugriffAmerican Chemical Society | 2021| -
Targeting Acute Myelogenous Leukemia Using Potent Human Dihydroorotate Dehydrogenase Inhibitors Based on the 2‑Hydroxypyrazolo[1,5‑a]pyridine Scaffold: SAR of the Biphenyl Moiety
Freier ZugriffAmerican Chemical Society | 2021| -
Fragment-Derived Selective Inhibitors of Dual-Specificity Kinases DYRK1A and DYRK1B
Freier ZugriffAmerican Chemical Society | 2021| -
Controlling Intramolecular Interactions in the Design of Selective, High-Affinity Ligands for the CREBBP Bromodomain
Freier ZugriffAmerican Chemical Society | 2021| -
Bioisosteric Discovery of NPA101.3, a Second-Generation RET/VEGFR2 Inhibitor Optimized for Single-Agent Polypharmacology
Freier ZugriffAmerican Chemical Society | 2020| -
Targeting Small GTPases and Their Prenylation in Diabetes Mellitus
Freier ZugriffAmerican Chemical Society | 2021|
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