Synthesis, evaluation, and crystallographic analysis of L-371,912: a potent and selective active-site thrombin inhibitor (Englisch)
- Neue Suche nach: Lyle, T. A.
- Neue Suche nach: Chen, Z.
- Neue Suche nach: Appleby, S. D.
- Neue Suche nach: Freidinger, R. M.
- Neue Suche nach: Gardell, S. J.
- Neue Suche nach: Lewis, S. D.
- Neue Suche nach: Li, Y.
- Neue Suche nach: Lyle, E. A.
- Neue Suche nach: Lynch, J. J.
- Neue Suche nach: Mulichak, A. M.
- Neue Suche nach: Lyle, T. A.
- Neue Suche nach: Chen, Z.
- Neue Suche nach: Appleby, S. D.
- Neue Suche nach: Freidinger, R. M.
- Neue Suche nach: Gardell, S. J.
- Neue Suche nach: Lewis, S. D.
- Neue Suche nach: Li, Y.
- Neue Suche nach: Lyle, E. A.
- Neue Suche nach: Lynch, J. J.
- Neue Suche nach: Mulichak, A. M.
In:
BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS
;
7
, 1
;
67-72
;
1997
-
ISSN:
- Aufsatz (Zeitschrift) / Print
-
Titel:Synthesis, evaluation, and crystallographic analysis of L-371,912: a potent and selective active-site thrombin inhibitor
-
Beteiligte:Lyle, T. A. ( Autor:in ) / Chen, Z. ( Autor:in ) / Appleby, S. D. ( Autor:in ) / Freidinger, R. M. ( Autor:in ) / Gardell, S. J. ( Autor:in ) / Lewis, S. D. ( Autor:in ) / Li, Y. ( Autor:in ) / Lyle, E. A. ( Autor:in ) / Lynch, J. J. ( Autor:in ) / Mulichak, A. M. ( Autor:in )
-
Erschienen in:BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS ; 7, 1 ; 67-72
-
Verlag:
-
Erscheinungsdatum:01.01.1997
-
Format / Umfang:6 pages
-
ISSN:
-
Medientyp:Aufsatz (Zeitschrift)
-
Format:Print
-
Sprache:Englisch
- Neue Suche nach: 572.5
- Weitere Informationen zu Dewey Decimal Classification
-
Klassifikation:
DDC: 572.5 -
Datenquelle:
© Metadata Copyright the British Library Board and other contributors. All rights reserved.
Inhaltsverzeichnis – Band 7, Ausgabe 1
Zeige alle Jahrgänge und Ausgaben
Die Inhaltsverzeichnisse werden automatisch erzeugt und basieren auf den im Index des TIB-Portals verfügbaren Einzelnachweisen der enthaltenen Beiträge. Die Anzeige der Inhaltsverzeichnisse kann daher unvollständig oder lückenhaft sein.
- 1
-
Synthesis and evaluation of the anticonvulsant activity of a series of 2-amino-1-phenyl-1-propanols derived from the metabolites of the antidepressant bupropionMusso, D.L. et al. | 1997
- 7
-
Bis-quinolinium cyclophanes: A novel class of potent blockers of the apamin-sensitive Ca2+-activated K+ channelRosa, J.Campos et al. | 1997
- 11
-
Studies on penam sulfones -- III. Synthesis and b-lactamase inhibitory activity of sodium (6R)-6-(a-hydroxybenzyl)-2b-methoxyiminomethyl- 2a-methyl-penam-3a-carboxylate 1,1-dioxide and sodium 2b-acyl-2a-methylpenam-3a-carboxylate 1,1-dioxideCzalkowski, D.P. et al. | 1997
- 11
-
Studies on penam sulfones - III. Synthesis and -lactamase inhibitory activity of sodium (6R)-6-(-hydroxybenzyl)-2-methoxyiminomethyl-2-methylpenam-3-carboxylate 1,1-dioxide and sodium 2-acyl-2-methylpenam-3-carboxylate 1,1-dioxideCzajkowski, D. P. / Reddy, A. V. N. / Setti, E. L. / Phillips, O. A. / Micetich, R. G. / Kunugita, C. / Maiti, S. N. et al. | 1997
- 15
-
Bleomycin model complex bearing a carbamoyl derived substituent capable of coordination to the chelated metal ion as a sixth ligandArai, T. et al. | 1997
- 19
-
SAR for MHC class II binding tetrapeptides: Correlation with potential binding siteCunningham, B.R. et al. | 1997
- 25
-
The synthesis and biological activity of some known and putative metabolites and of the atypical antipsychotic agent olanzapine (LY170053)Calligaro, D.O. et al. | 1997
- 25
-
The synthesis and biological activity of some known and putative metabolites of the atypical antipsychotic agent olanzapine (LY170053)Calligaro, D. O. / Fairhurst, J. / Hotten, T. M. / Moore, N. A. / Tupper, D. E. et al. | 1997
- 31
-
2,3-Substituted 2-azanorbornanes as polar -turn mimeticsHorwell, D. C. / Naylor, D. / Willems, H. M. G. et al. | 1997
- 31
-
2,3-Substituted 2-azanorbomanes as polar b-turn mimeticsHorwell, D.C. et al. | 1997
- 37
-
Structure-activity studies of CTL inhibitory peptides derived from HLA class I moleculesSchwartz, E.J. et al. | 1997
- 41
-
-((Tetronoyl)oxy)- and -((tetramoyl)oxy)methyl ketone inhibitors of the interleukin-1 converting enzyme (ICE)Graybill, T. L. / Prouty, C. P. / Speier, G. J. / Hoyer, D. / Dolle, R. E. / Helaszek, C. T. / Ator, M. A. / Uhl, J. / Strasters, J. et al. | 1997
- 41
-
a-((Tetronoyl)oxy)- and a-((tetramoyl)oxy)methyl ketone inhibitors of the interleukin-1b converting enzyme (ICE)Graybill, T.L. et al. | 1997
- 47
-
Synthesis and biological evaluation of 5,6-diarylimidazo(2.1-b)thiazole as selective COX-2 inhibitorsThérien, M. et al. | 1997
- 53
-
Characterization of the in vitro oxidative metabolites of the COX-2 selective inhibitor L-766,112Trimble, L. A. / Chauret, N. / Silva, J. M. / Nicoll-Griffith, D. A. / Li, C.-S. / Yergey, J. A. et al. | 1997
- 53
-
Characterization of the in vitro oxidative metabolites of the COX-2 selective inhibitor L-766,1122Trimble, L.A. et al. | 1997
- 57
-
A new series of selective COX-2 inhibitors: 5,6-diarylthiazolo(3,2-b)(1,2,4)-triazolesRoy, P. et al. | 1997
- 63
-
Highly preferential cleavage of unpaired guanines in DNA by a functionalized salen-nickel complexRoutler, S. et al. | 1997
- 67
-
Synthesis, evaluation, and crystallographic analysis of L-371,912: a potent and selective active-site thrombin inhibitorLyle, T. A. / Chen, Z. / Appleby, S. D. / Freidinger, R. M. / Gardell, S. J. / Lewis, S. D. / Li, Y. / Lyle, E. A. / Lynch, J. J. / Mulichak, A. M. et al. | 1997
- 67
-
Synthesis, evaluation, and crystallographic analysis of L-371,912: A potent selective active-site thrombin inhibitorLyle, T.A. et al. | 1997
- 73
-
Phosphorothioate oligonucleotides: Largely reduced (n-1)-mer and phosphodiester content through the use of dimeric phosphoramidite synthonsKrotz, A.H. et al. | 1997
- 79
-
S1 heterocyclic thrombin inhibitorsDominguez, C. et al. | 1997
- 85
-
Synthesis and hepatoprotective effects of soyasapogenol B derivativesSasaki, K. et al. | 1997
- 89
-
Imidazotriazinone inhibitors of the Ca2+-calmodulin sensitive phosphodiesterase (PDE 1)Hiasta, D.J. et al. | 1997
- 89
-
Imidazotriazinone inhibitors of the Ca^2^+-calmodulin sensitive phosphodiesterase (PDE I)Hlasta, D. J. / Bode, D. C. / Court, J. J. / Desai, R. C. / Pagani, E. D. / Silver, P. J. et al. | 1997
- 95
-
Combinatorial epitope search: pitfalls of library designYu, Z. / Chu, Y.-H. et al. | 1997
- 95
-
Combinatorial epitope search: Piffalls of library designYu, Z. et al. | 1997
-
Instructions to Contributors| 1997
-
Aims & Scope| 1997