Hydrogenative desulphurization of thienopyrrolizinones: An easy and selective access to (Z)-phenethylidenepyrrolizinones with in vitro cytotoxic activity (Englisch)
- Neue Suche nach: Perri, V.
- Neue Suche nach: Rochais, C.
- Neue Suche nach: Sopkova-de Oliveira Santos, J.
- Neue Suche nach: Legay, R.
- Neue Suche nach: Cresteil, T.
- Neue Suche nach: Dallemagne, P.
- Neue Suche nach: Rault, S.
- Neue Suche nach: Perri, V.
- Neue Suche nach: Rochais, C.
- Neue Suche nach: Sopkova-de Oliveira Santos, J.
- Neue Suche nach: Legay, R.
- Neue Suche nach: Cresteil, T.
- Neue Suche nach: Dallemagne, P.
- Neue Suche nach: Rault, S.
In:
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
;
45
, 3
;
1146-1150
;
2010
-
ISSN:
- Aufsatz (Zeitschrift) / Print
-
Titel:Hydrogenative desulphurization of thienopyrrolizinones: An easy and selective access to (Z)-phenethylidenepyrrolizinones with in vitro cytotoxic activity
-
Beteiligte:Perri, V. ( Autor:in ) / Rochais, C. ( Autor:in ) / Sopkova-de Oliveira Santos, J. ( Autor:in ) / Legay, R. ( Autor:in ) / Cresteil, T. ( Autor:in ) / Dallemagne, P. ( Autor:in ) / Rault, S. ( Autor:in )
-
Erschienen in:EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY ; 45, 3 ; 1146-1150
-
Verlag:
- Neue Suche nach: Elsevier Science B.V., Amsterdam.
-
Erscheinungsdatum:01.01.2010
-
Format / Umfang:5 pages
-
ISSN:
-
Medientyp:Aufsatz (Zeitschrift)
-
Format:Print
-
Sprache:Englisch
- Neue Suche nach: 615.1
- Weitere Informationen zu Dewey Decimal Classification
-
Klassifikation:
DDC: 615.1 -
Datenquelle:
© Metadata Copyright the British Library Board and other contributors. All rights reserved.
Inhaltsverzeichnis – Band 45, Ausgabe 3
Zeige alle Jahrgänge und Ausgaben
Die Inhaltsverzeichnisse werden automatisch erzeugt und basieren auf den im Index des TIB-Portals verfügbaren Einzelnachweisen der enthaltenen Beiträge. Die Anzeige der Inhaltsverzeichnisse kann daher unvollständig oder lückenhaft sein.
- 857
-
Design, synthesis and pharmacological screening of potential anticonvulsant agents using hybrid approachGhogare, J. G. / Bhandari, S. V. / Bothara, K. G. / Madgulkar, A. R. / Parashar, G. A. / Sonawane, B. G. / Inamdar, P. R. et al. | 2010
- 864
-
Synthesis and antiprotozoal activity of 4-arylcoumarinsPierson, J. T. / Dumetre, A. / Hutter, S. / Delmas, F. / Laget, M. / Finet, J. P. / Azas, N. / Combes, S. et al. | 2010
- 870
-
Synthesis of potent BACE-1 inhibitors incorporating a hydroxyethylene isostere as central coreWangsell, F. / Gustafsson, K. / Kvarnstrom, I. / Borkakoti, N. / Edlund, M. / Jansson, K. / Lindberg, J. / Hallberg, A. / Rosenquist, A. / Samuelsson, B. et al. | 2010
- 883
-
Synthesis, characterization and biocidal activity of new organotin complexes of 2-(3-oxocyclohex-1-enyl)benzoic acidVieira, F. T. / de Lima, G. M. / Maia, J. R. / Speziali, N. L. / Ardisson, J. D. / Rodrigues, L. / Correa, A. / Romero, O. B. et al. | 2010
- 890
-
Novel phosphoramidates with porphine and nitrogenous drug: One-pot synthesis and orientation to cancer cellsWang, Z. W. / Guo, C. C. / Xie, W. Z. / Liu, C. Z. / Xiao, C. G. / Tan, Z. et al. | 2010
- 896
-
5-Substituted [1]pyrindine derivatives with antiproliferative activityKolb, S. / Goddard, M. L. / Loukaci, A. / Mondesert, O. / Ducommun, B. / Braud, E. / Garbay, C. et al. | 2010
- 902
-
Conventional and microwave assisted synthesis of small molecule based biologically active heterocyclic amidine derivativesSondhi, S. M. / Rani, R. / Roy, P. / Agrawal, S. K. / Saxena, A. K. et al. | 2010
- 909
-
Synthesis and biological evaluation of [1,2,4]triazino[4,3-a] benzimidazole acetic acid derivatives as selective aldose reductase inhibitorsSahoo, P. K. / Behera, P. et al. | 2010
- 915
-
Synthesis and antibacterial activity of novel 3-O-carbamoyl derivatives of clarithromycin and 11,12-cyclic carbonate azithromycinZhang, L. / Song, L. / Liu, Z. / Li, H. / Lu, Y. / Li, Z. / Ma, S. et al. | 2010
- 923
-
Synthesis and biological activity of derivatives of the marine quinone avaroneBozic, T. / Novakovic, I. / Gasic, M. J. / Juranic, Z. / Stanojkovic, T. / Tufegdzic, S. / Kljajic, Z. / Sladic, D. et al. | 2010
- 930
-
Neural computational prediction of oral drug absorption based on CODES 2D descriptorsGuerra, A. / Campillo, N. E. / Paez, J. A. et al. | 2010
- 941
-
Curcuminoid analogs with potent activity against Trypanosoma and Leishmania speciesChangtam, C. / de Koning, H. P. / Ibrahim, H. / Sajid, M. S. / Gould, M. K. / Suksamrarn, A. et al. | 2010
- 957
-
New 1,3-oxazolo[4,5-c]quinoline derivatives: Synthesis and evaluation of antibacterial and antituberculosis propertiesEswaran, S. / Adhikari, A. V. / Ajay Kumar, R. et al. | 2010
- 967
-
CoMFA and molecular docking studies of benzoxazoles and benzothiazoles as CYP450 1A1 inhibitorsPan, J. / Liu, G. Y. / Cheng, J. / Chen, X. J. / Ju, X. L. et al. | 2010
- 973
-
Synthesis and antitumor activity of new dihydropyridine thioglycosides and their corresponding dehydrogenated formsAbbas, H. A. / El Sayed, W. A. / Fathy, N. M. et al. | 2010
- 983
-
Molecular modeling study of binding site selectivity of TQMP to G-quadruplex DNAAixiao, L. / Francois, M. / Florent, B. / Michel, D. / Baoshan, W. / Xiang, Z. / Ping, W. et al. | 2010
- 992
-
Synthesis, characterization and structure-activity relationship of novel N-phosphorylated E,E-3,5-bis(thienylidene)piperid-4-onesMakarov, M. V. / Leonova, E. S. / Rybalkina, E. Y. / Tongwa, P. / Khrustalev, V. N. / Timofeeva, T. V. / Odinets, I. L. et al. | 2010
- 1001
-
Synthesis of glycoside derivatives of hydroxyanthraquinone with ability to dissolve and inhibit formation of crystals of calcium oxalate. Potential compounds in kidney stone therapyFrackowiak, A. / Skibinski, P. / Gawel, W. / Zaczynska, E. / Czarny, A. / Gancarz, R. et al. | 2010
- 1008
-
Docking and 3D-QSAR studies of influenza neuraminidase inhibitors using three-dimensional holographic vector of atomic interaction field analysisSun, J. / Cai, S. / Yan, N. / Mei, H. et al. | 2010
- 1015
-
A theoretical study of the structure-radical scavenging activity of trans-resveratrol analogues and cis-resveratrol in gas phase and water environmentMikulski, D. / Gorniak, R. / Molski, M. et al. | 2010
- 1028
-
Synthesis and antimicrobial activities of 3-O-alkyl analogues of (+)-catechin: Improvement of stability and proposed action mechanismPark, K. D. / Cho, S. J. et al. | 2010
- 1034
-
New pH-dependent complexes, from mononuclear Pd(II) monomer to heteronuclear [Pd(II),K(I)]Polymer: DNA cleavage and cytotoxicity in vitroGao, E. J. / Zhu, M. C. / Huang, Y. / Liu, L. / Liu, H. Y. / Liu, F. C. / Ma, S. / Shi, C. Y. et al. | 2010
- 1042
-
New pyrazoles incorporating pyrazolylpyrazole moiety: Synthesis, anti-HCV and antitumor activityRiyadh, S. M. / Farghaly, T. A. / Abdallah, M. A. / Abdalla, M. M. / Abd El-Aziz, M. R. et al. | 2010
- 1051
-
Ruthenium(II)-arene complexes with functionalized pyridines: Synthesis, characterization and cytotoxic activityGrguric-Sipka, S. / Ivanovic, I. / Rakic, G. / Todorovic, N. / Gligorijevic, N. / Radulovic, S. / Arion, V. B. / Keppler, B. K. / Tesic, Z. L. et al. | 2010
- 1059
-
Antioxidant and antiviral activities of silybin fatty acid conjugatesGazak, R. / Purchartova, K. / Marhol, P. / Zivna, L. / Sedmera, P. / Valentova, K. / Kato, N. / Matsumura, H. / Kaihatsu, K. / Kren, V. et al. | 2010
- 1068
-
Synthesis of new spiroindolinones incorporating a benzothiazole moiety as antioxidant agentsKaral&imath / N. / Guzel, O. / Ozsoy, N. / Ozbey, S. / Salman, A. i. et al. | 2010
- 1078
-
Synthesis, antibacterial and antiviral properties of curcumin bioconjugates bearing dipeptide, fatty acids and folic acidSingh, R. K. / Rai, D. / Yadav, D. / Bhargava, A. / Balzarini, J. / De Clercq, E. et al. | 2010
- 1087
-
QSAR study on melanocortin-4 receptors by support vector machinePourbasheer, E. / Riahi, S. / Ganjali, M. R. / Norouzi, P. et al. | 2010
- 1094
-
Synthesis, antibacterial and antifungal activities of 6,5 fused steroidal oxazoles in cholestane seriesKhan, M. S. / Alam, M. / Tabassum, Z. / Ahmad, A. / Khan, A. U. et al. | 2010
- 1098
-
Pharmacophoric model building for antitubercular activity of the individual Schiff bases of small combinatorial libraryAbdel-Aal, W. S. / Hassan, H. Y. / Aboul-Fadl, T. / Youssef, A. F. et al. | 2010
- 1107
-
Synthesis of tropolone derivatives and evaluation of their in vitro neuroprotective activityKoufaki, M. / Theodorou, E. / Alexi, X. / Nikoloudaki, F. / Alexis, M. N. et al. | 2010
- 1113
-
QSAR study of isatin analogues as in vitro anti-cancer agentsSabet, R. / Mohammadpour, M. / Sadeghi, A. / Fassihi, A. et al. | 2010
- 1119
-
Predictive comparative QSAR modelling of (phenylpiperazinyl-alkyl) oxindoles as selective 5-HT1A antagonists by stepwise regression, PCRA, FA-MLR and PLS techniquesAdhikari, N. / Maiti, M. K. / Jha, T. et al. | 2010
- 1128
-
Synthesis, in vitro antibacterial and antifungal evaluations of new a-hydroxyphosphonate and new a-acetoxyphosphonate derivatives of tetrazolo [1, 5-a] quinolineKategaonkar, A. H. / Pokalwar, R. U. / Sonar, S. S. / Gawali, V. U. / Shingate, B. B. / Shingare, M. S. et al. | 2010
- 1133
-
Discovery of benzhydrylpiperazine derivatives as CB1 receptor inverse agonists via privileged structure-based approachMeng, T. / Wang, J. / Peng, H. / Fang, G. / Li, M. / Xiong, B. / Xie, X. / Zhang, Y. / Wang, X. / Shen, J. et al. | 2010
- 1140
-
Structure of aldehyde reductase in ternary complex with a 5-arylidene-2,4-thiazolidinedione aldose reductase inhibitorCarbone, V. / Giglio, M. / Chung, R. / Huyton, T. / Adams, J. / Maccari, R. / Ottana, R. / Hara, A. / El-Kabbani, O. et al. | 2010
- 1146
-
Hydrogenative desulphurization of thienopyrrolizinones: An easy and selective access to (Z)-phenethylidenepyrrolizinones with in vitro cytotoxic activityPerri, V. / Rochais, C. / Sopkova-de Oliveira Santos, J. / Legay, R. / Cresteil, T. / Dallemagne, P. / Rault, S. et al. | 2010
- 1151
-
Synthesis and antimicrobial studies on novel sulfonamides containing 4-azidomethyl coumarinBasanagouda, M. / Shivashankar, K. / Kulkarni, M. V. / Rasal, V. P. / Patel, H. / Mutha, S. S. / Mohite, A. A. et al. | 2010
- 1158
-
Design, synthesis, and biological evaluation of novel pyrimidine derivatives as CDK2 inhibitorsIbrahim, D. A. / El-Metwally, A. M. et al. | 2010
- 1167
-
Prediction of acetylcholinesterase inhibitors and characterization of correlative molecular descriptors by machine learning methodsLv, W. / Xue, Y. et al. | 2010
- 1173
-
Synthesis and antimicrobial activities of novel 1,5-diaryl pyrazolesRagavan, R. V. / Vijayakumar, V. / Kumari, N. S. et al. | 2010
- 1181
-
Synthesis, characterization and antibacterial activities of some new ferrocene-containing penemsLong, B. / He, C. / Yang, Y. / Xiang, J. et al. | 2010
- 1189
-
Identification of antibacterial and antifungal pharmacophore sites for potent bacteria and fungi inhibition: Indolenyl sulfonamide derivativesChohan, Z. H. / Youssoufi, M. H. / Jarrahpour, A. / Ben Hadda, T. et al. | 2010
- 1200
-
Antimicrobial study of newly synthesized 6-substituted indolo[1,2-c]quinazolinesRohini, R. / Muralidhar Reddy, P. / Shanker, K. / Hu, A. / Ravinder, V. et al. | 2010
- 1206
-
Synthesis, characterization and biological activity of some new 1,3,4-oxadiazole bearing 2-flouro-4-methoxy phenyl moietyChandrakantha, B. / Shetty, P. / Nambiyar, V. / Isloor, N. / Isloor, A. M. et al. | 2010
- 1211
-
6-Substituted 2-(N-trifluoroacetylamino)imidazopyridines induce cell cycle arrest and apoptosis in SK-LU-1 human cancer cell lineMartinez-Urbina, M. A. / Zentella, A. / Vilchis-Reyes, M. A. / Guzman, A. / Vargas, O. / Ramirez Apan, M. T. / Ventura Gallegos, J. L. / Diaz, E. et al. | 2010
- 1220
-
Synthesis and antioxidant properties of enone core based dendrimers with carbazole as surface groupRajakumar, P. / Venkatesan, N. / Sekar, K. / Nagaraj, S. / Rengasamy, R. et al. | 2010
- 1225
-
Synthesis and investigation of inhibition effect of fluorinated sulfonamide derivatives on carbonic anhydraseBenfodda, Z. / Guillen, F. / Romestand, B. / Dahmani, A. / Blancou, H. et al. | 2010
- 1230
-
New 14-membered octaazamacrocyclic complexes: Synthesis, spectral, antibacterial and antifungal studiesSingh, D. P. / Kumar, K. / Sharma, C. et al. | 2010
- 1237
-
Synthesis, cytotoxicity, antiviral activity and interferon inducing ability of 6-(2-aminoethyl)-6H-indolo[2,3-b]quinoxalinesShibinskaya, M. O. / Lyakhov, S. A. / Mazepa, A. V. / Andronati, S. A. / Turov, A. V. / Zholobak, N. M. / Spivak, N. Y. et al. | 2010
- 1244
-
An expeditious synthesis and anticancer activity of novel 4-(3prime-indolyl)oxazolesKumar, D. / Kumar, N. M. / Sundaree, S. / Johnson, E. O. / Shah, K. et al. | 2010
- 1250
-
Synthesis and evaluation of the a-glucosidase inhibitory activity of 3-[4-(phenylsulfonamido)benzoyl]-2H-1-benzopyran-2-one derivativesWang, S. / Yan, J. / Wang, X. / Yang, Z. / Lin, F. / Zhang, T. et al. | 2010
- 1256
-
Synthesis of highly functionalized barbituric acids and study of their interactions with p-glycoprotein and Mg2+ - Potential candidates for multi drug resistance modulationSingh, P. / Kaur, J. / Bhardwaj, A. et al. | 2010
- 1263
-
Simultaneous tritium labelling of two potent 5-HT4 ligandsSobrio, F. / Lemaitre, S. / Hinsberger, A. / Barre, L. / Rousseau, B. / Rault, S. et al. | 2010
- iii
-
Graphical contents list| 2010
-
Editorial board| 2010