2prime-Deoxy-2prime-a-fluoro-2prime-b-C-methyl 3prime,5prime-cyclic phosphate nucleotide prodrug analogs as inhibitors of HCV NS5B polymerase: Discovery of PSI-352938 (Englisch)
- Neue Suche nach: Reddy, P. G.
- Neue Suche nach: Bao, D.
- Neue Suche nach: Chang, W.
- Neue Suche nach: Chun, B. K.
- Neue Suche nach: Du, J.
- Neue Suche nach: Nagarathnam, D.
- Neue Suche nach: Rachakonda, S.
- Neue Suche nach: Ross, B. S.
- Neue Suche nach: Zhang, H. R.
- Neue Suche nach: Bansal, S.
- Neue Suche nach: Reddy, P. G.
- Neue Suche nach: Bao, D.
- Neue Suche nach: Chang, W.
- Neue Suche nach: Chun, B. K.
- Neue Suche nach: Du, J.
- Neue Suche nach: Nagarathnam, D.
- Neue Suche nach: Rachakonda, S.
- Neue Suche nach: Ross, B. S.
- Neue Suche nach: Zhang, H. R.
- Neue Suche nach: Bansal, S.
In:
BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS
;
20
, 24
;
7376-7380
;
2010
-
ISSN:
- Aufsatz (Zeitschrift) / Print
-
Titel:2prime-Deoxy-2prime-a-fluoro-2prime-b-C-methyl 3prime,5prime-cyclic phosphate nucleotide prodrug analogs as inhibitors of HCV NS5B polymerase: Discovery of PSI-352938
-
Beteiligte:Reddy, P. G. ( Autor:in ) / Bao, D. ( Autor:in ) / Chang, W. ( Autor:in ) / Chun, B. K. ( Autor:in ) / Du, J. ( Autor:in ) / Nagarathnam, D. ( Autor:in ) / Rachakonda, S. ( Autor:in ) / Ross, B. S. ( Autor:in ) / Zhang, H. R. ( Autor:in ) / Bansal, S. ( Autor:in )
-
Erschienen in:BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS ; 20, 24 ; 7376-7380
-
Verlag:
- Neue Suche nach: Elsevier Science B.V., Amsterdam.
-
Erscheinungsdatum:01.01.2010
-
Format / Umfang:5 pages
-
ISSN:
-
Medientyp:Aufsatz (Zeitschrift)
-
Format:Print
-
Sprache:Englisch
- Neue Suche nach: 572.5
- Weitere Informationen zu Dewey Decimal Classification
-
Klassifikation:
DDC: 572.5 -
Datenquelle:
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- 7488
-
Second generation analogs of rigid 6,7-spiro scaffolds targeting the bacterial ribosomeStathakis, Christos I. / Mavridis, Ioannis / Kythreoti, Georgia / Papakyriakou, Athanasios / Katsoulis, Ioannis A. / Cottin, Thomas / Anastasopoulou, Panoula / Vourloumis, Dionisios et al. | 2010
- 7493
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Synthesis of new acylsulfamoyl benzoxaboroles as potent inhibitors of HCV NS3 proteaseLi, Xianfeng / Zhang, Yong-Kang / Liu, Yang / Zhang, Suoming / Ding, Charles Z. / Zhou, Yasheen / Plattner, Jacob J. / Baker, Stephen J. / Liu, Liang / Bu, Wei et al. | 2010
- 7498
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Development of a sphingosine kinase 1 specific small-molecule inhibitorHengst, Jeremy A. / Wang, XuJun / Sk, Ugir H. / Sharma, Arun K. / Amin, Shantu / Yun, Jong K. et al. | 2010
- 7503
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N-Aryl-benzimidazolones as novel small molecule HSP90 inhibitorsBruncko, Milan / Tahir, Stephen K. / Song, Xiaohong / Chen, Jun / Ding, Hong / Huth, Jeffrey R. / Jin, Sha / Judge, Russell A. / Madar, David J. / Park, Chang H. et al. | 2010
- 7507
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Indium(III) chloride catalyzed three-component coupling reaction: A novel synthesis of 2-substituted aryl(indolyl)kojic acid derivatives as potent antifungal and antibacterial agentsReddy, B.V. Subba / Reddy, M. Ramana / Madan, Ch. / Kumar, K. Pranay / Rao, M. Srinivasa et al. | 2010
- 7512
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1,2,3-Triazolyl amino acids as AMPA receptor ligandsStanley, N.J. / Pedersen, D. Sejer / Nielsen, B. / Kvist, T. / Mathiesen, J.M. / Bräuner-Osborne, H. / Taylor, D.K. / Abell, A.D. et al. | 2010
- 7516
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Synthesis of potent, substituted carbazoles as selective androgen receptor modulators (SARMs)Miller, Chris P. / Bhaket, Pushpal / Muthukaman, Nagarajan / Lyttle, C. Richard / Shomali, Maysoun / Gallacher, Kyla / Slocum, Connie / Hattersley, Gary et al. | 2010
- 7521
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The identification of novel orally active mGluR5 antagonist GSK2210875Pilla, Maria / Andreoli, Michela / Tessari, Michela / Delle-Fratte, Sonia / Roth, Adelheid / Butler, Sharon / Brown, Fiona / Shah, Parita / Bettini, Ezio / Cavallini, Palmina et al. | 2010
- 7525
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Synthesis and pharmacological evaluation of the stereoisomers of 3-carba cyclic-phosphatidic acidGupte, Renuka / Siddam, Anjaih / Lu, Yan / Li, Wei / Fujiwara, Yuko / Panupinthu, Nattapon / Pham, Truc-Chi / Baker, Daniel L. / Parrill, Abby L. / Gotoh, Mari et al. | 2010
- 7529
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Inhibition of human neuraminidase 3 (NEU3) by C9-triazole derivatives of 2,3-didehydro-N-acetyl-neuraminic acidZou, Yao / Albohy, Amgad / Sandbhor, Mahendra / Cairo, Christopher W. et al. | 2010
- 7534
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Changes in flavonoid content and tyrosinase inhibitory activity in kenaf leaf extract after far-infrared treatmentRho, Ho Sik / Ahn, Soo Mi / Lee, Bum Chun / Kim, Myung Kyoo / Ghimeray, Amal Kumar / Jin, Cheng Wu / Cho, Dong Ha et al. | 2010
- 7537
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Synthesis and in vitro inhibitory activity of matrine derivatives towards pro-inflammatory cytokinesHu, Honggang / Wang, Shaozhan / Zhang, Chunmei / Wang, Liang / Ding, Li / Zhang, Junping / Wu, Qiuye et al. | 2010
- 7540
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N-(8-(3-Ethynylphenoxy)octyl-1-deoxynojirimycin suppresses growth and migration of human lung cancer cellsZhao, Yunxue / Liu, Wenjia / Zhou, Ying / Zhang, Xiumei / Murphy, Paul V. et al. | 2010
- 7544
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Two new cytotoxic labdane diterpenes from the rhizomes of Hedychium coronariumSuresh, G. / Prabhakar Reddy, P. / Suresh Babu, K. / Shaik, Thokhir Basha / Kalivendi, Shasi Vardhan et al. | 2010
- 7549
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SAR studies of gymnasterkoreayne derivatives with cancer chemopreventive activitiesShin, Dongyun / Yang, Jung-Eun / Lee, Saet Byoul / Nho, Chu Won et al. | 2010
- 7553
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Corrigendum to "Design, synthesis, and structure-activity relationship of novel orally efficacious pyrazole/sulfonamide based dihydroquinoline g-secretase inhibitors" [Bioorg. Med. Chem. Lett. 19 (2009) 4920]Truong, A. P. / Aubele, D. L. / Probst, G. D. / Neitzel, M. L. / Semko, C. M. / Bowers, S. / Dressen, D. / Hom, R. K. / Konradi, A. W. / Sham, H. L. et al. | 2010
- 7553
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Corrigendum to “Design, synthesis, and structure–activity relationship of novel orally efficacious pyrazole/sulfonamide based dihydroquinoline γ-secretase inhibitors” [Bioorg. Med. Chem. Lett. 19 (2009) 4920]Truong, Anh P. / Aubele, Danielle L. / Probst, Gary D. / Neitzel, Martin L. / Semko, Chris M. / Bowers, Simeon / Dressen, Darren / Hom, Roy K. / Konradi, Andrei W. / Sham, Hing L. et al. | 2010
- 7554
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Corrigendum to “New hydroxypyrimidinone-containing sulfonamides as carbonic anhydrase inhibitors also acting as MMP inhibitors” [Bioorg. Med. Chem. Lett. 20 (2010) 3623–3627]Esteves, M. Alexandra / Ortet, Osvaldo / Capelo, Anabela / Supuran, Claudiu T. / Marques, Sérgio M. / Santos, M. Amélia et al. | 2010
- 7555
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Corrigendum to “2-Arylbenzoxazoles as CETP inhibitors: Substitution of the benzoxazole moiety” [Bioorg. Med. Chem. Lett. 20 (2010) 346]Smith, Cameron J. / Ali, Amjad / Chen, Liya / Hammond, Milton L. / Anderson, Matt S. / Chen, Ying / Eveland, Suzanne S. / Guo, Qiu / Hyland, Sheryl A. / Milot, Denise P. et al. | 2010
- IFC
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Editorial board| 2010