Design, synthesis and biological evaluation of selective hybrid coumarin-thiazolidinedione aldose reductase-II inhibitors as potential antidiabetics (Englisch)
- Neue Suche nach: Kumar Pasala, Vijay
- Neue Suche nach: Gudipudi, Gopinath
- Neue Suche nach: Sankeshi, Venu
- Neue Suche nach: Basude, Manohar
- Neue Suche nach: Gundla, Rambabu
- Neue Suche nach: singh Jadav, Surendar
- Neue Suche nach: Srinivas, Burra
- Neue Suche nach: Yadaiah Goud, E.
- Neue Suche nach: Nareshkumar, Devasani
- Neue Suche nach: Kumar Pasala, Vijay
- Neue Suche nach: Gudipudi, Gopinath
- Neue Suche nach: Sankeshi, Venu
- Neue Suche nach: Basude, Manohar
- Neue Suche nach: Gundla, Rambabu
- Neue Suche nach: singh Jadav, Surendar
- Neue Suche nach: Srinivas, Burra
- Neue Suche nach: Yadaiah Goud, E.
- Neue Suche nach: Nareshkumar, Devasani
In:
Bioorganic Chemistry
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114
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2021
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ISSN:
- Aufsatz (Zeitschrift) / Elektronische Ressource
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Titel:Design, synthesis and biological evaluation of selective hybrid coumarin-thiazolidinedione aldose reductase-II inhibitors as potential antidiabetics
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Beteiligte:Kumar Pasala, Vijay ( Autor:in ) / Gudipudi, Gopinath ( Autor:in ) / Sankeshi, Venu ( Autor:in ) / Basude, Manohar ( Autor:in ) / Gundla, Rambabu ( Autor:in ) / singh Jadav, Surendar ( Autor:in ) / Srinivas, Burra ( Autor:in ) / Yadaiah Goud, E. ( Autor:in ) / Nareshkumar, Devasani ( Autor:in )
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Erschienen in:Bioorganic Chemistry ; 114
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Verlag:
- Neue Suche nach: Elsevier Inc.
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Erscheinungsdatum:04.05.2021
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ISSN:
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DOI:
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Medientyp:Aufsatz (Zeitschrift)
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Format:Elektronische Ressource
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Sprache:Englisch
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Schlagwörter:
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Datenquelle:
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Issue TOC| 2021
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Design, synthesis and biological evaluation of selective hybrid coumarin-thiazolidinedione aldose reductase-II inhibitors as potential antidiabeticsKumar Pasala, Vijay / Gudipudi, Gopinath / Sankeshi, Venu / Basude, Manohar / Gundla, Rambabu / singh Jadav, Surendar / Srinivas, Burra / Yadaiah Goud, E. / Nareshkumar, Devasani et al. | 2021
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The design and synthesis of transient receptor potential vanilloid 3 inhibitors with novel skeletonLv, Mengqi / Wu, Han / Qu, Yaxuan / Wu, Siyi / Wang, Junxia / Wang, Congcong / Luan, Yepeng / Zhang, Zhongyin et al. | 2021
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High activity, high selectivity and high biocompatibility BODIPY-pyrimidine derivatives for fluorescence target recognition and evaluation of inhibitory activityXu, Chi / Shao, Tingyu / Shao, Shihe / Jin, Guofan et al. | 2021
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Cyanobiphenyls: Novel H3 receptor ligands with cholinesterase and MAO B inhibitory activity as multitarget compounds for potential treatment of Alzheimer’s diseaseGodyń, Justyna / Zaręba, Paula / Łażewska, Dorota / Stary, Dorota / Reiner-Link, David / Frank, Annika / Latacz, Gniewomir / Mogilski, Szczepan / Kaleta, Maria / Doroz-Płonka, Agata et al. | 2021
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N-acylhydrazones confer inhibitory efficacy against New Delhi metallo-β-lactamase-1Gao, Han / Li, Jia-Qi / Kang, Peng-Wei / Chigan, Jia-Zhu / Wang, Huan / Liu, Lu / Xu, Yin-Sui / Zhai, Le / Yang, Ke-Wu et al. | 2021
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Polycyclic polyprenylated acylphloroglucinols with immunosuppressive activity from Hypericum perforatum and absolute configurations assignment of previously reported analoguesGuo, Yi / Cao, Yunfang / Qi, Changxing / Tong, Qingyi / Chen, Chunmei / Yang, Jing / Zhu, Hucheng / Zhang, Yonghui et al. | 2021
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Enhancing the tumor cell selectivity of a rhodamine-decorated iridium(III) complex by conjugating with indomethacin for COX-2 targeted photodynamic therapyLiu, Chuangjun / Xiang, Jingjing / Xiang, Chunbai / Li, Hongfeng et al. | 2021
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Novel thiazolidine derivatives as potent selective pro-apoptotic agentsHafez, Donia E. / Hafez, Eman / Eddiasty, Islam / Shih, Shou-Ping / Chien, Leng-Chiang / Hong, Yi-Jia / Lin, Hung-Yu / Keeton, Adam B. / Piazza, Gary A. / Abdel-Halim, Mohammad et al. | 2021
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A magnified aptamer fluorescence sensor based on the metal organic frameworks adsorbed DNA with enzyme catalysis amplification for ultra-sensitive determination of ATP and its logic gate operationYao, Jun / Yue, Tingting / Huang, Cheng / Wang, Heng et al. | 2021
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Discovery of 1,3,4,5-tetrasubstituted pyrazoles as anti-trypanosomatid agents: Identification of alterations in flagellar structure of L. amazonensisda Silva, Michael J.V. / Jacomini, Andrey P. / Gonçalves, Davana S. / Pianoski, Karlos Eduardo / Poletto, Julia / Lazarin-Bidóia, Danielle / Volpato, Hélito / Nakamura, Celso V. / Rosa, Fernanda A. et al. | 2021
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PROTACs technology for targeting non-oncoproteins: Advances and perspectivesWang, Chao / Zhang, Yujing / Xing, Dongming / Zhang, Renshuai et al. | 2021
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Optimization of pyrazole-based compounds with 1,2,4-triazole-3-thiol moiety as selective COX-2 inhibitors cardioprotective drug candidates: Design, synthesis, cyclooxygenase inhibition, anti-inflammatory, ulcerogenicity, cardiovascular evaluation, and molecular modeling studiesAbdellatif, Khaled R.A. / Abdelall, Eman K.A. / Elshemy, Heba A.H. / Philoppes, John N. / Hassanein, Emad H.M. / Kahk, Nesma M. et al. | 2021
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New cytotoxic dichapetalins in the leaves of Phyllanthus acidus: Identification, quantitative analysis, and preliminary toxicity assessmentGeng, Hui-Chun / Zhu, Hong-Tao / Yang, Wei-Nong / Wang, Dong / Yang, Chong-Ren / Zhang, Ying-Jun et al. | 2021
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Design, synthesis, in vitro and in silico studies of some novel thiazole-dihydrofuran derivatives as aromatase inhibitorsOsmaniye, Derya / Görgülü, Şennur / Sağlık, Begüm Nurpelin / Levent, Serkan / Özkay, Yusuf / Kaplancıklı, Zafer Asım et al. | 2021
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Anti-tumor compounds identification from gossypol Groebke imidazopyridine productWang, Wei / Lu, Yuzhi / Chen, Enhui / Shen, Kang / Li, Jun et al. | 2021
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Pharmacophore-based drug design of AChE and BChE dual inhibitors as potential anti-Alzheimer’s disease agentsGao, Hongwei / Jiang, Yingying / Zhan, Jiuyu / Sun, Yingni et al. | 2021
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Discovery of Novel Dihydropyrimidine and hydroxamic acid hybrids as potent Helicobacter pylori Urease inhibitorsMamidala, Ravinder / Bhimathati, Solomon Raj S. / Vema, Aparna et al. | 2021
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Potential drug development and therapeutic approaches for clinical intervention in COVID-19Dowarah, Jayanta / Marak, Brilliant N. / Yadav, Umesh Chand Singh / Singh, Ved Prakash et al. | 2021
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Synthesis of novel 5-(2,5-bis(2,2,2-trifluoroethoxy)phenyl)-1,3,4-oxadiazole-2-thiol derivatives as potential glucosidase inhibitorsGani, Ramesh S. / Kudva, Avinash K. / Timanagouda, Karabasanagouda / Raghuveer / Mujawar, Salma Begum Hussain / Joshi, Shrinivas D. / Raghu, Shamprasad Varija et al. | 2021
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Design, synthesis and biological evaluation of glycolamide, glycinamide, and β-amino carbonyl 1,2,4-triazole derivatives as DPP-4 inhibitorsFuh, Mao-Tsu / Tseng, Ching-Chun / Li, Sin-Min / Tsai, Shuo-En / Chuang, Tsung-Jui / Lu, Chih-Hao / Yang, Ya-Chen / Tsai, Henry J. / Wong, Fung Fuh et al. | 2021
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Bioactive sesquiterpenes from Inula heleniumZheng, Xiaoqin / Wu, Zi / Xu, Jie / Zhang, Xinxin / Tu, Yijun / Lei, Jiachuan / Yuan, Ruiying / Cheng, Haitao / Wang, Qiang / Yu, Jianqing et al. | 2021
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Investigation of indole functionalized pyrazoles and oxadiazoles as anti-inflammatory agents: Synthesis, in-vivo, in-vitro and in-silico analysisKumar, Devendra / Kumar, Ravi Ranjan / Pathania, Shelly / Singh, Pankaj Kumar / Kalra, Sourav / Kumar, Bhupinder et al. | 2021
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Structural exploration of multifunctional monoamine oxidase B inhibitors as potential drug candidates against Alzheimer’s diseaseZhang, Changjun / Lv, Yangjing / Bai, Renren / Xie, Yuanyuan et al. | 2021
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Synthesis, in vitro biological investigation, and molecular dynamics simulations of thiazolopyrimidine based compounds as corticotrophin releasing factor receptor-1 antagonistsElgiushy, Hossam R. / Abou-Taleb, Nageh A. / Holz, George G. / Chepurny, Oleg G. / Pirmettis, Ioannis / Kakabakos, Sotirios / Karageorgos, Vlasios / Liapakis, George / Albohy, Amgad / Abouzid, Khaled A.M. et al. | 2021
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3-Arylamino-quinoxaline-2-carboxamides inhibit the PI3K/Akt/mTOR signaling pathways to activate P53 and induce apoptosisChen, Nan-Ying / Lu, Ke / Yuan, Jing-Mei / Li, Xiao-Juan / Gu, Zi-Yu / Pan, Cheng-Xue / Mo, Dong-Liang / Su, Gui-Fa et al. | 2021
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Design, synthesis and biological evaluation of novel pyrazolopyrimidone derivatives as potent PDE1 inhibitorsZhang, Bei / Huang, Yue / Zhang, Si-Rui / Huang, Meng-Xing / Zhang, Chen / Luo, Hai-Bin et al. | 2021
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Identification of inhibitors targeting polyketide synthase 13 of Mycobacterium tuberculosis as antituberculosis drug leadsWang, Xiao / Zhao, Wenting / Wang, Bin / Ding, Wei / Guo, Hao / Zhao, Hongyi / Meng, Jianzhou / Liu, Sihan / Lu, Yu / Liu, Yishuang et al. | 2021
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An optimized BRD4 inhibitor effectively eliminates NF-κB-driven triple-negative breast cancer cellsYang, Guan-Jun / Song, Ying-Qi / Wang, Wanhe / Han, Quan-Bin / Ma, Dik-Lung / Leung, Chung-Hang et al. | 2021
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Discovery of the PARP (poly ADP-ribose polymerase) inhibitor 2-(1-(4,4-difluorocyclohexyl)piperidin-4-yl)-1H-benzo[d]imidazole-4-carboxamide for the treatment of cancerTang, Lin / Wu, Weibin / Zhang, Cunlong / Shi, Zhichao / Chen, Dawei / Zhai, Xin / Jiang, Yuyang et al. | 2021
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Identification of new building blocks by fragment screening for discovering GyrB inhibitorsYu, Ying / Guo, Junsong / Cai, Zhengjun / Ju, Yingchen / Xu, Jun / Gu, Qiong / Zhou, Huihao et al. | 2021
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Synthesis, biological evaluation, and molecular docking analysis of novel linker-less benzamide based potent and selective HDAC3 inhibitorsRoutholla, Ganesh / Pulya, Sravani / Patel, Tarun / Abdul Amin, Sk. / Adhikari, Nilanjan / Biswas, Swati / Jha, Tarun / Ghosh, Balaram et al. | 2021
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Euryfuranyl compounds from edible species of cuttlefish as potential anti-inflammatory leads attenuating NF-κB signaling cascade in lipopolysaccharide-activated macrophagesChakraborty, Kajal / Krishnan, Soumya / Joy, Minju et al. | 2021
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Artematrovirenins A–P, guaiane-type sesquiterpenoids with cytotoxicities against two hepatoma cell lines from Artemisia atrovirensSu, Li-Hua / Ma, Yun-Bao / Geng, Chang-An / Li, Tian-Ze / Huang, Xiao-Yan / Hu, Jing / Xin Zhang / Tang, Shuang / Shen, Cheng / Gao, Zhen et al. | 2021
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Application of a marine luminescent Vibrio sp. B4L for biosynthesis of silver nanoparticles with unique characteristics, biochemical properties, antibacterial and antibiofilm activitiesZamanpour, Noushin / Mohammad Esmaeily, Ali / Mashreghi, Mansour / Shahnavaz, Bahar / Reza Sharifmoghadam, Mohammad / Kompany, Ahmad et al. | 2021
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UV-fluorescence probe for detection Ni2+ with colorimetric/spectral dual-mode analysis method and its practical applicationZhang, Yingying / Zhao, Yanliang / Song, Bo / Liu, Kunming / Gu, Jiamin / Yue, Yiying / Xiong, Ranhua / Huang, Chaobo et al. | 2021
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Anti-diabetic potential of Masclura tricuspidata leaves: Prenylated isoflavonoids with α-glucosidase inhibitory and anti-glycation activityJo, Yang Hee / Lee, Solip / Yeon, Sang Won / Turk, Ayman / Lee, Jae Hyuk / Hong, Seong-Min / Han, Yoo Kyong / Lee, Ki Yong / Hwang, Bang Yeon / Kim, Sun Yeou et al. | 2021
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Structure-activity relationship study of dihydroartemisinin C-10 hemiacetal derivatives as Toll-like receptor 4 antagonistsWang, Shuo / Wang, Hongshuang / Lin, Cong / Zhang, Tianshu / Gao, Jingwei / Wu, Siru / Wang, Yibo / Li, Hongyuan / Min, Weihong / Liu, Chunlei et al. | 2021
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Rational design-aided discovery of novel 1,2,4-oxadiazole derivatives as potential EGFR inhibitorsUnadkat, Vishal / Rohit, Shishir / Parikh, Paranjay / Sanna, Vinod / Singh, Sanjay et al. | 2021
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3-Alkenyl-2-oxindoles: Synthesis, antiproliferative and antiviral properties against SARS-CoV-2Girgis, Adel S. / Panda, Siva S. / Srour, Aladdin M. / Abdelnaser, Anwar / Nasr, Soad / Moatasim, Yassmin / Kutkat, Omnia / El Taweel, Ahmed / Kandeil, Ahmed / Mostafa, Ahmed et al. | 2021
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Editorial Board| 2021