Novel propargylamine-based inhibitors of cholinesterases and monoamine oxidases: Synthesis, biological evaluation and docking study (Englisch)
- Neue Suche nach: Krátký, Martin
- Neue Suche nach: Vu, Quynh Anh
- Neue Suche nach: Štěpánková, Šárka
- Neue Suche nach: Maruca, Annalisa
- Neue Suche nach: Silva, Tiago Barros
- Neue Suche nach: Ambrož, Martin
- Neue Suche nach: Pflégr, Václav
- Neue Suche nach: Rocca, Roberta
- Neue Suche nach: Svrčková, Katarína
- Neue Suche nach: Alcaro, Stefano
- Neue Suche nach: Borges, Fernanda
- Neue Suche nach: Vinšová, Jarmila
- Neue Suche nach: Krátký, Martin
- Neue Suche nach: Vu, Quynh Anh
- Neue Suche nach: Štěpánková, Šárka
- Neue Suche nach: Maruca, Annalisa
- Neue Suche nach: Silva, Tiago Barros
- Neue Suche nach: Ambrož, Martin
- Neue Suche nach: Pflégr, Václav
- Neue Suche nach: Rocca, Roberta
- Neue Suche nach: Svrčková, Katarína
- Neue Suche nach: Alcaro, Stefano
- Neue Suche nach: Borges, Fernanda
- Neue Suche nach: Vinšová, Jarmila
In:
Bioorganic Chemistry
;
116
;
2021
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ISSN:
- Aufsatz (Zeitschrift) / Elektronische Ressource
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Titel:Novel propargylamine-based inhibitors of cholinesterases and monoamine oxidases: Synthesis, biological evaluation and docking study
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Beteiligte:Krátký, Martin ( Autor:in ) / Vu, Quynh Anh ( Autor:in ) / Štěpánková, Šárka ( Autor:in ) / Maruca, Annalisa ( Autor:in ) / Silva, Tiago Barros ( Autor:in ) / Ambrož, Martin ( Autor:in ) / Pflégr, Václav ( Autor:in ) / Rocca, Roberta ( Autor:in ) / Svrčková, Katarína ( Autor:in ) / Alcaro, Stefano ( Autor:in )
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Erschienen in:Bioorganic Chemistry ; 116
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Verlag:
- Neue Suche nach: Elsevier Inc.
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Erscheinungsdatum:18.08.2021
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ISSN:
-
DOI:
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Medientyp:Aufsatz (Zeitschrift)
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Format:Elektronische Ressource
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Sprache:Englisch
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Schlagwörter:
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Datenquelle:
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Design and synthesis of curcumin nanostructures: Evaluation of solubility, stability, antibacterial and antioxidant activitiesOmidi, Sakineh / Rafiee, Zeinab / Kakanejadifard, Ali et al. | 2021
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Interactions of isoorientin and its Semi-synthetic analogs with human serum albuminWang, Wenliang / Gao, Denghui / Zheng, Qiancheng / Zhao, Xi / Na, Risong / Wan, Xinsheng / Li, Qing X. et al. | 2021
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Design, synthesis, and biological evaluation of cyano-substituted 2,4-diarylaminopyrimidines as potent JAK3 inhibitors for the treatment of B-cell lymphomaWu, Bin / Yang, Song / Deng, Tuo / Wang, Changyuan / Jin, Yue / Yu, Jiawen / Xu, Youjun / Chen, Lixue / Li, Yanxia / Ma, Xiaodong et al. | 2021
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Hydrazonoyl bromide precursors as DHFR inhibitors for the synthesis of bis-thiazolyl pyrazole derivatives; antimicrobial activities, antibiofilm, and drug combination studies against MRSAIbrahim, Seham A. / Fayed, Eman A. / Rizk, Hala F. / Desouky, Said E. / Ragab, Ahmed et al. | 2021
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Synthesis, in vitro anticancer activity and in silico studies of certain pyrazole-based derivatives as potential inhibitors of cyclin dependent kinases (CDKs)Mohammed, Esraa Z. / Mahmoud, Walaa R. / George, Riham F. / Hassan, Ghaneya S. / Omar, Farghaly A. / Georgey, Hanan H. et al. | 2021
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Synthesis and biological evaluation of NO-donor containing photosensitizers to induce ferroptosis of cancer cellsGuo, Xiuhan / Yu, Haoze / Shen, Wanjie / Cai, Rui / Li, Yueqing / Li, Guangzhe / Zhao, Weijie / Wang, Shisheng et al. | 2021
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Panaxadiol as a major metabolite of AD-1 can significantly inhibit the proliferation and migration of breast cancer cells: In vitro and in vivo studyXu, Lei / Zhang, Xiaoshu / Xiao, Shengnan / Li, Xiaofei / Jiang, Hua / Wang, Ziyi / Sun, Baoshan / Zhao, Yuqing et al. | 2021
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Screening out anti-inflammatory or anti-viral targets in Xuanfei Baidu Tang through a new technique of reverse finding targetWang, Zixuan / Zhang, Jumei / Zhan, Jiuyu / Gao, Hongwei et al. | 2021
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Hybrids of 4-hydroxy derivatives of goniothalamin and piplartine bearing a diester or a 1,2,3-triazole linker as antiproliferative agentsGrigolo, Thiago A. / Braga, Carolyne B. / Ornelas, Catia / Russowsky, Dennis / Ferreira-Silva, Guilherme A. / Ionta, Marisa / Pilli, Ronaldo A. et al. | 2021
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Synthesis and biological evaluation of zwitterionic half-sandwich Rhodium(III) and Ruthenium(II) organometallic complexesGuo, Lihua / Hu, Xueyan / Yang, Yanjing / An, Wenyu / Gao, Jie / Liu, Qin / Liu, Zhe et al. | 2021
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Design, synthesis, and evaluation of HIV-1 entry inhibitors based on broadly neutralizing antibody 447-52D and gp120 V3loop interactionsSenapathi, Jagadeesh / Bommakanti, Akhila / Vangara, Srinivas / Kondapi, Anand K. et al. | 2021
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Spectroscopic and Small-angle X-ray scattering analysis of binding between Copper(II) −1-allylimidazole complex, a potential anti-tumor agent, and bovine serum albuminGałczyńska, Katarzyna / Ciepluch, Karol / Kurdziel, Krystyna / Biehl, Ralf / Arabski, Michał et al. | 2021
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Synthesis, in vitro anticancer activity and in silico studies of certain isoxazole-based carboxamides, ureates, and hydrazones as potential inhibitors of VEGFR2Abou-Seri, Sahar M. / Eissa, Amal A.M. / Behery, Mohamed G.M. / Omar, Farghaly A. et al. | 2021
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Development of 2′-aminospiro [pyrano[3,2–c]quinoline]-3′-carbonitrile derivatives as non-ATP competitive Src kinase inhibitors that suppress breast cancer cell migration and proliferationRamadan, Mohamed / A.M.M. Elshaier, Yaseen / Aly, Ashraf A. / Abdel-Aziz, Mohamed / Fathy, Hazem M. / Brown, Alan B. / Pridgen, Jacey R. / Dalby, Kevin N. / Kaoud, Tamer S. et al. | 2021
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Synthesis of N-methylpyridine-chlorofuranformamide analogs as novel OPG up-regulators and inhibitors of RANKL-induced osteoclastogenesisLiu, Chao / Li, Yining / Sheng, Ren / Han, Xiaowan / Bao, Li / Wang, Chenyin / Wang, Weizhi / Jiang, Xinhai / Han, Jiangxue / Lei, Lijuan et al. | 2021
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Epidermal growth factor receptor inhibitors as potential anticancer agents: An update of recent progressSharma, Bharti / Singh, Vikram Jeet / Chawla, Pooja A. et al. | 2021
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The AMPA receptor biophysical gating properties and binding site: Focus on novel curcumin-based diazepines as non-competitive antagonistsQneibi, Mohammad / Hamed, Othman / Jaradat, Nidal / Hawash, Mohammed / Al-Kerm, Rana / Al-Kerm, Rola / Sobuh, Shorooq / Tarazi, Sama et al. | 2021
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Synthesis and antibacterial evaluation of (E)-1-(1H-indol-3-yl) ethanone O-benzyl oxime derivatives against MRSA and VRSA strainsAkunuri, Ravikumar / Veerareddy, Vaishnavi / Kaul, Grace / Akhir, Abdul / Unnissa, Tanveer / Parupalli, Ramulu / Madhavi, Y.V. / Chopra, Sidharth / Nanduri, Srinivas et al. | 2021
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A new class of cytotoxic agents targets tubulin and disrupts microtubule dynamicsAl-Hamashi, Ayad A. / Koranne, Radhika / Dlamini, Samkeliso / Alqahtani, Abdulateef / Karaj, Endri / Rashid, Maisha S. / Knoff, Joseph R. / Dunworth, Matthew / Pflum, Mary Kay H. / Casero, Robert A. Jr et al. | 2021
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Trimeric and dimeric Aspidosperma-type alkaloids from leaves of Tabernaemontana divaricata 'Dwaft'Chen, Jing / Yu, Yang / Wu, Jing / Bao, Mei-Fen / Kongkiatpaiboon, Sumet / Schinnerl, Johann / Cai, Xiang-Hai et al. | 2021
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Design and synthesis of novel pyridopyrimidine derivatives with anchoring non-coplanar aromatic extensions of EGFR inhibitory activityEissa, Amal A.M. / Aljamal, Kholoud F.M. / Ibrahim, Hany S. / Abdelrasheed Allam, Heba et al. | 2021
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Exploration of novel anti-angiogenic PEDF-derived peptides with improved activitives by inhibiting proliferation, suppressing migration, and inducing 67LR internalizationShi, Wei / Li, Jiuhui / Zhou, Jiaqi / Li, Yuanyuan / Lin, Haiyan / Qian, Hai / Fan, Wen et al. | 2021
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A novel peptidomimetic therapeutic for selective suppression of lung cancer stem cells over non-stem cancer cellsShukla, Satya Prakash / Raymond, Aaron / Rustagi, Vineeta / Kedika, Samanth R. / Tran, Olivia / Wang, Liye / Guo, Bin / Udugamasooriya, D. Gomika et al. | 2021
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Discovery of 3,4-dichloro-N-(1H-indol-5-yl)benzamide: A highly potent, selective, and competitive hMAO-B inhibitor with high BBB permeability profile and neuroprotective actionElkamhawy, Ahmed / Kim, Hyeon Jeong / Elsherbeny, Mohamed H. / Paik, Sora / Park, Jong-Hyun / Gotina, Lizaveta / Abdellattif, Magda H. / Gouda, Noha A. / Cho, Jungsook / Lee, Kyeong et al. | 2021
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Design, synthesis, and molecular docking study of some 2-((7-chloroquinolin-4-yl) amino) benzohydrazide Schiff bases as potential Eg5 inhibitory agentsKavalapure, Rohini S. / Alegaon, Shankar G. / Venkatasubramanian, U. / Priya, A. Soundarya / Ranade, Shriram D. / Khanal, Pukar / Mishra, Sanjay / Patil, Dhanashree / Salve, Preeti S. / Jalalpure, Sunil S. et al. | 2021
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Interest of novel N-alkylpyridinium-indolizine hybrids in the field of Alzheimer's disease: Synthesis, characterization and evaluation of antioxidant activity, cholinesterase inhibition, and amyloid fibrillation interferenceBaussanne, Isabelle / Firstova, Olga / Dediu, Andreea Botezatu / Larosa, Camille / Furdui, Bianca / Ghinea, Ioana Ottilia / Thomas, Aline / Chierici, Sabine / Dinica, Rodica / Demeunynck, Martine et al. | 2021