5'-Alkyl-benzothiadiazides: A New Subgroup of AMPA Receptor Modulators with Improved Affinity (Englisch)
- Neue Suche nach: Phillips, Dean
- Neue Suche nach: Phillips, Dean
- Neue Suche nach: Sonnenberg, Jennifer
- Neue Suche nach: Arai, Amy C.
- Neue Suche nach: Vaswani, Rishi
- Neue Suche nach: Krutzik, Peter O.
- Neue Suche nach: Kleisli, Thomas
- Neue Suche nach: Kessler, Markus
- Neue Suche nach: Granger, Richard
- Neue Suche nach: Lynch, Gary
- Neue Suche nach: Richard Chamberlin, A.
In:
Bioorganic & medicinal chemistry
;
10
, 5
; 1229-1248
;
2002
-
ISSN:
- Aufsatz (Zeitschrift) / Print
-
Titel:5'-Alkyl-benzothiadiazides: A New Subgroup of AMPA Receptor Modulators with Improved Affinity
-
Beteiligte:Phillips, Dean ( Autor:in ) / Sonnenberg, Jennifer / Arai, Amy C. / Vaswani, Rishi / Krutzik, Peter O. / Kleisli, Thomas / Kessler, Markus / Granger, Richard / Lynch, Gary / Richard Chamberlin, A.
-
Erschienen in:Bioorganic & medicinal chemistry ; 10, 5 ; 1229-1248
-
Verlag:
- Neue Suche nach: Elsevier
-
Erscheinungsort:Amsterdam [u.a.]
-
Erscheinungsdatum:2002
-
ISSN:
-
ZDBID:
-
Medientyp:Aufsatz (Zeitschrift)
-
Format:Print
-
Sprache:Englisch
- Neue Suche nach: 35.70 / 44.33 / 44.40
- Weitere Informationen zu Basisklassifikation
-
Schlagwörter:
-
Klassifikation:
-
Datenquelle:
Inhaltsverzeichnis – Band 10, Ausgabe 5
Zeige alle Jahrgänge und Ausgaben
Die Inhaltsverzeichnisse werden automatisch erzeugt und basieren auf den im Index des TIB-Portals verfügbaren Einzelnachweisen der enthaltenen Beiträge. Die Anzeige der Inhaltsverzeichnisse kann daher unvollständig oder lückenhaft sein.
- 1197
-
An Analysis of the Binding of Cocaine Analogues to the Monoamine Transporters Using Tensor Decomposition 3-D QSARAppell, Michael et al. | 2002
- 1207
-
Coupling of Isoprenoid Triflates with Organoboron Nucleophiles: Synthesis and Biological Evaluation of Geranylgeranyl Diphosphate AnaloguesMu, Yongqi et al. | 2002
- 1221
-
Acetamidoquinone and acetamidohydroxy derivatives as inhibitors for both dihydroxyacetamido epoxidase and dehydrogenaseWhiteley, Chris G. et al. | 2002
- 1229
-
5prime-Alkyl-benzothiadiazides: A New Subgroup of AMPA Receptor Modulators with Improved AffinityPhillips, D. / Sonnenberg, J. / Arai, A. C. / Vaswani, R. / Krutzik, P. O. / Kleisli, T. / Kessler, M. / Granger, R. / Lynch, G. / Richard Chamberlin, A. et al. | 2002
- 1229
-
5'-Alkyl-benzothiadiazides: A New Subgroup of AMPA Receptor Modulators with Improved AffinityPhillips, Dean et al. | 2002
- 1249
-
Polyene substrates with unusual methylation patterns to probe the active sites of three catalytic antibodiesKim, Geun Tae et al. | 2002
- 1263
-
Synthesis and Biological Properties of Amino Acid Amide Ligand-Based Pyridinioalkanoyl Thioesters as Anti-HIV AgentsSong, Yongsheng et al. | 2002
- 1275
-
A Convenient Synthesis and Hepatoprotective Activity of Imidazo(1,2-c)pyrimido(5,4-e)pyrimidine, Tetraazaacenaphthene and Tetraazaphenalene from Cyclic Ketene Aminals Through Tandem Addition-Cyclization ReactionsRam, Vishnu J. et al. | 2002
- 1281
-
Novel Irreversible Butyrylcholinesterase Inhibitors: 2-Chloro-1-(substituted-phenyl)ethylphosphonic AcidsZhang, Nanjing et al. | 2002
- 1291
-
Structure-Activity relationships among novel phenoxybenzamine-Related b-ChloroethylaminesGiardinà, Dario et al. | 2002
- 1305
-
Fatty Acid Esters of Juvenoid Alcohols as Insect Hormonogen Agents (Juvenogens)Wimmer, Zdenek et al. | 2002
- 1313
-
The 1.76 °A Resolution Crystal Structure of Glycogen Phosphorylase b Complexed with Glucose, and CP320626, a Potential Antidiabetic DrugOikonomakos, Nikos G. et al. | 2002
- 1321
-
A Novel Approach towards Studying Non-Genotoxic Enediynes as Potential Anticancer TherapeuticsHakimelahi, Gholam Hossein et al. | 2002
- 1329
-
Recognition of Bulged DNA by a Neocarzinostatin Product via an Induced Fit MechanismYang, Catherine F. et al. | 2002
- 1337
-
Substituted Indoloquinolines as New Antifungal AgentsAblordeppey, Seth Y. et al. | 2002
- 1347
-
Discovery of diaminobutane derivatives as Ca2+-permeable AMPA receptor antagonistsYoneda, Yoshiyuki et al. | 2002
- 1361
-
QSAR Studies on Antimalarial Substituted Phenyl Analogues and Their Nw-OxidesAgrawal, Vijay K. et al. | 2002
- 1361
-
QSAR Studies on Antimalarial Substituted Phenyl Analogues and Their N-OxidesAgrawal, V. K. / Sharma, R. / Khadikar, P. V. et al. | 2002
- 1367
-
3-D-QSAR Analysis of N-(3-Acyloxy-2-benzylpropyl)-Nprime-dihydroxytetrahydrobenzazepine and Tetrahydroisoquinoline and N-(3-Acyloxy-2-benzylpropyl)-Nprime-(4-hydroxy-3-methoxybenzyl) Thioureas Analogues as Potent Vanilloid Receptor LigandsKim, K. H. et al. | 2002
- 1367
-
3-D-QSAR Analysis of N-(3-Acyloxy-2-benzylpropyl)-N'-dihydroxytetrahydrobenzazepine and Tetrahydroisoquinoline and N-(3-Acyloxy-2-benzylpropyl)-N'-(4-hydroxy-3-methoxybenzyl) Thioureas Analogues as Potent Vanilloid Receptor LigandsKim, Ki H. et al. | 2002
- 1373
-
Molecular Orbital Calculation for the Model Compounds of Kainoid Amino Acids, Agonists of Excitatory Amino Acid Receptors. Does the Kainoid C4-Substituent Directly Interact with the Receptors?Hashimoto, Kimiko et al. | 2002
- 1381
-
Aryl Cyclopentadienyl Tricarbonyl Rhenium Complexes: Novel Ligands for the Estrogen Receptor with Potential Use as Estrogen RadiopharmaceuticalsMull, Eric S. et al. | 2002
- 1399
-
Synthesis and Biological Activity of 1-Phenylsulfonyl-4-Phenylsulfonylaminopyrrolidine Derivatives as Thromboxane A2 Receptor AntagonistsMarusawa, Hiroshi et al. | 2002
- 1417
-
Certification of the Critical Importance of l-3-(2-Naphthyl)alanine at Position 3 of a Specific CXCR4 Inhibitor, T140, Leads to an Exploratory Performance of Its Downsizing StudyTamamura, Hirokazu et al. | 2002
- 1427
-
Binding of 1-Benzopyran-4-one Derivatives to Aldose Reductase: A Free Energy Perturbation StudyRastelli, Giulio et al. | 2002
- 1437
-
Discovery of new inhibitors of aldose reductase from molecular docking and database screeningRastelli, Giulio et al. | 2002
- 1451
-
Synthesis and 31P NMR characterization of new low toxic highly sensitive pH probes designed for in vivo acidic pH studiesMartel, Sophie et al. | 2002
- 1459
-
Novel anthracycline oligosaccharides: influence of chemical modifications of the carbohydrate moiety on biological activityCipollone, A. et al. | 2002
- 1471
-
Resolution of (RS)-Proglumide using Lipase from Candida cylindraceaeMuralidhar, R.V. et al. | 2002
- 1477
-
Experimental and Calculated Shift in pKa upon Binding of Phosphotyrosine Peptide to the SH2 Domain of p56lckde Mol, Nico J. et al. | 2002
- 1483
-
QSAR of HIV-1 integrase inhibitors by genetic function approximation methodMakhija, Mahindra T. et al. | 2002
- 1499
-
Synthesis and biological evaluation of novel thioapio dideoxynucleosidesMoon, Hyung Ryong et al. | 2002
- 1509
-
The Discovery of YM-60828: A Potent, Selective and Orally-Bioavailable Factor Xa InhibitorHirayama, Fukushi et al. | 2002
- 1525
-
I2-Imidazoline Binding Site Affinity of a Structurally Different Type of LigandsDardonville, Christophe et al. | 2002
- 1535
-
Orally Active Cephalosporins. Part 4: Synthesis, Structure-Activity Relationships and Oral Absorption of Novel 3-(4-Pyrazolylmethylthio)cephalosporins with Various C-7 Side ChainsYamamoto, Hirofumi et al. | 2002
- 1547
-
Absolute Stereostructure of Potent a-Glucosidase Inhibitor, Salacinol, with Unique Thiosugar Sulfonium Sulfate Inner Salt Structure from Salacia reticulataYoshikawa, Masayuki et al. | 2002
- 1555
-
Novel Non-Steroidal-Non-Anilide Type Androgen Antagonists with an Isoxazolone MoietyIshioka, Toshiyasu et al. | 2002
- 1567
-
Synthesis of Potential Thrombin Inhibitors. Incorporation of Tartaric Acid Templates as P2 Proline MimeticsDahlgren, Anders et al. | 2002
- 1581
-
Antioxidant activity of synthetic cytokinin analogues: 6-alkynyl- and 6-alkenylpurines as novel 15-Lipoxygenase inhibitorsBråthe, Anders et al. | 2002
- 1587
-
Mapping of Possible Binding Sequences of Two Beta-Sheet Breaker Peptides on Beta Amyloid Peptide of Alzheimer's DiseaseHetényi, Csaba et al. | 2002
- 1595
-
Structure-Activity Relationships of 1b-Methyl-2-(5-phenylpyrrolidin-3-ylthio)carbapenemsSato, Hiroki et al. | 2002
- 1611
-
Benzoyl and cinnamoyl nitrogen mustard derivatives of benzoheterocyclic analogues of the tallimustine: synthesis and antitumour activityBaraldi, Pier Giovanni et al. | 2002
- 1619
-
Powerful antioxidative agents based on garcinoic acid from Garcinia kolaTerashima, Kenji et al. | 2002
- 1627
-
9-Carboxymethyl-5H,10H-imidazo(1,2-a)indeno(1,2-e)pyrazin-4-one-2-c- arbocylic Acid (RPR117824): Selective Anticonvulsive and Neuroprotective AMPA AntagonistMignani, Serge et al. | 2002
- 1639
-
Novel Tn antigen-containing neoglycopeptides: synthesis and evaluation as anti tumor vaccinesCipolla, Laura et al. | 2002
-
Graphical Abstracts| 2002