(+--)-3-Amino-6-carboxamido-1,2,3,4-tetrahydrocarbazole: A Conformationally Restricted Analogue of 5-Carboxamidotryptamine with Selectivity for the Serotonin 5-HT1D Receptor (Englisch)
- Neue Suche nach: King, Frank D.
- Neue Suche nach: King, Frank D.
- Neue Suche nach: Brown, Anthony M.
- Neue Suche nach: Gaster, Laramie M.
- Neue Suche nach: Kaumann, Alberto J.
- Neue Suche nach: Medhurst, Andrew D.
- Neue Suche nach: Parker, Stephen G.
- Neue Suche nach: Parsons, Andrew A.
- Neue Suche nach: Patch, Tracey L.
- Neue Suche nach: Raval, Pravin
In:
Journal of medicinal chemistry
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36
, 21
; 3218
;
1993
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ISSN:
- Aufsatz (Zeitschrift) / Print
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Titel:(+--)-3-Amino-6-carboxamido-1,2,3,4-tetrahydrocarbazole: A Conformationally Restricted Analogue of 5-Carboxamidotryptamine with Selectivity for the Serotonin 5-HT1D Receptor
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Beteiligte:
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Erschienen in:Journal of medicinal chemistry ; 36, 21 ; 3218
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Verlag:
- Neue Suche nach: American Chemical Society
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Erscheinungsort:Easton, Pa.
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Erscheinungsdatum:1993
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ISSN:
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ZDBID:
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Medientyp:Aufsatz (Zeitschrift)
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Format:Print
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Sprache:Englisch
- Neue Suche nach: 770/4230
- Neue Suche nach: 44.42 / 44.42
- Weitere Informationen zu Basisklassifikation
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Datenquelle:
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Die Inhaltsverzeichnisse werden automatisch erzeugt und basieren auf den im Index des TIB-Portals verfügbaren Einzelnachweisen der enthaltenen Beiträge. Die Anzeige der Inhaltsverzeichnisse kann daher unvollständig oder lückenhaft sein.
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Pyrrolo[1,2-a]benzimidazole-based aziridinyl quinones. A new class of DNA cleaving agent exhibiting G and A base specificitySkibo, Edward B. / Schulz, William G. et al. | 1993
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Pyrrolo[1,2-]benzimidazole-Based Aziridinyl Quinones. A New Class of DNA Cleaving Agent Exhibiting G and A Base SpecificitySkibo, E. B. / Schulz, W. G. et al. | 1993
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Solution conformation of the antitumor drug streptonigrinHarding, Margaret M. / Long, Georgina V. / Brown, Christopher L. et al. | 1993
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Synthesis of A-Ring Fluorinated Derivatives of (17a,20E-Z)-(125I)Iodovinylestradiols: Effect on Receptor Binding and Receptor-Mediated Target Tissue Uptake1Ali, Hasrat et al. | 1993
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Synthesis of A-Ring Fluorinated Derivatives of (17,20E/Z)-[^1^2^5I]Iodovinylestradiols: Effect on Receptor Binding and Receptor-Mediated Target Tissue Uptake^1Ali, H. / Rousseau, J. / Van Lier, J. E. et al. | 1993
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Conformationally restrained analogs of sympathomimetic catecholamines. Synthesis, conformational analysis and adrenergic activity of isochroman derivativesMacchia, Bruno / Balsamo, Aldo / Breschi, Maria Cristina / Chiellini, Grazia / Lapucci, Annalina / Macchia, Marco / Manera, Clementina / Martinelli, Adriano / Martini, Claudia et al. | 1993
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Catalytic functionalization of polymers: a novel approach to site-specific delivery of misoprostol to the stomachTremont, Samuel J. / Collins, Paul W. / Perkins, William E. / Fenton, Rick L. / Forster, Denis / McGrath, Martin P. / Wagner, Grace M. / Gasiecki, Alan F. / Bianchi, Robert G. et al. | 1993
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Structural modification of 5-aryl-2,3-dihydroimidazo[2,1-a]isoquinoline platelet activating factor receptor antagonistsHoulihan, William J. / Cheon, Seung H. / Parrino, Vincent A. / Handley, Dean A. / Larson, Douglas A. et al. | 1993
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Structural Modification of 5-Aryl-2,3-dihydroimidazo[2,1-]isoquinoline Platelet Activating Factor Receptor AntagonistsHoulihan, W. J. / Cheon, S. H. / Parrino, V. A. / Handley, D. A. et al. | 1993
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2,4-Diaminothieno(2,3-d)pyrimidine Analogues of Trimetrexate and Piritrexim as Potential Inhibitors of Pneumocystis carinii and Toxoplasma gondii Dihydrofolate ReductaseRosowsky, Andre et al. | 1993
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A series of penicillin-derived C2-symmetric inhibitors of HIV-1 proteinase: structural and modeling studiesWonacott, Alan / Cooke, Robert / Hayes, Fiona R. / Hann, Michael M. / Jhoti, Harren / McMeekin, Peter / Mistry, Anil / Murray-Rust, Peter / Singh, Onkar M. P. / Weir, Malcolm P. et al. | 1993
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A series of penicillin-derived C2-symmetric inhibitors of HIV-1 proteinase: synthesis, mode of interaction, and structure-activity relationshipsHumber, David C. / Bamford, Mark J. / Bethell, Richard C. / Cammack, Nicholas / Cobley, Kevin / Evans, Derek N. / Gray, Norman M. / Hann, Michael M. / Orr, David C. et al. | 1993
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- 3137
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Azulenic retinoids: novel nonbenzenoid aromatic retinoids with anticancer activityAsato, Alfred E. / Peng, Ao / Hossain, Mohammad Z. / Mirzadegan, Taraneh / Bertram, John S. et al. | 1993
- 3148
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Synthesis and antibacterial activity of a new series of tetracyclic pyridone carboxylic acids. 2Jinbo, Yoshikazu / Taguchi, Masahiro / Inoue, Yoshimasa / Kondo, Hirosato / Miyasaka, Tomohiro / Tsujishita, Hideki / Sakamoto, Fumio / Tsukamoto, Goro et al. | 1993
- 3154
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14-[(p-Nitrocinnamoyl)amino]morphinones, 14-[(p-Nitrocinnamoyl)amino]-7,8-dihydromorphinones, and Their Codeinone Analogues: Synthesis and Receptor ActivitySebastian, A. / Bidlack, J. M. / Jiang, Q. / Deecher, D. et al. | 1993
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14.beta.-[(p-Nitrocinnamoyl)amino]morphinones, 14.beta.-[(p-nitrocinnamoyl)amino]-7,8-dihydromorphinones, and their codeinone analogs: synthesis and receptor activitySebastian, Alice / Bidlack, Jean M. / Jiang, Qi / Deecher, Darlene / Teitler, Milton / Glick, Stanley D. / Archer, Sydney et al. | 1993
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14b-((p-Nitrocinnamoyl)amino)morphinones, 14b-((p-Nitrocinnamoyl)amino)-7,8-dihydromorphinones, and Their Codeinone Analogues: Synthesis and Receptor ActivitySebastian, Alice et al. | 1993
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Synthesis of (R,S)-trans-8-hydroxy-2-[N-n-propyl-N-(3'-iodo-2'-propenyl)amino]tetralin (trans 8-OH-PIPAT): a new 5-HT1A receptor ligandZhuang, Zhi Ping / Kung, Mei Ping / Kung, Hank F. et al. | 1993
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The interaction of ammonium, sulfonium, and sulfide analogs of metoclopramide with the dopamine D2 receptorHarrold, Marc W. / Sriburi, Anong / Matsumoto, Kazuhisa / Miller, Duane D. / Farooqui, Tahira / Uretsky, Norman et al. | 1993
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The Interaction of Ammonium, Sulfonium, and Sulfide Analogues of Metoclopramide with the Dopamine D2 ReceptorHarrold, Marc W. et al. | 1993
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Voronoi modeling: the binding of triazines and pyrimidines to L. casei dihydrofolate reductaseBradley, Mary P. / Crippen, Gordon M. et al. | 1993
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Efficient inhibition of human leukocyte elastase and cathepsin G by saccharin derivativesGroutas, William C. / Houser-Archield, Nadene / Chong, Lee S. / Venkataraman, Radhika / Epp, Jeffrey B. / Huang, He / McClenahan, Jerald J. et al. | 1993
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TIPP(p): A Highly Potent and Stable Pseudopeptide d Opioid Receptor Antagonist with Extraordinary d SelectivitySchiller, Peter W. et al. | 1993
- 3182
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TIPP[psi]: A Highly Potent and Stable Pseudopeptide Opioid Receptor Antagonist with Extraordinary SelectivitySchiller, P. W. / Weltrowska, G. / Nguyen, T. M.-D. / Wilkes, B. C. et al. | 1993
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TIPP[.psi.]: a highly potent and stable pseudopeptide .delta. opioid receptor antagonist with extraordinary .delta. selectivitySchiller, Peter W. / Weltrowska, Grazyna / Nguyen, Thi M. D. / Wilkes, Brian C. / Chung, Nga N. / Lemieux, Carole et al. | 1993
- 3188
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Substituted 3-phenylpiperidines: new centrally acting dopamine autoreceptor antagonistsSonesson, Clas / Waters, Nicholas / Svensson, Kjell / Carlsson, Arvid / Smith, Martin W. / Piercey, Montford F. / Meier, Eddi / Wikstroem, Haakan et al. | 1993
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Synthesis, in vitro binding profile, and autoradiographic analysis of [3H]-cis-3-[(2-methoxybenzyl)amino]-2-phenylpiperidine, a highly potent and selective nonpeptide substance P receptor antagonist radioligandRosen, Terry / Seeger, Thomas F. / McLean, Stafford / Desai, Manoj C. / Guarino, Karen J. / Bryce, Dianne / Pratt, Kara / Heym, James / Chalabi, Philip M. et al. | 1993
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Troeger's base. An alternate synthesis and a structural analog with thromboxane A2 synthetase inhibitory activityJohnson, Roy A. / Gorman, Robert R. / Wnuk, Richard J. / Crittenden, Norman J. / Aiken, James W. et al. | 1993
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Tröger's Base. An Alternate Synthesis and a Structural Analog with Thromboxane A2 Synthetase Inhibitory ActivityJohnson, Roy A. et al. | 1993
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A potent, orally active, balanced affinity angiotensin II AT1 antagonist and AT2 binding inhibitorde Laszlo, Stephen E. / Quagliato, Carol S. / Greenlee, William J. / Patchett, Arthur A. / Chang, Raymond S. L. / Lotti, Victor J. / Chen, Tsing Bau / Scheck, Stacey A. / Faust, Kristi A. et al. | 1993
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3-(Alkylamino)-4H-pyrido[4,3-e]1,2,4-thiadiazine 1,1-dioxides as powerful inhibitors of insulin release from rat pancreatic B-cells: a new class of potassium channel openers?Pirotte, Bernard / de Tullio, Pascal / Lebrun, Philippe / Antoine, Marie Helene / Fontaine, Jeanine / Masereel, Bernard / Schynts, Marc / Dupont, Leon / Herchuelz, Andre / Delarge, Jacques et al. | 1993
- 3214
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Book Reviews| 1993
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Medicinal Chemistry for the 21st Century. A 'Chemistry for the 21st Century' MonographMewshaw, Richard E. et al. | 1993
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Optical Resolution Procedures for Chemical Compounds. Volume 4. Compounds Containing a Sulfur or Selenium Stereocenter. Parts I and IINewman, Paul et al. | 1993
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Microbial Reagents in Organic SynthesisLevy, Mark et al. | 1993
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Biotransformations. Volume 5. A Survey of the Biotransformations of Drugs and Chemicals in AnimalsStaff et al. | 1993
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Advances in Neurology. Volume 60. Parkinson's Disease. From Basic Research to TreatmentStaff et al. | 1993
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Heme Oxygenase: Clinical Applications and FunctionsMaines, Mahin D. et al. | 1993
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Annual Review of Neuroscience. Volume 16Ferkany, John Wm et al. | 1993
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Synthetic Fluorine ChemistryKirk, Kenneth L. et al. | 1993
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Synthesis and Biological Activity of N^5-(p-Sulfophenyl)alkyl and N^6-Sulfoalkyl Derivatives and Adenosine: Water-Soluble and Peripherally Selective Adenosine AgonistsJacobson, K. A. / Nikodijevic, O. / Ji, X.-D. / Berkich, D. A. et al. | 1993
- 3218
-
Synthesis and biological activity of N6-(p-sulfophenyl)alkyl and N6-sulfoalkyl derivatives of adenosine: water-soluble and peripherally selective adenosine agonists. [Erratum to document cited in CA117(23):234413y]Jacobson, Kenneth A. / Nikodijevic, Olga / Ji, Xiao Duo / Berkich, Deborah A. / Eveleth, David / Dean, Reginald L. / Hiramatsu, Kenichiro / Kassell, Neal F. / Van Galen, Philip J. M. et al. | 1993
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(+--)-3-Amino-6-carboxamido-1,2,3,4-tetrahydrocarbazole: A Conformationally Restricted Analogue of 5-Carboxamidotryptamine with Selectivity for the Serotonin 5-HT1D ReceptorKing, Frank D. et al. | 1993
- 3218
-
(.+-.)-3-Amino-6-carboxamido-1,2,3,4-tetrahydrocarbazole: A conformationally restricted analog of 5-carboxamidotryptamine with selectivity for the serotonin 5-HT1D receptor. [Erratum to document cited in CA119(11):117079z]King, Frank D. / Brown, Anthony M. / Gaster, Laramie M. / Kaumann, Alberto J. / Medhurst, Andrew D. / Parker, Stephen G. / Parsons, Andrew A. / Patch, Tracey L. / Raval, Pravin et al. | 1993
- 3218
-
Synthesis and Biological Activity of N8- (p-Sulfophenyl)alkyl and N6-Sulfoalkyl Derivatives and Adenosine: Water-Soluble and Peripherally Selective Adenosine AgonistsJacobson, Kenneth A. et al. | 1993
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Masthead| 1993