The discovery of GSK221149A: A potent and selective oxytocin antagonist (Englisch)
- Neue Suche nach: Liddle, John
- Neue Suche nach: Liddle, John
- Neue Suche nach: Allen, Michael J.
- Neue Suche nach: Borthwick, Alan D.
- Neue Suche nach: Brooks, David P.
- Neue Suche nach: Davies, David E.
- Neue Suche nach: Edwards, Richard M.
- Neue Suche nach: Exall, Anne M.
- Neue Suche nach: Hamlett, Chris
- Neue Suche nach: Irving, Wendy R.
- Neue Suche nach: Mason, Andrew M.
- Neue Suche nach: Mccafferty, Gerald P.
- Neue Suche nach: Nerozzi, Fabrizio
- Neue Suche nach: Peace, Simon
- Neue Suche nach: Philp, Joanne
- Neue Suche nach: Pollard, Derek
- Neue Suche nach: Pullen, Mark A.
- Neue Suche nach: Shabbir, Shaila S.
- Neue Suche nach: Sollis, Steve L.
- Neue Suche nach: Westfall, Timothy D.
In:
Bioorganic & medicinal chemistry letters
;
18
, 1
; 90-94
;
2008
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ISSN:
- Aufsatz (Zeitschrift) / Print
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Titel:The discovery of GSK221149A: A potent and selective oxytocin antagonist
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Beteiligte:Liddle, John ( Autor:in ) / Allen, Michael J. / Borthwick, Alan D. / Brooks, David P. / Davies, David E. / Edwards, Richard M. / Exall, Anne M. / Hamlett, Chris / Irving, Wendy R. / Mason, Andrew M.
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Erschienen in:Bioorganic & medicinal chemistry letters ; 18, 1 ; 90-94
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Verlag:
- Neue Suche nach: Elsevier
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Erscheinungsort:Amsterdam [u.a.]
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Erscheinungsdatum:2008
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ISSN:
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ZDBID:
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Medientyp:Aufsatz (Zeitschrift)
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Format:Print
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Sprache:Englisch
- Neue Suche nach: 35.70 / 44.33 / 44.42
- Weitere Informationen zu Basisklassifikation
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Schlagwörter:
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Klassifikation:
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Datenquelle:
Inhaltsverzeichnis – Band 18, Ausgabe 1
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Sulfonamide derivatives of bridgehead substituted bicyclo[4.2.1]nonanes as γ-secretase inhibitorsSparey, Tim / Clarke, Earl / Hannam, Joanne / Harrison, Timothy / Madin, Andrew / Shearman, Mark / Sohal, Bindi et al. | 2007
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Sulfonamide derivatives of bridgehead substituted bicyclo[4.2.1]nonanes as g-secretase inhibitorsSparey, T. / Clarke, E. / Hannam, J. / Harrison, T. / Madin, A. / Shearman, M. / Sohal, B. et al. | 2008
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Identification of novel inhibitors of bacterial surface enzyme Staphylococcus aureus Sortase AChenna, Bala Chandra / Shinkre, Bidhan A. / King, Jason R. / Lucius, Aaron L. / Narayana, Sthanam V.L. / Velu, Sadanandan E. et al. | 2007
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Identification of aminopyrazolopyridine ureas as potent VEGFR/PDGFR multitargeted kinase inhibitorsDai, Yujia / Hartandi, Kresna / Soni, Niru B. / Pease, Lori J. / Reuter, David R. / Olson, Amanda M. / Osterling, Donald J. / Doktor, Stella Z. / Albert, Daniel H. / Bouska, Jennifer J. et al. | 2007
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Design, synthesis, and studies of small molecule STAT3 inhibitorsBhasin, Deepak / Cisek, Katryna / Pandharkar, Trupti / Regan, Nicholas / Li, Chenglong / Pandit, Bulbul / Lin, Jiayuh / Li, Pui-Kai et al. | 2007
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Synthesis and antiplasmodial activity of new 4-aryl-2-trichloromethylquinazolinesVerhaeghe, Pierre / Azas, Nadine / Gasquet, Monique / Hutter, Sébastien / Ducros, Christophe / Laget, Michèle / Rault, Sylvain / Rathelot, Pascal / Vanelle, Patrice et al. | 2007
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Enantioselective actions of 4-amino-3-hydroxybutanoic acid and (3-amino-2-hydroxypropyl)methylphosphinic acid at recombinant GABAC receptorsHinton, Tina / Chebib, Mary / Johnston, Graham A.R. et al. | 2007
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Syntheses and in vitro evaluation of arylsulfone-based MMP inhibitors with heterocycle-derived zinc-binding groups (ZBGs)Zhang, Yue-Mei / Fan, Xiaodong / Yang, Shyh-Ming / Scannevin, Robert H. / Burke, Sharon L. / Rhodes, Kenneth J. / Jackson, Paul F. et al. | 2007
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1-Hydroxy-2-pyridinone-based MMP inhibitors: Synthesis and biological evaluation for the treatment of ischemic strokeZhang, Yue-Mei / Fan, Xiaodong / Chakaravarty, Devraj / Xiang, Bangping / Scannevin, Robert H. / Huang, Zhihong / Ma, Jianya / Burke, Sharon L. / Karnachi, Prabha / Rhodes, Kenneth J. et al. | 2007
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Potent pyrrolidine- and piperidine-based BACE-1 inhibitorsIserloh, U. / Wu, Y. / Cumming, J.N. / Pan, J. / Wang, L.Y. / Stamford, A.W. / Kennedy, M.E. / Kuvelkar, R. / Chen, X. / Parker, E.M. et al. | 2007
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Discovery of an orally efficaceous 4-phenoxypyrrolidine-based BACE-1 inhibitorIserloh, U. / Pan, J. / Stamford, A.W. / Kennedy, M.E. / Zhang, Q. / Zhang, L. / Parker, E.M. / McHugh, N.A. / Favreau, L. / Strickland, C. et al. | 2007
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Multi-target-directed coumarin derivatives: hAChE and BACE1 inhibitors as potential anti-Alzheimer compoundsPiazzi, Lorna / Cavalli, Andrea / Colizzi, Francesco / Belluti, Federica / Bartolini, Manuela / Mancini, Francesca / Recanatini, Maurizio / Andrisano, Vincenza / Rampa, Angela et al. | 2007
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Substrate specificity and screening of the integral membrane protease PlaAgarkov, Anton / Chauhan, Sadhana / Lory, Pedro J. / Gilbertson, Scott R. / Motin, Vladimir L. et al. | 2007
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Synthesis, characterization and evaluation of benzimidazole derivative and its precursors as inhibitors of MDA-MB-231 human breast cancer cell proliferationThimmegowda, N.R. / Nanjunda Swamy, S. / Ananda Kumar, C.S. / Sunil Kumar, Y.C. / Chandrappa, S. / Yip, George W. / Rangappa, K.S. et al. | 2007
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Eco-friendly and efficient one-pot synthesis of alkyl- or aryl-14H-dibenzo[a,j]xanthenes in waterDabiri, Minoo / Baghbanzadeh, Mostafa / Nikcheh, Maryam Shakouri / Arzroomchilar, Elham et al. | 2007
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Instructions to contributors| 2007
- IFC
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Editorial board| 2007