(−)-Cercosporamide derivatives as novel antihyperglycemic agents (Englisch)
- Neue Suche nach: Furukawa, Akihiro
- Neue Suche nach: Furukawa, Akihiro
- Neue Suche nach: Arita, Tsuyoshi
- Neue Suche nach: Satoh, Susumu
- Neue Suche nach: Araki, Kazushi
- Neue Suche nach: Kuroha, Masanori
- Neue Suche nach: Ohsumi, Jun
In:
Bioorganic & medicinal chemistry letters
;
19
, 3
; 724-726
;
2009
-
ISSN:
- Aufsatz (Zeitschrift) / Print
-
Titel:(−)-Cercosporamide derivatives as novel antihyperglycemic agents
-
Beteiligte:Furukawa, Akihiro ( Autor:in ) / Arita, Tsuyoshi / Satoh, Susumu / Araki, Kazushi / Kuroha, Masanori / Ohsumi, Jun
-
Erschienen in:Bioorganic & medicinal chemistry letters ; 19, 3 ; 724-726
-
Verlag:
- Neue Suche nach: Elsevier
-
Erscheinungsort:Amsterdam [u.a.]
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Erscheinungsdatum:2009
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ISSN:
-
ZDBID:
-
Medientyp:Aufsatz (Zeitschrift)
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Format:Print
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Sprache:Englisch
- Neue Suche nach: 35.70 / 44.33 / 44.42
- Weitere Informationen zu Basisklassifikation
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Schlagwörter:
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Klassifikation:
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Datenquelle:
Inhaltsverzeichnis – Band 19, Ausgabe 3
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2-(6-Phenyl-1H-indazol-3-yl)-1H-benzo[d]imidazoles: Design and synthesis of a potent and isoform selective PKC-z inhibitorTrujillo, J. I. / Kiefer, J. R. / Huang, W. / Thorarensen, A. / Xing, L. / Caspers, N. L. / Day, J. E. / Mathis, K. J. / Kretzmer, K. K. / Reitz, B. A. et al. | 2009
- 912
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2-Aminoimidazoles inhibitors of TGF-β receptor 1Bonafoux, Dominique / Chuaqui, Claudio / Boriack-Sjodin, P. Ann / Fitch, Chris / Hankins, Gretchen / Josiah, Serene / Black, Cheryl / Hetu, Gregg / Ling, Leona / Lee, Wen-Cherng et al. | 2008
- 912
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2-Aminoimidazoles inhibitors of TGF-b receptor 1Bonafoux, D. / Chuaqui, C. / Boriack-Sjodin, P. A. / Fitch, C. / Hankins, G. / Josiah, S. / Black, C. / Hetu, G. / Ling, L. / Lee, W. C. et al. | 2009
- 917
-
Synthesis and biological evaluation of phloridzin analogs as human concentrative nucleoside transporter 3 (hCNT3) inhibitorsGupte, Amol / Buolamwini, John K. et al. | 2008
- 922
-
Stereo-controlled synthesis of novel photoreactive γ-secretase inhibitorsYang, Guangli / Yin, Ye Ingrid / Chun, Jiong / Shelton, Christopher C. / Ouerfelli, Ouathek / Li, Yue-Ming et al. | 2008
- 922
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Stereo-controlled synthesis of novel photoreactive g-secretase inhibitorsYang, G. / Yin, Y. I. / Chun, J. / Shelton, C. C. / Ouerfelli, O. / Li, Y. M. et al. | 2009
- 926
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(S)-N-(5-Chlorothiophene-2-sulfonyl)-β,β-diethylalaninol a Notch-1-sparing γ-secretase inhibitorCole, Derek C. / Stock, Joseph R. / Kreft, Anthony F. / Antane, Madelene / Aschmies, Suzan H. / Atchison, Kevin P. / Casebier, David S. / Comery, Thomas A. / Diamantidis, George / Ellingboe, John W. et al. | 2008
- 926
-
(S)-N-(5-Chlorothiophene-2-sulfonyl)-b,b-diethylalaninol a Notch-1-sparing g-secretase inhibitorCole, D. C. / Stock, J. R. / Kreft, A. F. / Antane, M. / Aschmies, S. H. / Atchison, K. P. / Casebier, D. S. / Comery, T. A. / Diamantidis, G. / Ellingboe, J. W. et al. | 2009
- 930
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Potent and selective inhibitors of Helicobacter pylori glutamate racemase (MurI): Pyridodiazepine aminesGeng, Bolin / Basarab, Gregory / Comita-Prevoir, Janelle / Gowravaram, Madhusudhan / Hill, Pamela / Kiely, Andrew / Loch, James / MacPherson, Lawrence / Morningstar, Marshall / Mullen, George et al. | 2008
- 937
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In vitro anti-inflammatory activity of lignans isolated from Magnolia fargesiiKim, Jae Yeon / Lim, Hyo Jin / Lee, Da Yeon / Kim, Ji Sun / Kim, Do Hee / Lee, Hwa Jin / Kim, Hee Doo / Jeon, Raok / Ryu, Jae-Ha et al. | 2008
- 941
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3-Aminoxypropionate-based linker system for cyclization activation in prodrug designGe, Yiyu / Wu, Xinghua / Zhang, Dazhi / Hu, Longqin et al. | 2008
- 945
-
Synthesis and antimicrobial activities of halogenated bis(hydroxyphenyl)methanesOh, Ki-Bong / Lee, Ji Hye / Lee, Jong Wook / Yoon, Kyung-Mi / Chung, Soon-Chun / Jeon, Heung Bae / Shin, Jongheon / Lee, Hyi-Seung et al. | 2008
- 949
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Synthesis of spiro[chroman-2,4′-piperidin]-4-one derivatives as acetyl-CoA carboxylase inhibitorsShinde, Pundlik / Srivastava, Sanjay K. / Odedara, Rajendra / Tuli, Davinder / Munshi, Siralee / Patel, Jitendra / Zambad, Shitalkumar P. / Sonawane, Rajesh / Gupta, Ramesh C. / Chauthaiwale, Vijay et al. | 2008
- 949
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Synthesis of spiro[chroman-2,4prime-piperidin]-4-one derivatives as acetyl-CoA carboxylase inhibitorsShinde, P. / Srivastava, S. K. / Odedara, R. / Tuli, D. / Munshi, S. / Patel, J. / Zambad, S. P. / Sonawane, R. / Gupta, R. C. / Chauthaiwale, V. et al. | 2009
- 954
-
Synthesis and structure–activity relationships of novel, substituted 5,6-dihydrodibenzo[a,g]quinolizinium P2X7 antagonistsLee, Ga Eun / Lee, Ho-Sung / Lee, So Deok / Kim, Jung-Ho / Kim, Won-Ki / Kim, Yong-Chul et al. | 2008
- 959
-
HY251, a novel cell cycle inhibitor isolated from Aralia continentalis, induces G1 phase arrest via p53-dependent pathway in HeLa cellsOh, Ha Lim / Lim, Haeyoung / Cho, Youl-Hee / Koh, Hyun Chul / Kim, Hojung / Lim, Yoongho / Lee, Chul-Hoon et al. | 2008
- 962
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Positive allosteric modulators of the metabotropic glutamate receptor subtype 4 (mGluR4). Part II: Challenges in hit-to-leadWilliams, Richard / Niswender, Colleen M. / Luo, Qingwei / Le, Uyen / Conn, P. Jeffrey / Lindsley, Craig W. et al. | 2008
- 967
-
Potent and selective adenosine A2A receptor antagonists: 1,2,4-Triazolo[1,5-c]pyrimidinesNeustadt, Bernard R. / Liu, Hong / Hao, Jinsong / Greenlee, William J. / Stamford, Andrew W. / Foster, Carolyn / Arik, Leyla / Lachowicz, Jean / Zhang, Hongtao / Bertorelli, Rosalia et al. | 2008
- 972
-
Type II NADH dehydrogenase of the respiratory chain of Plasmodium falciparum and its inhibitorsDong, Carolyn K. / Patel, Vishal / Yang, Jimmy C. / Dvorin, Jeffrey D. / Duraisingh, Manoj T. / Clardy, Jon / Wirth, Dyann F. et al. | 2008
- 976
-
Anthranilimide-based glycogen phosphorylase inhibitors for the treatment of type 2 diabetes: 1. Identification of 1-amino-1-cycloalkyl carboxylic acid headgroupsSparks, Steven M. / Banker, Pierette / Bickett, David M. / Carter, H. Luke / Clancy, Daphne C. / Dickerson, Scott H. / Dwornik, Kate A. / Garrido, Dulce M. / Golden, Pamela L. / Nolte, Robert T. et al. | 2008
- 981
-
Anthranilimide-based glycogen phosphorylase inhibitors for the treatment of Type 2 diabetes: 2. Optimization of serine and threonine ether amino acid residuesSparks, Steven M. / Banker, Pierette / Bickett, David M. / Clancy, Daphne C. / Dickerson, Scott H. / Garrido, Dulce M. / Golden, Pamela L. / Peat, Andrew J. / Sheckler, Lauren R. / Tavares, Francis X. et al. | 2008
- 986
-
Synthesis, in vitro antitrypanosomal and antibacterial activity of phenoxy, phenylthio or benzyloxy substituted quinolonesMa, Xiang / Zhou, Weicheng / Brun, Reto et al. | 2008
- 990
-
Discovery and optimization of highly ligand-efficient oxytocin receptor antagonists using structure-based drug designBellenie, Benjamin R. / Barton, Nicholas P. / Emmons, Amanda J. / Heer, Jag P. / Salvagno, Cristian et al. | 2008
- 995
-
Development of dual-acting prodrugs for circumventing multidrug resistanceAbu Ajaj, Khalid / Kratz, Felix et al. | 2008
- 1001
-
Replacing alkyl sulfonamide with aromatic sulfonamide in sulfonamide-type RXR agonists favors switch towards antagonist activityMorishita, Ken-ichi / Yakushiji, Nobumasa / Ohsawa, Fuminori / Takamatsu, Kayo / Matsuura, Nobuyasu / Makishima, Makoto / Kawahata, Masatoshi / Yamaguchi, Kentaro / Tai, Akihiro / Sasaki, Kenji et al. | 2008
- 1004
-
Discovery and optimization of imidazo[1,2-a]pyridine inhibitors of insulin-like growth factor-1 receptor (IGF-1R)Emmitte, Kyle A. / Wilson, Brian J. / Baum, Erich W. / Emerson, Holly K. / Kuntz, Kevin W. / Nailor, Kristen E. / Salovich, James M. / Smith, Stephon C. / Cheung, Mui / Gerding, Roseanne M. et al. | 2008
- 1009
-
New analogues of agmatine with higher affinity to imidazoline receptorsTreder, Adam P. / Andruszkiewicz, Ryszard / Zgoda, Włodzimierz / Ford, Celeste / Hudson, Alan L. et al. | 2008
- 1012
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N,N-Dimethylsphingosine conjugates of poly-l-glutamic acid: Synthesis, characterization, and initial biological evaluationGhosh, Sukhen C. / Auzenne, Edmond / Khodadadian, Mojgan / Farquhar, David / Klostergaard, Jim et al. | 2008
- 1018
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Discovery of thiophene inhibitors of polo-like kinaseEmmitte, Kyle A. / Andrews, C. Webb / Badiang, Jennifer G. / Davis-Ward, Ronda G. / Dickson, Hamilton D. / Drewry, David H. / Emerson, Holly K. / Epperly, Andrea H. / Hassler, Daniel F. / Knick, Victoria B. et al. | 2008
- 1022
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1,2,3-Triazole derivatives as new cannabinoid CB1 receptor antagonistsHou, Duen-Ren / Alam, Safiul / Kuan, Ting-Chun / Ramanathan, Mani / Lin, Tsung-Pang / Hung, Ming-Shiu et al. | 2008
- 1026
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Identification of amidoheteroaryls as potent inhibitors of mutant (V600E) B-Raf kinase with in vivo activityLyne, Paul D. / Aquila, Brian / Cook, Donald J. / Dakin, Les A. / Ezhuthachan, Jay / Ioannidis, Stephanos / Pontz, Timothy / Su, Mei / Ye, Qing / Zheng, Xiaolan et al. | 2008
- 1030
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Development of pH-responsive core–shell nanocarriers for delivery of therapeutic and diagnostic agentsXu, Shangjie / Luo, Ying / Graeser, Ralph / Warnecke, André / Kratz, Felix / Hauff, Peter / Licha, Kai / Haag, Rainer et al. | 2008
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Instructions to contributors| 2009
- IFC
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Editorial board| 2009