Bioorganic and Medicinal Chemistry
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 7525
-
Graphical contents list| 2008
- 7535
-
Discovery of betamethasone 17α-carbamates as dissociated glucocorticoid receptor modulators in the ratAli, Amjad / Balkovec, James M. / Greenlee, Mark et al. | 2008
- 7535
-
Discovery of betamethasone 17a-carbamates as dissociated glucocorticoid receptor modulators in the ratAli, A. / Balkovec, J. M. / Greenlee, M. et al. | 2008
- 7543
-
Design, synthesis and in vitro antitumor activity of 4-aminoquinoline and 4-aminoquinazoline derivatives targeting EGFR tyrosine kinaseAbouzid, Khaled / Shouman, Samia et al. | 2008
- 7552
-
Structure–activity relationship studies on a novel class of antiproliferative agents derived from Lavendustin A. Part I: Ring A modificationsNussbaumer, Peter / Winiski, Anthony P. et al. | 2008
- 7561
-
Nakijiquinones G–I, new sesquiterpenoid quinones from marine spongeTakahashi, Yohei / Kubota, Takaaki / Ito, Junji et al. | 2008
- 7565
-
1,3,4-Oxadiazole-3(2H)-carboxamide derivatives as potential novel class of monoamine oxidase (MAO) inhibitors: Synthesis, evaluation, and role of urea moietyKe, Shaoyong / Li, Zhong / Qian, Xuhong et al. | 2008
- 7573
-
Synthesis and cellular effects of cycloterpenals: Cyclohexadienal-based activators of neurite outgrowthBench, Bennie J. / Tichy, Shane E. / Perez, Lisa M. et al. | 2008
- 7582
-
9-N-Substituted berberine derivatives: Stabilization of G-quadruplex DNA and down-regulation of oncogene c-mycMa, Yan / Ou, Tian-Miao / Hou, Jin-Qiang et al. | 2008
- 7592
-
Inhibitory effects of polymethoxy flavones isolated from Citrus reticulate on degranulation in rat basophilic leukemia RBL-2H3: Enhanced inhibition by their combinationItoh, Tomohiro / Ohguchi, Kenji / Iinuma, Munekazu et al. | 2008
- 7599
-
In silico prediction of novel phosphodiesterase type-5 inhibitors derived from Sildenafil, Vardenafil and TadalafilAntunes, João E. / Freitas, Matheus P. / da Cunha, Elaine F.F. et al. | 2008
- 7607
-
Microwave-assisted solid phase synthesis, PEGylation, and biological activity studies of glucagon-like peptide-1(7–36) amideChi, Yushi / Zhang, Huibin / Huang, Wenlong et al. | 2008
- 7615
-
A concise approach to 1,11-didechloro-6-methyl-4′-O-demethyl rebeccamycin and its binding to human serum albumin: Fluorescence spectroscopy and molecular modeling methodCui, Fengling / Qin, Lixia / Zhang, Guisheng et al. | 2008
- 7615
-
A concise approach to 1,11-didechloro-6-methyl-4prime-O-demethyl rebeccamycin and its binding to human serum albumin: Fluorescence spectroscopy and molecular modeling methodCui, F. / Qin, L. / Zhang, G. et al. | 2008
- 7622
-
Determination and characterization of new benzimidazoles with activity against Trypanosoma cruzi by UV spectroscopy and HPLCBrain-Isasi, Stephanie / Quezada, Cristián / Pessoa, Hernán et al. | 2008
- 7631
-
Inhibition of oxidative metabolism of tocopherols with ω-N-heterocyclic derivatives of vitamin EOhnmacht, Stephan / Nava, Phillip / West, Ryan et al. | 2008
- 7639
-
Synthesis and antiproliferative evaluation of amide-containing flavone and isoflavone derivativesChen, I-Li / Chen, Jhy-Yih / Shieh, Po-Chuen et al. | 2008
- 7646
-
2-Phenoxy-indan-1-one derivatives as acetylcholinesterase inhibitors: A study on the importance of modifications at the side chain on the activityShen, Yanhong / Sheng, Rong / Zhang, Jing et al. | 2008
- 7654
-
Synthesis and pharmacological evaluation of pentacyclic 6a,7-dihydrodiindole and 2,3-dihydrodiindole derivatives as novel melatoninergic ligandsAttia, Mohamed I. / Witt-Enderby, Paula A. / Julius, Justin et al. | 2008
- 7662
-
Synthesis and evaluation in vitro and in vivo of a 11C-labeled cyclooxygenase-2 (COX-2) inhibitorWuest, Frank / Kniess, Torsten / Bergmann, Ralf et al. | 2008
- 7671
-
Design, synthesis and preliminary biological evaluation of acridine compounds as potential agents for a combined targeted chemo-radionuclide therapy approach to melanomaDesbois, Nicolas / Gardette, Maryline / Papon, Janine et al. | 2008
- 7691
-
Solid-phase synthesis and biological evaluation of a parallel library of 2,3-dihydro-1,5-benzothiazepinesAnsari, Farzana Latif / Iftikhar, Fatima / Ihsan-ul-Haq et al. | 2008
- 7698
-
Synthesis and silencing properties of siRNAs possessing lipophilic groups at their 3prime-terminiUeno, Y. / Kawada, K. / Naito, T. et al. | 2008
- 7698
-
Synthesis and silencing properties of siRNAs possessing lipophilic groups at their 3′-terminiUeno, Yoshihito / Kawada, Koshi / Naito, Tomoharu et al. | 2008
- 7705
-
TX-2152: A conformationally rigid and electron-rich diyne analogue of FTY720 with in vivo antiangiogenic activityNakayama, Shinichi / Uto, Yoshihiro / Tanimoto, Kanako et al. | 2008
- 7715
-
Synthesis, biological evaluation, and molecular modeling studies of methylene imidazole substituted biaryls as inhibitors of human 17α-hydroxylase-17,20-lyase (CYP17)—Part II: Core rigidification and influence of substituents at the methylene bridgeHu, Qingzhong / Negri, Matthias / Jahn-Hoffmann, Kerstin et al. | 2008
- 7715
-
Synthesis, biological evaluation, and molecular modeling studies of methylene imidazole substituted biaryls as inhibitors of human 17a-hydroxylase-17,20-lyase (CYP17)-Part II: Core rigidification and influence of substituents at the methylene bridgeHu, Q. / Negri, M. / Jahn-Hoffmann, K. et al. | 2008
- 7728
-
Design, synthesis and biological evaluation of new tryptamine and tetrahydro-β-carboline-based selective inhibitors of CDK4Jenkins, Paul R. / Wilson, James / Emmerson, Daniel et al. | 2008
- 7728
-
Design, synthesis and biological evaluation of new tryptamine and tetrahydro-b-carboline-based selective inhibitors of CDK4Jenkins, P. R. / Wilson, J. / Emmerson, D. et al. | 2008
- 7740
-
Synthesis and preliminary pharmacological evaluation of novel derivatives of l-β-threo-benzylaspartate as inhibitors of the neuronal glutamate transporter EAAT3Mavencamp, Terri L. / Rhoderick, Joseph F. / Bridges, Richard J. et al. | 2008
- 7740
-
Synthesis and preliminary pharmacological evaluation of novel derivatives of l-b-threo-benzylaspartate as inhibitors of the neuronal glutamate transporter EAAT3Mavencamp, T. L. / Rhoderick, J. F. / Bridges, R. J. et al. | 2008
- 7749
-
Development of a receptor-based 3D-QSAR study for the analysis of MMP2, MMP3, and MMP9 inhibitorsTuccinardi, Tiziano / Nuti, Elisa / Ortore, Gabriella et al. | 2008
- 7759
-
New tacrine-dihydropyridine hybrids that inhibit acetylcholinesterase, calcium entry, and exhibit neuroprotection propertiesLeón, Rafael / Ríos, Cristóbal de los / Marco-Contelles, José et al. | 2008
- 7770
-
HP-Lattice QSAR for dynein proteins: Experimental proteomics (2D-electrophoresis, mass spectrometry) and theoretic study of a Leishmania infantum sequenceDea-Ayuela, María Auxiliadora / Pérez-Castillo, Yunierkis / Meneses-Marcel, Alfredo et al. | 2008
- 7777
-
Novel dimeric aryldiketo containing inhibitors of HIV-1 integrase: Effects of the phenyl substituent and the linker orientationZeng, Li-Fan / Jiang, Xiao-Hua / Sanchez, Tino et al. | 2008
- 7788
-
Array-based fluorescence assay for serine/threonine kinases using specific chemical reactionAkita, Shoji / Umezawa, Naoki / Kato, Nobuki et al. | 2008
- 7795
-
Inhibitory effect of the alkyl side chain of caffeic acid analogues on lipopolysaccharide-induced nitric oxide production in RAW264.7 macrophagesUwai, Koji / Osanai, Yuu / Imaizumi, Takuma et al. | 2008
- 7804
-
Synthesis, DNA-binding ability and evaluation of antitumour activity of triazolo[1,2,4]benzothiadiazine linked pyrrolo[2,1-c][1,4]benzodiazepine conjugatesKamal, Ahmed / Khan, M. Naseer A. / Srikanth, Y.V.V. et al. | 2008
- 7811
-
Synthesis of stable and selective inhibitors of human galectins-1 and -3Giguère, Denis / Bonin, Marc-André / Cloutier, Philipe et al. | 2008
- 7824
-
Syntheses and biological evaluation of topoisomerase I-targeting agents related to 11-[2-(N,N-dimethylamino)ethyl]-2,3-dimethoxy-8,9-methylenedioxy-11H-isoquino[4,3-c]cinnolin-12-one (ARC-31)Satyanarayana, Mavurapu / Feng, Wei / Cheng, Liang et al. | 2008
- 7832
-
Studies on the antifungal properties of N-thiolated b-lactamsO'Driscoll, M. / Greenhalgh, K. / Young, A. et al. | 2008
- 7832
-
Studies on the antifungal properties of N-thiolated β-lactamsO’Driscoll, Marci / Greenhalgh, Kerriann / Young, Ashley et al. | 2008
- 7838
-
Chemical synthesis of scyllo-inosamine and catabolism studies in Sinorhizobium melilotiSchoffers, Elke / Gurung, Sing R. / Kohler, Petra R.A. et al. | 2008
- 7843
-
Inhibitory effects of benzyl benzoate and its derivatives on angiotensin II-induced hypertensionOhno, Osamu / Ye, Mao / Koyama, Tomoyuki et al. | 2008
- 7853
-
Heme activates artemisinin more efficiently than hemin, inorganic iron, or hemoglobinZhang, Shiming / Gerhard, Glenn S. et al. | 2008
- 7862
-
Erratum to “Achiral, selective CCK2 receptor antagonists based on a 1,3,5-benzotriazepine-2,4-dione template” [Bioorg. Med. Chem. 16 (2008) 2974–2983]Spencer, John / Gaffen, John / Griffin, Eric et al. | 2008
- I
-
Instructions to contributors| 2008
- IFC
-
Editorial board| 2008