Bioorganic and Medicinal Chemistry
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 5279
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Graphical contents list| 2011
- 5291
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Synthesis, structural, and biological evaluation of bis-heteroarylmaleimides and bis-heterofused imidesFerri, Nicola / Radice, Tiziano / Antonino, Manuela et al. | 2011
- 5300
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Antifungal thiopeptide cyclothiazomycin B1 exhibits growth inhibition accompanying morphological changes via binding to fungal cell wall chitinMizuhara, Naoko / Kuroda, Manabu / Ogita, Akira et al. | 2011
- 5311
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Synthesis of benzo[3,4]azepino[1,2-b]isoquinolin-9-ones from 3-arylisoquinolines via ring closing metathesis and evaluation of topoisomerase I inhibitory activity, cytotoxicity and docking studyVan, Hue Thi My / Khadka, Daulat Bikram / Yang, Su Hui et al. | 2011
- 5321
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Chemical modifications of resveratrol for improved protein kinase C alpha activityDas, Joydip / Pany, Satyabrata / Majhi, Anjoy et al. | 2011
- 5334
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5a-Carba-b-d-glucopyranose derivatives as novel sodium-dependent glucose cotransporter 2 (SGLT2) inhibitors for the treatment of type 2 diabetesOhtake, Y. / Sato, T. / Matsuoka, H. et al. | 2011
- 5334
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5a-Carba-β-d-glucopyranose derivatives as novel sodium-dependent glucose cotransporter 2 (SGLT2) inhibitors for the treatment of type 2 diabetesOhtake, Yoshihito / Sato, Tsutomu / Matsuoka, Hiroharu et al. | 2011
- 5342
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Biochemical characterization of a novel type-II VEGFR2 kinase inhibitor: Comparison of binding to non-phosphorylated and phosphorylated VEGFR2Iwata, Hidehisa / Imamura, Shinichi / Hori, Akira et al. | 2011
- 5352
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Synthesis and biological evaluation of Matijing-Su derivatives as potent anti-HBV agentsQiu, Jingying / Xu, Bixue / Huang, Zhengming et al. | 2011
- 5361
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Design and synthesis of new prostaglandin D2 receptor antagonistsIwahashi, Maki / Takahashi, Eiji / Tanaka, Motoyuki et al. | 2011
- 5372
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SAR studies of acidic dual γ-secretase/PPARγ modulatorsHieke, Martina / Ness, Julia / Steri, Ramona et al. | 2011
- 5372
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SAR studies of acidic dual g-secretase/PPARg modulatorsHieke, M. / Ness, J. / Steri, R. et al. | 2011
- 5383
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Synthesis of pheophorbide-a conjugates with anticancer drugs as potential cancer diagnostic and therapeutic agentsYou, Hyun / Yoon, Hyo-Eun / Yoon, Jung-Hoon et al. | 2011
- 5392
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Isolation, identification, and biological evaluation of HIF-1-modulating compounds from Brazilian green propolisHattori, Hisanori / Okuda, Kensuke / Murase, Tetsuji et al. | 2011
- 5402
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Pachastrissamine (jaspine B) and its stereoisomers inhibit sphingosine kinases and atypical protein kinase CYoshimitsu, Yuji / Oishi, Shinya / Miyagaki, Jun et al. | 2011
- 5409
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Design and synthesis of 1,3-biarylsulfanyl derivatives as new anti-breast cancer agentsKumar, Atul / Tripathi, Vishwa Deepak / Kumar, Promod et al. | 2011
- 5420
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Assessment of dopamine D1 receptor affinity and efficacy of three tetracyclic conformationally-restricted analogs of SKF38393Clark, Alia H. / McCorvy, John D. / Watts, Val J. et al. | 2011
- 5432
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6,7-Dihydro-5H-cyclopenta[d]pyrazolo[1,5-a]pyrimidines and their derivatives as novel corticotropin-releasing factor 1 receptor antagonistsSaito, Tetsuji / Obitsu, Tetsuo / Kondo, Takashi et al. | 2011
- 5446
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Synthesis and characterization of tritylthioethanamine derivatives with potent KSP inhibitory activityRodriguez, Delany / Ramesh, Chinnasamy / Henson, Lauren H. et al. | 2011
- 5454
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Design, synthesis, and biological evaluation of imidazoline derivatives as p53–MDM2 binding inhibitorsHu, Chunqi / Li, Xin / Wang, Weisi et al. | 2011
- 5462
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Extended targeting potential and improved synthesis of Microcin C analogs as antibacterialsVondenhoff, Gaston H.M. / Dubiley, Svetlana / Severinov, Konstantin et al. | 2011
- 5468
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Novel macrocyclic C-aryl glucoside SGLT2 inhibitors as potential antidiabetic agentsKim, Min Ju / Lee, Suk Ho / Park, So Ok et al. | 2011
- 5480
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Synthesis and biological evaluation of a peptide–paclitaxel conjugate which targets the integrin αvβ6Li, Shunzi / Gray, Bethany Powell / McGuire, Michael J. et al. | 2011
- 5480
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Synthesis and biological evaluation of a peptide-paclitaxel conjugate which targets the integrin avb6Li, S. / Gray, B. P. / McGuire, M. J. et al. | 2011
- 5490
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2-({6-[(3R)-3-amino-3-methylpiperidine-1-yl]-1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydro-5H-pyrrolo[3,2-d]pyrimidine-5-yl}methyl)-4-fluorobenzonitrile (DSR-12727): A potent, orally active dipeptidyl peptidase IV inhibitor without mechanism-based inactivation of CYP3ANishio, Yukihiro / Kimura, Hidenori / Sawada, Naoyuki et al. | 2011
- 5500
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Substituted lactam and cyclic azahemiacetals modulate Pseudomonas aeruginosa quorum sensingMalladi, Venkata L.A. / Sobczak, Adam J. / Maricic, Natalie et al. | 2011
- 5507
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Inhibition of LuxS by S-ribosylhomocysteine analogues containing a [4-aza]ribose ringMalladi, Venkata L.A. / Sobczak, Adam J. / Meyer, Tiffany M. et al. | 2011
- 5520
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Synthesis and photobiological study of a novel chlorin photosensitizer BCPD-18MA for photodynamic therapyZhang, Jialiang / Deng, Li / Yao, Jianzhong et al. | 2011
- 5529
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Synthesis and SAR requirements of adamantane–colchicine conjugates with both microtubule depolymerizing and tubulin clustering activitiesZefirova, Olga N. / Nurieva, Evgeniya V. / Shishov, Dmitrii V. et al. | 2011
- 5539
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Discovery, synthesis, and structure–activity relationship of 6-aminomethyl-7,8-dihydronaphthalenes as human melanin-concentrating hormone receptor 1 antagonistsKamata, Makoto / Yamashita, Toshiro / Imaeda, Toshihiro et al. | 2011
- 5553
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Synthesis and biological evaluation of HQCAs with aryl or benzyl substituents on N-1 position as potential HIV-1 integrase inhibitorsHe, Qiu-Qin / Zhang, Xuan / Wu, Hai-Qiu et al. | 2011
- 5559
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Inhibitory effects of chalcone glycosides isolated from Brassica rapa L. ‘hidabeni’ and their synthetic derivatives on LPS-induced NO production in microgliaHara, Hirokazu / Nakamura, Yoko / Ninomiya, Masayuki et al. | 2011
- 5569
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N-(1,3-Diaryl-3-oxopropyl)amides as a new template for xanthine oxidase inhibitorsNepali, Kunal / Agarwal, Amit / Sapra, Sameer et al. | 2011
- 5577
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Synthesis and protective effects of aralkyl alcoholic 2-acetamido-2-deoxy-b-d-pyranosides on hypoglycemia and serum limitation induced apoptosis in PC12 cellMeng, Y. / Guo, Y. / Ling, Y. et al. | 2011
- 5577
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Synthesis and protective effects of aralkyl alcoholic 2-acetamido-2-deoxy-β-d-pyranosides on hypoglycemia and serum limitation induced apoptosis in PC12 cellMeng, Ying / Guo, Yibing / Ling, Yong et al. | 2011
- 5585
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The structure–activity relationship of urea derivatives as anti-tuberculosis agentsBrown, Joshua R. / North, Elton J. / Hurdle, Julian G. et al. | 2011
- 5596
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Design, synthesis, and biological evaluation of curcumin analogues as multifunctional agents for the treatment of Alzheimer’s diseaseChen, Shang-Ying / Chen, Yuan / Li, Yan-Ping et al. | 2011
- 5605
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Synthesis, antitubercular activity, and SAR study of N-substituted-phenylamino-5-methyl-1H-1,2,3-triazole-4-carbohydrazidesJordão, Alessandro K. / Sathler, Plínio C. / Ferreira, Vitor F. et al. | 2011
- 5612
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De novo design, synthesis and biological evaluation of 1,4-dihydroquinolin-4-ones and 1,2,3,4-tetrahydroquinazolin-4-ones as potent kinesin spindle protein (KSP) inhibitorsJiang, Cheng / Yang, Lei / Wu, Wu-Tong et al. | 2011
- 5628
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Synthesis and pharmacological evaluation of 1-alkyl-N-[2-ethyl-2-(4-fluorophenyl)butyl]piperidine-4-carboxamide derivatives as novel antihypertensive agentsWatanuki, Susumu / Matsuura, Keisuke / Tomura, Yuichi et al. | 2011
- 5639
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A novel 3-arylethynyl-substituted pyrido[2,3,-b]pyrazine derivatives and pharmacophore model as Wnt2/β-catenin pathway inhibitors in non-small-cell lung cancer cell linesGong, Young-Dae / Dong, Mi-Sook / Lee, Sang-Bum et al. | 2011
- 5639
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A novel 3-arylethynyl-substituted pyrido[2,3,-b]pyrazine derivatives and pharmacophore model as Wnt2/b-catenin pathway inhibitors in non-small-cell lung cancer cell linesGong, Y. D. / Dong, M. S. / Lee, S. B. et al. | 2011
- 5648
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Synthesis and biological evaluation of 2′,4′- and 3′,4′-bridged nucleoside analoguesNicolaou, K.C. / Ellery, Shelby P. / Rivas, Fatima et al. | 2011
- 5648
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Synthesis and biological evaluation of 2prime,4prime- and 3prime,4prime-bridged nucleoside analoguesNicolaou, K. C. / Ellery, S. P. / Rivas, F. et al. | 2011
- 5670
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Anthraquinone derivatives induce G2/M cell cycle arrest and apoptosis in NTUB1 cellsTu, Huang-Yao / Huang, A-Mei / Teng, Chi-Huang et al. | 2011
- 5679
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Synthesis and glycosidase inhibitory profiles of functionalised morpholines and oxazepanesBurland, Peter A. / Osborn, Helen M.I. / Turkson, Andrea et al. | 2011
- 5693
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Isolation and structural identification of a direct-acting mutagen derived from N-nitroso-N-methylpentylamine and Fenton’s reagent with copper ionMiura, Motofumi / Inami, Keiko / Yoshida, Masafumi et al. | 2011
- 5698
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Fluorinated cannabinoid CB2 receptor ligands: Synthesis and in vitro binding characteristics of 2-oxoquinoline derivativesTurkman, Nashaat / Shavrin, Aleksander / Ivanov, Roman A. et al. | 2011
- 5708
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Synthesis, antibacterial activities and molecular docking studies of Schiff bases derived from N-(2/4-benzaldehyde-amino) phenyl-N′-phenyl-thioureaZhang, Hong-Jia / Qin, Xuan / Liu, Kai et al. | 2011
- 5708
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Synthesis, antibacterial activities and molecular docking studies of Schiff bases derived from N-(2/4-benzaldehyde-amino) phenyl-Nprime-phenyl-thioureaZhang, H. J. / Qin, X. / Liu, K. et al. | 2011
- 5716
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A novel amino-benzosuberone derivative is a picomolar inhibitor of mammalian aminopeptidase N/CD13Maiereanu, Carmen / Schmitt, Céline / Schifano-Faux, Nadège et al. | 2011
- 5734
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Norcantharimide analogues possessing terminal phosphate esters and their anti-cancer activityRobertson, Mark J. / Gordon, Christopher P. / Gilbert, Jayne et al. | 2011
- 5742
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Corrigendum to “Discovery of potent, selective, and orally bioavailable quinoline-based dipeptidyl peptidase IV inhibitors targeting Lys554” [Bioorg. Med. Chem. 19 (2011) 4482–4498]Maezaki, Hironobu / Banno, Yoshihiro / Miyamoto, Yasufumi et al. | 2011
- IFC
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Editorial board| 2011