Bioorganic and Medicinal Chemistry
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 2135
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Graphical contents list| 2008
- 2148
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Fluorinated methylenecyclopropane analogues of nucleosides. Synthesis and antiviral activity of (Z)- and (E)-9-{[(2-fluoromethyl-2-hydroxymethyl)-cyclopropylidene]methyl}adenine and -guanineLi, Chengwei / Prichard, Mark N. / Korba, Brent E. et al. | 2007
- 2156
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Fused bicyclic pyrrolizinones as new scaffolds for human NK1 antagonistsMorriello, Gregori J. / DeVita, Robert J. / Mills, Sander G. et al. | 2007
- 2171
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A combined NMR and molecular dynamics simulation study to determine the conformational properties of agonists and antagonists against experimental autoimmune encephalomyelitisMantzourani, Efthimia D. / Blokar, Klemen / Tselios, Theodore V. et al. | 2007
- 2183
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Novel 2-(4-methylsulfonylphenyl)pyrimidine derivatives as highly potent and specific COX-2 inhibitorsOrjales, Aurelio / Mosquera, Ramón / López, Beatriz et al. | 2007
- 2200
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Structure–activity study of 2,3-benzodiazepin-4-ones noncompetitive AMPAR antagonists: Identification of the 1-(4-amino-3-methylphenyl)-3,5-dihydro-7,8-ethylenedioxy-4H-2,3-benzodiazepin-4-one as neuroprotective agentMicale, Nicola / Colleoni, Simona / Postorino, Giovanna et al. | 2007
- 2212
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α- and β-Substituted phosphonate analogs of LPA as autotaxin inhibitorsCui, Peng / McCalmont, William F. / Tomsig, Jose L. et al. | 2007
- 2212
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a- and b-Substituted phosphonate analogs of LPA as autotaxin inhibitorsCui, P. / McCalmont, W. F. / Tomsig, J. L. et al. | 2008
- 2226
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Imidazolidines as new anti-Trypanosoma cruzi agents: Biological evaluation and structure–activity relationshipsCaterina, M. Cristina / Perillo, Isabel A. / Boiani, Lucía et al. | 2007
- 2235
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Docking and hydropathic scoring of polysubstituted pyrrole compounds with antitubulin activityTripathi, Ashutosh / Fornabaio, Micaela / Kellogg, Glen E. et al. | 2007
- 2243
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Discovery of sulfonylalkylamides: A new class of orally active factor Xa inhibitorsImaeda, Yasuhiro / Miyawaki, Toshio / Sakamoto, Hiroki et al. | 2007
- 2261
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Structural requirements for the stability of novel cephalosporins to AmpC β-lactamase based on 3D-structureMurano, Kenji / Yamanaka, Toshio / Toda, Ayako et al. | 2007
- 2261
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Structural requirements for the stability of novel cephalosporins to AmpC b-lactamase based on 3D-structureMurano, K. / Yamanaka, T. / Toda, A. et al. | 2008
- 2276
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Activation and inhibition of DNA methyltransferases by S-adenosyl-l-homocysteine analoguesKumar, Ritesh / Srivastava, Richa / Singh, Ramendra Kumar et al. | 2007
- 2286
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Requirement of β-alanine components in sequence-specific DNA alkylation by pyrrole–imidazole conjugates with seven-base pair recognitionBando, Toshikazu / Minoshima, Masafumi / Kashiwazaki, Gengo et al. | 2007
- 2286
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Requirement of b-alanine components in sequence-specific DNA alkylation by pyrrole-imidazole conjugates with seven-base pair recognitionBando, T. / Minoshima, M. / Kashiwazaki, G. et al. | 2008
- 2292
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The number and distances of positive charges of polyamine side chains in a series of perylene diimides significantly influence their ability to induce G-quadruplex structures and inhibit human telomeraseFranceschin, Marco / Lombardo, Caterina Maria / Pascucci, Emanuela et al. | 2007
- 2305
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Nδ-Methylated l-arginine derivatives and their effects on the nitric oxide generating systemKotthaus, Jürke / Schade, Dennis / Töpker-Lehmann, Katrin et al. | 2007
- 2305
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Nd-Methylated l-arginine derivatives and their effects on the nitric oxide generating systemKotthaus, J. / Schade, D. / Topker-Lehmann, K. et al. | 2008
- 2313
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Parallel synthesis of a series of potentially brain penetrant aminoalkyl benzoimidazolesMicco, Iolanda / Nencini, Arianna / Quinn, Joanna et al. | 2007
- 2329
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Synthesis, cytostatic and anti-HCV activity of 6-(N-substituted aminomethyl)-, 6-(O-substituted hydroxymethyl)- and 6-(S-substituted sulfanylmethyl)purine nucleosidesŠilhár, Peter / Hocek, Michal / Pohl, Radek et al. | 2007
- 2367
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Synthesis and evaluation of antitumoral activity of ester and amide derivatives of 2-arylamino-6-trifluoromethyl-3-pyridinecarboxylic acidsOnnis, Valentina / Cocco, Maria T. / Lilliu, Valentina et al. | 2007
- 2379
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Synthesis and anticonvulsant evaluation of N-substituted isoquinoline AMPA receptor antagonistsGitto, Rosaria / De Luca, Laura / Pagano, Benedetta et al. | 2007
- 2385
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Bornyl (3,4,5-trihydroxy)-cinnamate - An optimized human neutrophil elastase inhibitor designed by free energy calculationsSteinbrecher, Thomas / Hrenn, Andrea / Dormann, Korinna L. et al. | 2007
- 2391
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Molecular modeling study and synthesis of novel pyrrolo[2,3-d]pyrimidines and pyrrolotriazolopyrimidines of expected antitumor and radioprotective activitiesAbou El Ella, Dalal A. / Ghorab, Mostafa M. / Noaman, Eman et al. | 2007
- 2403
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Synthesis and structure–immunosuppressive activity relationships of bakuchiol and its derivativesChen, Hongli / Du, Xiaolong / Tang, Wei et al. | 2007
- 2412
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Glyconanobiotics: Novel carbohydrated nanoparticle antibiotics for MRSA and Bacillus anthracisAbeylath, Sampath C. / Turos, Edward / Dickey, Sonja et al. | 2007
- 2419
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1,3-Dipropyl-8-(1-phenylacetamide-1H-pyrazol-3-yl)-xanthine derivatives as highly potent and selective human A2B adenosine receptor antagonistsTabrizi, Mojgan Aghazadeh / Baraldi, Pier Giovanni / Preti, Delia et al. | 2007
- 2431
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Synthesis and biological evaluation of pyrroloiminoquinone derivativesPassarella, Daniele / Belinghieri, Francesca / Scarpellini, Michele et al. | 2007
- 2439
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Three-dimensional quantitative structure–activity relationship studies on novel series of benzotriazine based compounds acting as Src inhibitors using CoMFA and CoMSIAGueto, Carlos / Ruiz, José L. / Torres, Juan E. et al. | 2007
- 2448
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Functional assay and structure–activity relationships of new third-generation P-glycoprotein inhibitorsMüller, Henrik / Pajeva, Ilza K. / Globisch, Christoph et al. | 2007
- 2463
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Structure–activity relationships in the inhibition of monoamine oxidase B by 1-methyl-3-phenylpyrrolesOgunrombi, Modupe O. / Malan, Sarel F. / Terre’Blanche, Gisella et al. | 2007
- 2473
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Stereospecific synthesis and bio-activity of novel β3-adrenoceptor agonists and inverse agonistsPerrone, Maria Grazia / Santandrea, Ernesto / Bleve, Laura et al. | 2007
- 2473
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Stereospecific synthesis and bio-activity of novel b3-adrenoceptor agonists and inverse agonistsPerrone, M. G. / Santandrea, E. / Bleve, L. et al. | 2008
- 2489
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ω-(2-Naphthyloxy) amino alkanes as a novel class of anti-hyperglycemic and lipid lowering agentsChaturvedi, Devdutt / Ray, Suprabhat / Srivastava, Arvind K. et al. | 2007
- 2499
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SAR studies of capsazepinoid bronchodilators. Part 1: The importance of the catechol moiety and aspects of the B-ring structureDalence-Guzmán, Marı´a F. / Berglund, Magnus / Skogvall, Staffan et al. | 2007
- 2513
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SAR studies of capsazepinoid bronchodilators. Part 2: Chlorination and catechol replacement in the A-ringBerglund, Magnus / Dalence-Guzmán, María F. / Skogvall, Staffan et al. | 2007
- 2529
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SAR studies of capsazepinoid bronchodilators 3: The thiourea part (coupling region) and the 2-(4-chlorophenyl)ethyl moiety (C-region)Berglund, Magnus / Dalence-Guzmán, María F. / Skogvall, Staffan et al. | 2007
- 2541
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Synthesis and antiproliferative activity of benzyl and phenethyl analogs of makaluvaminesShinkre, Bidhan A. / Raisch, Kevin P. / Fan, Liming et al. | 2007
- 2550
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Synthesis and biological evaluation of imidazol-2-one derivatives as potential antitumor agentsXue, Na / Yang, Xiaochun / Wu, Rui et al. | 2007
- 2558
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Synthesis and antimycobacterial evaluation of newer 1-cyclopropyl-1,4-dihydro-6-fluoro-7-(substituted secondary amino)-8-methoxy-5-(sub)-4-oxoquinoline-3-carboxylic acidsSenthilkumar, Palaniappan / Dinakaran, Murugesan / Banerjee, Debjani et al. | 2007
- 2570
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Novel quinazolinone derivatives as 5-HT7 receptor ligandsNa, Yong Ho / Hong, Sung Ho / Lee, Jung Hyang et al. | 2007
- 2579
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Rate enhancement of the oxidative folding of lysozyme by the use of aromatic thiol containing redox buffersGurbhele-Tupkar, Minakshi C. / Perez, Lissette R. / Silva, Yenia et al. | 2007
- 2591
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Activity of Mannich bases of 7-hydroxycoumarin against FlaviviridaeMazzei, Mauro / Nieddu, Erika / Miele, Mariangela et al. | 2007
- 2606
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Improved syntheses and applicability of different DOTA building blocks for multiply derivatized scaffoldsWängler, C. / Wängler, B. / Eisenhut, M. et al. | 2007
- 2617
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Novel AMPA and kainate receptor antagonists containing the pyrazolo[1,5-c]quinazoline ring system: Synthesis and structure–activity relationshipsVarano, Flavia / Catarzi, Daniela / Colotta, Vittoria et al. | 2007
- 2627
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Alachalasins A–G, new cytochalasins from the fungus Stachybotrys charatumZhang, Yonggang / Tian, Renrong / Liu, Shuchun et al. | 2007
- 2635
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Designed modification of partial agonist of ORL1 nociceptin receptor for conversion into highly potent antagonistLi, Jinglan / Isozaki, Kaname / Okada, Kazushi et al. | 2007
- 2645
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Low molecular weight lignin suppresses activation of NF-κB and HIV-1 promoterMitsuhashi, Shinya / Kishimoto, Takao / Uraki, Yasumitsu et al. | 2007
- 2645
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Low molecular weight lignin suppresses activation of NF-kB and HIV-1 promoterMitsuhashi, S. / Kishimoto, T. / Uraki, Y. et al. | 2008
- 2651
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Synthesis of novel oxazolidinone antimicrobial agentsEbner, David C. / Culhane, Jeffrey C. / Winkelman, Tyler N. et al. | 2007
- 2657
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Synthesis, nitric oxide release, and anti-leukemic activity of glutathione-activated nitric oxide prodrugs: Structural analogues of PABA/NO, an anti-cancer lead compoundChakrapani, Harinath / Wilde, Thomas C. / Citro, Michael L. et al. | 2007
- 2665
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Structural insights into hydroxycoumarin-induced apoptosis in U-937 cellsRiveiro, Maria E. / Moglioni, Albertina / Vazquez, Ramiro et al. | 2007
- 2676
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Synthesis and solution conformation studies of 3-substituted uridine and pseudouridine derivativesChang, Yu-Cheng / Herath, Jayatilake / Wang, Tony H.-H. et al. | 2007
- 2687
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Amphiphilic chitosan nanosphere: Studies on formation, toxicity, and guest molecule incorporationYoksan, Rangrong / Chirachanchai, Suwabun et al. | 2007
- 2697
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Selective COX-2 inhibitors. Part 2: Synthesis and biological evaluation of 4-benzylideneamino- and 4-phenyliminomethyl-benzenesulfonamidesLin, Shwu-Jiuan / Tsai, Wei-Jern / Chiou, Wen-Fei et al. | 2007
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Instructions to contributors| 2008
- IFC
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Editorial board| 2008