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Volume 67,
Issue 11
Volume 67,
Issue 10
Volume 67,
Issue 9
Volume 67,
Issue 8
Volume 67,
Issue 7
Volume 67,
Issue 6
Volume 67,
Issue 5
Volume 67,
Issue 4
Volume 67,
Issue 3
Volume 67,
Issue 2
Volume 67,
Issue 1
Volume 66,
Issue 24
Volume 66,
Issue 23
Volume 66,
Issue 22
Volume 66,
Issue 21
Volume 66,
Issue 20
Volume 66,
Issue 19
Volume 66,
Issue 18
Volume 66,
Issue 17
Volume 66,
Issue 16
Volume 66,
Issue 15
Volume 66,
Issue 14
Volume 66,
Issue 13
Volume 66,
Issue 12
Volume 66,
Issue 11
Volume 66,
Issue 10
Volume 66,
Issue 9
Volume 66,
Issue 8
Volume 66,
Issue 7
Volume 66,
Issue 6
Volume 66,
Issue 5
Volume 66,
Issue 4
Volume 66,
Issue 3
Volume 66,
Issue 2
Volume 66,
Issue 1
Volume 65,
Issue 20
Volume 65,
Issue 19
Volume 65,
Issue 18
Volume 65,
Issue 17
Volume 65,
Issue 16
Volume 65,
Issue 15
Volume 65,
Issue 14
Volume 65,
Issue 13
Volume 65,
Issue 12
Volume 65,
Issue 11
Volume 65,
Issue 10
Volume 65,
Issue 9
Volume 65,
Issue 8
Volume 65,
Issue 7
Volume 65,
Issue 6
Volume 65,
Issue 5
Volume 65,
Issue 4
Volume 65,
Issue 3
Volume 65,
Issue 2
Volume 65,
Issue 1
Volume 64,
Issue 24
Volume 64,
Issue 23
Volume 64,
Issue 22
Volume 64,
Issue 21
Volume 64,
Issue 20
Volume 64,
Issue 19
Volume 64,
Issue 18
Volume 64,
Issue 17
Volume 64,
Issue 16
Volume 64,
Issue 15
Volume 64,
Issue 14
Volume 64,
Issue 13
Volume 64,
Issue 12
Volume 64,
Issue 11
Volume 64,
Issue 10
Volume 64,
Issue 9
Volume 64,
Issue 8
Volume 64,
Issue 7
Volume 64,
Issue 6
Volume 64,
Issue 5
Volume 64,
Issue 4
Volume 64,
Issue 3
Volume 64,
Issue 2
Volume 64,
Issue 1
Volume 63,
Issue 24
Volume 63,
Issue 23
Volume 63,
Issue 22
Volume 63,
Issue 21
Volume 63,
Issue 20
Volume 63,
Issue 19
Volume 63,
Issue 18
Volume 63,
Issue 17
Volume 63,
Issue 16
Volume 63,
Issue 15
Volume 63,
Issue 14
Volume 63,
Issue 13
Volume 63,
Issue 12
Volume 63,
Issue 11
Volume 63,
Issue 10
Volume 63,
Issue 9
Volume 63,
Issue 8
Volume 63,
Issue 7
Volume 63,
Issue 6
Volume 63,
Issue 5
Volume 63,
Issue 4
Volume 63,
Issue 3
Volume 63,
Issue 2
Volume 63,
Issue 1
Volume 62,
Issue 24
Volume 62,
Issue 23
Volume 62,
Issue 22
Volume 62,
Issue 21
Volume 62,
Issue 20
Volume 62,
Issue 19
Volume 62,
Issue 18
Volume 62,
Issue 17
Volume 62,
Issue 16
Volume 62,
Issue 15
Volume 62,
Issue 14
Volume 62,
Issue 13
Volume 62,
Issue 12
Volume 62,
Issue 11
Volume 62,
Issue 10
Volume 62,
Issue 9
Volume 62,
Issue 8
Volume 62,
Issue 7
Volume 62,
Issue 6
Volume 62,
Issue 5
Volume 62,
Issue 4
Volume 62,
Issue 3
Volume 62,
Issue 2
Volume 62,
Issue 1
Volume 61,
Issue 24
Volume 61,
Issue 23
Volume 61,
Issue 22
Volume 61,
Issue 21
Volume 61,
Issue 20
Volume 61,
Issue 19
Volume 61,
Issue 18
Volume 61,
Issue 17
Volume 61,
Issue 16
Volume 61,
Issue 15
Volume 61,
Issue 14
Volume 61,
Issue 13
Volume 61,
Issue 12
Volume 61,
Issue 11
Volume 61,
Issue 10
Volume 61,
Issue 9
Volume 61,
Issue 8
Volume 61,
Issue 7
Volume 61,
Issue 6
Volume 61,
Issue 5
Volume 61,
Issue 4
Volume 61,
Issue 3
Volume 61,
Issue 2
Volume 61,
Issue 1
Volume 60,
Issue 24
Volume 60,
Issue 23
Volume 60,
Issue 22
Volume 60,
Issue 21
Volume 60,
Issue 20
Volume 60,
Issue 19
Volume 60,
Issue 18
Volume 60,
Issue 17
Volume 60,
Issue 16
Volume 60,
Issue 15
Volume 60,
Issue 14
Volume 60,
Issue 13
Volume 60,
Issue 12
Volume 60,
Issue 11
Volume 60,
Issue 10
Volume 60,
Issue 9
Volume 60,
Issue 8
Volume 60,
Issue 7
Volume 60,
Issue 6
Volume 60,
Issue 5
Volume 60,
Issue 4
Volume 60,
Issue 3
Volume 60,
Issue 2
Volume 60,
Issue 1
Volume 59,
Issue 24
Volume 59,
Issue 23
Volume 59,
Issue 22
Volume 59,
Issue 21
Volume 59,
Issue 20
Volume 59,
Issue 19
Volume 59,
Issue 18
Volume 59,
Issue 17
Volume 59,
Issue 16
Volume 59,
Issue 15
Volume 59,
Issue 14
Volume 59,
Issue 13
Volume 59,
Issue 12
Volume 59,
Issue 11
Volume 59,
Issue 10
Volume 59,
Issue 9
Volume 59,
Issue 8
Volume 59,
Issue 7
Volume 59,
Issue 6
Volume 59,
Issue 5
Volume 59,
Issue 4
Volume 59,
Issue 3
Volume 59,
Issue 2
Volume 59,
Issue 1
Volume 58,
Issue 24
Volume 58,
Issue 23
Volume 58,
Issue 22
Volume 58,
Issue 21
Volume 58,
Issue 20
Volume 58,
Issue 19
Volume 58,
Issue 18
Volume 58,
Issue 17
Volume 58,
Issue 16
Volume 58,
Issue 15
Volume 58,
Issue 14
Volume 58,
Issue 13
Volume 58,
Issue 12
Volume 58,
Issue 11
Volume 58,
Issue 10
Volume 58,
Issue 9
Volume 58,
Issue 8
Volume 58,
Issue 7
Volume 58,
Issue 6
Volume 58,
Issue 5
Volume 58,
Issue 4
Volume 58,
Issue 3
Volume 58,
Issue 2
Volume 58,
Issue 1
Volume 57,
Issue 24
Volume 57,
Issue 23
Volume 57,
Issue 22
Volume 57,
Issue 21
Volume 57,
Issue 20
Volume 57,
Issue 19
Volume 57,
Issue 18
Volume 57,
Issue 17
Volume 57,
Issue 16
Volume 57,
Issue 15
Volume 57,
Issue 14
Volume 57,
Issue 13
Volume 57,
Issue 12
Volume 57,
Issue 11
Volume 57,
Issue 10
Volume 57,
Issue 9
Volume 57,
Issue 8
Volume 57,
Issue 7
Volume 57,
Issue 6
Volume 57,
Issue 5
Volume 57,
Issue 4
Volume 57,
Issue 3
Volume 57,
Issue 2
Volume 57,
Issue 1
Volume 56,
Issue 24
Volume 56,
Issue 23
Volume 56,
Issue 22
Volume 56,
Issue 21
Volume 56,
Issue 20
Volume 56,
Issue 19
Volume 56,
Issue 18
Volume 56,
Issue 17
Volume 56,
Issue 16
Volume 56,
Issue 15
Volume 56,
Issue 14
Volume 56,
Issue 13
Volume 56,
Issue 12
Volume 56,
Issue 11
Volume 56,
Issue 10
Volume 56,
Issue 9
Volume 56,
Issue 8
Volume 56,
Issue 7
Volume 56,
Issue 6
Volume 56,
Issue 5
Volume 56,
Issue 4
Volume 56,
Issue 3
Volume 56,
Issue 2
Volume 56,
Issue 1
Volume 55,
Issue 24
Volume 55,
Issue 23
Volume 55,
Issue 22
Volume 55,
Issue 21
Volume 55,
Issue 20
Volume 55,
Issue 19
Volume 55,
Issue 18
Volume 55,
Issue 17
Volume 55,
Issue 16
Volume 55,
Issue 15
Volume 55,
Issue 14
Volume 55,
Issue 13
Volume 55,
Issue 12
Volume 55,
Issue 11
Volume 55,
Issue 10
Volume 55,
Issue 9
Volume 55,
Issue 8
Volume 55,
Issue 7
Volume 55,
Issue 6
Volume 55,
Issue 5
Volume 55,
Issue 4
Volume 55,
Issue 3
Volume 55,
Issue 2
Volume 55,
Issue 1
Volume 54,
Issue 24
Volume 54,
Issue 23
Volume 54,
Issue 22
Volume 54,
Issue 21
Volume 54,
Issue 20
Volume 54,
Issue 19
Volume 54,
Issue 18
Volume 54,
Issue 17
Volume 54,
Issue 16
Volume 54,
Issue 15
Volume 54,
Issue 14
Volume 54,
Issue 13
Volume 54,
Issue 12
Volume 54,
Issue 11
Volume 54,
Issue 10
Volume 54,
Issue 9
Volume 54,
Issue 8
Volume 54,
Issue 7
Volume 54,
Issue 6
Volume 54,
Issue 5
Volume 54,
Issue 4
Volume 54,
Issue 3
Volume 54,
Issue 2
Volume 54,
Issue 1
Volume 53,
Issue 24
Volume 53,
Issue 23
Volume 53,
Issue 22
Volume 53,
Issue 21
Volume 53,
Issue 20
Volume 53,
Issue 19
Volume 53,
Issue 18
Volume 53,
Issue 17
Volume 53,
Issue 16
Volume 53,
Issue 15
Volume 53,
Issue 14
Volume 53,
Issue 13
Volume 53,
Issue 12
Volume 53,
Issue 11
Volume 53,
Issue 10
Volume 53,
Issue 9
Volume 53,
Issue 8
Volume 53,
Issue 7
Volume 53,
Issue 6
Volume 53,
Issue 5
Volume 53,
Issue 4
Volume 53,
Issue 3
Volume 53,
Issue 2
Volume 53,
Issue 1
Volume 52,
Issue 24
Volume 52,
Issue 23
Volume 52,
Issue 22
Volume 52,
Issue 21
Volume 52,
Issue 20
Volume 52,
Issue 19
Volume 52,
Issue 18
Volume 52,
Issue 17
Volume 52,
Issue 16
Volume 52,
Issue 15
Volume 52,
Issue 14
Volume 52,
Issue 13
Volume 52,
Issue 12
Volume 52,
Issue 11
Volume 52,
Issue 10
Volume 52,
Issue 9
Volume 52,
Issue 8
Volume 52,
Issue 7
Volume 52,
Issue 6
Volume 52,
Issue 5
Volume 52,
Issue 4
Volume 52,
Issue 3
Volume 52,
Issue 2
Volume 52,
Issue 1
Volume 51,
Issue 24
Volume 51,
Issue 23
Volume 51,
Issue 22
Volume 51,
Issue 21
Volume 51,
Issue 20
Volume 51,
Issue 19
Volume 51,
Issue 18
Volume 51,
Issue 17
Volume 51,
Issue 16
Volume 51,
Issue 15
Volume 51,
Issue 14
Volume 51,
Issue 13
Volume 51,
Issue 12
Volume 51,
Issue 11
Volume 51,
Issue 10
Volume 51,
Issue 9
Volume 51,
Issue 8
Volume 51,
Issue 7
Volume 51,
Issue 6
Volume 51,
Issue 5
Volume 51,
Issue 4
Volume 51,
Issue 3
Volume 51,
Issue 2
Volume 51,
Issue 1
Volume 50,
Issue 26
Volume 50,
Issue 25
Volume 50,
Issue 24
Volume 50,
Issue 23
Volume 50,
Issue 22
Volume 50,
Issue 21
Volume 50,
Issue 20
Volume 50,
Issue 19
Volume 50,
Issue 18
Volume 50,
Issue 17
Volume 50,
Issue 16
Volume 50,
Issue 15
Volume 50,
Issue 14
Volume 50,
Issue 13
Volume 50,
Issue 12
Volume 50,
Issue 11
Volume 50,
Issue 10
Volume 50,
Issue 9
Volume 50,
Issue 8
Volume 50,
Issue 7
Volume 50,
Issue 6
Volume 50,
Issue 5
Volume 50,
Issue 4
Volume 50,
Issue 3
Volume 50,
Issue 2
Volume 50,
Issue 1
Volume 49,
Issue 26
Volume 49,
Issue 25
Volume 49,
Issue 24
Volume 49,
Issue 23
Volume 49,
Issue 22
Volume 49,
Issue 21
Volume 49,
Issue 20
Volume 49,
Issue 19
Volume 49,
Issue 18
Volume 49,
Issue 17
Volume 49,
Issue 16
Volume 49,
Issue 15
Volume 49,
Issue 14
Volume 49,
Issue 13
Volume 49,
Issue 12
Volume 49,
Issue 11
Volume 49,
Issue 10
Volume 49,
Issue 9
Volume 49,
Issue 8
Volume 49,
Issue 7
Volume 49,
Issue 6
Volume 49,
Issue 5
Volume 49,
Issue 4
Volume 49,
Issue 3
Volume 49,
Issue 2
Volume 49,
Issue 1
Volume 48,
Issue 26
Volume 48,
Issue 25
Volume 48,
Issue 24
Volume 48,
Issue 23
Volume 48,
Issue 22
Volume 48,
Issue 21
Volume 48,
Issue 20
Volume 48,
Issue 19
Volume 48,
Issue 18
Volume 48,
Issue 17
Volume 48,
Issue 16
Volume 48,
Issue 15
Volume 48,
Issue 14
Volume 48,
Issue 13
Volume 48,
Issue 12
Volume 48,
Issue 11
Volume 48,
Issue 10
Volume 48,
Issue 9
Volume 48,
Issue 8
Volume 48,
Issue 7
Volume 48,
Issue 6
Volume 48,
Issue 5
Volume 48,
Issue 4
Volume 48,
Issue 3
Volume 48,
Issue 2
Volume 48,
Issue 1
Volume 47,
Issue 27
Volume 47,
Issue 26
Volume 47,
Issue 25
Volume 47,
Issue 24
Volume 47,
Issue 23
Volume 47,
Issue 22
Volume 47,
Issue 21
Volume 47,
Issue 20
Volume 47,
Issue 19
Volume 47,
Issue 18
Volume 47,
Issue 17
Volume 47,
Issue 16
Volume 47,
Issue 15
Volume 47,
Issue 14
Volume 47,
Issue 13
Volume 47,
Issue 12
Volume 47,
Issue 11
Volume 47,
Issue 10
Volume 47,
Issue 9
Volume 47,
Issue 8
Volume 47,
Issue 7
Volume 47,
Issue 6
Volume 47,
Issue 5
Volume 47,
Issue 4
Volume 47,
Issue 3
Volume 47,
Issue 2
Volume 47,
Issue 1
Volume 46,
Issue 26
Volume 46,
Issue 25
Volume 46,
Issue 24
Volume 46,
Issue 23
Volume 46,
Issue 22
Volume 46,
Issue 21
Volume 46,
Issue 20
Volume 46,
Issue 19
Volume 46,
Issue 18
Volume 46,
Issue 17
Volume 46,
Issue 16
Volume 46,
Issue 15
Volume 46,
Issue 14
Volume 46,
Issue 13
Volume 46,
Issue 12
Volume 46,
Issue 11
Volume 46,
Issue 10
Volume 46,
Issue 9
Volume 46,
Issue 8
Volume 46,
Issue 7
Volume 46,
Issue 6
Volume 46,
Issue 5
Volume 46,
Issue 4
Volume 46,
Issue 3
Volume 46,
Issue 2
Volume 46,
Issue 1
Volume 45,
Issue 26
Volume 45,
Issue 25
Volume 45,
Issue 24
Volume 45,
Issue 23
Volume 45,
Issue 22
Volume 45,
Issue 21
Volume 45,
Issue 20
Volume 45,
Issue 19
Volume 45,
Issue 18
Volume 45,
Issue 17
Volume 45,
Issue 16
Volume 45,
Issue 15
Volume 45,
Issue 14
Volume 45,
Issue 13
Volume 45,
Issue 12
Volume 45,
Issue 11
Volume 45,
Issue 10
Volume 45,
Issue 9
Volume 45,
Issue 8
Volume 45,
Issue 7
Volume 45,
Issue 6
Volume 45,
Issue 5
Volume 45,
Issue 4
Volume 45,
Issue 3
Volume 45,
Issue 2
Volume 45,
Issue 1
Volume 44,
Issue 26
Volume 44,
Issue 25
Volume 44,
Issue 24
Volume 44,
Issue 23
Volume 44,
Issue 22
Volume 44,
Issue 21
Volume 44,
Issue 20
Volume 44,
Issue 19
Volume 44,
Issue 18
Volume 44,
Issue 17
Volume 44,
Issue 16
Volume 44,
Issue 15
Volume 44,
Issue 14
Volume 44,
Issue 13
Volume 44,
Issue 12
Volume 44,
Issue 11
Volume 44,
Issue 10
Volume 44,
Issue 9
Volume 44,
Issue 8
Volume 44,
Issue 7
Volume 44,
Issue 6
Volume 44,
Issue 5
Volume 44,
Issue 4
Volume 44,
Issue 3
Volume 44,
Issue 2
Volume 44,
Issue 1
Volume 43,
Issue 26
Volume 43,
Issue 25
Volume 43,
Issue 24
Volume 43,
Issue 23
Volume 43,
Issue 22
Volume 43,
Issue 21
Volume 43,
Issue 20
Volume 43,
Issue 19
Volume 43,
Issue 18
Volume 43,
Issue 17
Volume 43,
Issue 16
Volume 43,
Issue 15
Volume 43,
Issue 14
Volume 43,
Issue 13
Volume 43,
Issue 12
Volume 43,
Issue 11
Volume 43,
Issue 10
Volume 43,
Issue 9
Volume 43,
Issue 8
Volume 43,
Issue 7
Volume 43,
Issue 6
Volume 43,
Issue 5
Volume 43,
Issue 4
Volume 43,
Issue 3
Volume 43,
Issue 2
Volume 43,
Issue 1
Volume 42,
Issue 26
Volume 42,
Issue 25
Volume 42,
Issue 24
Volume 42,
Issue 23
Volume 42,
Issue 22
Volume 42,
Issue 21
Volume 42,
Issue 20
Volume 42,
Issue 19
Volume 42,
Issue 18
Volume 42,
Issue 17
Volume 42,
Issue 16
Volume 42,
Issue 15
Volume 42,
Issue 14
Volume 42,
Issue 13
Volume 42,
Issue 12
Volume 42,
Issue 11
Volume 42,
Issue 10
Volume 42,
Issue 9
Volume 42,
Issue 8
Volume 42,
Issue 7
Volume 42,
Issue 6
Volume 42,
Issue 5
Volume 42,
Issue 4
Volume 42,
Issue 3
Volume 42,
Issue 2
Volume 42,
Issue 1
Volume 41,
Issue 27
Volume 41,
Issue 26
Volume 41,
Issue 25
Volume 41,
Issue 24
Volume 41,
Issue 23
Volume 41,
Issue 22
Volume 41,
Issue 21
Volume 41,
Issue 20
Volume 41,
Issue 19
Volume 41,
Issue 18
Volume 41,
Issue 17
Volume 41,
Issue 16
Volume 41,
Issue 15
Volume 41,
Issue 14
Volume 41,
Issue 13
Volume 41,
Issue 12
Volume 41,
Issue 11
Volume 41,
Issue 10
Volume 41,
Issue 9
Volume 41,
Issue 8
Volume 41,
Issue 7
Volume 41,
Issue 6
Volume 41,
Issue 5
Volume 41,
Issue 4
Volume 41,
Issue 3
Volume 41,
Issue 2
Volume 41,
Issue 1
Volume 40,
Issue 26
Volume 40,
Issue 25
Volume 40,
Issue 24
Volume 40,
Issue 23
Volume 40,
Issue 22
Volume 40,
Issue 21
Volume 40,
Issue 20
Volume 40,
Issue 19
Volume 40,
Issue 18
Volume 40,
Issue 17
Volume 40,
Issue 16
Volume 40,
Issue 15
Volume 40,
Issue 14
Volume 40,
Issue 13
Volume 40,
Issue 12
Volume 40,
Issue 11
Volume 40,
Issue 10
Volume 40,
Issue 9
Volume 40,
Issue 8
Volume 40,
Issue 7
Volume 40,
Issue 6
Volume 40,
Issue 5
Volume 40,
Issue 4
Volume 40,
Issue 3
Volume 40,
Issue 2
Volume 40,
Issue 1
Volume 39,
Issue 26
Volume 39,
Issue 25
Volume 39,
Issue 24
Volume 39,
Issue 23
Volume 39,
Issue 22
Volume 39,
Issue 21
Volume 39,
Issue 20
Volume 39,
Issue 19
Volume 39,
Issue 18
Volume 39,
Issue 17
Volume 39,
Issue 16
Volume 39,
Issue 15
Volume 39,
Issue 14
Volume 39,
Issue 13
Volume 39,
Issue 12
Volume 39,
Issue 11
Volume 39,
Issue 10
Volume 39,
Issue 9
Volume 39,
Issue 8
Volume 39,
Issue 7
Volume 39,
Issue 6
Volume 39,
Issue 5
Volume 39,
Issue 4
Volume 39,
Issue 3
Volume 39,
Issue 2
Volume 39,
Issue 1
Volume 38,
Issue 26
Volume 38,
Issue 25
Volume 38,
Issue 24
Volume 38,
Issue 23
Volume 38,
Issue 22
Volume 38,
Issue 21
Volume 38,
Issue 20
Volume 38,
Issue 19
Volume 38,
Issue 18
Volume 38,
Issue 17
Volume 38,
Issue 16
Volume 38,
Issue 15
Volume 38,
Issue 14
Volume 38,
Issue 13
Volume 38,
Issue 12
Volume 38,
Issue 11
Volume 38,
Issue 10
Volume 38,
Issue 9
Volume 38,
Issue 8
Volume 38,
Issue 7
Volume 38,
Issue 6
Volume 38,
Issue 5
Volume 38,
Issue 4
Volume 38,
Issue 3
Volume 38,
Issue 2
Volume 38,
Issue 1
Volume 37,
Issue 26
Volume 37,
Issue 25
Volume 37,
Issue 24
Volume 37,
Issue 23
Volume 37,
Issue 22
Volume 37,
Issue 21
Volume 37,
Issue 20
Volume 37,
Issue 19
Volume 37,
Issue 18
Volume 37,
Issue 17
Volume 37,
Issue 16
Volume 37,
Issue 15
Volume 37,
Issue 14
Volume 37,
Issue 13
Volume 37,
Issue 12
Volume 37,
Issue 11
Volume 37,
Issue 10
Volume 37,
Issue 9
Volume 37,
Issue 8
Volume 37,
Issue 7
Volume 37,
Issue 6
Volume 37,
Issue 5
Volume 37,
Issue 4
Volume 37,
Issue 3
Volume 37,
Issue 2
Volume 37,
Issue 1
Volume 36,
Issue 26
Volume 36,
Issue 25
Volume 36,
Issue 24
Volume 36,
Issue 23
Volume 36,
Issue 22
Volume 36,
Issue 21
Volume 36,
Issue 20
Volume 36,
Issue 19
Volume 36,
Issue 18
Volume 36,
Issue 17
Volume 36,
Issue 16
Volume 36,
Issue 15
Volume 36,
Issue 14
Volume 36,
Issue 13
Volume 36,
Issue 12
Volume 36,
Issue 11
Volume 36,
Issue 10
Volume 36,
Issue 9
Volume 36,
Issue 8
Volume 36,
Issue 7
Volume 36,
Issue 6
Volume 36,
Issue 5
Volume 36,
Issue 4
Volume 36,
Issue 3
Volume 36,
Issue 2
Volume 36,
Issue 1
Volume 35,
Issue 26
Volume 35,
Issue 25
Volume 35,
Issue 24
Volume 35,
Issue 23
Volume 35,
Issue 22
Volume 35,
Issue 21
Volume 35,
Issue 20
Volume 35,
Issue 19
Volume 35,
Issue 18
Volume 35,
Issue 17
Volume 35,
Issue 16
Volume 35,
Issue 15
Volume 35,
Issue 14
Volume 35,
Issue 13
Volume 35,
Issue 12
Volume 35,
Issue 11
Volume 35,
Issue 10
Volume 35,
Issue 9
Volume 35,
Issue 8
Volume 35,
Issue 7
Volume 35,
Issue 6
Volume 35,
Issue 5
Volume 35,
Issue 4
Volume 35,
Issue 3
Volume 35,
Issue 2
Volume 35,
Issue 1
Volume 34,
Issue 12
Volume 34,
Issue 11
Volume 34,
Issue 10
Volume 34,
Issue 9
Volume 34,
Issue 8
Volume 34,
Issue 7
Volume 34,
Issue 6
Volume 34,
Issue 5
Volume 34,
Issue 4
Volume 34,
Issue 3
Volume 34,
Issue 2
Volume 34,
Issue 1
Volume 33,
Issue 12
Volume 33,
Issue 11
Volume 33,
Issue 10
Volume 33,
Issue 9
Volume 33,
Issue 8
Volume 33,
Issue 7
Volume 33,
Issue 6
Volume 33,
Issue 5
Volume 33,
Issue 4
Volume 33,
Issue 3
Volume 33,
Issue 2
Volume 33,
Issue 1
Volume 32,
Issue 12
Volume 32,
Issue 11
Volume 32,
Issue 10
Volume 32,
Issue 9
Volume 32,
Issue 8
Volume 32,
Issue 7
Volume 32,
Issue 6
Volume 32,
Issue 5
Volume 32,
Issue 4
Volume 32,
Issue 3
Volume 32,
Issue 2
Volume 32,
Issue 1
Volume 31,
Issue 12
Volume 31,
Issue 11
Volume 31,
Issue 10
Volume 31,
Issue 9
Volume 31,
Issue 8
Volume 31,
Issue 7
Volume 31,
Issue 6
Volume 31,
Issue 5
Volume 31,
Issue 4
Volume 31,
Issue 3
Volume 31,
Issue 2
Volume 31,
Issue 1
Volume 30,
Issue 12
Volume 30,
Issue 11
Volume 30,
Issue 10
Volume 30,
Issue 9
Volume 30,
Issue 8
Volume 30,
Issue 7
Volume 30,
Issue 6
Volume 30,
Issue 5
Volume 30,
Issue 4
Volume 30,
Issue 3
Volume 30,
Issue 2
Volume 30,
Issue 1
Volume 29,
Issue 12
Volume 29,
Issue 11
Volume 29,
Issue 10
Volume 29,
Issue 9
Volume 29,
Issue 8
Volume 29,
Issue 7
Volume 29,
Issue 6
Volume 29,
Issue 5
Volume 29,
Issue 4
Volume 29,
Issue 3
Volume 29,
Issue 2
Volume 29,
Issue 1
Volume 28,
Issue 12
Volume 28,
Issue 11
Volume 28,
Issue 10
Volume 28,
Issue 9
Volume 28,
Issue 8
Volume 28,
Issue 7
Volume 28,
Issue 6
Volume 28,
Issue 5
Volume 28,
Issue 4
Volume 28,
Issue 3
Volume 28,
Issue 2
Volume 28,
Issue 1
Volume 27,
Issue 12
Volume 27,
Issue 11
Volume 27,
Issue 10
Volume 27,
Issue 9
Volume 27,
Issue 8
Volume 27,
Issue 7
Volume 27,
Issue 6
Volume 27,
Issue 5
Volume 27,
Issue 4
Volume 27,
Issue 3
Volume 27,
Issue 2
Volume 27,
Issue 1
Volume 26,
Issue 12
Volume 26,
Issue 11
Volume 26,
Issue 10
Volume 26,
Issue 9
Volume 26,
Issue 8
Volume 26,
Issue 7
Volume 26,
Issue 6
Volume 26,
Issue 5
Volume 26,
Issue 4
Volume 26,
Issue 3
Volume 26,
Issue 2
Volume 26,
Issue 1
Volume 25,
Issue 12
Volume 25,
Issue 11
Volume 25,
Issue 10
Volume 25,
Issue 9
Volume 25,
Issue 8
Volume 25,
Issue 7
Volume 25,
Issue 6
Volume 25,
Issue 5
Volume 25,
Issue 4
Volume 25,
Issue 3
Volume 25,
Issue 2
Volume 25,
Issue 1
Volume 24,
Issue 12
Volume 24,
Issue 11
Volume 24,
Issue 10
Volume 24,
Issue 9
Volume 24,
Issue 8
Volume 24,
Issue 7
Volume 24,
Issue 6
Volume 24,
Issue 5
Volume 24,
Issue 4
Volume 24,
Issue 3
Volume 24,
Issue 2
Volume 24,
Issue 1
Volume 23,
Issue 12
Volume 23,
Issue 11
Volume 23,
Issue 10
Volume 23,
Issue 9
Volume 23,
Issue 8
Volume 23,
Issue 7
Volume 23,
Issue 6
Volume 23,
Issue 5
Volume 23,
Issue 4
Volume 23,
Issue 3
Volume 23,
Issue 2
Volume 23,
Issue 1
Volume 22,
Issue 12
Volume 22,
Issue 11
Volume 22,
Issue 10
Volume 22,
Issue 9
Volume 22,
Issue 8
Volume 22,
Issue 7
Volume 22,
Issue 6
Volume 22,
Issue 5
Volume 22,
Issue 4
Volume 22,
Issue 3
Volume 22,
Issue 2
Volume 22,
Issue 1
Volume 21,
Issue 12
Volume 21,
Issue 11
Volume 21,
Issue 10
Volume 21,
Issue 9
Volume 21,
Issue 8
Volume 21,
Issue 7
Volume 21,
Issue 6
Volume 21,
Issue 5
Volume 21,
Issue 4
Volume 21,
Issue 3
Volume 21,
Issue 2
Volume 21,
Issue 1
Volume 20,
Issue 12
Volume 20,
Issue 11
Volume 20,
Issue 10
Volume 20,
Issue 9
Volume 20,
Issue 8
Volume 20,
Issue 7
Volume 20,
Issue 6
Volume 20,
Issue 5
Volume 20,
Issue 4
Volume 20,
Issue 3
Volume 20,
Issue 2
Volume 20,
Issue 1
Volume 19,
Issue 12
Volume 19,
Issue 11
Volume 19,
Issue 10
Volume 19,
Issue 9
Volume 19,
Issue 8
Volume 19,
Issue 7
Volume 19,
Issue 6
Volume 19,
Issue 5
Volume 19,
Issue 4
Volume 19,
Issue 3
Volume 19,
Issue 2
Volume 19,
Issue 1
Volume 18,
Issue 12
Volume 18,
Issue 11
Volume 18,
Issue 10
Volume 18,
Issue 9
Volume 18,
Issue 8
Volume 18,
Issue 7
Volume 18,
Issue 6
Volume 18,
Issue 5
Volume 18,
Issue 4
Volume 18,
Issue 3
Volume 18,
Issue 2
Volume 18,
Issue 1
Volume 17,
Issue 12
Volume 17,
Issue 11
Volume 17,
Issue 10
Volume 17,
Issue 9
Volume 17,
Issue 8
Volume 17,
Issue 7
Volume 17,
Issue 6
Volume 17,
Issue 5
Volume 17,
Issue 4
Volume 17,
Issue 3
Volume 17,
Issue 2
Volume 17,
Issue 1
Volume 16,
Issue 12
Volume 16,
Issue 11
Volume 16,
Issue 10
Volume 16,
Issue 9
Volume 16,
Issue 8
Volume 16,
Issue 7
Volume 16,
Issue 6
Volume 16,
Issue 5
Volume 16,
Issue 4
Volume 16,
Issue 3
Volume 16,
Issue 2
Volume 16,
Issue 1
Volume 15,
Issue 12
Volume 15,
Issue 11
Volume 15,
Issue 10
Volume 15,
Issue 9
Volume 15,
Issue 8
Volume 15,
Issue 7
Volume 15,
Issue 6
Volume 15,
Issue 5
Volume 15,
Issue 4
Volume 15,
Issue 3
Volume 15,
Issue 2
Volume 15,
Issue 1
Volume 14,
Issue 12
Volume 14,
Issue 11
Volume 14,
Issue 10
Volume 14,
Issue 9
Volume 14,
Issue 8
Volume 14,
Issue 7
Volume 14,
Issue 6
Volume 14,
Issue 5
Volume 14,
Issue 4
Volume 14,
Issue 3
Volume 14,
Issue 2
Volume 14,
Issue 1
Volume 13,
Issue 6
Volume 13,
Issue 5
Volume 13,
Issue 4
Volume 13,
Issue 3
Volume 13,
Issue 2
Volume 13,
Issue 1
Volume 12,
Issue 6
Volume 12,
Issue 5
Volume 12,
Issue 4
Volume 12,
Issue 3
Volume 12,
Issue 2
Volume 12,
Issue 1
Volume 11,
Issue 6
Volume 11,
Issue 5
Volume 11,
Issue 4
Volume 11,
Issue 3
Volume 11,
Issue 2
Volume 11,
Issue 1
Volume 10,
Issue 6
Volume 10,
Issue 5
Volume 10,
Issue 4
Volume 10,
Issue 3
Volume 10,
Issue 2
Volume 10,
Issue 1
Volume 9,
Issue 6
Volume 9,
Issue 5
Volume 9,
Issue 4
Volume 9,
Issue 3
Volume 9,
Issue 2
Volume 9,
Issue 1
Volume 8,
Issue 6
Volume 8,
Issue 5
Volume 8,
Issue 4
Volume 8,
Issue 3
Volume 8,
Issue 2
Volume 8,
Issue 1
Volume 7,
Issue 6
Volume 7,
Issue 5
Volume 7,
Issue 4
Volume 7,
Issue 3
Volume 7,
Issue 2
Volume 7,
Issue 1
Volume 6,
Issue 6
Volume 6,
Issue 5
Volume 6,
Issue 4
Volume 6,
Issue 3
Volume 6,
Issue 2
Volume 6,
Issue 1
Volume 4,
Issue 3
Volume 4,
Issue 2
Volume 4,
Issue 1
Volume 3,
Issue 3
Volume 3,
Issue 2
Volume 3,
Issue 1
Volume 2,
Issue 6
Volume 2,
Issue 5
Volume 2,
Issue 4
Volume 2,
Issue 3
Volume 2,
Issue 2
Volume 2,
Issue 1
Volume 1,
Issue 6
Volume 1,
Issue 5
Volume 1,
Issue 4
Volume 1,
Issue 3
Volume 1,
Issue 2
Volume 1,
Issue 1
>
Table of contents
1685
Memorial Issue in Honor of Dr. Paul A. J. Janssen Preface
Galemmo,, Robert A.
/ Janssens, Frans E.
/ Lewi, Paul J.
et al.
| 2005
1686
In Memoriam: Dr. Paul A. J. Janssen (1926−2003)
Galemmo,, Robert A.
/ Janssens, Frans E.
/ Lewi, Paul J.
et al.
| 2005
1687
A Personal Perspective on Dr. Paul Janssen
Black, James
et al.
| 2005
1689
From 4,5,6,7-Tetrahydro-5-methylimidazo[4,5,1-jk](1,4)benzodiazepin-2(1H)-one (TIBO) to Etravirine (TMC125): Fifteen Years of Research on Non-Nucleoside Inhibitors of HIV-1 Reverse Transcriptase †
De Corte, Bart L.
et al.
| 2005
1697
Identification of Substituted 6-Amino-4-phenyltetrahydroquinoline Derivatives: Potent Antagonists for the Follicle-Stimulating Hormone Receptor
van Straten, Nicole C. R.
/ van Berkel, Twan H. J.
/ Demont, Dennis R.
et al.
| 2005
1701
Synthesis and Pharmacological Evaluation of Huprine−Tacrine Heterodimers: Subnanomolar Dual Binding Site Acetylcholinesterase Inhibitors
Camps, Pelayo
/ Formosa, Xavier
/ Muñoz-Torrero, Diego
et al.
| 2005
1705
Novel Atypical Antipsychotic Agents: Rational Design, an Efficient Palladium-Catalyzed Route, and Pharmacological Studies
Campiani, Giuseppe
/ Butini, Stefania
/ Fattorusso, Caterina
et al.
| 2005
1709
Discovery of New Tetracyclic Tetrahydrofuran Derivatives as Potential Broad-Spectrum Psychotropic Agents
Fernández, Javier
/ Alonso, José M.
/ Andrés, José I.
et al.
| 2005
1713
A Bivalent Ligand (KDAN-18) Containing δ-Antagonist and κ-Agonist Pharmacophores Bridges δ2 and κ1 Opioid Receptor Phenotypes †
Daniels, David J.
/ Kulkarni, Amol
/ Xie, Zhihua
et al.
| 2005
1713
A Bivalent Ligand (KDAN-18) Containing delta-Antagonist and kappa-Agonist Pharmacophores Bridges delta~2 and kappa~1 Opioid Receptor Phenotypes
Daniels, D. J.
/ Kulkarni, A.
/ Xie, Z.
et al.
| 2005
1713
A Bivalent Ligand (KDAN-18) Containing d-Antagonist and k-Agonist Pharmacophores Bridges d2 and k1 Opioid Receptor Phenotypes
Daniels, D.J.
et al.
| 2005
1717
2-Hydroxy-4,6-diamino-[1,3,5]triazines: A Novel Class of VEGF-R2 (KDR) Tyrosine Kinase Inhibitors
Baindur, Nand
/ Chadha, Naresh
/ Brandt, Benjamin M.
et al.
| 2005
1721
Novel Pyridyl Ring C5 Substituted Analogues of Epibatidine and 3-(1-Methyl-2(S)-pyrrolidinylmethoxy)pyridine (A-84543) as Highly Selective Agents for Neuronal Nicotinic Acetylcholine Receptors Containing beta2 Subunits
Wei, Z.-L.
/ Xiao, Y.
/ Yuan, H.
et al.
| 2005
1721
Novel Pyridyl Ring C5 Substituted Analogues of Epibatidine and 3-(1-Methyl-2(S)- pyrrolidinylmethoxy)pyridine (A-84543) as Highly Selective Agents for Neuronal Nicotinic Acetylcholine Receptors Containing b2 Subunits
Wei, Z.-L.
et al.
| 2005
1721
Novel Pyridyl Ring C5 Substituted Analogues of Epibatidine and 3-(1-Methyl-2(S)- pyrrolidinylmethoxy)pyridine (A-84543) as Highly Selective Agents for Neuronal Nicotinic Acetylcholine Receptors Containing β2 Subunits
Wei, Zhi-Liang
/ Xiao, Yingxian
/ Yuan, Hongbin
et al.
| 2005
1725
Novel Indolylindazolylmaleimides as Inhibitors of Protein Kinase C-β: Synthesis, Biological Activity, and Cardiovascular Safety †
Zhang, Han-Cheng
/ Derian, Claudia K.
/ McComsey, David F.
et al.
| 2005
1725
Novel Indolylindazolylmaleimides as Inhibitors of Protein Kinase C-beta: Synthesis, Biological Activity, and Cardiovascular Safety
Zhang, H.-C.
/ Derian, C. K.
/ McComsey, D. F.
et al.
| 2005
1725
Novel Indolylindazolylmaleimides as Inhibitors of Protein Kinase C-b: Synthesis, Biological Activity, and Cardiovascular Safety
Zhang, H.-C.
et al.
| 2005
1729
Discovery of 1-(3‘-Aminobenzisoxazol-5‘-yl)-3-trifluoromethyl-N-[2-fluoro-4- [(2‘-dimethylaminomethyl)imidazol-1-yl]phenyl]-1H-pyrazole-5-carboxyamide Hydrochloride (Razaxaban), a Highly Potent, Selective, and Orally Bioavailable Factor Xa Inhibitor
Quan, Mimi L.
/ Lam, Patrick Y. S.
/ Han, Qi
et al.
| 2005
1745
(N)-Methanocarba 2,N 6 -Disubstituted Adenine Nucleosides as Highly Potent and Selective A3 Adenosine Receptor Agonists
Tchilibon, Susanna
/ Joshi, Bhalchandra V.
/ Kim, Soo-Kyung
et al.
| 2005
1759
Solvent Constraints on the Property Space of Acetylcholine. I. Isotropic Solvents
Vistoli, Giulio
/ Pedretti, Alessandro
/ Villa, Luigi
et al.
| 2005
1768
Fluoro-Olefins as Peptidomimetic Inhibitors of Dipeptidyl Peptidases
Van der Veken, Pieter
/ Senten, Kristel
/ Kertèsz, István
et al.
| 2005
1781
Medicinal Chemistry Driven Approaches Toward Novel and Selective Serotonin 5-HT6 Receptor Ligands
Holenz, Jörg
/ Mercè, Ramon
/ Díaz, José Luis
et al.
| 2005
1796
Synthesis and Evaluation of Imidazolylmethylenetetrahydronaphthalenes and Imidazolylmethyleneindanes: Potent Inhibitors of Aldosterone Synthase
Ulmschneider, Sarah
/ Müller-Vieira, Ursula
/ Mitrenga, Markus
et al.
| 2005
1806
Nanomolar Inhibitors of CNS Epinephrine Biosynthesis: (R)-(+)-3-Fluoromethyl-7-(N-substituted aminosulfonyl)-1,2,3,4-tetrahydroisoquinolines as Potent and Highly Selective Inhibitors of Phenylethanolamine N-Methyltransferase
Grunewald, Gary L.
/ Romero, F. Anthony
/ Criscione, Kevin R.
et al.
| 2005
1806
Nanomolar Inhibitors of CNS Epinephrine Biosynthesis: (R)-(+)-3-Fluoromethyl-7-(N-substituted aminosulfonyl)-1,2,3,4-tetrahydroisoquinolines as Potent and Highly Selective Inhibitors of Phenylethanolamine N-Methyltransferase1
Grunewald, G.L.
et al.
| 2005
1813
Discovery and Selection of TMC114, a Next Generation HIV-1 Protease Inhibitor §
Surleraux, Dominique L. N. G.
/ Tahri, Abdellah
/ Verschueren, Wim G.
et al.
| 2005
1823
Bioisosteric Replacements of the Pyrazole Moiety of Rimonabant: Synthesis, Biological Properties, and Molecular Modeling Investigations of Thiazoles, Triazoles, and Imidazoles as Potent and Selective CB1 Cannabinoid Receptor Antagonists
Lange, Jos H. M.
/ van Stuivenberg, Herman H.
/ Coolen, Hein K. A. C.
et al.
| 2005
1839
Novel 3D Pharmacophore of α-MSH/γ-MSH Hybrids Leads to Selective Human MC1R and MC3R Analogues †
Cai, Minying
/ Mayorov, Alexander V.
/ Cabello, Christopher
et al.
| 2005
1839
Novel 3D Pharmacophore of alpha-MSH/gamma-MSH Hybrids Leads to Selective Human MC1R and MC3R Analogues
Cai, M.
/ Mayorov, A. V.
/ Cabello, C.
et al.
| 2005
1839
Novel 3D Pharmacophore of a-MSH-g-MSH Hybrids Leads to Selective Human MC1R and MC3R Analogues
Cai, M.
et al.
| 2005
1849
Discovery of a Potent, Selective, and Efficacious Class of Reversible alpha-Ketoheterocycle Inhibitors of Fatty Acid Amide Hydrolase Effective as Analgesics
Boger, D. L.
/ Miyauchi, H.
/ Du, W.
et al.
| 2005
1849
Discovery of a Potent, Selective, and Efficacious Class of Reversible α-Ketoheterocycle Inhibitors of Fatty Acid Amide Hydrolase Effective as Analgesics ∇
Boger, Dale L.
/ Miyauchi, Hiroshi
/ Du, Wu
et al.
| 2005
1849
Discovery of a Potent, Selective, and Efficacious Class of Reversible a-Ketoheterocycle Inhibitors of Fatty Acid Amide Hydrolase Effective as Analgesics
Boger, D.L.
et al.
| 2005
1857
Identification and Biological Evaluation of 4-(3-Trifluoromethylpyridin-2-yl)piperazine-1-carboxylic Acid (5-Trifluoromethylpyridin-2-yl)amide, a High Affinity TRPV1 (VR1) Vanilloid Receptor Antagonist
Swanson, Devin M.
/ Dubin, Adrienne E.
/ Shah, Chandra
et al.
| 2005
1873
Checkpoint Kinase Inhibitors: SAR and Radioprotective Properties of a Series of 2-Arylbenzimidazoles
Arienti, Kristen L.
/ Brunmark, Anders
/ Axe, Frank U.
et al.
| 2005
1886
Synthesis and Discovery of Pyrazine−Pyridine Biheteroaryl as a Novel Series of Potent Vascular Endothelial Growth Factor Receptor-2 Inhibitors
Kuo, Gee-Hong
/ Wang, Aihua
/ Emanuel, Stuart
et al.
| 2005
1901
In Search of a Novel Anti-HIV Drug: Multidisciplinary Coordination in the Discovery of 4-[[4-[[4-[(1E)-2-Cyanoethenyl]-2,6-dimethylphenyl]amino]-2- pyrimidinyl]amino]benzonitrile (R278474, Rilpivirine)
Janssen, Paul A. J.
/ Lewi, Paul J.
/ Arnold, Eddy
et al.
| 2005
1910
Design, Synthesis, and SAR of a Novel Pyrazinone Series with Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitory Activity
Heeres, Jan
/ de Jonge, Marc R.
/ Koymans, Lucien M. H.
et al.
| 2005
1919
Development of Molecular Probes for the Identification of Extra Interaction Sites in the Mid-Gorge and Peripheral Sites of Butyrylcholinesterase (BuChE). Rational Design of Novel, Selective, and Highly Potent BuChE Inhibitors †
Campiani, Giuseppe
/ Fattorusso, Caterina
/ Butini, Stefania
et al.
| 2005
1930
Design and Optimization of Tricyclic Phtalimide Analogues as Novel Inhibitors of HIV-1 Integrase
Verschueren, Wim G.
/ Dierynck, Inge
/ Amssoms, Katie I. E.
et al.
| 2005
1941
Comparison of Sulfamate and Sulfamide Groups for the Inhibition of Carbonic Anhydrase-II by Using Topiramate as a Structural Platform †
Maryanoff, Bruce E.
/ McComsey, David F.
/ Costanzo, Michael J.
et al.
| 2005
1948
4-Benzyl and 4-Benzoyl-3-dimethylaminopyridin-2(1H)-ones: In Vitro Evaluation of New C-3-Amino-Substituted and C-5,6-Alkyl-Substituted Analogues against Clinically Important HIV Mutant Strains
Benjahad, Abdellah
/ Croisy, Martine
/ Monneret, Claude
et al.
| 2005
1965
Design of HIV-1 Protease Inhibitors Active on Multidrug-Resistant Virus
Surleraux, Dominique L. N. G.
/ de Kock, Herman A.
/ Verschueren, Wim G.
et al.
| 2005
1974
Concentration and pH Dependent Aggregation of Hydrophobic Drug Molecules and Relevance to Oral Bioavailability
Frenkel, Yulia Volovik
/ Clark,, Arthur D.
/ Das, Kalyan
et al.
| 2005
1984
In-Depth Study of Tripeptide-Based α-Ketoheterocycles as Inhibitors of Thrombin. Effective Utilization of the S1 ‘ Subsite and Its Implications to Structure-Based Drug Design
Costanzo, Michael J.
/ Almond, Harold R.
/ Hecker, Leonard R.
et al.
| 2005
1984
In-Depth Study of Tripeptide-Based a-Ketoheterocycles as Inhibitors of Thrombin. Effective Utilization of the S1' Subsite and Its Implications to Structure-Based Drug Design1
Costanzo, M.J.
et al.
| 2005
1984
In-Depth Study of Tripeptide-Based alpha-Ketoheterocycles as Inhibitors of Thrombin. Effective Utilization of the S~1' Subsite and Its Implications to Structure-Based Drug Design
Costanzo, M. J.
/ Almond, H. R.
/ Hecker, L. R.
et al.
| 2005
2009
Novel Diamino Derivatives of [1,2,4]Triazolo[1,5-a][1,3,5]triazine as Potent and Selective Adenosine A2a Receptor Antagonists
Vu, Chi B.
/ Pan, Deborah
/ Peng, Bo
et al.
| 2005
2019
Synthesis of New Quinoxaline-2-carboxylate 1,4-Dioxide Derivatives as Anti-Mycobacterium t uberculosis Agents
Jaso, Andrés
/ Zarranz, Belén
/ Aldana, Ignacio
et al.
| 2005
2026
Binding Thermodynamics as a Tool To Investigate the Mechanisms of Drug−Receptor Interactions: Thermodynamics of Cytoplasmic Steroid/Nuclear Receptors in Comparison with Membrane Receptors
Gilli, Paola
/ Gilli, Gastone
/ Borea, Pier Andrea
et al.
| 2005
2036
Biological Properties of d- and l-1-Deoxyazasugars
Kato, Atsushi
/ Kato, Noriko
/ Kano, Erika
et al.
| 2005
2045
A Series of Ligands Displaying a Remarkable Agonistic−Antagonistic Profile at the Adenosine A1 Receptor
Chang, Lisa C. W.
/ von Frijtag Drabbe Künzel, Jacobien K.
/ Mulder-Krieger, Thea
et al.
| 2005
2054
Discovery of a New Series of Centrally Active Tricyclic Isoxazoles Combining Serotonin (5-HT) Reuptake Inhibition with alpha~2-Adrenoceptor Blocking Activity
Andres, J. I.
/ Alcazar, J.
/ Alonso, J. M.
et al.
| 2005
2054
Discovery of a New Series of Centrally Active Tricyclic Isoxazoles Combining Serotonin (5-HT) Reuptake Inhibition with a2-Adrenoceptor Blocking Activity
Andres, J.I.
et al.
| 2005
2054
Discovery of a New Series of Centrally Active Tricyclic Isoxazoles Combining Serotonin (5-HT) Reuptake Inhibition with α2 -Adrenoceptor Blocking Activity
Andrés, J. Ignacio
/ Alcázar, Jesús
/ Alonso, José M.
et al.
| 2005
2072
Synthesis of Novel Diarylpyrimidine Analogues and Their Antiviral Activity against Human Immunodeficiency Virus Type 1
Guillemont, Jerome
/ Pasquier, Elisabeth
/ Palandjian, Patrice
et al.
| 2005
2080
Synthesis of New Benzoxazinone Derivatives as Neuropeptide Y5 Antagonists for the Treatment of Obesity #
Torrens, Antoni
/ Mas, Josep
/ Port, Adriana
et al.
| 2005
2093
Organometallic Anticancer Agents: Cellular Uptake and Cytotoxicity Studies on Thiol Derivatives of the Antitumor Agent Molybdocene Dichloride
Waern, Jenny B.
/ Dillon, Carolyn T.
/ Harding, Margaret M.
et al.
| 2005
2100
N-Substituted Piperidinyl Alkyl Imidazoles: Discovery of Methimepip as a Potent and Selective Histamine H3 Receptor Agonist
Kitbunnadaj, Ruengwit
/ Hashimoto, Takeshi
/ Poli, Enzo
et al.
| 2005
2108
Development of Spin-Labeled Probes for Adenosine Receptors †
Ilaš, Janez
/ Pečar, Slavko
/ Hockemeyer, Jörg
et al.
| 2005
2115
Genotype Dependent QSAR for HIV-1 Protease Inhibition
Boutton, Carlo W.
/ De Bondt, Hendrik L.
/ De Jonge, Marc R.
et al.
| 2005
2121
Carbonic Anhydrase Inhibitors: Synthesis and Inhibition of Cytosolic/Membrane-Associated Carbonic Anhydrase Isozymes I, II, and IX with Sulfonamides Incorporating Hydrazino Moieties
Winum, Jean-Yves
/ Dogné, Jean-Michel
/ Casini, Angela
et al.
| 2005
2126
Pyrroloquinolone PDE5 Inhibitors with Improved Pharmaceutical Profiles for Clinical Studies on Erectile Dysfunction
Jiang, Weiqin
/ Guan, Jihua
/ Macielag, Mark J.
et al.
| 2005
2134
Synthesis, Structure−Activity Relationship, and Receptor Pharmacology of a New Series of Quinoline Derivatives Acting as Selective, Noncompetitive mGlu1 Antagonists
Mabire, Dominique
/ Coupa, Sophie
/ Adelinet, Christophe
et al.
| 2005
2154
Norpiperidine Imidazoazepines as a New Class of Potent, Selective, and Nonsedative H1 Antihistamines
Janssens, Frans
/ Leenaerts, Jos
/ Diels, Gaston
et al.
| 2005
2167
Synthesis and Biological Evaluation of 1,2,4-Triazinylphenylalkylthiazolecarboxylic Acid Esters as Cytokine-Inhibiting Antedrugs with Strong Bronchodilating Effects in an Animal Model of Asthma
Freyne, Eddy J.
/ Lacrampe, Jean F.
/ Deroose, Frederik
et al.
| 2005
2176
Structure Based Activity Prediction of HIV-1 Reverse Transcriptase Inhibitors
de Jonge, Marc R.
/ Koymans, Lucien M. H.
/ Vinkers, H. Maarten
et al.
| 2005
2184
Synthesis and in Vitro and in Vivo Structure−Activity Relationships of Novel Antifungal Triazoles for Dermatology
Meerpoel, Lieven
/ Backx, Leo J. J.
/ Van der Veken, Louis J. E.
et al.
| 2005
2194
Discovery of CC Chemokine Receptor-3 (CCR3) Antagonists with Picomolar Potency
De Lucca, George V.
/ Kim, Ui Tae
/ Vargo, Brian J.
et al.
| 2005
2212
Muscarinic Allosteric Enhancers of Ligand Binding: Pivotal Pharmacophoric Elements in Hexamethonio-Type Agents
Muth, Mathias
/ Sennwitz, Matthias
/ Mohr, Klaus
et al.
| 2005
2218
Design, Synthesis and Structure−Activity Relationships of Novel Taxane-Based Multidrug Resistance Reversal Agents
Ojima, Iwao
/ Borella, Christopher P.
/ Wu, Xinyuan
et al.
| 2005
2229
4-Phenoxypiperidines: Potent, Conformationally Restricted, Non-Imidazole Histamine H3 Antagonists
Dvorak, Curt A.
/ Apodaca, Richard
/ Barbier, Ann J.
et al.
| 2005
2239
Development of Low Molecular Weight HIV-1 Protease Dimerization Inhibitors
Hwang, You Seok
/ Chmielewski, Jean
et al.
| 2005
2243
Discovery of Novel Quinoline-Based Estrogen Receptor Ligands Using Peptide Interaction Profiling
Hoekstra, William J.
/ Patel, Hari S.
/ Liang, Xi
et al.
| 2005
2248
Design and Synthesis of N-[(4-Methoxyphenoxy)carbonyl]-N-[[4-[2-(5- methyl-2-phenyl-4-oxazolyl)ethoxy]phenyl]methyl]glycine [Muraglitazar/BMS-298585], a Novel Peroxisome Proliferator-Activated Receptor α/γ Dual Agonist with Efficacious Glucose and Lipid-Lowering Activities
Devasthale, Pratik V.
/ Chen, Sean
/ Jeon, Yoon
et al.
| 2005
2248
Design and Synthesis of N-((4-Methoxyphenoxy)carbonyl)-N-((4-(2-(5- methyl-2-phenyl-4-oxazolyl)ethoxy)phenyl)methyl)glycine (Muraglitazar-BMS-298585), a Novel Peroxisome Proliferator-Activated Receptor a-g Dual Agonist with Efficacious Glucose and Lipid-Lowering Activities
Devasthale, P.V.
et al.
| 2005
2248
Design and Synthesis of N-[(4-Methoxyphenoxy)carbonyl]-N-[[4-[2-(5-methyl-2-phenyl-4-oxazolyl)ethoxy]phenyl]methyl]glycine [Muraglitazar/BMS-298585], a Novel Peroxisome Proliferator-Activated Receptor alpha/gamma Dual Agonist with Efficacious Glucose and Lipid-Lowering Activities
Devasthale, P. V.
/ Chen, S.
/ Jeon, Y.
et al.
| 2005