Syntheses of a Selective Peroxisome Proliferator Activated Receptor Modulator and Practical New Preparations of 2-(4-Alkoxyphenyl)-ethylamines (English)
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In:
ORGANIC PROCESS RESEARCH AND DEVELOPMENT
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13
, 2
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280-284
;
2009
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ISSN:
- Article (Journal) / Print
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Title:Syntheses of a Selective Peroxisome Proliferator Activated Receptor Modulator and Practical New Preparations of 2-(4-Alkoxyphenyl)-ethylamines
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Contributors:Magnus, N.A. ( author ) / Astleford, B.A. ( author ) / Brennan, J. ( author ) / Stout, J.R. ( author ) / Tharp-Taylor, R.W. ( author )
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Published in:ORGANIC PROCESS RESEARCH AND DEVELOPMENT ; 13, 2 ; 280-284
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Publisher:
- New search for: ROYAL SOCIETY OF
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Place of publication:AMERICAN CHEMICAL SOCIETY &
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Publication date:2009-01-01
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Size:5 pages
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ISSN:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 547
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Classification:
DDC: 547 -
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Table of contents – Volume 13, Issue 2
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 127
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Special Issue Dedicated to Chris Schmid, Former Associate Editor of Organic Process Research and Development, Who Died in 2007Laird, Trevor et al. | 2009
- 128
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Christopher Randall Schmid 1959−2007| 2009
- 131
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The Role of New Technologies in Defining a Manufacturing Process for PPARα Agonist LY518674Argentine, Mark D. / Braden, Timothy M. / Czarnik, Jeffrey / Conder, Edward W. / Dunlap, Steven E. / Fennell, Jared W. / LaPack, Mark A. / Rothhaar, Roger R. / Scherer, R. Brian / Schmid, Christopher R. et al. | 2009
- 131
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The Role of New Technologies in Defining a Manufacturing Process for PPAR alpha Agonist LY518674Argentine, M.D. / Braden, T.M. / Czarnik, J. / Conder, E.W. / Dunlap, S.E. / Fennell, J.W. / LaPack, M.A. / Rothhaar, R.R. / Scherer, R.B. / Schmid, C.R. et al. | 2009
- 144
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Optimization of Organolithium ReactionsRathman, Terry ‘Li’ / Bailey, William F. et al. | 2009
- 152
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Improved Synthesis of 1-(Azidomethyl)-3,5-bis-(trifluoromethyl)benzene: Development of Batch and Microflow Azide ProcessesKopach, Michael E. / Murray, Michael M. / Braden, Timothy M. / Kobierski, Michael E. / Williams, Otis L. et al. | 2009
- 161
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Global Green Chemistry Metrics Analysis Algorithm and Spreadsheets: Evaluation of the Material Efficiency Performances of Synthesis Plans for Oseltamivir Phosphate (Tamiflu) as a Test CaseAndraos, John et al. | 2009
- 186
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Development of a Practical and Efficient Synthesis of CP-945,598-01, a CB1 Antagonist for the Treatment of ObesityRagan, John A. / Bourassa, Dennis E. / Blunt, Jon / Breen, Darragh / Busch, Frank R. / Cordi, Eric M. / Damon, David B. / Do, Nga / Engtrakul, Alanya / Lynch, Denis et al. | 2009
- 198
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Development of a Practical Synthesis of an Aminoindanol-Derived M1 AgonistHansen, Marvin M. / Borders, Sandra S. K. / Clayton, Marcella T. / Heath, Perry C. / Kolis, Stanley P. / Larsen, Samuel D. / Linder, Ryan J. / Reutzel-Edens, Susan M. / Smith, Justin C. / Tameze, Shella L. et al. | 2009
- 209
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Practical Synthesis of Chiral 2-Morpholine: (4-Benzylmorpholin-2-(S)-yl)-(tetrahydropyran-4-yl)methanone Mesylate, a Useful Pharmaceutical IntermediateKopach, Michael E. / Singh, Utpal K. / Kobierski, Michael E. / Trankle, William G. / Murray, Michael M. / Pietz, Mark A. / Forst, Mindy B. / Stephenson, Gregory A. / Mancuso, Vincent / Giard, Thierry et al. | 2009
- 225
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Impact of Entropic Effects in the Classical Resolution of a 2-ArylpyrrolidineBarnes, David M. / Barkalow, Jufang / Chen, Yong / Gupta, Ashok / Haight, Anthony R. / Hengeveld, John E. / Kerdesky, Francis A. J. / Kotecki, Brian J. / Macri, Bryan / Pal, Agnes et al. | 2009
- 230
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Development of a Practical Synthesis of a p38 MAP Kinase InhibitorThiel, Oliver R. / Achmatowicz, Michal / Bernard, Charles / Wheeler, Philip / Savarin, Cecile / Correll, Tiffany L. / Kasparian, Annie / Allgeier, Alan / Bartberger, Michael D. / Tan, Helming et al. | 2009
- 242
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Crystallization Process Development for a Stable Polymorph of Treprostinil Diethanolamine (UT-15C) by SeedingBatra, Hitesh / Penmasta, Raju / Phares, Kenneth / Staszewski, James / Tuladhar, Sudersan M. / Walsh, David A. et al. | 2009
- 250
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Second-Generation Process for the HCV Protease Inhibitor BILN 2061: A Greener Approach to Ru-Catalyzed Ring-Closing MetathesisFarina, Vittorio / Shu, Chutian / Zeng, Xingzhong / Wei, Xudong / Han, Zhengxu / Yee, Nathan K. / Senanayake, Chris H. et al. | 2009
- 255
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Development of an Acyl Sulfonamide Anti-Proliferative Agent, LY573636·NaYates, Matthew H. / Kallman, Neil J. / Ley, Christopher P. / Wei, Jeffrey N. et al. | 2009
- 263
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Preparation, Use, and Safety of O-MesitylenesulfonylhydroxylamineMendiola, Javier / Rincón, Juan A. / Mateos, Carlos / Soriano, José Francisco / de Frutos, Óscar / Niemeier, Jeffry K. / Davis, Edward M. et al. | 2009
- 268
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An Efficient Synthesis of a Multipotent Eicosanoid Pathway ModulatorYates, Matthew H. / Koenig, Thomas M. / Kallman, Neil J. / Ley, Christopher P. / Mitchell, David et al. | 2009
- 276
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Identifying Scale Sensitivity for API Crystallizations from Desupersaturation MeasurementsSingh, Utpal K. / Pietz, Mark A. / Kopach, Michael E. et al. | 2009
- 280
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Syntheses of a Selective Peroxisome Proliferator Activated Receptor Modulator and Practical New Preparations of 2-(4-Alkoxyphenyl)ethylaminesMagnus, Nicholas A. / Astleford, Bret A. / Brennan, John / Stout, James R. / Tharp-Taylor, Roger W. et al. | 2009
- 285
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Approaches to Assessment, Testing Decisions, and Analytical Determination of Genotoxic Impurities in Drug SubstancesPierson, Duane A. / Olsen, Bernard A. / Robbins, David K. / DeVries, Keith M. / Varie, David L. et al. | 2009
- 292
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Enzymatic Resolution of N-Substituted- beta -prolinesMendiola, J. / Garcia-Cerrada, S. / de Frutos, O. / de la Puente, M.L. / Gu, R.L. / Khau, V.V. et al. | 2009
- 292
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Enzymatic Resolution of N-Substituted-β-prolinesMendiola, Javier / García-Cerrada, Susana / de Frutos, Óscar / de la Puente, María Luz / Gu, Rui Lin / Khau, Vien V. et al. | 2009
- 297
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Process Development for Sodelglitazar: A PPAR PanagonistBrown, Andrew D. / Davis, Roman D. / Fitzgerald, Russ N. / Glover, Bobby N. / Harvey, Kim A. / Jones, Lynda A. / Liu, Bing / Patterson, Daniel E. / Sharp, Matthew J. et al. | 2009
- 303
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Process Development and Scale-Up of a PPARγ Agonist: Selection of the Manufacture RouteBullock, Kae M. / Burton, Delphilia / Corona, John / Diederich, Ann / Glover, Bobby / Harvey, Kim / Mitchell, Mark B. / Trone, Mark D. / Yule, Robert / Zhang, Yong et al. | 2009
- 303
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Process Development and Scale-Up of a PPAR gamma Agonist: Selection of the Manufacture RouteBullock, K.M. / Burton, D. / Corona, J. / Diederich, A. / Glover, B. / Harvey, K. / Mitchell, M.B. / Trone, M.D. / Yule, R. / Zhang, Y. et al. | 2009
- 310
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A Practical Method for Functionalized Peptide or Amide Bond Formation in Aqueous−Ethanol Media with EDC as ActivatorPu, Yangwei John / Vaid, Radhe K. / Boini, Sathish K. / Towsley, Robert W. / Doecke, Christopher W. / Mitchell, David et al. | 2009
- 315
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Development of an Efficient Palladium-Catalyzed Intramolecular Carbometalation Reaction for the Synthesis of a Dibenzoxapine Containing Tetra-substituted Exocyclic AlkeneRichey, Rachel N. / Yu, Hannah et al. | 2009
- 321
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The Newman−Kwart Rearrangement Revisited: Continuous Process under Supercritical ConditionsTilstam, Ulf / Defrance, Thierry / Giard, Thierry / Johnson, Martin D. et al. | 2009
- 324
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Preparation of a Corticotropin-Releasing Factor Antagonist by Nucleophilic Aromatic Substitution and Copper-Mediated Ether FormationCaron, Stéphane / Do, Nga M. / Sieser, Janice E. / Whritenour, David C. / Hill, Paul D. et al. | 2009
- 331
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A Scalable Synthesis of the INOS Inhibitor PHA-399733Wuts, Peter G. M. / Ashford, Scott W. / Conway, Brian / Havens, Jeffrey L. / Taylor, Bill / Hritzko, Ben / Xiang, Yanqiao / Zakarias, Peter S. et al. | 2009
- 336
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Synthesis of 2-Methyl-2,5-diazabicyclo[2.2.1]heptane, Side Chain to DanofloxacinBraish, Tamim F. et al. | 2009
- 336
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Synthesis of 2-Methyl-2,5-diazabicyclo[2.2.1]heptane, Side Chain to Danofloxacin(1)Braish, Tamim F. et al. | 2009
- 341
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Microwave-Irradiated Synthesis of Nitrophen Using PEG 400 as Phase Transfer Catalyst and SolventYadav, Ganapati D. / Motirale, Bhavana G. et al. | 2009
- 349
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A Practical Palladium-Catalyzed Telomerization for the Synthesis of Functionalized AlcoholsJackstell, Ralf / Grotevendt, Anne / Andreu, Mario Gomez / Beller, Matthias et al. | 2009
- 354
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Heavy-Metal-Free Reduction Methodology for Large-Scale Synthesis Applicable to Heterocyclic and ArylhydrazinesNorris, Timothy / Bezze, Chiara / Franz, Samuela Zambelli / Stivanello, Mariano et al. | 2009
- 358
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Large-Scale Preparation of (+)-p-Menth-2-ene-1,8-diol, a Key Intermediate in the Synthesis of Delta -9-TetrahydrocannabinolCabaj, J.E. / Lukesh, J.M. / Pariza, R.J. / Zizelman, P.M. et al. | 2009
- 358
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Large-Scale Preparation of (+)-p-Menth-2-ene-1,8-diol, a Key Intermediate in the Synthesis of Δ-9-TetrahydrocannabinolCabaj, John E. / Lukesh, Julie M. / Pariza, Richard J. / Zizelman, Paul M. et al. | 2009
- 362
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Good Manufacturing Practices for Pharmaceuticals (Drugs and the Pharmaceutical Sciences, 6th ed., Vol. 169)Robinson, D. et al. | 2009
- 362
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Book Review of Good Manufacturing Practices for PharmaceuticalsRobinson, Derek et al. | 2009