Development and evaluation of a 68Ga labeled pamoic acid derivative for in vivo visualization of necrosis using positron emission tomography (English)
- New search for: Prinsen, K.
- New search for: Li, J.
- New search for: Vanbilloen, H.
- New search for: Vermaelen, P.
- New search for: Devos, E.
- New search for: Mortelmans, L.
- New search for: Bormans, G.
- New search for: Ni, Y.
- New search for: Verbruggen, A.
- New search for: Prinsen, K.
- New search for: Li, J.
- New search for: Vanbilloen, H.
- New search for: Vermaelen, P.
- New search for: Devos, E.
- New search for: Mortelmans, L.
- New search for: Bormans, G.
- New search for: Ni, Y.
- New search for: Verbruggen, A.
In:
BIOORGANIC AND MEDICINAL CHEMISTRY
;
18
, 14
;
5274-5281
;
2010
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ISSN:
- Article (Journal) / Print
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Title:Development and evaluation of a 68Ga labeled pamoic acid derivative for in vivo visualization of necrosis using positron emission tomography
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Contributors:Prinsen, K. ( author ) / Li, J. ( author ) / Vanbilloen, H. ( author ) / Vermaelen, P. ( author ) / Devos, E. ( author ) / Mortelmans, L. ( author ) / Bormans, G. ( author ) / Ni, Y. ( author ) / Verbruggen, A. ( author )
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Published in:BIOORGANIC AND MEDICINAL CHEMISTRY ; 18, 14 ; 5274-5281
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Publisher:
- New search for: Elsevier Science B.V., Amsterdam.
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Publication date:2010-01-01
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Size:8 pages
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ISSN:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 615.19
- Further information on Dewey Decimal Classification
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Classification:
DDC: 615.19 -
Source:
© Metadata Copyright the British Library Board and other contributors. All rights reserved.
Table of contents – Volume 18, Issue 14
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 4855
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Graphical contents list| 2010
- 4872
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Publisher’s Note| 2010
- 4873
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Coumarinyl-substituted sulfonamides strongly inhibit several human carbonic anhydrase isoforms: solution and crystallographic investigationsWagner, Jason / Avvaru, Balendu Sankara / Robbins, Arthur H. / Scozzafava, Andrea / Supuran, Claudiu T. / McKenna, Robert et al. | 2010
- 4879
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Antineoplastic agents 582. Part 1: Isolation and structure of a cyclobutane-type sesquiterpene cancer cell growth inhibitor from Coprinus cinereus (Coprinaceae)Pettit, George R. / Meng, Yanhui / Pettit, Robin K. / Herald, Delbert L. / Hogan, Fiona / Cichacz, Zbigniew A. et al. | 2010
- 4884
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Target-specific control of lymphoid-specific protein tyrosine phosphatase (Lyp) activityWalton, Zandra E. / Bishop, Anthony C. et al. | 2010
- 4892
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Structural characteristics of green tea catechins for formation of protein carbonyl in human serum albuminIshii, Takeshi / Mori, Taiki / Ichikawa, Tatsuya / Kaku, Maiko / Kusaka, Koji / Uekusa, Yoshinori / Akagawa, Mitsugu / Aihara, Yoshiyuki / Furuta, Takumi / Wakimoto, Toshiyuki et al. | 2010
- 4897
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Syntheses and herbicidal activity of new triazolopyrimidine-2-sulfonamides as acetohydroxyacid synthase inhibitorChen, Chao-Nan / Chen, Qiong / Liu, Yu-Chao / Zhu, Xiao-Lei / Niu, Cong-Wei / Xi, Zhen / Yang, Guang-Fu et al. | 2010
- 4905
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2-Phenyl-1-[4-(2-piperidine-1-yl-ethoxy)benzyl]-1H-benzimidazoles as ligands for the estrogen receptor: Synthesis and pharmacological evaluationDettmann, Sandra / Szymanowitz, Katrin / Wellner, Anja / Schiedel, Anke / Müller, Christa E. / Gust, Ronald et al. | 2010
- 4917
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Development of chemical probes: Toward the mode of action of a methylene-linked di(aryl acetate) E1Smith, Mark E.B. / Gunn, Richard M. / Rosivatz, Evelyn / Mak, Lok H. / Woscholski, Rüdiger / Hailes, Helen C. et al. | 2010
- 4928
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Constrained peptidomimetics as antiplasmodial falcipain-2 inhibitorsBova, Floriana / Ettari, Roberta / Micale, Nicola / Carnovale, Caterina / Schirmeister, Tanja / Gelhaus, Christoph / Leippe, Matthias / Grasso, Silvana / Zappalà, Maria et al. | 2010
- 4939
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Synthesis and CYP24A1 inhibitory activity of N-(2-(1H-imidazol-1-yl)-2-phenylethyl)arylamidesAboraia, Ahmed S. / Yee, Sook Wah / Gomaa, Mohamed Sayed / Shah, Nikhil / Robotham, Anna C. / Makowski, Bart / Prosser, David / Brancale, Andrea / Jones, Glenville / Simons, Claire et al. | 2010
- 4947
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Callyaerins A–F and H, new cytotoxic cyclic peptides from the Indonesian marine sponge Callyspongia aerizusaIbrahim, Sabrin R.M. / Min, Cho Cho / Teuscher, Franka / Ebel, Rainer / Kakoschke, Christel / Lin, Wenhan / Wray, Victor / Edrada-Ebel, RuAngelie / Proksch, Peter et al. | 2010
- 4957
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Identification and evaluation of apoptotic compounds from Garcinia paucinervisGao, Xue-Mei / Yu, Ting / Lai, Fanny Shuk Fan / Zhou, Yan / Liu, Xin / Qiao, Chun-Feng / Song, Jing-Zheng / Chen, Shi-Lin / Luo, Kathy Qian / Xu, Hong-Xi et al. | 2010
- 4965
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Synthesis of novel pyrazolic analogues of chalcones and their 3-aryl-4-(3-aryl-4,5-dihydro-1H-pyrazol-5-yl)-1-phenyl-1H-pyrazole derivatives as potential antitumor agentsInsuasty, Braulio / Tigreros, Alexis / Orozco, Fabián / Quiroga, Jairo / Abonía, Rodrigo / Nogueras, Manuel / Sanchez, Adolfo / Cobo, Justo et al. | 2010
- 4975
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Evaluation of N-substitution in 6,7-benzomorphan compoundsPasquinucci, Lorella / Prezzavento, Orazio / Marrazzo, Agostino / Amata, Emanuele / Ronsisvalle, Simone / Georgoussi, Zafiroula / Fourla, Danai-Dionysia / Scoto, Giovanna M. / Parenti, Carmela / Aricò, Giuseppina et al. | 2010
- 4983
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Novel structure–activity relationships and selectivity profiling of cage dimeric 1,4-dihydropyridines as multidrug resistance (MDR) modulatorsCoburger, Claudius / Wollmann, Jörg / Krug, Martin / Baumert, Christiane / Seifert, Marianne / Molnár, Joséf / Lage, Hermann / Hilgeroth, Andreas et al. | 2010
- 4991
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Synthesis, molecular modeling, and biological evaluation of cinnamic acid metronidazole ester derivatives as novel anticancer agentsQian, Yong / Zhang, Hong-Jia / Zhang, Hao / Xu, Chen / Zhao, Jing / Zhu, Hai-Liang et al. | 2010
- 4997
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Hypoxic selectivity and solubility—investigating the properties of A-ring substituted nitro seco-1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-ones (nitroCBIs) as hypoxia-activated prodrugs for antitumor therapyTercel, Moana / Yang, Shangjin / Atwell, Graham J. / Smith, Eileen / Gu, Yongchuan / Anderson, Robert F. / Denny, William A. / Wilson, William R. / Pruijn, Frederik B. et al. | 2010
- 5007
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Synthesis and pharmacological evaluation of pyrazine N-acylhydrazone derivatives designed as novel analgesic and anti-inflammatory drug candidatesSilva, Yolanda Karla Cupertino da / Augusto, Cristina Villarinho / Barbosa, Maria Letícia de Castro / Melo, Gabriela Muniz de Albuquerque / Queiroz, Aline Cavalcanti de / Dias, Thays de Lima Matos Freire / Júnior, Walfrido Bispo / Barreiro, Eliezer J. / Lima, Lídia Moreira / Alexandre-Moreira, Magna Suzana et al. | 2010
- 5016
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A novel achiral seco-cyclopropylpyrido[e]indolone (CPyI) analog of CC-1065 and the duocarmycins: Synthesis, DNA interactions, in vivo anticancer and anti-parasitic evaluationChavda, Sameer / Babu, Balaji / Yanow, Stephanie K. / Jardim, Armando / Spithill, Terry W. / Kiakos, Konstantinos / Kluza, Jerome / Hartley, John A. / Lee, Moses et al. | 2010
- 5025
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Spectroscopic characterization of the inclusion complexes of luteolin with native and derivatized b-cyclodextrinJullian, C. / Cifuentes, C. / Alfaro, M. / Miranda, S. / Barriga, G. / Olea-Azar, C. et al. | 2010
- 5025
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Spectroscopic characterization of the inclusion complexes of luteolin with native and derivatized β-cyclodextrinJullian, Carolina / Cifuentes, Constanza / Alfaro, Muriel / Miranda, Sebastián / Barriga, Germán / Olea-Azar, Claudio et al. | 2010
- 5032
-
Synthesis of a series of caffeic acid phenethyl amide (CAPA) fluorinated derivatives: Comparison of cytoprotective effects to caffeic acid phenethyl ester (CAPE)Yang, John / Marriner, Gwendolyn A. / Wang, Xinyu / Bowman, Phillip D. / Kerwin, Sean M. / Stavchansky, Salomon et al. | 2010
- 5039
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Hybrid diarylbenzopyrimidine non-nucleoside reverse transcriptase inhibitors as promising new leads for improved anti-HIV-1 chemotherapyZeng, Zhao-Sen / He, Qiu-Qin / Liang, Yong-Hong / Feng, Xiao-Qing / Chen, Fen-Er / Clercq, Erik De / Balzarini, Jan / Pannecouque, Christophe et al. | 2010
- 5048
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Design and synthesis of novel benzimidazole derivatives as inhibitors of hepatitis B virusLuo, Yu / Yao, Jia-Ping / Yang, Li / Feng, Chun-Lan / Tang, Wei / Wang, Gui-Feng / Zuo, Jian-Pin / Lu, Wei et al. | 2010
- 5056
-
Virtual fragment screening for novel inhibitors of 6-phosphogluconate dehydrogenaseRuda, Gian Filippo / Campbell, Gordon / Alibu, Vincent P. / Barrett, Michael P. / Brenk, Ruth / Gilbert, Ian H. et al. | 2010
- 5063
-
Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitorsChimenti, Franco / Secci, Daniela / Bolasco, Adriana / Chimenti, Paola / Granese, Arianna / Carradori, Simone / Maccioni, Elias / Cardia, M. Cristina / Yáñez, Matilde / Orallo, Francisco et al. | 2010
- 5071
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Morphinans and isoquinolines: Acetylcholinesterase inhibition, pharmacophore modeling, and interaction with opioid receptorsSchuster, Daniela / Spetea, Mariana / Music, Melisa / Rief, Silvia / Fink, Monika / Kirchmair, Johannes / Schütz, Johannes / Wolber, Gerhard / Langer, Thierry / Stuppner, Hermann et al. | 2010
- 5081
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Pteridine–sulfonamide conjugates as dual inhibitors of carbonic anhydrases and dihydrofolate reductase with potential antitumor activityMarques, Sérgio M. / Enyedy, Éva A. / Supuran, Claudiu T. / Krupenko, Natalia I. / Krupenko, Sergey A. / Amélia Santos, M. et al. | 2010
- 5090
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Synthesis of 5-arylidene-2-amino-4-azolones and evaluation of their anticancer activitySubtel’na, Ivanna / Atamanyuk, Dmytro / Szymańska, Ewa / Kieć-Kononowicz, Katarzyna / Zimenkovsky, Borys / Vasylenko, Olexandr / Gzella, Andrzej / Lesyk, Roman et al. | 2010
- 5103
-
Tryptamine-derived alkaloids from Annonaceae exerting neurotrophin-like properties on primary dopaminergic neuronsSchmidt, Fanny / Douaron, Gael Le / Champy, Pierre / Amar, Majid / Séon-Méniel, Blandine / Raisman-Vozari, Rita / Figadère, Bruno et al. | 2010
- 5114
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Substituted 2-(3′,4′,5′-trimethoxybenzoyl)-benzo[b]thiophene derivatives as potent tubulin polymerization inhibitorsRomagnoli, Romeo / Baraldi, Pier Giovanni / Carrion, Maria Dora / Cruz-Lopez, Olga / Tolomeo, Manlio / Grimaudo, Stefania / Cristina, Antonietta Di / Pipitone, Maria Rosaria / Balzarini, Jan / Brancale, Andrea et al. | 2010
- 5114
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Substituted 2-(3prime,4prime,5prime-trimethoxybenzoyl)-benzo[b]thiophene derivatives as potent tubulin polymerization inhibitorsRomagnoli, R. / Baraldi, P. G. / Carrion, M. D. / Cruz-Lopez, O. / Tolomeo, M. / Grimaudo, S. / Cristina, A. D. / Pipitone, M. R. / Balzarini, J. / Brancale, A. et al. | 2010
- 5123
-
STD-NMR studies of two acceptor substrates of GlfT2, a galactofuranosyltransferase from Mycobacterium tuberculosis: Epitope mapping studiesSzczepina, Monica G. / Zheng, Ruixiang B. / Completo, Gladys C. / Lowary, Todd L. / Pinto, B. Mario et al. | 2010
- 5129
-
Studies on the anti-hepatitis C virus activity of newly synthesized tropolone derivatives: Identification of NS3 helicase inhibitors that specifically inhibit subgenomic HCV replicationNajda-Bernatowicz, Andżelika / Krawczyk, Mariusz / Stankiewicz-Drogoń, Anna / Bretner, Maria / Boguszewska-Chachulska, Anna M. et al. | 2010
- 5137
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Novel antimicrobial peptides that exhibit activity against select agents and other drug resistant bacteriaVenugopal, Divakaramenon / Klapper, David / Srouji, Antoine H. / Bhonsle, Jayendra B. / Borschel, Richard / Mueller, Allen / Russell, Amanda L. / Williams, Brittany C. / Hicks, Rickey P. et al. | 2010
- 5148
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Identification of novel bacterial histidine biosynthesis inhibitors using docking, ensemble rescoring, and whole-cell assaysHenriksen, S.T. / Liu, J. / Estiu, G. / Oltvai, Z.N. / Wiest, O. et al. | 2010
- 5157
-
2-Acylamino-4,6-diphenylpyridine derivatives as novel GPR54 antagonists with good brain exposure and in vivo efficacy for plasma LH level in male ratsKobayashi, Toshitake / Sasaki, Satoshi / Tomita, Naoki / Fukui, Seiji / Nakayama, Masaharu / Kiba, Atsushi / Kusaka, Masami / Matsumoto, Shin-ichi / Yamaguchi, Masashi / Itoh, Fumio et al. | 2010
- 5172
-
Synthesis and antiproliferative evaluation of certain iminonaphtho[2,3-b]furan derivativesTseng, Chih-Hua / Chen, Yeh-Long / Yang, Sheng-Huei / Peng, Shin-I / Cheng, Chih-Mei / Han, Chein-Hwa / Lin, Shinne-Ren / Tzeng, Cherng-Chyi et al. | 2010
- 5183
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Synthesis and biological evaluation of cytotoxic activity of novel anthracene l-rhamnopyranosidesSong, Gaopeng / Liu, Hongchun / Zhang, Wei / Geng, Meiyu / Li, Yingxia et al. | 2010
- 5194
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New 2-arylnaphthalenediols and triol inhibitors of HIV-1 integrase—Discovery of a new polyhydroxylated antiviral agentMaurin, Cédric / Lion, Cédric / Bailly, Fabrice / Touati, Nadia / Vezin, Hervé / Mbemba, Gladys / Mouscadet, Jean François / Debyser, Zeger / Witvrouw, Myriam / Cotelle, Philippe et al. | 2010
- 5202
-
Synthesis and biodistribution of [11C]A-836339, a new potential radioligand for PET imaging of cannabinoid type 2 receptors (CB2)Horti, Andrew G. / Gao, Yongjun / Ravert, Hayden T. / Finley, Paige / Valentine, Heather / Wong, Dean F. / Endres, Christopher J. / Savonenko, Alena V. / Dannals, Robert F. et al. | 2010
- 5208
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Discovery of orally available spirodiketopiperazine-based CCR5 antagonistsNishizawa, Rena / Nishiyama, Toshihiko / Hisaichi, Katsuya / Hirai, Keisuke / Habashita, Hiromu / Takaoka, Yoshikazu / Tada, Hideaki / Sagawa, Kenji / Shibayama, Shiro / Maeda, Kenji et al. | 2010
- 5224
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Structure–activity relationship of brominated 3-alkyl-5-methylene-2(5H)-furanones and alkylmaleic anhydrides as inhibitors of Salmonella biofilm formation and quorum sensing regulated bioluminescence in Vibrio harveyiSteenackers, Hans P. / Levin, Jeremy / Janssens, Joost C. / Weerdt, Ami De / Balzarini, Jan / Vanderleyden, Jos / De Vos, Dirk E. / De Keersmaecker, Sigrid C. et al. | 2010
- 5234
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Characterization of multivalent lactose quantum dots and its application in carbohydrate–protein interactions study and cell imagingYang, Yang / Yu, Min / Yan, Ting-Ting / Zhao, Zhi-Hui / Sha, Yin-Lin / Li, Zhong-Jun et al. | 2010
- 5241
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(−)-N-Formylanonaine from Michelia alba as a human tyrosinase inhibitor and antioxidantWang, Hui-Min / Chen, Chung-Yi / Chen, Chun-Yen / Ho, Mei-Ling / Chou, Yi-Ting / Chang, Hou-Chien / Lee, Chih-Hung / Wang, Chau-Zen / Chu, I-Ming et al. | 2010
- 5248
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Cell-penetration by Co(III)cyclen-based peptide-cleaving catalysts selective for pathogenic proteins of amyloidosesChei, Woo Suk / Lee, Joo-Won / Kim, Jae Bum / Suh, Junghun et al. | 2010
- 5254
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New antimalarials with a triterpenic scaffold from Momordica balsaminaRamalhete, Cátia / Lopes, Dinora / Mulhovo, Silva / Molnár, Joseph / Rosário, Virgílio E. / Ferreira, Maria-José U. et al. | 2010
- 5261
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Design, synthesis and evaluation of 2-amino-4-m-bromoanilino-6-arylmethyl-7H-pyrrolo[2,3-d]pyrimidines as tyrosine kinase inhibitors and antiangiogenic agentsGangjee, Aleem et al. | 2010
- 5261
-
Design, synthesis and evaluation of 2-amino-4-m-bromoanilino-6-arylmethyl-7H-pyrrolo[2,3-d]pyrimidines as tyrosine kinase inhibitors and antiangiogenic agents1Gangjee, Aleem / Zhao, Ying / Raghavan, Sudhir / Ihnat, Michael A. / Disch, Bryan C. et al. | 2010
- 5274
-
Development and evaluation of a 68Ga labeled pamoic acid derivative for in vivo visualization of necrosis using positron emission tomographyPrinsen, Kristof / Li, Junjie / Vanbilloen, Hubert / Vermaelen, Peter / Devos, Ellen / Mortelmans, Luc / Bormans, Guy / Ni, Yicheng / Verbruggen, Alfons et al. | 2010
- 5282
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Synthesis and biological study of 3-(phenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidines as potent and selective serotonin 5-HT6 receptor antagonistsIvachtchenko, Alexandre V. / Golovina, Elena S. / Kadieva, Madina G. / Koryakova, Angela G. / Kovalenko, Sergiy M. / Mitkin, Oleg D. / Okun, Ilya M. / Ravnyeyko, Irina M. / Tkachenko, Sergey E. / Zaremba, Oleg V. et al. | 2010
- 5291
-
Synthesis and characterization of selective dopamine D2 receptor antagonists. 2. Azaindole, benzofuran, and benzothiophene analogs of L-741,626Vangveravong, Suwanna / Taylor, Michelle / Xu, Jinbin / Cui, Jinquan / Calvin, Wesley / Babic, Sonja / Luedtke, Robert R. / Mach, Robert H. et al. | 2010
- 5301
-
Synthesis and cytotoxic activity of a new potential DNA bisintercalator: 1,4-Bis{3-[N-(4-chlorobenzo[g]phthalazin-1-yl)aminopropyl]}piperazineGalisteo, Juan / Navarro, Pilar / Campayo, Lucrecia / Yunta, María J.R. / Gómez-Contreras, Fernando / Villa-Pulgarin, Janny A. / Sierra, Beatriz G. / Mollinedo, Faustino / Gonzalez, Jorge / Garcia-España, Enrique et al. | 2010
- 5310
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Terpioside B, a difucosyl GSL from the marine sponge Terpios sp. is a potent inhibitor of NO releaseCostantino, Valeria / Fattorusso, Ernesto / Mangoni, Alfonso / Teta, Roberta / Panza, Elisabetta / Ianaro, Angela et al. | 2010
- 5316
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Novel anti-viability ceramide analogs: Design, synthesis, and structure–activity relationship studies of substituted (S)-2-(benzylideneamino)-3-hydroxy-N-tetradecylpropanamidesLiu, Jiawang / Antoon, James W. / Ponnapakkam, Adharsh / Beckman, Barbara S. / Foroozesh, Maryam et al. | 2010
- 5323
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Development of tryptase inhibitors derived from thalidomideTetsuhashi, Masashi / Ishikawa, Minoru / Hashimoto, Mariko / Hashimoto, Yuichi / Aoyama, Hiroshi et al. | 2010
- 5339
-
Synthesis of 5-deoxy-β-d-galactofuranosides as tools for the characterization of β-d-galactofuranosidasesBordoni, Andrea / de Lederkremer, Rosa M. / Marino, Carla et al. | 2010
- 5339
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Synthesis of 5-deoxy-b-d-galactofuranosides as tools for the characterization of b-d-galactofuranosidasesBordoni, A. / de Lederkremer, R. M. / Marino, C. et al. | 2010
- 5346
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Discovery of potent and orally active tricyclic-based FBPase inhibitorsTsukada, Tomoharu / Kanno, Osamu / Yamane, Takahiro / Tanaka, Jun / Yoshida, Taishi / Okuno, Akira / Shiiki, Takeshi / Takahashi, Mizuki / Nishi, Takahide et al. | 2010
- 5352
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Design, synthesis, and biological evaluation of resveratrol analogues as aromatase and quinone reductase 2 inhibitors for chemoprevention of cancerSun, Bin / Hoshino, Juma / Jermihov, Katie / Marler, Laura / Pezzuto, John M. / Mesecar, Andrew D. / Cushman, Mark et al. | 2010
- 5367
-
1H-1,2,3-Triazol-1-yl thiodigalactoside derivatives as high affinity galectin-3 inhibitorsSalameh, Bader A. / Cumpstey, Ian / Sundin, Anders / Leffler, Hakon / Nilsson, Ulf J. et al. | 2010
- 5379
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Anti-influenza activity of phenethylphenylphthalimide analogs derived from thalidomideIwai, Yuma / Takahashi, Hitoshi / Hatakeyama, Dai / Motoshima, Kazunori / Ishikawa, Minoru / Sugita, Kazuyuki / Hashimoto, Yuichi / Harada, Yuichi / Itamura, Shigeyuki / Odagiri, Takato et al. | 2010
- 5391
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Identification of chalcones as in vivo liver monofunctional phase II enzymes inducersCabrera, Mauricio / Lavaggi, María Laura / Croce, Fiorela / Celano, Laura / Thomson, Leonor / Fernández, Marcelo / Pintos, Cristina / Raymondo, Stella / Bollati, Mariela / Monge, Antonio et al. | 2010
- 5400
-
Development of a new radioligand for cholecystokinin receptor subtype 2 scintigraphy: From molecular modeling to in vivo evaluationBrillouet, Séverine / Dorbes, Sandra / Courbon, Frédéric / Picard, Claude / Delord, Jean Pierre / Benoist, Eric / Poirot, Marc / Mestre-Voegtlé, Béatrice / Silvente-Poirot, Sandrine et al. | 2010
- 5413
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Improved P2 phenylglycine-based hepatitis C virus NS3 protease inhibitors with alkenylic prime-side substituentsLampa, Anna / Ehrenberg, Angelica E. / Gustafsson, Sofia S. / Vema, Aparna / Åkerblom, Eva / Lindeberg, Gunnar / Karlén, Anders / Danielson, U. Helena / Sandström, Anja et al. | 2010
- 5425
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An integrative in silico methodology for the identification of modulators of macrophage migration inhibitory factor (MIF) tautomerase activityEl Turk, Farah / Fauvet, Bruno / Ouertatani-Sakouhi, Hajer / Lugari, Adrien / Betzi, Stephane / Roche, Philippe / Morelli, Xavier / Lashuel, Hilal A. et al. | 2010
- 5441
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Synthesis and structure–activity relationships of N-aryl-piperidine derivatives as potent (partial) agonists for human histamine H3 receptorIshikawa, Makoto / Furuuchi, Takeshi / Yamauchi, Miki / Yokoyama, Fumikazu / Kakui, Nobukazu / Sato, Yasuo et al. | 2010
- 5449
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Identification of novel inhibitors for a low molecular weight protein tyrosine phosphatase via virtual screeningHoman, Kristoff T. / Balasubramaniam, Deepa / Zabell, Adam P.R. / Wiest, Olaf / Helquist, Paul / Stauffacher, Cynthia V. et al. | 2010
- IFC
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Editorial board| 2010