1,2,3-Triazole-, arylamino- and thio-substituted 1,4-naphthoquinones: Potent antitumor activity, electrochemical aspects, and bioisosteric replacement of C-ring-modified lapachones (English)
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- New search for: de Melo, I. M. M.
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In:
BIOORGANIC AND MEDICINAL CHEMISTRY
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22
, 5
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1608-1619
;
2014
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ISSN:
- Article (Journal) / Print
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Title:1,2,3-Triazole-, arylamino- and thio-substituted 1,4-naphthoquinones: Potent antitumor activity, electrochemical aspects, and bioisosteric replacement of C-ring-modified lapachones
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Contributors:da Cruz, E. H. G. ( author ) / Hussene, C. M. B. ( author ) / Dias, G. G. ( author ) / Diogo, E. B. T. ( author ) / de Melo, I. M. M. ( author ) / Rodrigues, B. L. ( author ) / da Silva, M. G. ( author ) / Valenca, W. O. ( author ) / Camara, C. A. ( author ) / de Oliveira, R. N. ( author )
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Published in:BIOORGANIC AND MEDICINAL CHEMISTRY ; 22, 5 ; 1608-1619
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Publisher:
- New search for: Elsevier Science B.V., Amsterdam.
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Publication date:2014-01-01
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Size:12 pages
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ISSN:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 615.19
- Further information on Dewey Decimal Classification
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Classification:
DDC: 615.19 -
Source:
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Table of contents – Volume 22, Issue 5
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1507
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Graphical contents list| 2014
- 1515
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Synthesis, nitric oxide release, and α-glucosidase inhibition of nitric oxide donating apigenin and chrysin derivativesWang, Qi-Qin / Cheng, Ning / Yi, Wen-Bing / Peng, Sheng-Ming / Zou, Xiao-Qing et al. | 2014
- 1515
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Synthesis, nitric oxide release, and @a-glucosidase inhibition of nitric oxide donating apigenin and chrysin derivativesWang, Q. Q. / Cheng, N. / Yi, W. B. / Peng, S. M. / Zou, X. Q. et al. | 2014
- 1522
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Synthesis of 6-tetrazolyl-substituted sulfocoumarins acting as highly potent and selective inhibitors of the tumor-associated carbonic anhydrase isoforms IX and XIIGrandane, Aiga / Tanc, Muhammet / Zalubovskis, Raivis / Supuran, Claudiu T. et al. | 2014
- 1529
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Design, synthesis and preliminary bioactivity studies of 1,2-dihydrobenzo[d]isothiazol-3-one-1,1-dioxide hydroxamic acid derivatives as novel histone deacetylase inhibitorsHan, Leiqiang / Wang, Lei / Hou, Xuben / Fu, Huansheng / Song, Weiguo / Tang, Weiping / Fang, Hao et al. | 2014
- 1539
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Synthesis, selective cytotoxicities and probable mechanism of action of 7-methoxy-3-arylflavone-8-acetic acidsZhou, Zhong-Zhen / Gu, Chun-Ping / Deng, Yan-Hong / Yan, Guang-Hua / Li, Xiao-Fang / Yu, Le / Chen, Wen-Hua / Liu, Shu-Wen et al. | 2014
- 1548
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Structure-based optimization of cyclopropyl urea derivatives as potent soluble epoxide hydrolase inhibitors for potential decrease of renal injury without hypotensive actionTakai, Kentaro / Nakajima, Tomoko / Takanashi, Yosuke / Sone, Toshihiko / Nariai, Tetsuro / Chiyo, Naoki / Nakatani, Shogo / Ishikawa, Chihiro / Yamaguchi, Nobuyuki / Fujita, Katsuya et al. | 2014
- 1558
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Synthesis of 2,6-disubstituted benzylamine derivatives as reversible selective inhibitors of copper amine oxidasesLucchesini, Francesco / Pocci, Marco / Alfei, Silvana / Bertini, Vincenzo / Buffoni, Franca et al. | 2014
- 1568
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Antiprotozoan lead discovery by aligning dry and wet screening: Prediction, synthesis, and biological assay of novel quinoxalinonesMartins Alho, Miriam A. / Marrero-Ponce, Yovani / Barigye, Stephen J. / Meneses-Marcel, Alfredo / Machado Tugores, Yanetsy / Montero-Torres, Alina / Gómez-Barrio, Alicia / Nogal, Juan J. / García-Sánchez, Rory N. / Vega, María Celeste et al. | 2014
- 1586
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Carbonic anhydrase inhibitors: Synthesis and inhibition of the human carbonic anhydrase isoforms I, II, IX and XII with benzene sulfonamides incorporating 4- and 3-nitrophthalimide moietiesSethi, Kalyan K. / Verma, Saurabh M. / Tanç, Muhammet / Purper, Gaultier / Calafato, Gaetan / Carta, Fabrizio / Supuran, Claudiu T. et al. | 2014
- 1596
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Discovery and SAR study of hydroxyacetophenone derivatives as potent, non-steroidal farnesoid X receptor (FXR) antagonistsLiu, Peng / Xu, Xing / Chen, Lili / Ma, Lei / Shen, Xu / Hu, Lihong et al. | 2014
- 1608
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1,2,3-Triazole-, arylamino- and thio-substituted 1,4-naphthoquinones: Potent antitumor activity, electrochemical aspects, and bioisosteric replacement of C-ring-modified lapachonesda Cruz, Eduardo H.G. / Hussene, Caio M.B. / Dias, Gleiston G. / Diogo, Emilay B.T. / de Melo, Isadora M.M. / Rodrigues, Bernardo L. / da Silva, Mauro G. / Valença, Wagner O. / Camara, Celso A. / de Oliveira, Ronaldo N. et al. | 2014
- 1620
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A comparative study of ATP analogs for phosphorylation-dependent kinase–substrate crosslinkingGarre, Satish / Senevirathne, Chamara / Pflum, Mary Kay H. et al. | 2014
- 1626
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2-Acylamino-5-nitro-1,3-thiazoles: Preparation and in vitro bioevaluation against four neglected protozoan parasitesNava-Zuazo, Carlos / Chávez-Silva, Fabiola / Moo-Puc, Rosa / Chan-Bacab, Manuel Jesús / Ortega-Morales, Benjamín Otto / Moreno-Díaz, Hermenegilda / Díaz-Coutiño, Daniel / Hernández-Núñez, Emanuel / Navarrete-Vázquez, Gabriel et al. | 2014
- 1634
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2,6-Diaminopurine nucleoside derivative of 9-ethyloxy-2-oxo-1,3-diazaphenoxazine (2-amino-Adap) for recognition of 8-oxo-dG in DNATaniguchi, Yosuke / Fukabori, Keitaro / Kikukawa, Yoshiya / Koga, Yohei / Sasaki, Shigeki et al. | 2014
- 1642
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Lead modification: Amino acid appended indoles as highly effective 5-LOX inhibitorsPrasher, Parteek / Pooja / Singh, Palwinder et al. | 2014
- 1649
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Discovery of a novel series of indoline carbamate and indolinylpyrimidine derivatives as potent GPR119 agonistsSato, Kenjiro / Sugimoto, Hiromichi / Rikimaru, Kentaro / Imoto, Hiroshi / Kamaura, Masahiro / Negoro, Nobuyuki / Tsujihata, Yoshiyuki / Miyashita, Hirohisa / Odani, Tomoyuki / Murata, Toshiki et al. | 2014
- 1667
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Anion inhibition study of the β-carbonic anhydrase (CahB1) from the cyanobacterium Coleofasciculus chthonoplastes (ex-Microcoleus chthonoplastes)Vullo, Daniela / Kupriyanova, Elena V. / Scozzafava, Andrea / Capasso, Clemente / Supuran, Claudiu T. et al. | 2014
- 1667
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Anion inhibition study of the @b-carbonic anhydrase (CahB1) from the cyanobacterium Coleofasciculus chthonoplastes (ex-Microcoleus chthonoplastes)Vullo, D. / Kupriyanova, E. V. / Scozzafava, A. / Capasso, C. / Supuran, C. T. et al. | 2014
- 1672
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Synthesis and biological evaluation of 2,5-di(7-indolyl)-1,3,4-oxadiazoles, and 2- and 7-indolyl 2-(1,3,4-thiadiazolyl)ketones as antimicrobialsKandemir, Hakan / Ma, Cong / Kutty, Samuel K. / Black, David StC. / Griffith, Renate / Lewis, Peter J. / Kumar, Naresh et al. | 2014
- 1680
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Synthesis of a novel series of thiazole-based histone acetyltransferase inhibitorsSecci, Daniela / Carradori, Simone / Bizzarri, Bruna / Bolasco, Adriana / Ballario, Paola / Patramani, Zoi / Fragapane, Paola / Vernarecci, Stefano / Canzonetta, Claudia / Filetici, Patrizia et al. | 2014
- 1690
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Synthesis and anticancer activity of focused compound libraries from the natural product lead, oroidinDyson, Lauren / Wright, Anthony D. / Young, Kelly A. / Sakoff, Jennette A. / McCluskey, Adam et al. | 2014
- 1700
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Synthesis, [18F] radiolabeling, and evaluation of poly (ADP-ribose) polymerase-1 (PARP-1) inhibitors for in vivo imaging of PARP-1 using positron emission tomographyZhou, Dong / Chu, Wenhua / Xu, Jinbin / Jones, Lynne A. / Peng, Xin / Li, Shihong / Chen, Delphine L. / Mach, Robert H. et al. | 2014
- 1708
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Discovery and optimization of a new class of pyruvate kinase inhibitors as potential therapeutics for the treatment of methicillin-resistant Staphylococcus aureus infectionsKumar, Nag S. / Dullaghan, Edie M. / Finlay, B. Brett / Gong, Huansheng / Reiner, Neil E. / Jon Paul Selvam, J. / Thorson, Lisa M. / Campbell, Sara / Vitko, Nicholas / Richardson, Anthony R. et al. | 2014
- 1726
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Reaction intermediate analogues as bisubstrate inhibitors of pantothenate synthetaseXu, Zhixiang / Yin, Wei / Martinelli, Leonardo K. / Evans, Joanna / Chen, Jinglei / Yu, Yang / Wilson, Daniel J. / Mizrahi, Valerie / Qiao, Chunhua / Aldrich, Courtney C. et al. | 2014
- 1736
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Design, synthesis, radiolabeling and in vivo evaluation of potential positron emission tomography (PET) radioligands for brain imaging of the 5-HT7 receptorLacivita, Enza / Niso, Mauro / Hansen, Hanne D. / Di Pilato, Pantaleo / Herth, Matthias M. / Lehel, Szabolcs / Ettrup, Anders / Montenegro, Lisa / Perrone, Roberto / Berardi, Francesco et al. | 2014
- 1751
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Discovery of simplified N2-substituted pyrazolo[3,4-d]pyrimidine derivatives as novel adenosine receptor antagonists: Efficient synthetic approaches, biological evaluations and molecular docking studiesVenkatesan, Gopalakrishnan / Paira, Priyankar / Cheong, Siew Lee / Vamsikrishna, Kosaraju / Federico, Stephanie / Klotz, Karl-Norbert / Spalluto, Giampiero / Pastorin, Giorgia et al. | 2014
- 1766
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Chemical constituents of Plectranthus amboinicus and the synthetic analogs possessing anti-inflammatory activityChen, Yuan-Siao / Yu, Hui-Ming / Shie, Jiun-Jie / Cheng, Ting-Jen Rachel / Wu, Chung-Yi / Fang, Jim-Min / Wong, Chi-Huey et al. | 2014
- 1773
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Synthesis of novel, peptidic kinase inhibitors with cytostatic/cytotoxic activitySzymanski, Wiktor / Zwolinska, Magdalena / Klossowski, Szymon / Młynarczuk-Biały, Izabela / Biały, Łukasz / Issat, Tadeusz / Malejczyk, Jacek / Ostaszewski, Ryszard et al. | 2014
- 1782
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Structure activity relationship studies of 3-arylsulfonyl-pyrido[1,2-a]pyrimidin-4-imines as potent 5-HT6 antagonistsHu, Shuanghua / Huang, Yazhong / Wu, Yong-Jin / He, Huan / Grant-Young, Katherine A. / Bertekap, Robert L. / Whiterock, Valerie / Brassil, Patrick / Lentz, Kimberley / Sivaprakasam, Prasanna et al. | 2014
- IFC
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Editorial board| 2014