Spirostanol saponins from Tacca vietnamensis and their anti-inflammatory activity (English)
- New search for: Yen, P. H.
- New search for: Chi, V. T.
- New search for: Kiem, P. V.
- New search for: Tai, B. H.
- New search for: Quang, T. H.
- New search for: Nhiem, N. X.
- New search for: Anh, H. L.
- New search for: Ban, N. K.
- New search for: Thanh, B. V.
- New search for: Minh, C. V.
- New search for: Yen, P. H.
- New search for: Chi, V. T.
- New search for: Kiem, P. V.
- New search for: Tai, B. H.
- New search for: Quang, T. H.
- New search for: Nhiem, N. X.
- New search for: Anh, H. L.
- New search for: Ban, N. K.
- New search for: Thanh, B. V.
- New search for: Minh, C. V.
In:
BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS ONLINE
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26
, 15
;
3780-3784
;
2016
-
ISSN:
- Article (Journal) / Print
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Title:Spirostanol saponins from Tacca vietnamensis and their anti-inflammatory activity
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Contributors:Yen, P. H. ( author ) / Chi, V. T. ( author ) / Kiem, P. V. ( author ) / Tai, B. H. ( author ) / Quang, T. H. ( author ) / Nhiem, N. X. ( author ) / Anh, H. L. ( author ) / Ban, N. K. ( author ) / Thanh, B. V. ( author ) / Minh, C. V. ( author )
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Published in:BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS ONLINE ; 26, 15 ; 3780-3784
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Publisher:
- New search for: Elsevier Science B.V., Amsterdam.
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Publication date:2016-01-01
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Size:5 pages
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ISSN:
-
Type of media:Article (Journal)
-
Type of material:Print
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Language:English
- New search for: 572.5
- Further information on Dewey Decimal Classification
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Classification:
DDC: 572.5 -
Source:
© Metadata Copyright the British Library Board and other contributors. All rights reserved.
Table of contents – Volume 26, Issue 15
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 3381
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From bosentan (Tracleer®) to macitentan (Opsumit®): The medicinal chemistry perspectiveBoss, Christoph / Bolli, Martin H. / Gatfield, John et al. | 2016
- 3395
-
Poly(ADP-ribose): From chemical synthesis to drug designDrenichev, Mikhail S. / Mikhailov, Sergey N. et al. | 2016
- 3404
-
Polyphenolic compounds with anti-tumour potential from Corchorus olitorius (L.) Tiliaceae, a Nigerian leaf vegetableTaiwo, Bamigboye J. / Taiwo, Grace O. / Olubiyi, Olujide O. / Fatokun, Amos A. et al. | 2016
- 3411
-
Insights into the structure–activity relationship of the anticancer compound ZJ-101, a derivative of marine natural product superstolide A: A critical role played by the conjugated trienyl lactone moietyQian, Shan / Shah, Aashay K. / Head, Sarah A. / Liu, Jun O. / Jin, Zhendong et al. | 2016
- 3414
-
Aryl or heteroaryl substituted aminal derivatives of HCV NS5A inhibitor MK-8742Yu, Wensheng / Coburn, Craig A. / Nair, Anilkumar G. / Wong, Michael / Rosenblum, Stuart B. / Zhou, Guowei / Dwyer, Michael P. / Tong, Ling / Hu, Bin / Zhong, Bin et al. | 2016
- 3421
-
Design, synthesis and anticancer activity of novel hybrid compounds between benzofuran and N-aryl piperazineMao, Ze-Wei / Zheng, Xi / Lin, Yu-Ping / Hu, Chun-Yan / Wang, Xiu-Li / Wan, Chun-Ping / Rao, Gao-Xiong et al. | 2016
- 3425
-
Anti-inflammatory polyphenol constituents derived from Cissus pteroclada HayataLi, Yi-jie / Xu, Cheng-ting / Lin, Dan-dan / Qin, Jiang-ke / Ye, Gao-jie / Deng, Qing-hua et al. | 2016
- 3429
-
Quinoxaline-based inhibitors of Ebola and Marburg VP40 egressLoughran, H. Marie / Han, Ziying / Wrobel, Jay E. / Decker, Sarah E. / Ruthel, Gordon / Freedman, Bruce D. / Harty, Ronald N. / Reitz, Allen B. et al. | 2016
- 3436
-
A cascade screening approach for the identification of Bcr-Abl myristate pocket binders active against wild type and T315I mutantRadi, Marco / Schneider, Ralf / Fallacara, Anna Lucia / Botta, Lorenzo / Crespan, Emmanuele / Tintori, Cristina / Maga, Giovanni / Kissova, Miroslava / Calgani, Alessia / Richters, André et al. | 2016
- 3441
-
Design and synthesis of 1H-pyrazolo[3,4-c]pyridine derivatives as a novel structural class of potent GPR119 agonistsMatsuda, Daisuke / Kobashi, Yohei / Mikami, Ayako / Kawamura, Madoka / Shiozawa, Fumiyasu / Kawabe, Kenichi / Hamada, Makoto / Oda, Koji / Nishimoto, Shinichi / Kimura, Kayo et al. | 2016
- 3447
-
Synthesis, characterization and antimicrobial activity of novel Schiff base tethered boronate esters of 1,2-O-isopropylidene-α-d-xylofuranoseReddy, Eda Rami / Trivedi, Rajiv / Sudheer Kumar, Buddana / Sirisha, Katukuri / Sarma, Akella Venkata Subrahmanya / Sridhar, Balasubramanian / Prakasham, Reddy Shetty et al. | 2016
- 3453
-
Development of novel 1,4-benzodiazepine-based Michael acceptors as antitrypanosomal agentsEttari, Roberta / Previti, Santo / Cosconati, Sandro / Maiorana, Santina / Schirmeister, Tanja / Grasso, Silvana / Zappalà, Maria et al. | 2016
- 3457
-
A chromatography-free isolation of rohitukine from leaves of Dysoxylum binectariferum: Evaluation for in vitro cytotoxicity, Cdk inhibition and physicochemical propertiesKumar, Vikas / Guru, Santosh K. / Jain, Shreyans K. / Joshi, Prashant / Gandhi, Sumit G. / Bharate, Sandip B. / Bhushan, Shashi / Bharate, Sonali S. / Vishwakarma, Ram A. et al. | 2016
- 3464
-
Structural modification of luteolin from Flos Chrysanthemi leads to increased tumor cell growth inhibitory activityYang, Chao / Chen, Hui / Lu, Shihai / Zhang, Meng / Tian, Wei / Wang, Mingping / Zhang, Ling / Song, Yunlong / Shen, Aijun / Zhou, Youjun et al. | 2016
- 3468
-
Conversion of adenine to 5-amino-4-pyrimidinylimidazole caused by acetyl capping during solid phase oligonucleotide synthesisRodriguez, Andrew A. / Cedillo, Isaiah / McPherson, Andrew K. et al. | 2016
- 3472
-
New structure–activity relationships of N-acetamide substituted pyrazolopyrimidines as pharmacological ligands of TSPOLi, Jun / Schulte, Michael L. / Nickels, Michael L. / Manning, H. Charles et al. | 2016
- 3478
-
An evaluation of Minor Groove Binders as anti-lung cancer therapeuticsScott, Fraser J. / Puig-Sellart, Mireia / Khalaf, Abedawn I. / Henderson, Catherine J. / Westrop, Gareth / Watson, David G. / Carter, Katharine / Grant, M. Helen / Suckling, Colin J. et al. | 2016
- 3487
-
Synthesis and evaluation of 2-pyridinylpyrimidines as inhibitors of HIV-1 structural protein assemblyKožíšek, Milan / Štěpánek, Ondřej / Parkan, Kamil / Berenguer Albiñana, Carlos / Pávová, Marcela / Weber, Jan / Krӓusslich, Hans-Georg / Konvalinka, Jan / Machara, Aleš et al. | 2016
- 3491
-
Coumarin sulfonamides derivatives as potent and selective COX-2 inhibitors with efficacy in suppressing cancer proliferation and metastasisLu, Xiao-Yuan / Wang, Zhong-Chang / Ren, Shen-Zhen / Shen, Fa-Qian / Man, Ruo-Jun / Zhu, Hai-Liang et al. | 2016
- 3499
-
Exploration of GGTase-I substrate requirements. Part 1: Synthesis and biochemical evaluation of novel aryl-modified geranylgeranyl diphosphate analogsTemple, Kayla J. / Wright, Elia N. / Fierke, Carol A. / Gibbs, Richard A. et al. | 2016
- 3503
-
Exploration of GGTase-I substrate requirements. Part 2: Synthesis and biochemical analysis of novel saturated geranylgeranyl diphosphate analogsTemple, Kayla J. / Wright, Elia N. / Fierke, Carol A. / Gibbs, Richard A. et al. | 2016
- 3508
-
Hydroxychalcone inhibitors of Streptococcus mutans glucosyl transferases and biofilms as potential anticaries agentsNijampatnam, Bhavitavya / Casals, Luke / Zheng, Ruowen / Wu, Hui / Velu, Sadanandan E. et al. | 2016
- 3514
-
Synthetic phospholipids as specific substrates for plasma endothelial lipasePapillon, Julien P.N. / Pan, Meihui / Brousseau, Margaret E. / Gilchrist, Mark A. / Lou, Changgang / Singh, Alok K. / Stawicki, Todd / Thompson, James E. et al. | 2016
- 3518
-
Synthesis and evaluation of a series of 4-azaindole-containing p21-activated kinase-1 inhibitorsLee, Wendy / Crawford, James J. / Aliagas, Ignacio / Murray, Lesley J. / Tay, Suzanne / Wang, Weiru / Heise, Christopher E. / Hoeflich, Klaus P. / La, Hank / Mathieu, Simon et al. | 2016
- 3525
-
Synthesis and antimicrobial evaluation of novel ethyl 2-(2-(4-substituted)acetamido)-4-subtituted-thiazole-5-carboxylate derivativesPawar, Chandrakant D. / Sarkate, Aniket P. / Karnik, Kshipra S. / Bahekar, Sushilkumar S. / Pansare, Dattatraya N. / Shelke, Rohini N. / Jawale, Chetan S. / Shinde, Devanand B. et al. | 2016
- 3529
-
Synthesis and evaluation of (+)-decursin derivatives as inhibitors of the Wnt/β-catenin pathwayLee, Jee-Hyun / Kim, Min-Ah / Park, Seoyoung / Cho, Soo-Hyun / Yun, Eunju / O, Yu-Seok / Kim, Jiseon / Goo, Ja-Il / Yun, Mi-Young / Choi, Yongseok et al. | 2016
- 3533
-
Structure–activity relationships of vanillic acid ester analogs in inhibitory effect of antigen-mediated degranulation in rat basophilic leukemia RBL-2H3 cellsIshimata, Nao / Ito, Hideyuki / Tai, Akihiro et al. | 2016
- 3537
-
New insights into 3-(aminomethyl)naphthoquinones: Evaluation of cytotoxicity, electrochemical behavior and search for structure–activity correlationda Silva, Gustavo B. / Neves, Amanda P. / Vargas, Maria D. / Marinho-Filho, José D.B. / Costa-Lotufo, Letícia V. et al. | 2016
- 3543
-
Structure–activity relationship study at C9 position of kaitocephalinYasuno, Yoko / Hamada, Makoto / Yoshida, Yuya / Shimamoto, Keiko / Shigeri, Yasushi / Akizawa, Toshifumi / Konishi, Motomi / Ohfune, Yasufumi / Shinada, Tetsuro et al. | 2016
- 3547
-
Kinetic investigation of human 5-lipoxygenase with arachidonic acidMittal, Monica / Kumar, Ramakrishnan B. / Balagunaseelan, Navisraj / Hamberg, Mats / Jegerschöld, Caroline / Rådmark, Olof / Haeggström, Jesper Z. / Rinaldo-Matthis, Agnes et al. | 2016
- 3552
-
Synthesis of a fluorescence resonance energy transfer-based probe containing a tricyclic nucleoside analog for single nucleotide polymorphism typingHayai, Aya / Maeda, Yusuke / Ueno, Yoshihito et al. | 2016
- 3556
-
Lanostane triterpenoids from Ganoderma curtisii and their NO production inhibitory activities of LPS-induced microgliaJiao, Yang / Xie, Ting / Zou, Lu-Hui / Wei, Qian / Qiu, Li / Chen, Li-Xia et al. | 2016
- 3562
-
Discovery of 4-(4-aminopyrazolo[1,5-a][1,3,5]triazin-8-yl)benzamides as novel, highly potent and selective, orally bioavailable inhibitors of Tyrosine Threonine Kinase, TTKLaufer, Radoslaw / Li, Sze-Wan / Liu, Yong / Ng, Grace / Lang, Yunhui / Feher, Miklos / Brokx, Richard / Beletskaya, Irina / Hodgson, Richard / Mao, Guodong et al. | 2016
- 3567
-
Synthesis, characterization and anti-cancer activity of a peptide nucleolipid bioconjugateRana, Niki / Huang, Suiying / Patel, Pradeepkumar / Samuni, Uri / Sabatino, David et al. | 2016
- 3572
-
An evolved oxazolidinone with selective potency against Mycobacterium tuberculosis and gram positive bacteriaKaushik, Amit / Heuer, Abigail M. / Bell, Drew T. / Culhane, Jeffrey C. / Ebner, David C. / Parrish, Nicole / Ippoliti, J. Thomas / Lamichhane, Gyanu et al. | 2016
- 3577
-
Facile synthesis of acacetin and its derivativesZhao, Yuan / Cai, Li / Sui, Qiang / Lin, Feng / Jiang, Wen / Chen, Jianli / Lu, Weigeng / Gao, Qi et al. | 2016
- 3581
-
Optimization of pyrazole-containing 1,2,4-triazolo-[3,4-b]thiadiazines, a new class of STAT3 pathway inhibitorsLaPorte, Matthew G. / Wang, Zhuzhu / Colombo, Raffaele / Garzan, Atefeh / Peshkov, Vsevolod A. / Liang, Mary / Johnston, Paul A. / Schurdak, Mark E. / Sen, Malabika / Camarco, Daniel P. et al. | 2016
- 3586
-
Synthesis and biological activity of novel ester derivatives of N 3-(4-metoxyfumaroyl)-(S)-2,3-diaminopropanoic acid containing amide and keto function as inhibitors of glucosamine-6-phosphate synthasePawlak, Dorota / Schielmann, Marta / Wojciechowski, Marek / Andruszkiewicz, Ryszard et al. | 2016
- 3590
-
Four new minor brominated indole related alkaloids with antibacterial activities from Laurencia similisLi, Mei-Chen / Sun, Wen-Shuang / Cheng, Wei / Liu, Dong / Liang, Hong / Zhang, Qing-Ying / Lin, Wen-Han et al. | 2016
- 3594
-
Enriching screening libraries with bioactive fragment spaceZhang, Na / Zhao, Hongtao et al. | 2016
- 3598
-
Design, synthesis, and evaluation of water-soluble morpholino-decorated paclitaxel prodrugs with remarkably decreased toxicityFeng, Siliang / Chen, Kuncheng / Wang, Chenhong / Jiang, Xifeng / Dong, Huajin / Gong, Zehui / Liu, Keliang et al. | 2016
- 3603
-
Discovery of N-(3-fluoro-4-methylsulfonamidomethylphenyl)urea as a potent TRPV1 antagonistic templateAnn, Jihyae / Sun, Wei / Zhou, Xing / Jung, Aeran / Baek, Jisoo / Lee, Sunho / Kim, Changhoon / Yoon, Suyoung / Hong, Sunhye / Choi, Sun et al. | 2016
- 3608
-
New sesquiterpene lactones, vernonilides A and B, from the seeds of Vernonia anthelmintica in Uyghur and their antiproliferative activitiesIto, Takuya / Aimaiti, Simayijiang / Win, Nwet Nwet / Kodama, Takeshi / Morita, Hiroyuki et al. | 2016
- 3612
-
Synthesis and cytotoxic activities of semisynthetic zearalenone analoguesTadpetch, Kwanruthai / Kaewmee, Benyapa / Chantakaew, Kittisak / Kantee, Kawalee / Rukachaisirikul, Vatcharin / Phongpaichit, Souwalak et al. | 2016
- 3617
-
Synthesis of riccardin D derivatives as potent antimicrobial agentsSun, Bin / Zhang, Ming / Li, Ying / Hu, Qing-wen / Zheng, Hong-bo / Chang, Wen-qiang / Lou, Hong-xiang et al. | 2016
- 3621
-
Synthesis of lignan conjugates via cyclopropanation: Antimicrobial and antioxidant studiesRaghavendra, Kanchipura Ramachandrappa / Renuka, Nagamallu / Kameshwar, Vivek H. / Srinivasan, Bharath / Ajay Kumar, Kariyappa / Shashikanth, Sheena et al. | 2016
- 3626
-
Synthesis, nematocidal activity and docking study of novel chiral 1-(3-chloropyridin-2-yl)-3-(trifluoromethyl)-1H-pyrazole-4-carboxamide derivativesLiu, Xing-Hai / Zhao, Wen / Shen, Zhong-Hua / Xing, Jia-Hua / Yuan, Jing / Yang, Guo / Xu, Tian-Ming / Peng, Wei-Li et al. | 2016
- 3629
-
[Dmt1]DALDA analogues modified with tyrosine analogues at position 1Cai, Yunxin / Lu, Dandan / Chen, Zhen / Ding, Yi / Chung, Nga N. / Li, Tingyou / Schiller, Peter W. et al. | 2016
- 3632
-
Synthesis and bioactivity of pyrazole and triazole derivatives as potential PDE4 inhibitorsLi, Ya-Sheng / Tian, Hao / Zhao, Dong-Sheng / Hu, De-Kun / Liu, Xing-Yu / Jin, Hong-Wei / Song, Gao-Peng / Cui, Zi-Ning et al. | 2016
- 3636
-
Rational design and synthesis of novel anti-prostate cancer agents bearing a 3,5-bis-trifluoromethylphenyl moietyFerla, Salvatore / Bassetto, Marcella / Pertusati, Fabrizio / Kandil, Sahar / Westwell, Andrew D. / Brancale, Andrea / McGuigan, Christopher et al. | 2016
- 3641
-
Synthesis and evaluation of fluorescent Pam3Cys peptide conjugatesGential, Geoffroy P.P. / Ho, Nataschja I. / Chiodo, Fabrizio / Meeuwenoord, Nico / Ossendorp, Ferry / Overkleeft, Herman S. / van der Marel, Gijs A. / Filippov, Dmitri V. et al. | 2016
- 3646
-
Synthesis and antitubercular activity of new 1,3,4-oxadiazoles bearing pyridyl and thiazolyl scaffoldsDhumal, Sambhaji T. / Deshmukh, Amarsinh R. / Bhosle, Manisha R. / Khedkar, Vijay M. / Nawale, Laxman U. / Sarkar, Dhiman / Mane, Ramrao A. et al. | 2016
- 3652
-
Synthesis and cytotoxic evaluation of novel indenoisoquinoline-substituted triazole hybridsPham Thi, Tham / Le Nhat, Thuy Giang / Ngo Hanh, Thuong / Luc Quang, Tan / Pham The, Chinh / Dang Thi, Tuyet Anh / Nguyen, Ha Thanh / Nguyen, Thu Ha / Hoang Thi, Phuong / Van Nguyen, Tuyen et al. | 2016
- 3658
-
Biofunction-assisted DNA detection through RNase H-enhanced 3′ processing of a premature tRNA probe in a wheat germ extractOgawa, Atsushi / Tabuchi, Junichiro / Doi, Yasunori / Takamatsu, Masashi et al. | 2016
- 3662
-
Characterization of three amidinotransferases involved in the biosynthesis of ketomemicinsOgasawara, Yasushi / Fujimori, Michiko / Kawata, Junpei / Dairi, Tohru et al. | 2016
- 3665
-
Efficient transmembrane anion transport mediated by a bis(imidazolyl)-functionalized bis(choloyl) conjugateLi, Zhi / Deng, Li-Qun / Chen, Yun / Wu, Tao / Chen, Wen-Hua et al. | 2016
- 3669
-
Identification of novel 2-aminothiazole conjugated nitrofuran as antitubercular and antibacterial agentsRan, Kai / Gao, Chao / Deng, Hongxia / Lei, Qian / You, Xinyu / Wang, Ningyu / Shi, Yaojie / Liu, Zhihao / Wei, Wei / Peng, Cuiting et al. | 2016
- 3675
-
Design, synthesis and in vitro evaluation of benzothiazole-based ureas as potential ABAD/17β-HSD10 modulators for Alzheimer’s disease treatmentHroch, Lukas / Benek, Ondrej / Guest, Patrick / Aitken, Laura / Soukup, Ondrej / Janockova, Jana / Musil, Karel / Dohnal, Vlastimil / Dolezal, Rafael / Kuca, Kamil et al. | 2016
- 3679
-
Design, synthesis and biological evaluation of novel 3-alkylsulfanyl-4-amino-1,2,4-triazole derivativesZhao, Pei-Liang / Chen, Peng / Li, Qiu / Hu, Meng-Jin / Diao, Peng-Cheng / Pan, En-Shan / You, Wen-Wei et al. | 2016
- 3684
-
Click-based synthesis and antitubercular evaluation of dibenzofuran tethered thiazolyl-1,2,3-triazolyl acetamidesSurineni, Goverdhan / Yogeeswari, Perumal / Sriram, Dharmarajan / Kantevari, Srinivas et al. | 2016
- 3690
-
Conjugation of mono and di-GalNAc sugars enhances the potency of antisense oligonucleotides via ASGR mediated delivery to hepatocytesKinberger, Garth A. / Prakash, Thazha P. / Yu, Jinghua / Vasquez, Guillermo / Low, Audrey / Chappell, Alfred / Schmidt, Karsten / Murray, Heather M. / Gaus, Hans / Swayze, Eric E. et al. | 2016
- 3694
-
Synthesis of [11C]MK-1064 as a new PET radioligand for imaging of orexin-2 receptorGao, Mingzhang / Wang, Min / Zheng, Qi-Huang et al. | 2016
- 3700
-
Application of the Huisgen cycloaddition and ‘click’ reaction toward various 1,2,3-triazoles as HIV non-nucleoside reverse transcriptase inhibitorsPribut, Nicole / Veale, Clinton G.L. / Basson, Adriaan E. / van Otterlo, Willem A.L. / Pelly, Stephen C. et al. | 2016
- 3705
-
The effect of desolvation on the binding of inhibitors to HIV-1 protease and cyclin-dependent kinases: Causes of resistanceFong, Clifford W. et al. | 2016
- 3714
-
New peptide deformylase inhibitors design, synthesis and pharmacokinetic assessmentLv, Fengping / Chen, Chen / Tang, Yang / Wei, Jianhai / Zhu, Tong / Hu, Wenhao et al. | 2016
- 3719
-
Azadirachta indica triterpenoids promote osteoblast differentiation and mineralization in vitro and in vivoKushwaha, Priyanka / Khedgikar, Vikram / Haldar, Saikat / Gautam, Jyoti / Mulani, Fayaj A. / Thulasiram, Hirekodathakallu V. / Trivedi, Ritu et al. | 2016
- 3725
-
The chemical synthesis and preliminary biological studies of phosphodiester and phosphorothioate analogues of 2-methoxy-lysophosphatidylethanolamineSowińska, Agata / Rytczak, Przemysław / Gendaszewska-Darmach, Edyta / Drzazga, Anna / Koziołkiewicz, Maria / Okruszek, Andrzej et al. | 2016
- 3730
-
New indolizine–chalcones as potent inhibitors of human farnesyltransferase: Design, synthesis and biological evaluationMoise, Iuliana-Monica / Ghinet, Alina / Belei, Dalila / Dubois, Joëlle / Farce, Amaury / Bîcu, Elena et al. | 2016
- 3735
-
Spirooxindoles as novel 3D-fragment scaffolds: Synthesis and screening against CYP121 from M. tuberculosisDavis, Holly J. / Kavanagh, Madeline E. / Balan, Tudor / Abell, Chris / Coyne, Anthony G. et al. | 2016
- 3741
-
Evaluation of bisbenzamidines as inhibitors for matriptase-2Beckmann, Anna-Madeleine / Gilberg, Erik / Gattner, Susanne / Huang, Tien L. / Vanden Eynde, Jean Jacques / Mayence, Annie / Bajorath, Jürgen / Stirnberg, Marit / Gütschow, Michael et al. | 2016
- 3746
-
Novel substituted isoxazole FXR agonists with cyclopropyl, hydroxycyclobutyl and hydroxyazetidinyl linkers: Understanding and improving key determinants of pharmacological propertiesKinzel, Olaf / Steeneck, Christoph / Schlüter, Thomas / Schulz, Andreas / Gege, Christian / Hahn, Ulrike / Hambruch, Eva / Hornberger, Martin / Spalwisz, Adriana / Frick, Katharina et al. | 2016
- 3754
-
Benzamide capped peptidomimetics as non-ATP competitive inhibitors of CDK2 using the REPLACE strategyPremnath, Padmavathy Nandha / Craig, Sandra N. / Liu, Shu / McInnes, Campbell et al. | 2016
- 3761
-
Synthesis of 1H-pyrrolo[3,2-h]quinoline-8-amine derivatives that target CTG trinucleotide repeatsMatsumoto, Jun / Li, Jinxing / Dohno, Chikara / Nakatani, Kazuhiko et al. | 2016
- 3765
-
Design, synthesis and biological evaluation of novel chiral oxazino-indoles as potential and selective neuroprotective agents against Aβ25–35-induced neuronal damageChen, Jing / Tao, Ling-Xue / Xiao, Wei / Ji, Sha-Sha / Wang, Jian-Rong / Li, Xu-Wen / Zhang, Hai-Yan / Guo, Yue-Wei et al. | 2016
- 3770
-
Antibacterial activities of fluorescent nano assembled triphenylamine phosphonium ionic liquidsBrunel, Frédéric / Lautard, Christelle / Garzino, Frédéric / Giorgio, Suzanne / Raimundo, Jean M. / Bolla, Jean M. / Camplo, Michel et al. | 2016
- 3774
-
Synthesis and biological analysis of novel glycoside derivatives of l-AEP, as targeted antibacterial agentsBovill, Richard / Evans, Philip G. / Howse, Gemma L. / Osborn, Helen M.I. et al. | 2016
- 3780
-
Spirostanol saponins from Tacca vietnamensis and their anti-inflammatory activityYen, Pham Hai / Chi, Vu Thi Quynh / Kiem, Phan Van / Tai, Bui Huu / Quang, Tran Hong / Nhiem, Nguyen Xuan / Anh, Hoang Le Tuan / Ban, Ninh Khac / Thanh, Bui Van / Minh, Chau Van et al. | 2016
- 3785
-
Natural cholinesterase inhibitors from Myristica cinnamomea KingAbdul Wahab, Siti Mariam / Sivasothy, Yasodha / Liew, Sook Yee / Litaudon, Marc / Mohamad, Jamaludin / Awang, Khalijah et al. | 2016
- 3793
-
Discovery of potent macrocyclic HCV NS5A inhibitorsYu, Wensheng / Vibulbhan, Bancha / Rosenblum, Stuart B. / Martin, Gregory S. / Vellekoop, A. Samuel / Holst, Christian L. / Coburn, Craig A. / Wong, Michael / Selyutin, Oleg / Ji, Tao et al. | 2016
- 3800
-
Alkyl substituted aminal derivatives of HCV NS5A inhibitor MK-8742Yu, Wensheng / Coburn, Craig A. / Nair, Anilkumar G. / Wong, Michael / Tong, Ling / Dwyer, Michael P. / Hu, Bin / Zhong, Bin / Hao, Jinglai / Yang, De-Yi et al. | 2016
- 3806
-
Protective effect of α-mangostin against iodixanol-induced apoptotic damage in LLC-PK1 cellsLee, Dahae / Choi, Young Ok / Kim, Ki Hyun / Chin, Young-Won / Namgung, Hojin / Yamabe, Noriko / Jung, Kiwon et al. | 2016
- 3810
-
Synthesis and evaluation of substituted 4-(N-benzylamino)cinnamate esters as potential anti-cancer agents and HIV-1 integrase inhibitorsFaridoon / Edkins, Adrienne L. / Isaacs, Michelle / Mnkandhla, Dumisani / Hoppe, Heinrich C. / Kaye, Perry T. et al. | 2016
- 3813
-
Identification of novel EZH2 inhibitors through pharmacophore-based virtual screening and biological assaysWu, Yunlong / Hu, Junchi / Ding, Hong / Chen, Limin / Zhang, Yuanyuan / Liu, Rongfeng / Xu, Pan / Du, Daohai / Lu, Wenchao / Liu, Jingqiu et al. | 2016
- 3818
-
Synthesis and biological activities of novel 1,3,4-thiadiazole-containing pyrazole oxime derivativesDai, Hong / Li, Gang / Chen, Jia / Shi, Yujun / Ge, Shushan / Fan, Chongguang / He, Haibing et al. | 2016
- 3822
-
Further optimization of the M1 PAM VU0453595: Discovery of novel heterobicyclic core motifs with improved CNS penetrationPanarese, Joseph D. / Cho, Hykeyung P. / Adams, Jeffrey J. / Nance, Kellie D. / Garcia-Barrantes, Pedro M. / Chang, Sichen / Morrison, Ryan D. / Blobaum, Anna L. / Niswender, Colleen M. / Stauffer, Shaun R. et al. | 2016
- 3826
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Cupriphilic compounds to aid in proteasome inhibitionMukherjee, Sreya / Sparks, Robert / Metcalf, Rainer / Brooks, Wesley / Daniel, Kenyon / Guida, Wayne C. et al. | 2016
- 3830
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Corrigendum to “Assessing the oral bioavailability of difluorosialic acid prodrugs, potent viral neuraminidase inhibitors, using a snapshot PK screening assay” [Bioorg. Med. Chem. Lett. 25 (2015) 2505–2509]Arns, Steve / Tan, Jason / Sun, Sharon / Galey, Adam / Zisman, Natalia / Ross, Fiona / Udechukwu, Jenna / Dercho, Samantha / Gusti, Vionarica / Paquette, Jay et al. | 2015
- IFC
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Editorial board| 2016