Metronidazole-triazole conjugates: Activity against Clostridium difficile and parasites (Unknown)
- New search for: Jarrad, Angie M.
- New search for: Karoli, Tomislav
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- New search for: Tay, Chin Yen
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- New search for: Elliott, Alysha G.
- New search for: Miyamoto, Yukiko
- New search for: Ramu, Soumya
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- New search for: Jarrad, Angie M.
- New search for: Karoli, Tomislav
- New search for: Debnath, Anjan
- New search for: Tay, Chin Yen
- New search for: Huang, Johnny X.
- New search for: Kaeslin, Geraldine
- New search for: Elliott, Alysha G.
- New search for: Miyamoto, Yukiko
- New search for: Ramu, Soumya
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In:
European journal of medicinal chemistry
;
101
;
96-102
;
2015
-
ISSN:
- Article (Journal) / Print
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Title:Metronidazole-triazole conjugates: Activity against Clostridium difficile and parasites
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Contributors:Jarrad, Angie M. ( author ) / Karoli, Tomislav ( author ) / Debnath, Anjan ( author ) / Tay, Chin Yen ( author ) / Huang, Johnny X. ( author ) / Kaeslin, Geraldine ( author ) / Elliott, Alysha G. ( author ) / Miyamoto, Yukiko ( author ) / Ramu, Soumya ( author ) / Kavanagh, Angela M. ( author )
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Published in:European journal of medicinal chemistry ; 101 ; 96-102
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Publisher:
- New search for: Elsevier Science B.V., Amsterdam.
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Publication date:2015-01-01
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Size:7 pages
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ISSN:
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Type of media:Article (Journal)
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Type of material:Print
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Language:Unknown
- New search for: 615.1
- Further information on Dewey Decimal Classification
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Classification:
DDC: 615.1 -
Source:
© Metadata Copyright the British Library Board and other contributors. All rights reserved.
Table of contents – Volume 101
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 1
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Novel dialkylphosphorylhydrazones: Synthesis, leishmanicidal evaluation and theoretical investigation of the proposed mechanism of actionda Matta, Carolina Barbosa Brito / de Queiroz, Aline Cavalcanti / Santos, Mariana Silva / Alexandre-Moreira, Magna Suzana / Gonçalves, Vinicius Tomaz / Del Cistia, Catarina de Nigris / Sant'Anna, Carlos Mauricio R. / DaCosta, João Batista N. et al. | 2015
- 13
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Properties of myelin altered peptide ligand cyclo(87-99)(Ala91,Ala96)MBP87-99 render it a promising drug lead for immunotherapy of multiple sclerosisDeraos, George / Rodi, Maria / Kalbacher, Hubert / Chatzantoni, Kokona / Karagiannis, Fotios / Synodinos, Loukas / Plotas, Panayiotis / Papalois, Apostolos / Dimisianos, Nikolaos / Papathanasopoulos, Panagiotis et al. | 2015
- 24
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Leishmanicidal, antiproteolytic, and mutagenic evaluation of alkyltriazoles and alkylphosphocholinesGontijo, Vanessa Silva / Espuri, Patrícia Ferreira / Alves, Rosemeire Brondi / de Camargos, Luiz Fernando / Santos, Fábio Vieira dos / de Souza Judice, Wagner Alves / Marques, Marcos José / Freitas, Rossimiriam Pereira et al. | 2015
- 34
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Sequence-activity relationship, and mechanism of action of mastoparan analogues against extended-drug resistant Acinetobacter baumanniiVila-Farrés, Xavier / López-Rojas, Rafael / Pachón-Ibáñez, Maria Eugenia / Teixidó, Meritxell / Pachón, Jerónimo / Vila, Jordi / Giralt, Ernest et al. | 2015
- 41
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Synthesis of 3,4-diaminobenzoyl derivatives as factor Xa inhibitorsYang, Jiabin / Su, Guoqiang / Ren, Yu / Chen, Yang et al. | 2015
- 52
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Synthesis, antiplasmodial activity and mechanistic studies of pyrimidine-5-carbonitrile and quinoline hybridsKaur, H. / Balzarini, J. / de Kock, C. / Smith, P.J. / Chibale, K. / Singh, K. et al. | 2015
- 63
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Identification of N-acylhydrazone derivatives as novel lactate dehydrogenase A inhibitorsRupiani, Sebastiano / Buonfiglio, Rosa / Manerba, Marcella / Di Ianni, Lorenza / Vettraino, Marina / Giacomini, Elisa / Masetti, Matteo / Falchi, Federico / Di Stefano, Giuseppina / Roberti, Marinella et al. | 2015
- 71
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Design, synthesis, nitric oxide release and antibacterial evaluation of novel nitrated ocotillol-type derivativesBi, Yi / Yang, Xiao / Zhang, Tingting / Liu, Zeyun / Zhang, Xiaochen / Lu, Jing / Cheng, Keguang / Xu, Jinyi / Wang, Hongbo / Lv, Guangyao et al. | 2015
- 81
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Synthesis, characterization, evaluation and molecular dynamics studies of 5, 6–diphenyl–1,2,4–triazin–3(2H)–one derivatives bearing 5–substituted 1,3,4–oxadiazole as potential anti–inflammatory and analgesic agentsBanerjee, Anupam G. / Das, Nirupam / Shengule, Sushant A. / Srivastava, Radhey Shyam / Shrivastava, Sushant Kumar et al. | 2015
- 96
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Metronidazole-triazole conjugates: Activity against Clostridium difficile and parasitesJarrad, A.M. / Karoli, T. / Debnath, A. / Tay, C.Y. / Huang, J.X. / Kaeslin, G. / Elliott, A.G. / Miyamoto, Y. / Ramu, S. et al. | 2015
- 103
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Design, synthesis, and biological evaluation of new N4-Substituted 2′-deoxy-2′-fluoro-4′-azido cytidine derivatives as potent anti-HBV agentsLv, Zhigang / He, Wu / Tian, Xianhai / Kang, Jinfeng / Liu, Yangxue / Peng, Youmei / Zheng, Liyun / Wang, Qingduan / Yu, Wenquan / Chang, Junbiao et al. | 2015
- 111
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Synthesis, cytotoxicity and antimicrobial activity of thiourea derivatives incorporating 3-(trifluoromethyl)phenyl moietyBielenica, Anna / Stefańska, Joanna / Stępień, Karolina / Napiórkowska, Agnieszka / Augustynowicz-Kopeć, Ewa / Sanna, Giuseppina / Madeddu, Silvia / Boi, Stefano / Giliberti, Gabriele / Wrzosek, Małgorzata et al. | 2015
- 126
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The interaction of 4-thiazolidinone derivatives containing indolin-2-one moiety with P-glycoprotein studied using K562 cell linesWang, Feng / Liu, Zijian / Wang, Jian / Tao, Jun / Gong, Ping / Bao, Xue / Zhao, Yanfang / Wang, Yulin et al. | 2015
- 133
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Synthesis and biological evaluation of novel myrtucommulones and structural analogues that target mPGES-1 and 5-lipoxygenaseWiechmann, K. / Muller, H. / Huch, V. / Hartmann, D. / Werz, O. / Jauch, J. et al. | 2015
- 150
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Design, synthesis, pharmacological evaluation and molecular dynamics of @b-amino acids morphan-derivatives as novel ligands for opioid receptorsNieto, C.T. / Gonzalez-Nunez, V. / Rodriguez, R.E. / Diez, D. / Garrido, N.M. et al. | 2015
- 150
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Design, synthesis, pharmacological evaluation and molecular dynamics of β-amino acids morphan-derivatives as novel ligands for opioid receptorsNieto, Carlos T. / Gonzalez-Nunez, Veronica / Rodríguez, Raquel E. / Diez, David / Garrido, Narciso M. et al. | 2015
- 163
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Novel benzidine and diaminofluorene prolinamide derivatives as potent hepatitis C virus NS5A inhibitorsBae, I.H. / Kim, H.S. / You, Y. / Chough, C. / Choe, W. / Seon, M.K. / Lee, S.G. / Keum, G. / Jang, S.K. et al. | 2015
- 179
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Synthesis and evaluation of novel pleuromutilin derivatives with a substituted pyrimidine moietyYi, Y. / Yang, G. / Zhang, C. / Chen, J. / Liang, J. / Shang, R. et al. | 2015
- 185
-
Synthesis and biological evaluation of a new series of 2-amino-3-aroyl thiophene derivatives as agonist allosteric modulators of the A1 adenosine receptor. A position-dependent effect studyRomagnoli, Romeo / Baraldi, Pier Giovanni / Lopez-Cara, Carlota / Cruz-Lopez, Olga / Moorman, Allan R. / Massink, Arnault / IJzerman, Adriaan P. / Vincenzi, Fabrizio / Borea, Pier Andrea / Varani, Katia et al. | 2015
- 205
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Design, synthesis and antiproliferative activity of novel heterobivalent hybrids based on imidazo[2,1-b][1,3,4]thiadiazole and imidazo[2,1-b][1,3]thiazole scaffoldsRomagnoli, R. / Baraldi, P.G. / Prencipe, F. / Balzarini, J. / Liekens, S. / Estevez, F. et al. | 2015
- 218
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Design, synthesis and evaluation of new GEQ derivatives as inhibitors of InhA enzyme and Mycobacterium tuberculosis growthChollet, Aurélien / Mori, Giorgia / Menendez, Christophe / Rodriguez, Frédéric / Fabing, Isabelle / Pasca, Maria Rosalia / Madacki, Jan / Korduláková, Jana / Constant, Patricia / Quémard, Annaïk et al. | 2015
- 236
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Enhancement of premature stop codon readthrough in the CFTR gene by Ataluren (PTC124) derivativesPibiri, Ivana / Lentini, Laura / Melfi, Raffaella / Gallucci, Giulia / Pace, Andrea / Spinello, Angelo / Barone, Giampaolo / Di Leonardo, Aldo et al. | 2015
- 245
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Synthesis and anti-metastatic effects of novel chiral ionone alkaloid derivativesFang, Hai-Jun / Shou, Xiao-Ai / Liu, Qian / Gan, Chun-Chun / Duan, Hong-Quan / Qin, Nan et al. | 2015
- 254
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Hybrid compounds with two redox centres: Modular synthesis of chalcogen-containing lapachones and studies on their antitumor activityVieira, André A. / Brandão, Igor R. / Valença, Wagner O. / de Simone, Carlos A. / Cavalcanti, Bruno C. / Pessoa, Claudia / Carneiro, Teiliane R. / Braga, Antonio L. / da Silva, Eufrânio N. et al. | 2015
- 266
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Primaquine–pyrimidine hybrids: Synthesis and dual-stage antiplasmodial activityKaur, Hardeep / Machado, Marta / de Kock, Carmen / Smith, Peter / Chibale, Kelly / Prudêncio, Miguel / Singh, Kamaljit et al. | 2015
- 274
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Advances in tetrahydropyrido[1,2-a]isoindolone (valmerins) series: Potent glycogen synthase kinase 3 and cyclin dependent kinase 5 inhibitorsBoulahjar, Rajâa / Ouach, Aziz / Bourg, Stéphane / Bonnet, Pascal / Lozach, Olivier / Meijer, Laurent / Guguen-Guillouzo, Christiane / Le Guevel, Rémy / Lazar, Saïd / Akssira, Mohamed et al. | 2015
- 288
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Discovery of N-aryl-naphthylamines as in vitro inhibitors of the interaction between HIV integrase and the cofactor LEDGFp75Cuzzucoli Crucitti, G. / Pescatori, L. / Messore, A. / Madia, V.N. / Pupo, G. / Saccoliti, F. / Scipione, L. / Tortorella, S. / Di Leva, F.S. et al. | 2015
- 295
-
Understanding the chemistry behind the antioxidant activities of butylated hydroxytoluene (BHT): A reviewYehye, Wageeh A. / Rahman, Noorsaadah Abdul / Ariffin, Azhar / Abd Hamid, Sharifah Bee / Alhadi, Abeer A. / Kadir, Farkaad A. / Yaeghoobi, Marzieh et al. | 2015
- 313
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Imidazolidine-4-one derivatives in the search for novel chemosensitizers of Staphylococcus aureus MRSA: Synthesis, biological evaluation and molecular modeling studiesMatys, Anna / Podlewska, Sabina / Witek, Karolina / Witek, Jagna / Bojarski, Andrzej J. / Schabikowski, Jakub / Otrębska-Machaj, Ewa / Latacz, Gniewomir / Szymańska, Ewa / Kieć-Kononowicz, Katarzyna et al. | 2015
- 326
-
Molecular docking design and one-pot expeditious synthesis of novel 2,5-diarylpyrazolo[1,5-a]pyrimidin-7-amines as anti-inflammatory agentsAggarwal, Ranjana / Singh, Gulshan / Kaushik, Pawan / Kaushik, Dhirender / Paliwal, Deepika / Kumar, Ajay et al. | 2015
- 334
-
Probing the ‘bipolar’ nature of the carbonic anhydrase active site: Aromatic sulfonamides containing 1,3-oxazol-5-yl moiety as picomolar inhibitors of cytosolic CA I and CA II isoformsKrasavin, Mikhail / Korsakov, Mikhail / Dorogov, Mikhail / Tuccinardi, Tiziano / Dedeoglu, Nurcan / Supuran, Claudiu T. et al. | 2015
- 348
-
Design, synthesis and anticancer properties of novel oxaazaspiro[4,5]trienones as potent apoptosis inducers through mitochondrial disruptionYugandhar, D. / Nayak, V.L. / Archana, S. / Shekar, K.C. / Srivastava, A.K. et al. | 2015
- 358
-
Synthesis of bicoumarin thiophosphate derivatives as steroid sulfatase inhibitorsDemkowicz, Sebastian / Kozak, Witold / Daśko, Mateusz / Masłyk, Maciej / Gielniewski, Bartłomiej / Rachon, Janusz et al. | 2015
- 367
-
Bifunctional compounds targeting both D"2 and non-@a7 nACh receptors: Design, synthesis and pharmacological characterizationMatera, C. / Pucci, L. / Fiorentini, C. / Fucile, S. / Missale, C. / Grazioso, G. / Clementi, F. / Zoli, M. / De Amici, M. et al. | 2015
- 367
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Bifunctional compounds targeting both D2 and non-α7 nACh receptors: Design, synthesis and pharmacological characterizationMatera, Carlo / Pucci, Luca / Fiorentini, Chiara / Fucile, Sergio / Missale, Cristina / Grazioso, Giovanni / Clementi, Francesco / Zoli, Michele / De Amici, Marco / Gotti, Cecilia et al. | 2015
- 384
-
Discovery and characterization of aryl isonitriles as a new class of compounds versus methicillin- and vancomycin-resistant Staphylococcus aureusDavis, Dexter C. / Mohammad, Haroon / Kyei-Baffour, Kwaku / Younis, Waleed / Creemer, Cassidy Noel / Seleem, Mohamed N. / Dai, Mingji et al. | 2015
- 391
-
Incorporation of a Michael acceptor enhances the antitumor activity of triterpenoic acidsHeller, L. / Schwarz, S. / Perl, V. / Kowitsch, A. / Siewert, B. / Csuk, R. et al. | 2015
- 400
-
Glucose conjugated platinum(II) complex: Antitumor superiority to oxaliplatin, combination effect and mechanism of actionLi, Hong / Gao, Xiangqian / Liu, Ran / Wang, Yu / Zhang, Menghua / Fu, Zheng / Mi, Yi / Wang, Yiqiang / Yao, Zhi / Gao, Qingzhi et al. | 2015
- 409
-
Multistage virtual screening and identification of novel HIV-1 protease inhibitors by integrating SVM, shape, pharmacophore and docking methodsWei, Yu / Li, Jinlong / Chen, Zeming / Wang, Fengwei / Huang, Weiqiang / Hong, Zhangyong / Lin, Jianping et al. | 2015
- 419
-
Synthesis and evaluation of isatin-β-thiosemicarbazones as novel agents against antibiotic-resistant Gram-positive bacterial speciesZhang, Xu-Meng / Guo, Hui / Li, Zai-Shun / Song, Fu-Hang / Wang, Wei-Min / Dai, Huan-Qin / Zhang, Li-Xin / Wang, Jian-Guo et al. | 2015
- 419
-
Synthesis and evaluation of isatin-@b-thiosemicarbazones as novel agents against antibiotic-resistant Gram-positive bacterial speciesZhang, X.M. / Guo, H. / Li, Z.S. / Song, F.H. / Wang, W.M. / Dai, H.Q. / Zhang, L.X. / Wang, J.G. et al. | 2015
- 431
-
N-heterocyclic carbenes (NHC) with 1,2,4-oxadiazole-substituents related to natural products: Synthesis, structure and potential antitumor activity of some corresponding gold(I) and silver(I) complexesMaftei, Catalin V. / Fodor, Elena / Jones, Peter G. / Freytag, Matthias / Franz, M. Heiko / Kelter, Gerhard / Fiebig, Heinz-Herbert / Tamm, Matthias / Neda, Ion et al. | 2015
- 442
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Design and synthesis of some new pyrazolyl-pyrazolines as potential anti-inflammatory, analgesic and antibacterial agentsViveka, S. / Dinesha / Shama, P. / Nagaraja, G.K. / Ballav, S. / Kerkar, S. et al. | 2015
- 452
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CORAL: Prediction of binding affinity and efficacy of thyroid hormone receptor ligandsToropova, A.P. / Toropov, A.A. / Benfenati, E. et al. | 2015
- 462
-
Design, synthesis and biological activities of novel oxazolo[4,5-g]quinazolin-2(1H)-one derivatives as EGFR inhibitorsYin, S. / Zhou, L. / Lin, J. / Xue, L. / Zhang, C. et al. | 2015
- 476
-
Coumarins as anticancer agents: A review on synthetic strategies, mechanism of action and SAR studiesThakur, A. / Singla, R. / Jaitak, V. et al. | 2015
- 496
-
Chalcone scaffolds as anti-infective agents: Structural and molecular target perspectivesMahapatra, Debarshi Kar / Bharti, Sanjay Kumar / Asati, Vivek et al. | 2015
- 525
-
Synthesis and biological evaluation of 6-substituted indolizinoquinolinediones as catalytic DNA topoisomerase I inhibitorsYu, L.M. / Zhang, X.R. / Li, X.B. / Yang, Y. / Wei, H.Y. / He, X.X. / Gu, L.Q. / Huang, Z.S. / Pommier, Y. et al. | 2015
- 534
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Ferroquine and its derivatives: New generation of antimalarial agentsWani, Waseem A. / Jameel, Ehtesham / Baig, Umair / Mumtazuddin, Syed / Hun, Lee Ting et al. | 2015
- 552
-
Synthesis of new 4-phenylpyrimidine-2(1H)-thiones and their potency to inhibit COX-1 and COX-2Seebacher, Werner / Faist, Johanna / Presser, Armin / Weis, Robert / Saf, Robert / Kaserer, Teresa / Temml, Veronika / Schuster, Daniela / Ortmann, Sabine / Otto, Nadine et al. | 2015
- 560
-
Reversal of P-gp and BCRP-mediated MDR by tariquidar derivativesLi, X.Q. / Wang, L. / Lei, Y. / Hu, T. / Zhang, F.L. / Cho, C.H. / To, K.K.W. et al. | 2015
- 573
-
Design, synthesis and evaluation of semi-synthetic triazole-containing caffeic acid analogues as 5-lipoxygenase inhibitorsDe Lucia, Daniela / Lucio, Oscar Méndez / Musio, Biagia / Bender, Andreas / Listing, Monika / Dennhardt, Sophie / Koeberle, Andreas / Garscha, Ulrike / Rizzo, Roberta / Manfredini, Stefano et al. | 2015
- 584
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Synthesis and biological evaluation of new curcumin analogues as antioxidant and antitumor agents: Molecular modeling studyBayomi, Said M. / El-Kashef, Hassan A. / El-Ashmawy, Mahmoud B. / Nasr, Magda N.A. / El-Sherbeny, Magda A. / Abdel-Aziz, Naglaa I. / El-Sayed, Magda A.-A. / Suddek, Ghada M. / El-Messery, Shahenda M. / Ghaly, Mariam A. et al. | 2015
- 595
-
Design, synthesis and evaluation of novel polypharmacological antichlamydial agentsSunduru, N. / Salin, O. / Gylfe, A. / Elofsson, M. et al. | 2015
- 604
-
Preliminary research on 1-(4-bromo-2-nitroimidazol-1-yl)-3-[18F]fluoropropan-2-ol as a novel brain hypoxia PET tracer in a rodent model of strokeNieto, Elena / Delgado, Mercedes / Sobrado, Mónica / de Ceballos, María L. / Alajarín, Ramón / García-García, Luis / Kelly, James / Lizasoain, Ignacio / Pozo, Miguel A. / Álvarez-Builla, Julio et al. | 2015
- 616
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Small lipidated anti-obesity compounds derived from neuromedin UMicewicz, Ewa D. / Bahattab, Omar S.O. / Willars, Gary B. / Waring, Alan J. / Navab, Mohamad / Whitelegge, Julian P. / McBride, William H. / Ruchala, Piotr et al. | 2015
- 627
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4-Fluoro-3′,4′,5′-trimethoxychalcone as a new anti-invasive agent. From discovery to initial validation in an in vivo metastasis modelRoman, Bart I. / De Ryck, Tine / Patronov, Atanas / Slavov, Svetoslav H. / Vanhoecke, Barbara W.A. / Katritzky, Alan R. / Bracke, Marc E. / Stevens, Christian V. et al. | 2015
- 640
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N-Alkyl/aryl-4-(3-substituted-3-phenylpropyl)piperazine-1-carbothioamide as dual-action vaginal microbicides with reverse transcriptase inhibitionBala, Veenu / Mandalapu, Dhanaraju / Gupta, Sonal / Jangir, Santosh / Kushwaha, Bhavana / Chhonker, Yashpal S. / Chandasana, Hardik / Krishna, Shagun / Rawat, Kavita / Krishna, Atul et al. | 2015
- 651
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Synthesis, pharmacological evaluation and docking studies of pyrrole structure-based CB"2 receptor antagonistsRagusa, G. / Gomez-Canas, M. / Morales, P. / Hurst, D.P. / Deligia, F. / Pazos, R. / Pinna, G.A. / Fernandez-Ruiz, J. / Goya, P. et al. | 2015
- 668
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Melanoma-targeted delivery system (part 1): Design, synthesis and evaluation of releasable disulfide drug by glutathioneEl Aissi, R. / Chezal, J.M. / Tarrit, S. / Chavignon, O. / Moreau, E. et al. | 2015
- 681
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Structure-kinetics relationships of Capadenoson derivatives as adenosine A1 receptor agonistsLouvel, Julien / Guo, Dong / Soethoudt, Marjolein / Mocking, Tamara A.M. / Lenselink, Eelke B. / Mulder-Krieger, Thea / Heitman, Laura H. / IJzerman, Adriaan P. et al. | 2015
- 692
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Combating highly resistant emerging pathogen Mycobacterium abscessus and Mycobacterium tuberculosis with novel salicylanilide esters and carbamatesBaranyai, Z. / Kratky, M. / Vinsova, J. / Szabo, N. / Senoner, Z. / Horvati, K. / Stolarikova, J. / David, S. / Bosze, S. et al. | 2015
- 705
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Design, synthesis of benzocoumarin-pyrimidine hybrids as novel class of antitubercular agents, their DNA cleavage and X-ray studiesReddy, Dinesh S. / Hosamani, Kallappa M. / Devarajegowda, Hirihalli C. et al. | 2015
- 716
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Discovery and optimization of adamantane carboxylic acid derivatives as potent diacylglycerol acyltransferase 1 inhibitors for the potential treatment of obesity and diabetesPagire, S.H. / Pagire, H.S. / Lee, G.B. / Han, S.J. / Kwak, H.J. / Kim, J.Y. / Kim, K.Y. / Rhee, S.D. / Ryu, J.I. et al. | 2015
- 736
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Synthesis and in vitro characterization of novel fluorinated derivatives of the TSPO 18 kDa ligand SSR180575Damont, A. / Marguet, F. / Puech, F. / Dolle, F. et al. | 2015
- 746
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Synthesis, leishmanicidal, trypanocidal and cytotoxic activity of quinoline-hydrazone hybridsCoa, J.C. / Castrillon, W. / Cardona, W. / Carda, M. / Ospina, V. / Munoz, J.A. / Velez, I.D. / Robledo, S.M. et al. | 2015
- 754
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Design, synthesis, in-vitro antiproliferative activity and kinase profile of new picolinamide based 2-amido and ureido quinoline derivativesEl-Damasy, Ashraf Kareem / Seo, Seon Hee / Cho, Nam-Chul / Kang, Soon Bang / Pae, Ae Nim / Kim, Key-Sun / Keum, Gyochang et al. | 2015
- 769
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Design, synthesis and anticancer activity of Michael-type thiol adducts of α-santonin analogue with exocyclic methyleneKhazir, Jabeena / Riley, Darren L. / Chashoo, Gousia / Mir, Bilal Ahmad / Liles, David / Islam, Md. Ataul / Singh, Shashank K. / Vishwakarma, Ram A. / Pilcher, Lynne A. et al. | 2015
- 769
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Design, synthesis and anticancer activity of Michael-type thiol adducts of @a-santonin analogue with exocyclic methyleneKhazir, J. / Riley, D.L. / Chashoo, G. / Mir, B.A. / Liles, D. / Islam, Md.A. / Singh, S.K. / Vishwakarma, R.A. / Pilcher, L.A. et al. | 2015
- 780
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Synthesis and biological evaluation of novel aromatic-heterocyclic biphenyls as potent anti-leukemia agentsDong, Jinyun / Pan, Xiaoyan / Wang, Jinfeng / Su, Ping / Zhang, Lin / Wei, Fen / Zhang, Jie et al. | 2015
- 790
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Design, synthesis and biological evaluation of 1,3-diphenyl-1H-pyrazole derivatives containing benzimidazole skeleton as potential anticancer and apoptosis inducing agentsReddy, T. Srinivasa / Kulhari, Hitesh / Reddy, V. Ganga / Bansal, Vipul / Kamal, Ahmed / Shukla, Ravi et al. | 2015
- 806
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Lowering the pKa of a bisimidazoline lead with halogen atoms results in improved activity and selectivity against Trypanosoma brucei in vitroRíos Martínez, Carlos H. / Nué Martínez, J. Jonathan / Ebiloma, Godwin U. / de Koning, Harry P. / Alkorta, Ibon / Dardonville, Christophe et al. | 2015
- 818
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Synthesis and structure–activity relationship study of a new series of antiparasitic aryloxyl thiosemicarbazones inhibiting Trypanosoma cruzi cruzainEspíndola, José Wanderlan Pontes / Cardoso, Marcos Veríssimo de Oliveira / Filho, Gevanio Bezerra de Oliveira / Oliveira e Silva, Dayane Albuquerque / Moreira, Diogo Rodrigo Magalhaes / Bastos, Tanira Matutino / Simone, Carlos Alberto de / Soares, Milena Botelho Pereira / Villela, Filipe Silva / Ferreira, Rafaela Salgado et al. | 2015
- 836
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Synthesis and cytotoxic activity evaluation of some novel 1-(3-(aryl-4,5-dihydroisoxazol-5-yl)methyl)-4-trihalomethyl-1H-pyrimidin-2-ones in human cancer cellsLobo, Marcio M. / Viau, Cassiana M. / dos Santos, Josiane M. / Bonacorso, Helio G. / Martins, Marcos A.P. / Amaral, Simone S. / Saffi, Jenifer / Zanatta, Nilo et al. | 2015
- iii
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Graphical contents list| 2015
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Editorial board| 2015