Solvent effect on copper-catalyzed azide–alkyne cycloaddition (CuAAC): Synthesis of novel triazolyl substituted quinolines as potential anticancer agents (English)
- New search for: Ellanki, Amarender Reddy
- New search for: Ellanki, Amarender Reddy
- New search for: Islam, Aminul
- New search for: Rama, Veera Swamy
- New search for: Pulipati, Ranga Prasad
- New search for: Rambabu, D.
- New search for: Rama Krishna, G.
- New search for: Malla Reddy, C.
- New search for: Mukkanti, K.
- New search for: Vanaja, G.R.
- New search for: Kalle, Arunasree M.
- New search for: Shiva Kumar, K.
- New search for: Pal, Manojit
In:
Bioorganic & medicinal chemistry letters
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22
, 10
; 3455-3460
;
2012
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ISSN:
- Article (Journal) / Print
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Title:Solvent effect on copper-catalyzed azide–alkyne cycloaddition (CuAAC): Synthesis of novel triazolyl substituted quinolines as potential anticancer agents
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Contributors:
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Published in:Bioorganic & medicinal chemistry letters ; 22, 10 ; 3455-3460
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2012
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ISSN:
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ZDBID:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.42
- Further information on Basic classification
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Keywords:
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Source:
Table of contents – Volume 22, Issue 10
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 3377
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Graphical contents list| 2012
- 3387
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The discovery of potent and selective pyridopyrimidin-7-one based inhibitors of B-RafV600E kinaseRen, Li / Ahrendt, Kateri A. / Grina, Jonas / Laird, Ellen R. / Buckmelter, Alex J. / Hansen, Joshua D. / Newhouse, Brad / Moreno, David / Wenglowsky, Steve / Dinkel, Victoria et al. | 2012
- 3392
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Discovery of a series of 2-(1H-pyrazol-1-yl)pyridines as ALK5 inhibitors with potential utility in the prevention of dermal scarringBoys, Mark L. / Bian, Feng / Kramer, James B. / Chio, Christopher L. / Ren, Xiao-Dan / Chen, Huifen / Barrett, Stephen D. / Sexton, Karen E. / Iula, Donna M. / Filzen, Gary F. et al. | 2012
- 3398
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Ianthellamide A, a selective kynurenine-3-hydroxylase inhibitor from the Australian marine sponge Ianthella quadrangulataFeng, Yunjiang / Bowden, Bruce F. / Kapoor, Vimal et al. | 2012
- 3402
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Synthesis of indolizidinone analogues of cytotoxic alkaloids: Monocyclic precursors are also activeBoto, Alicia / Miguélez, Javier / Marín, Raquel / Díaz, Mario et al. | 2012
- 3408
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Tetrahydro-naphthols as orally available TRPV1 inhibitorsUrbahns, Klaus / Yura, Takeshi / Gupta, Jang B. / Tajimi, Masaomi / Fujishima, Hiroshi / Masuda, Tsutomu / Yamamoto, Noriyuki / Ikegami, Yuka / Marumo, Makiko / Yasoshima, Kayo et al. | 2012
- 3412
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Acylated Gly-(2-cyano)pyrrolidines as inhibitors of fibroblast activation protein (FAP) and the issue of FAP/prolyl oligopeptidase (PREP)-selectivityRyabtsova, Oxana / Jansen, Koen / Van Goethem, Sebastiaan / Joossens, Jurgen / Cheng, Jonathan D. / Lambeir, Anne-Marie / De Meester, Ingrid / Augustyns, Koen / Van der Veken, Pieter et al. | 2012
- 3418
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Synthesis and characterization of folic acid modified water-soluble chitosan derivatives for folate-receptor-mediated targetingJing, Huihui / Guo, Zhide / Guo, Wenyan / Yang, Wenjiang / Xu, Peng / Zhang, Xianzhong et al. | 2012
- 3425
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Conjugates of 5-isoquinolinesulfonylamides and oligo-d-arginine possess high affinity and selectivity towards Rho kinase (ROCK)Lavogina, Darja / Kalind, Katrin / Bredihhina, Jevgenia / Hurt, Madis / Vaasa, Angela / Kasari, Marje / Enkvist, Erki / Raidaru, Gerda / Uri, Asko et al. | 2012
- 3431
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Novel triazolopyridylbenzamides as potent and selective p38α inhibitorsAiguadé, Josep / Balagué, Cristina / Carranco, Inés / Caturla, Francisco / Domínguez, María / Eastwood, Paul / Esteve, Cristina / González, Jacob / Lumeras, Wenceslao / Orellana, Adelina et al. | 2012
- 3431
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Novel triazolopyridylbenzamides as potent and selective p38a inhibitorsAiguade, J. / Balague, C. / Carranco, I. / Caturla, F. / Dominguez, M. / Eastwood, P. / Esteve, C. / Gonzalez, J. / Lumeras, W. / Orellana, A. et al. | 2012
- 3437
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Discovery of cariprazine (RGH-188): A novel antipsychotic acting on dopamine D3/D2 receptorsÁgai-Csongor, Éva / Domány, György / Nógrádi, Katalin / Galambos, János / Vágó, István / Keserű, György Miklós / Greiner, István / Laszlovszky, István / Gere, Anikó / Schmidt, Éva et al. | 2012
- 3441
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Practical access to four stereoisomers of naftidrofuryl and their binding affinity towards 5-hydroxytryptamine 2A receptorHao, Jia / Chen, Bo / Yao, Yiwu / Hossain, Murad / Nagatomo, Takafumi / Yao, Hequan / Kong, Lingyi / Sun, Hongbin et al. | 2012
- 3445
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A novel pyrimidine derivatives with aryl urea, thiourea and sulfonamide moieties: Synthesis, anti-inflammatory and antimicrobial evaluationKeche, Ashish P. / Hatnapure, Girish D. / Tale, Rajesh H. / Rodge, Atish H. / Birajdar, Satish S. / Kamble, Vandana M. et al. | 2012
- 3449
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Synthesis and biological evaluation of some novel thiazole substituted benzotriazole derivativesGaikwad, Nitin D. / Patil, Sachin V. / Bobade, Vivek D. et al. | 2012
- 3455
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Solvent effect on copper-catalyzed azide–alkyne cycloaddition (CuAAC): Synthesis of novel triazolyl substituted quinolines as potential anticancer agentsEllanki, Amarender Reddy / Islam, Aminul / Rama, Veera Swamy / Pulipati, Ranga Prasad / Rambabu, D. / Rama Krishna, G. / Malla Reddy, C. / Mukkanti, K. / Vanaja, G.R. / Kalle, Arunasree M. et al. | 2012
- 3460
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Identification of ETP-46321, a potent and orally bioavailable PI3K a, d inhibitorMartinez Gonzalez, S. / Hernandez, A. I. / Varela, C. / Rodriguez-Aristegui, S. / Lorenzo, M. / Rodriguez, A. / Rivero, V. / Martin, J. I. / Saluste, C. G. / Ramos-Lima, F. et al. | 2012
- 3460
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Identification of ETP-46321, a potent and orally bioavailable PI3K α, δ inhibitorMartínez González, Sonia / Hernández, Ana Isabel / Varela, Carmen / Rodríguez-Arístegui, Sonsoles / Lorenzo, Milagros / Rodríguez, Antonio / Rivero, Virginia / Martín, José Ignacio / Saluste, Carl Gustav / Ramos-Lima, Francisco et al. | 2012
- 3467
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Continued optimization of the MLPCN probe ML071 into highly potent agonists of the hM1 muscarinic acetylcholine receptorMelancon, Bruce J. / Gogliotti, Rocco D. / Tarr, James C. / Saleh, Sam A. / Chauder, Brian A. / Lebois, Evan P. / Cho, Hyekyung P. / Utley, Thomas J. / Sheffler, Douglas J. / Bridges, Thomas M. et al. | 2012
- 3473
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Synthesis, biological evaluation and structure–activity relationships of glycyrrhetinic acid derivatives as novel anti-hepatitis B virus agentsWang, Li-Jun / Geng, Chang-An / Ma, Yun-Bao / Huang, Xiao-Yan / Luo, Jie / Chen, Hao / Zhang, Xue-Mei / Chen, Ji-Jun et al. | 2012
- 3480
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Synthesis and anti-norovirus activity of pyranobenzopyrone compoundsPokhrel, Laxman / Kim, Yunjeong / Nguyen, Thi D.T. / Prior, Allan M. / Lu, Jianyu / Chang, Kyeong-Ok / Hua, Duy H. et al. | 2012
- 3485
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The effect of vindoline C-16 substituents on the biomimetic coupling reaction: Synthesis and cytotoxicity evaluation of the corresponding vinorelbine analoguesSong, Weibin / Hu, Lingjun / Meng, Yuhui / Ma, Lei / Guo, Dean / Liu, Xuan / Hu, Lihong et al. | 2012
- 3488
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Synthesis and biological evaluation of new potent and selective HCV NS5A inhibitorsShi, Junxing / Zhou, Longhu / Amblard, Franck / Bobeck, Drew R. / Zhang, Hongwang / Liu, Peng / Bondada, Lavanya / McBrayer, Tamara R. / Tharnish, Phillip M. / Whitaker, Tony et al. | 2012
- 3492
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Crystal structures of AKR1C3 containing an N-(aryl)amino-benzoate inhibitor and a bifunctional AKR1C3 inhibitor and androgen receptor antagonist. Therapeutic leads for castrate resistant prostate cancerChen, Mo / Adeniji, Adegoke O. / Twenter, Barry M. / Winkler, Jeffrey D. / Christianson, David W. / Penning, Trevor M. et al. | 2012
- 3498
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The central valine concept provides an entry in a new class of non peptide inhibitors of the p53–MDM2 interactionFuret, Pascal / Chène, Patrick / De Pover, Alain / Valat, Thérèse Stachyra / Lisztwan, Joanna Hergovich / Kallen, Joerg / Masuya, Keiichi et al. | 2012
- 3503
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Serendipity in discovery of proteasome inhibitorsDunn, Derek / Iqbal, Mohamed / Husten, Jean / Ator, Mark A. / Chatterjee, Sankar et al. | 2012
- 3506
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Structure–activity relationship in the antitumor activity of 6-, 8- or 6,8-substituted 3-benzylamino-β-carboline derivativesIkeda, Reiko / Kimura, Takanori / Tsutsumi, Tatsuya / Tamura, Syunsuke / Sakai, Norio / Konakahara, Takeo et al. | 2012
- 3506
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Structure-activity relationship in the antitumor activity of 6-, 8- or 6,8-substituted 3-benzylamino-b-carboline derivativesIkeda, R. / Kimura, T. / Tsutsumi, T. / Tamura, S. / Sakai, N. / Konakahara, T. et al. | 2012
- 3516
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Long-acting peptidomimetics based DPP-IV inhibitorsJadav, Pradip / Bahekar, Rajesh / Shah, Shailesh R. / Patel, Dipam / Joharapurkar, Amit / Kshirsagar, Samadhan / Jain, Mukul / Shaikh, Mubeen / Sairam, Kalapatapu V.V.M. et al. | 2012
- 3522
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Enzymatic polymerisation involving 2′-amino-LNA nucleotidesJohannsen, Marie W. / Veedu, Rakesh N. / Madsen, Andreas Stahl / Wengel, Jesper et al. | 2012
- 3522
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Enzymatic polymerisation involving 2prime-amino-LNA nucleotidesJohannsen, M. W. / Veedu, R. N. / Madsen, A. S. / Wengel, J. et al. | 2012
- 3527
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Novel desosamine-modified 14- and 15-membered macrolides without antibacterial activityJakopović, Ivana Palej / Krajačić, Mirjana Bukvić / Škugor, Maja Matanović / Štimac, Vlado / Pešić, Dijana / Vujasinović, Ines / Alihodžić, Sulejman / Paljetak, Hana Čipčić / Kragol, Goran et al. | 2012
- 3531
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The discovery of 2-fluoro-N-(3-fluoro-4-(5-((4-morpholinobutyl)amino)-1,3,4-oxadiazol-2-yl)phenyl)benzamide, a full agonist of the alpha-7 nicotinic acetylcholine receptor showing efficacy in the novel object recognition model of cognition enhancementSkidmore, John / Atcha, Zeenat / Boucherat, Emmanuelle / Castelletti, Laura / Chen, Deborah W. / Coppo, Frank T. / Cutler, Leanne / Dunsdon, Rachel M. / Heath, Bronagh M. / Hutchings, Rio et al. | 2012
- 3535
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Modulation of thermo-transient receptor potential (thermo-TRP) channels by thymol-based compoundsOrtar, Giorgio / Morera, Ludovica / Schiano Moriello, Aniello / Morera, Enrico / Nalli, Marianna / Di Marzo, Vincenzo / De Petrocellis, Luciano et al. | 2012
- 3540
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Substrate specificity of galactokinase from Streptococcus pneumoniae TIGR4 towards galactose, glucose, and their derivativesZou, Yang / Wang, Wenjun / Cai, Li / Chen, Leilei / Xue, Mengyang / Zhang, Xiaomei / Shen, Jie / Chen, Min et al. | 2012
- 3544
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Synthesis and SAR studies of imidazo-[1,2-a]-pyrazine Aurora kinase inhibitors with improved off-target kinase selectivityVoss, Matthew E. / Rainka, Matthew P. / Fleming, Mike / Peterson, Lisa H. / Belanger, David B. / Siddiqui, M. Arshad / Hruza, Alan / Voigt, Johannes / Gray, Kimberly / Basso, Andrea D. et al. | 2012
- 3550
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Derivatives of 8-hydroxyquinoline—antibacterial agents that target intra- and extracellular Gram-negative pathogensEnquist, Per-Anders / Gylfe, Åsa / Hägglund, Ulrik / Lindström, Pia / Norberg-Scherman, Henrik / Sundin, Charlotta / Elofsson, Mikael et al. | 2012
- 3554
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Synthesis and acrosin inhibitory activity of methyl 5-substituted-1H-benzo[d]imidazol-2-yl carbamate derivativesLiu, Xuefei / Chen, Qianqian / Zhu, Ju / Fan, Yongzheng / Ding, Lili / Zhao, Juntao / Han, Guangqian / Tian, Wei / Qi, Jingjing / Zhou, Youjun et al. | 2012
- 3560
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Identification of a series of 1,3,4-oxadiazol-2-amines as potent alpha-7 agonists with efficacy in the novel object recognition model of cognitionSkidmore, John / Atcha, Zeenat / Boucherat, Emmanuelle / Castelletti, Laura / Chen, Deborah W. / Coppo, Frank T. / Cutler, Leanne / Dunsdon, Rachel M. / Heath, Bronagh M. / Hutchings, Rio et al. | 2012
- 3564
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A carbosilane dendrimer and a silacyclopentadiene analog carrying peripheral lactoses as drug-delivery systemsAizawa, Hiroaki / Otomo, Kentaro / Honsho, Nobuaki / Shimazaki, Tomoyuki / Villeneuve, Masumi / Matsuoka, Koji / Hatano, Ken / Terunuma, Daiyo et al. | 2012
- 3567
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Synthesis and biological activity of 2-aminothiazoles as novel inhibitors of PGE2 production in cellsSmith, Breland / Chang, Hui-Hua / Medda, Federico / Gokhale, Vijay / Dietrich, Justin / Davis, Angela / Meuillet, Emmanuelle J. / Hulme, Christopher et al. | 2012
- 3571
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Identification of a selective small molecule inhibitor of breast cancer stem cellsGermain, Andrew R. / Carmody, Leigh C. / Morgan, Barbara / Fernandez, Cristina / Forbeck, Erin / Lewis, Timothy A. / Nag, Partha P. / Ting, Amal / VerPlank, Lynn / Feng, Yuxiong et al. | 2012
- IFC
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Editorial board| 2012