Recent advances in the chemistry and biology of anti-inflammatory and specialized pro-resolving mediators biosynthesized from n-3 docosapentaenoic acid (English)
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In:
Bioorganic & medicinal chemistry letters
;
27
, 11
; 2259-2266
;
2017
-
ISSN:
- Article (Journal) / Print
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Title:Recent advances in the chemistry and biology of anti-inflammatory and specialized pro-resolving mediators biosynthesized from n-3 docosapentaenoic acid
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Contributors:
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Published in:Bioorganic & medicinal chemistry letters ; 27, 11 ; 2259-2266
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Publisher:
- New search for: Elsevier
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Place of publication:Amsterdam [u.a.]
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Publication date:2017
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ISSN:
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ZDBID:
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DOI:
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Type of media:Article (Journal)
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Type of material:Print
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Language:English
- New search for: 35.70 / 44.33 / 44.42
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Source:
Table of contents – Volume 27, Issue 11
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
- 2239
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Pharmacological property optimization for allosteric ligands: A medicinal chemistry perspectiveJohnstone, Shawn / Albert, Jeffrey S. et al. | 2017
- 2259
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Recent advances in the chemistry and biology of anti-inflammatory and specialized pro-resolving mediators biosynthesized from n-3 docosapentaenoic acidVik, Anders / Dalli, Jesmond / Hansen, Trond Vidar et al. | 2017
- 2267
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Cytotoxic steroidal saponins from Trillium kamtschaticumQin, Xu-Jie / Si, Yong-Ai / Chen, Yu / Liu, Hui / Ni, Wei / Yan, Huan / Shu, Tong / Ji, Yun-Heng / Liu, Hai-Yang et al. | 2017
- 2274
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Structure-related protein tyrosine phosphatase 1B inhibition by naringenin derivativesJung, Hyun Ah / Paudel, Pradeep / Seong, Su Hui / Min, Byung-Sun / Choi, Jae Sue et al. | 2017
- 2281
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Design, synthesis and evaluation of 1,3,6-trisubstituted-4-oxo-1,4-dihydroquinoline-2-carboxylic acid derivatives as ETA receptor selective antagonists using FRET assayKhadtare, Nikhil / Stephani, Ralph / Korlipara, Vijaya et al. | 2017
- 2286
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Brefeldin A enhances docetaxel-induced growth inhibition and apoptosis in prostate cancer cells in monolayer and 3D culturesHuang, Huarong / Liu, Ting / Guo, Junxi / Yu, Lin / Wu, Xiaofeng / He, Yan / Li, Dongli / Liu, Junlei / Zhang, Kun / Zheng, Xi et al. | 2017
- 2292
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Copalic acid analogs down-regulate androgen receptor and inhibit small chaperone proteinIdippily, Nethrie D. / Zheng, Qiaoyun / Gan, Chunfang / Quamine, Aicha / Ashcraft, Morgan M. / Zhong, Bo / Su, Bin et al. | 2017
- 2296
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Optimization of M4 positive allosteric modulators (PAMs): The discovery of VU0476406, a non-human primate in vivo tool compound for translational pharmacologyMelancon, Bruce J. / Wood, Michael R. / Noetzel, Meredith J. / Nance, Kellie D. / Engelberg, Eileen M. / Han, Changho / Lamsal, Atin / Chang, Sichen / Cho, Hyekyung P. / Byers, Frank W. et al. | 2017
- 2302
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Stereoselective synthesis of enantiopure N-substituted pyrrolidin-2,5-dione derivatives by 1,3-dipolar cycloaddition and assessment of their in vitro antioxidant and antibacterial activitiesGhannay, Siwar / Bakari, Sana / Ghabi, Ameni / Kadri, Adel / Msaddek, Moncef / Aouadi, Kaïss et al. | 2017
- 2308
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Novel non-trimethoxylphenyl piperlongumine derivatives selectively kill cancer cellsZhang, Youjun / Ma, Hao / Wu, Yuelin / Wu, Zhongli / Yao, Zhengguang / Zhang, Wannian / Zhuang, Chunlin / Miao, Zhenyuan et al. | 2017
- 2313
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Approaches towards the development of chimeric DPP4/ACE inhibitors for treating metabolic syndromeSattigeri, Jitendra A. / Sethi, Sachin / Davis, Joseph A. / Ahmed, Shahadat / Rayasam, Geeta V. / Jadhav, Balasaheb G. / Chilla, Satya M. / Datta, Dhrubajyoti / Gadhave, A. / Tulasi, Vamshi K. et al. | 2017
- 2319
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Acetanilide and bromoacetyl-lysine derivatives as activators for human histone deacetylase 8Mukhtar, Yusif M. / Huang, Yajun / Liu, Jiajia / Chen, Di / Zheng, Weiping et al. | 2017
- 2324
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Identification of low micromolar dual inhibitors for aldose reductase (ALR2) and poly (ADP-ribose) polymerase (PARP-1) using structure based design approachChadha, Navriti / Silakari, Om et al. | 2017
- 2331
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Potent and selective oxytocin receptor agonists without disulfide bridgesAdachi, Yusuke / Sakimura, Katsuya / Shimizu, Yuji / Nakayama, Masaharu / Terao, Yasuko / Yano, Takahiko / Asami, Taiji et al. | 2017
- 2336
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4-Connected azabicyclo[5.3.0]decane Smac mimetics-Zn2+ chelators as dual action antitumoral agentsManzoni, Leonardo / Samela, Alessandro / Barbini, Stefano / Cairati, Silvia / Penconi, Marta / Arosio, Daniela / Lecis, Daniele / Seneci, Pierfausto et al. | 2017
- 2345
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Synthesis, structural characterization and biological activity of novel Knoevenagel condensates on DLD-1 human colon carcinomaRišiaňová, Lucia / Fischer-Fodor, Eva / Valentová, Jindra / Tatomir, Corina / Corina Decea, Nicoleta / Virag, Piroska / Pechová, Iveta / Devínsky, Ferdinand / Miklášová, Natalia et al. | 2017
- 2350
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Functional evaluation of synthetic flavonoids and chalcones for potential antiviral and anticancer propertiesMateeva, Nelly / Eyunni, Suresh V.K. / Redda, Kinfe K. / Ononuju, Ucheze / Hansberry, Tony D. II / Aikens, Cecilia / Nag, Anita et al. | 2017
- 2357
-
Synthesis and evaluation of pyridinium polyoxometalates as anti-HIV-1 agentsWang, Shunyi / Sun, Wuji / Hu, Qin / Yan, Hong / Zeng, Yi et al. | 2017
- 2360
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Design, synthesis and anticancer activity of novel nopinone-based thiosemicarbazone derivativesWang, Yunyun / Gu, Wen / Shan, Yu / Liu, Fei / Xu, Xu / Yang, Yiqin / Zhang, Qiangjian / Zhang, Yan / Kuang, Hongbo / Wang, Zhonglong et al. | 2017
- 2364
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Recent progress on the treatment of Ebola virus disease with Favipiravir and other related strategiesZhang, Tao / Zhai, Min / Ji, Jianbo / Zhang, Jian / Tian, Ye / Liu, Xinyong et al. | 2017
- 2369
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Design and synthesis of 1,2,3-triazolo-phenanthrene hybrids as cytotoxic agentsKumar, Niggula Praveen / Nekkanti, Shalini / Sujana Kumari, S. / Sharma, Pankaj / Shankaraiah, Nagula et al. | 2017
- 2377
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Novel pyrazoles and pyrazolo[1,2-a]pyridazines as selective COX-2 inhibitors; Ultrasound-assisted synthesis, biological evaluation, and DFT calculationsGhareb, Nagat / Elshihawy, Hosam A. / Abdel-Daim, Mohamed M. / Helal, Mohamed A. et al. | 2017
- 2384
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Discovery of indazole aldosterone synthase (CYP11B2) inhibitors as potential treatments for hypertensionHoyt, Scott B. / Taylor, Jerry / London, Clare / Ali, Amjad / Ujjainwalla, Feroze / Tata, Jim / Struthers, Mary / Cully, Doris / Wisniewski, Tom / Ren, Ning et al. | 2017
- 2389
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Rapid, microwave-accelerated synthesis and anti-osteoporosis activities evaluation of Morusin scaffolds and Morusignin L scaffoldsLin, Bing / Huang, Jun-Fei / Liu, Xiong-Wei / Ma, Xi-Tao / Liu, Xiong-Li / Lu, Yi / Zhou, Ying / Guo, Feng-Min / Feng, Ting-Ting et al. | 2017
- 2397
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Syntheses of benzophenone-xanthone hybrid polyketides and their antibacterial activitiesKodama, Takeshi / Ito, Takuya / Dibwe, Dya Fita / Woo, So-Yeun / Morita, Hiroyuki et al. | 2017
- 2401
-
Synthesis of novel 5,6-dehydrokawain analogs as osteogenic inducers and their action mechanismsKumagai, Momochika / Nishikawa, Keisuke / Mishima, Takashi / Yoshida, Izumi / Ide, Masahiro / Koizumi, Keiko / Nakamura, Munetomo / Morimoto, Yoshiki et al. | 2017
- 2407
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Synthesis of octapeptin C4 and biological profiling against NDM-1 and polymyxin-resistant bacteriaBecker, Bernd / Butler, Mark S. / Hansford, Karl A. / Gallardo-Godoy, Alejandra / Elliott, Alysha G. / Huang, Johnny X. / Edwards, David J. / Blaskovich, Mark A.T. / Cooper, Matthew A. et al. | 2017
- 2410
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Generation of a cysteine sulfinic acid analog for incorporation in peptides using solid phase peptide synthesisCorpuz, Nixon / Schwans, Jason P. et al. | 2017
- 2415
-
pH-Dependant fluorescence switching of an i-motif structure incorporating an isomeric azobenzene/pyrene fluorophoreJoo, Han Na / Van Thi Nguyen, Thuy / Chae, Hyeon Kyeong / Seo, Young Jun et al. | 2017
- 2420
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Discovery and optimization of selective FGFR4 inhibitors via scaffold hoppingWang, Yikai / Chen, Zhengxia / Dai, Meibi / Sun, Peipei / Wang, Chunqiu / Gao, Yang / Zhao, Haixia / Zeng, Wenqin / Shen, Liang / Mao, Weifeng et al. | 2017
- 2424
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Efficient and practical synthesis of FondaparinuxDing, Yili / Vara Prasad, Chamakura V.N.S. / Bai, Hua / Wang, Bingyun et al. | 2017
- 2428
-
First insight into structure-activity relationships of selective meprin β inhibitorsRamsbeck, Daniel / Hamann, Antje / Schlenzig, Dagmar / Schilling, Stephan / Buchholz, Mirko et al. | 2017
- 2432
-
Design, synthesis, and X-ray structural studies of BACE-1 inhibitors containing substituted 2-oxopiperazines as P1′-P2′ ligandsGhosh, Arun K. / Brindisi, Margherita / Yen, Yu-Chen / Cárdenas, Emilio L. / Ella-Menye, Jean-Rene / Kumaragurubaran, Nagaswamy / Huang, Xiangping / Tang, Jordan / Mesecar, Andrew D. et al. | 2017
- 2439
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Pharmacological evaluation of a novel series of urea, thiourea and guanidine derivatives as P2X7 receptor antagonistsWong, Erick C.N. / Reekie, Tristan A. / Werry, Eryn L. / O'Brien-Brown, James / Bowyer, Sarah L. / Kassiou, Michael et al. | 2017
- 2443
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Cytochrome P450 binding studies of novel tacrine derivatives: Predicting the risk of hepatotoxicityMcEneny-King, Alanna / Osman, Wesseem / Edginton, Andrea N. / Rao, Praveen P.N. et al. | 2017
- 2450
-
Synthesis, antiplatelet and antithrombotic activities of resveratrol derivatives with NO-donor propertiesDutra, Luiz Antonio / Guanaes, Jéssica Frade O. / Johmann, Nadine / Lopes Pires, Maria Elisa / Chin, Chung Man / Marcondes, Sisi / Dos Santos, Jean Leandro et al. | 2017
- 2454
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Synthesis of isoflavene-thiosemicarbazone hybrids and evaluation of their anti-tumor activityYee, Eugene M.H. / Brandl, Miriam B. / Black, David StC / Vittorio, Orazio / Kumar, Naresh et al. | 2017
- 2459
-
Computer-aided discovery of two novel chalcone-like compounds active and selective against Leishmania infantumGomes, Marcelo N. / Alcântara, Laura M. / Neves, Bruno J. / Melo-Filho, Cleber C. / Freitas-Junior, Lucio H. / Moraes, Carolina B. / Ma, Rui / Franzblau, Scott G. / Muratov, Eugene / Andrade, Carolina Horta et al. | 2017
- 2465
-
A calcineurin antifungal strategy with analogs of FK506Nambu, Mitchell / Covel, Jonathan A. / Kapoor, Mili / Li, Xiaoming / Moloney, Molly K. / Numa, Mehdi M. / Soltow, Quinlyn A. / Trzoss, Michael / Webb, Peter / Webb, Robert R. II et al. | 2017
- 2472
-
Virtual screen to NMR (VS2NMR): Discovery of fragment hits for the CBP bromodomainSpiliotopoulos, Dimitrios / Zhu, Jian / Wamhoff, Eike-Christian / Deerain, Nicholas / Marchand, Jean-Rémy / Aretz, Jonas / Rademacher, Christoph / Caflisch, Amedeo et al. | 2017
- 2479
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Synthesis and evaluation of 4,6-disubstituted pyrimidines as CNS penetrant pan-muscarinic antagonists with a novel chemotypeBender, Aaron M. / Weiner, Rebecca L. / Luscombe, Vincent B. / Cho, Hyekyung P. / Niswender, Colleen M. / Engers, Darren W. / Bridges, Thomas M. / Conn, P. Jeffrey / Lindsley, Craig W. et al. | 2017
- 2484
-
New modified 2-aminobenzimidazole nucleosides: Synthesis and evaluation of their activity against herpes simplex virus type 1Kharitonova, Maria I. / Denisova, Alexandra O. / Andronova, Valeria L. / Kayushin, Alexei L. / Konstantinova, Irina D. / Kotovskaya, Svetlana K. / Galegov, Georgiy A. / Charushin, Valery N. / Miroshnikov, Anatoly I. et al. | 2017
- 2488
-
Design of antitumor agents containing carbohydrate based on GLUT1, and evaluation of antiproliferative activityZhang, Renshuai / Song, Lairong / Jiang, Bo / Wang, Lijun / Wu, Ning / Guo, Shuju / Shi, Dayong et al. | 2017
- 2493
-
Self-assembly of glutamic acid linked paclitaxel dimers into nanoparticles for chemotherapyWang, Zhanfeng / Zhuang, Miao / Sun, Tingting / Wang, Xin / Xie, Zhigang et al. | 2017
- 2497
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Practical application of 3-substituted-2,6-difluoropyridines in drug discovery: Facile synthesis of novel protein kinase C theta inhibitorsKatoh, Taisuke / Tomata, Yoshihide / Setoh, Masaki / Sasaki, Satoshi / Takai, Takafumi / Yoshitomi, Yayoi / Yukawa, Tomoya / Nakagawa, Hideyuki / Fukumoto, Shoji / Tsukamoto, Tetsuya et al. | 2017
- 2502
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One drug for two targets: Biological evaluation of antiretroviral agents endowed with antiproliferative activityBotta, Lorenzo / Maccari, Giorgio / Calandro, Pierpaolo / Tiberi, Marika / Brai, Annalaura / Zamperini, Claudio / Canducci, Filippo / Chiariello, Mario / Martí-Centelles, Rosa / Falomir, Eva et al. | 2017
- 2506
-
Identification of acylation products in SHAPE chemistryLin, Chaoqi / Poyer, Salomé / Zargarian, Loussiné / Salpin, Jean-Yves / Fossé, Philippe / Mauffret, Olivier / Xie, Juan et al. | 2017
- 2510
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Iodine catalyzed three component synthesis of 1-((2-hydroxy naphthalen-1-yl)(phenyl)(methyl))pyrrolidin-2-one derivatives: Rationale as potent PI3K inhibitors and anticancer agentsMuralidharan, Vivek Panyam / Alagumuthu, Manikandan / Iyer, Sathiyanarayanan Kulathu et al. | 2017
- 2515
-
Synthesis and biological evaluation of pyrimidine derivatives with diverse azabicyclic ether/amine as novel GPR119 agonistYang, Zunhua / Fang, Yuanying / Park, Haeil et al. | 2017
- 2520
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Discovery of LRRK2 inhibitors by using an ensemble of virtual screening methodsGancia, Emanuela / De Groot, Marcel / Burton, Brenda / Clark, David E. et al. | 2017
- 2528
-
Photo-controlled release of fipronil from a coumarin triggered precursorGao, Zhenhong / Yuan, Pengtao / Wang, Donghui / Xu, Zhiping / Li, Zhong / Shao, Xusheng et al. | 2017
- 2536
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Generation of tricyclic imidazo[1,2-a]pyrazines as novel PI3K inhibitors by application of a conformational restriction strategyMartínez González, Sonia / Rodríguez-Arístegui, Sonsoles / Hernández, Ana Isabel / Varela, Carmen / González Cantalapiedra, Esther / Álvarez, Rosa María / Rodríguez Hergueta, Antonio / Bischoff, James R. / Albarrán, María Isabel / Cebriá, Antonio et al. | 2017
- 2544
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Synthesis and structure–activity relationship study of pyrazolo[3,4-d]pyrimidines as tyrosine kinase RET inhibitorsWang, Chengyan / Liu, Hongchun / Song, Zilan / Ji, Yinchun / Xing, Li / Peng, Xia / Wang, Xisheng / Ai, Jing / Geng, Meiyu / Zhang, Ao et al. | 2017
- 2549
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Rational design and synthesis of 2-anilinopyridinyl-benzothiazole Schiff bases as antimitotic agentsShaik, Thokhir B. / Hussaini, S.M. Ali / Nayak, V. Lakshma / Sucharitha, M. Lakshmi / Malik, M. Shaheer / Kamal, Ahmed et al. | 2017
- 2559
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Improvement of hERG-ROMK index of spirocyclic ROMK inhibitors through scaffold optimization and incorporation of novel pharmacophoresDong, Shuzhi / VanGelder, Kelsey / Shi, Zhi-Cai / Yu, Yang / Wu, Zhicai / Ferguson, Ron / Guo, Zack Zhiqiang / Tang, Haifeng / Frie, Jessica / Fu, Qinghong et al. | 2017
- 2567
-
Synthesis of both enantiomers of 1,2,3,4-tetrahydroisoquinoline derivative IPPAM-1 and enantio-dependency of its positive allosteric modulation of prostacyclin receptorYamamoto, Kohki / Suzuki, Toshifumi / Imamura, Riyo / Nagano, Tetsuo / Okabe, Takayoshi / Miyachi, Hiroyuki et al. | 2017
- 2571
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Investigation of the inhibitory mechanism of apomorphine against MDM2–p53 interactionIshiba, Hiroyuki / Noguchi, Taro / Shu, Keitou / Ohno, Hiroaki / Honda, Kaori / Kondoh, Yasumitsu / Osada, Hiroyuki / Fujii, Nobutaka / Oishi, Shinya et al. | 2017
- 2575
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New derivatives of ursolic acid through the biotransformation by Bacillus megaterium CGMCC 1.1741 as inhibitors on nitric oxide productionZhang, Chao / Xu, Shao-Hua / Ma, Bai-Ling / Wang, Wei-wei / Yu, Bo-Yang / Zhang, Jian et al. | 2017
- 2579
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Novel bioactive molecules from Lentzea violacea strain AS 08 using one strain-many compounds (OSMAC) approachHussain, Aehtesham / Rather, Muzafar A. / Dar, Mohd S. / Aga, Mushtaq A. / Ahmad, Nisar / Manzoor, Aabid / Qayum, Arem / Shah, Aiyatullah / Mushtaq, Saleem / Ahmad, Zahoor et al. | 2017
- 2583
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6-Nitro-2,3-dihydroimidazo[2,1-b][1,3]thiazoles: Facile synthesis and comparative appraisal against tuberculosis and neglected tropical diseasesThompson, Andrew M. / Blaser, Adrian / Palmer, Brian D. / Anderson, Robert F. / Shinde, Sujata S. / Launay, Delphine / Chatelain, Eric / Maes, Louis / Franzblau, Scott G. / Wan, Baojie et al. | 2017
- 2590
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Efficient synthesis of a multi-substituted diphenylmethane skeleton as a steroid mimeticMisawa, Takashi / Tanaka, Katsuya / Demizu, Yosuke / Kurihara, Masaaki et al. | 2017
- 2594
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Tricyclic 4,4-dimethyl-3,4-dihydrochromeno[3,4-d]imidazole derivatives as microsomal prostaglandin E2 synthase-1 (mPGES-1) inhibitors: SAR and in vivo efficacy in hyperalgesia pain modelMuthukaman, Nagarajan / Tambe, Macchindra / Shaikh, Mahamadhanif / Pisal, Dnyandeo / Deshmukh, Sanjay / Tondlekar, Shital / Sarode, Neelam / Narayana, Lakshminarayana / Gajera, Jitendra M. / Kattige, Vidya G. et al. | 2017
- 2602
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Antiplasmodial β-triketones from the flowers of the Australian tree Angophora woodsianaSenadeera, Sarath P.D. / Duffy, Sandra / Avery, Vicky M. / Carroll, Anthony R. et al. | 2017
- 2608
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Picrasidine G decreases viability of MDA-MB 468 EGFR-overexpressing triple-negative breast cancer cells through inhibition of EGFR/STAT3 signaling pathwayYamashita, Naoya / Kondo, Manami / Zhao, Shuai / Li, Wei / Koike, Kazuo / Nemoto, Kiyomitsu / Kanno, Yuichiro et al. | 2017
- 2613
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Identification and structure activity relationship of novel flavone derivatives that inhibit the production of nitric oxide and PGE2 in LPS-induced RAW 264.7 cellsAn, Ji-Young / Lee, Hwi-Ho / Shin, Ji-Sun / Yoo, Hyung-Seok / Park, Jong Seon / Son, Seung Hwan / Kim, Sang Won / Yu, Jihyun / Lee, Jun / Lee, Kyung-Tae et al. | 2017
- 2617
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Developing DYRK inhibitors derived from the meridianins as a means of increasing levels of NFAT in the nucleusShaw, Simon J. / Goff, Dane A. / Lin, Nan / Singh, Rajinder / Li, Wei / McLaughlin, John / Baltgalvis, Kristen A. / Payan, Donald G. / Kinsella, Todd M. et al. | 2017
- 2622
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Discovery of novel aminobenzisoxazole derivatives as orally available factor IXa inhibitorsSakurada, Isao / Endo, Toshiya / Hikita, Katsuyoshi / Hirabayashi, Tomokazu / Hosaka, Yoshitaka / Kato, Yutaka / Maeda, Yoshitaka / Matsumoto, Shigeki / Mizuno, Takashi / Nagasue, Hiroshi et al. | 2017
- 2629
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The identification of novel acid isostere based inhibitors of the VPS10P family sorting receptor SortilinAndersen, Jacob Lauwring / Lindberg, Samsa / Langgård, Morten / Maltas, Philip J. / Rønn, Lars Christian Biilmann / Bundgaard, Christoffer / Strandbygaard, Dorthe / Thirup, Søren / Watson, Stephen P et al. | 2017
- 2634
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Discovery of benzophosphadiazine drug candidate IDX375: A novel hepatitis C allosteric NS5B RdRp inhibitorPaparin, Jean-Laurent / Amador, Agnès / Badaroux, Eric / Bot, Stéphanie / Caillet, Catherine / Convard, Thierry / Da Costa, Daniel / Dukhan, David / Griffe, Ludovic / Griffon, Jean-François et al. | 2017
- 2641
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Synthesis and nematicidal activities of 1,2,3-benzotriazin-4-one derivatives containing thiourea and acylthiourea against Meloidogyne incognitaChang, Yaning / Zhang, Jingwei / Chen, Xiulei / Li, Zhong / Xu, Xiaoyong et al. | 2016
- IFC
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Editorial board| 2017