Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 1541
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Graphical contents list| 2009
- 1559
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Biochemical basis for differences in metabolism-dependent genotoxicity by two diazinylpiperazine-based 5-HT2C receptor agonistsKalgutkar, Amit S. / Bauman, Jonathan N. / McClure, Kim F. et al. | 2009
- 1564
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Identification of novel and orally active spiroindoline NPY Y5 receptor antagonistsSakamoto, Toshihiro / Moriya, Minoru / Haga, Yuji et al. | 2009
- 1569
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Simultaneous detection of alkaline phosphatase and β-galactosidase activity using SERRSIngram, Andrew / Moore, Barry D. / Graham, Duncan et al. | 2009
- 1569
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Simultaneous detection of alkaline phosphatase and b-galactosidase activity using SERRSIngram, A. / Moore, B. D. / Graham, D. et al. | 2009
- 1572
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Bioactive metabolites produced by Chaetomium globosum, an endophytic fungus isolated from Ginkgo bilobaQin, Jian-Chun / Zhang, Ya-Mei / Gao, Jin-Ming et al. | 2009
- 1575
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Novel N-substituted 2-phenyl-1-sulfonylamino-cyclopropane carboxylates as selective ADAMTS-5 (Aggrecanase-2) inhibitorsShiozaki, Makoto / Maeda, Katsuya / Miura, Tomoya et al. | 2009
- 1581
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Production of chromopyrrolic acid by coexpression of inkOD in a heterologous host Streptomyces albusChae, Choong-Sik / Park, Jin-Soo / Chung, Soon-Chun et al. | 2009
- 1584
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Benzo(h)quinoline derivatives as G-quadruplex binding agentsParitala, Hanumantharao / Firestine, Steven M. et al. | 2009
- 1588
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5-Aminomethylbenzimidazoles as potent ITK antagonistsRiether, Doris / Zindell, Renée / Kowalski, Jennifer A. et al. | 2009
- 1592
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Deciphering the antitumoral activity of quinacrine: Binding to and inhibition of Bcl-xLOrzáez, Mar / Mondragón, Laura / García-Jareño, Alicia et al. | 2009
- 1596
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Identification of the first fluorescent α-amidoboronic acids that change fluorescent properties upon sugar bindingJin, Shan / Zhu, Chunyuan / Li, Minyong et al. | 2009
- 1596
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Identification of the first fluorescent a-amidoboronic acids that change fluorescent properties upon sugar bindingJin, S. / Zhu, C. / Li, M. et al. | 2009
- 1600
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Benzimidazolone-based serotonin 5-HT1A or 5-HT7R ligands: Synthesis and biological evaluationBadarau, Eduard / Suzenet, Franck / Bojarski, Andrzej J. et al. | 2009
- 1604
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Morpholine containing CB2 selective agonistsZindell, Renée / Riether, Doris / Bosanac, Todd et al. | 2009
- 1610
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[2-(4-Phenyl-4-piperidinyl)ethyl]amine based CCR5 antagonists: derivatizations at the N-terminal of the piperidine ringDuan, Maosheng / Aquino, Christopher / Ferris, Robert et al. | 2009
- 1614
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Enhancement of DNA cleavage activity of an unnatural ferrocene-amino acid conjugateHiggins, Pamela J. / Gellett, Amanda M. et al. | 2009
- 1618
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Approaches to the simultaneous inactivation of metallo- and serine-b-lactamasesGanta, S. R. / Perumal, S. / Pagadala, S. R. et al. | 2009
- 1618
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Approaches to the simultaneous inactivation of metallo- and serine-β-lactamasesGanta, Sudhakar Reddy / Perumal, Senthil / Pagadala, Sundar Ram Reddy et al. | 2009
- 1623
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Synthesis and biological evaluation of platensimycin analogsShen, Hong C. / Ding, Fa-Xiang / Singh, Sheo B. et al. | 2009
- 1628
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Identification and SAR of novel diaminopyrimidines. Part 1: The discovery of RO-4, a dual P2X3/P2X2/3 antagonist for the treatment of painCarter, David S. / Alam, Muzaffar / Cai, Haiying et al. | 2009
- 1632
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Identification and SAR of novel diaminopyrimidines. Part 2: The discovery of RO-51, a potent and selective, dual P2X3/P2X2/3 antagonist for the treatment of painJahangir, Alam / Alam, Muzaffar / Carter, David S. et al. | 2009
- 1636
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Aryl diketoacids (ADK) selectively inhibit duplex DNA-unwinding activity of SARS coronavirus NTPase/helicaseLee, Chaewoon / Lee, Jin Moo / Lee, Na-Ra et al. | 2009
- 1639
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New prostaglandin derivative for glaucoma treatmentPerrino, Elena / Uliva, Caterina / Lanzi, Cecilia et al. | 2009
- 1643
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Evaluation of synthetic sphingolipid analogs as ligands for peroxisome proliferator-activated receptorsTsuji, Kiyomi / Satoh, Shigeru / Mitsutake, Susumu et al. | 2009
- 1647
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Porphyrins containing nitric oxide donors: Synthesis and cancer cell-oriented NO releaseLiu, Wukun / Liu, Chaozhou / Gong, Changjun et al. | 2009
- 1650
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Inhibitory activity of prostaglandin E2 production by the synthetic 2′-hydroxychalcone analogues: Synthesis and SAR studyTran, Thanh-Dao / Park, Haeil / Kim, Hyun Pyo et al. | 2009
- 1650
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Inhibitory activity of prostaglandin E2 production by the synthetic 2prime-hydroxychalcone analogues: Synthesis and SAR studyTran, T. D. / Park, H. / Kim, H. P. et al. | 2009
- 1654
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Discovery of tetrahydro-cyclopenta[b]indole as selective LXRs modulatorRatni, Hassen / Blum-Kaelin, Denise / Dehmlow, Henrietta et al. | 2009
- 1658
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5-Aminopyrimidin-2-ylnitriles as Cathepsin K inhibitorsMorley, Andrew D. / Kenny, Peter W. / Burton, Brenda et al. | 2009
- 1662
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Carbonic anhydrase activators: Activation of the β-carbonic anhydrase Nce103 from the yeast Saccharomyces cerevisiae with amines and amino acidsIsik, Semra / Kockar, Feray / Aydin, Meltem et al. | 2009
- 1662
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Carbonic anhydrase activators: Activation of the b-carbonic anhydrase Nce103 from the yeast Saccharomyces cerevisiae with amines and amino acidsIsik, S. / Kockar, F. / Aydin, M. et al. | 2009
- 1666
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Fluorinated 9H-xanthene-9-carboxylic acid oxazol-2-yl-amides as potent, orally available mGlu1 receptor enhancersVieira, Eric / Huwyler, Jörg / Jolidon, Synèse et al. | 2009
- 1670
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Discovery of substituted 2,4,4-triarylimidazoline derivatives as potent and selective neuropeptide Y Y5 receptor antagonistsSato, Nagaaki / Jitsuoka, Makoto / Ishikawa, Shiho et al. | 2009
- 1675
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Iodine-catalyzed one-pot synthesis and antimalarial activity evaluation of symmetrically and asymmetrically substituted 3,6-diphenyl[1,2,4,5]tetraoxanesKumar, Nitin / Khan, Shabana I. / Sharma, Mukul et al. | 2009
- 1678
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Preparation and characterization of antioxidant nanospheres from multiple α-lipoic acid-containing compoundsLee, Bong Seop / Yuan, Xiangpeng / Xu, Qijin et al. | 2009
- 1678
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Preparation and characterization of antioxidant nanospheres from multiple a-lipoic acid-containing compoundsLee, B. S. / Yuan, X. / Xu, Q. et al. | 2009
- 1682
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Preparation and characterization of N-(3-pyridinyl) spirocyclic diamines as ligands for nicotinic acetylcholine receptorsSippy, Kevin B. / Anderson, David J. / Bunnelle, William H. et al. | 2009
- 1686
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M3 muscarinic acetylcholine receptor antagonists: SAR and optimization of bi-aryl aminesBudzik, Brian / Wang, Yonghui / Shi, Dongchuan et al. | 2009
- 1691
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Design and synthesis of novel tri-aryl CB2 selective cannabinoid ligandsBhattacharjee, Himanshu / Gurley, Steven N. / Moore, Bob M. II et al. | 2009
- 1694
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Design of potent thiophene inhibitors of polo-like kinase 1 with improved solubility and reduced protein bindingEmmitte, Kyle A. / Adjebang, George M. / Andrews, C. Webb et al. | 2009
- 1698
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Synthesis and antibacterial activity of 4″,11-di-O-arylalkylcarbamoyl azithromycin derivativesMa, Shutao / Jiao, Bo / Liu, Zhaopeng et al. | 2009
- 1698
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Synthesis and antibacterial activity of 4Prime,11-di-O-arylalkylcarbamoyl azithromycin derivativesMa, S. / Jiao, B. / Liu, Z. et al. | 2009
- 1702
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2,4-Diaminopyridine d-opioid receptor agonists and their associated hERG pharmacologyOwen, D. R. / Rodriguez-Lens, M. / Corless, M. D. et al. | 2009
- 1702
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2,4-Diaminopyridine δ-opioid receptor agonists and their associated hERG pharmacologyOwen, Dafydd R. / Rodriguez-Lens, Margarita / Corless, Martin D. et al. | 2009
- 1707
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[18F]FEAC and [18F]FEDAC: Two novel positron emission tomography ligands for peripheral-type benzodiazepine receptor in the brainYanamoto, Kazuhiko / Kumata, Katsushi / Yamasaki, Tomoteru et al. | 2009
- 1711
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Pyrano[2,3-e]isoindol-2-ones, new angelicin heteroanaloguesBarraja, Paola / Spanò, Virginia / Patrizia, Diana et al. | 2009
- 1715
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Potent inhibitors of Huntingtin protein aggregation in a cell-based assayRinderspacher, Alison / Cremona, Maria Laura / Liu, Yidong et al. | 2009
- 1718
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Development of multitargeted inhibitors of both the insulin-like growth factor receptor (IGF-IR) and members of the epidermal growth factor family of receptor tyrosine kinasesHubbard, Robert D. / Bamaung, Nwe Y. / Fidanze, Steve D. et al. | 2009
- 1722
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Identification of a selective thieno[2,3-c]pyridine inhibitor of COT kinase and TNF-a productionCusack, K. / Allen, H. / Bischoff, A. et al. | 2009
- 1722
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Identification of a selective thieno[2,3-c]pyridine inhibitor of COT kinase and TNF-α productionCusack, Kevin / Allen, Hamish / Bischoff, Agnieszka et al. | 2009
- 1726
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Synthesis and biological evaluation on novel analogs of 9-methylstreptimidone, an inhibitor of NF-κBIshikawa, Yuichi / Tachibana, Miyuki / Matsui, Chino et al. | 2009
- 1726
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Synthesis and biological evaluation on novel analogs of 9-methylstreptimidone, an inhibitor of NF-kBIshikawa, Y. / Tachibana, M. / Matsui, C. et al. | 2009
- 1729
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Discovery of non-peptidergic MrgX1 and MrgX2 receptor agonists and exploration of an initial SAR using solid-phase synthesisMalik, Leila / Kelly, Nicholas M. / Ma, Jian-Nong et al. | 2009
- 1733
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Design, synthesis, and evaluation of peptidomimetics containing Freidinger lactams as STAT3 inhibitorsGomez, Cindy / Bai, Longchuan / Zhang, Jian et al. | 2009
- 1737
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Comparative QSAR modelling of 2-phenylindole-3-carbaldehyde derivatives as potential antimitotic agentsHalder, Amit Kumar / Adhikari, Nilanjan / Jha, Tarun et al. | 2009
- 1740
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Synthesis and biological evaluation of sulfonylurea and thiourea derivatives substituted with benzenesulfonamide groups as potential hypoglycemic agentsZhang, Hui-bin / Zhang, Ya-an / Wu, Guan-zhong et al. | 2009
- 1745
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N-Benzyl-indolo carboxylic acids: Design and synthesis of potent and selective adipocyte fatty-acid binding protein (A-FABP) inhibitorsBarf, Tjeerd / Lehmann, Fredrik / Hammer, Kristin et al. | 2009
- 1749
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First small molecular inhibitors of T. brucei dolicholphosphate mannose synthase (DPMS), a validated drug target in African sleeping sicknessSmith, Terry K. / Young, Benjamin L. / Denton, Helen et al. | 2009
- 1753
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Synthesis and structure–activity relationships of novel benzofuran farnesyltransferase inhibitorsAsoh, Kohsuke / Kohchi, Masami / Hyoudoh, Ikumi et al. | 2009
- 1758
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4,4-Difluorinated analogues of l-arginine and NG-hydroxy-l-arginine as mechanistic probes for nitric oxide synthaseMartin, Nathaniel I. / Woodward, Joshua J. / Winter, Michael B. et al. | 2009
- 1763
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Antiproliferative effects of peracetylated naphthoxylosidesNilsson, Ulrika / Jacobsson, Mårten / Johnsson, Richard et al. | 2009
- 1767
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Atropisomeric small molecule Bcl-2 ligands: Determination of bioactive conformationPorter, John / Payne, Andrew / Whitcombe, Ian et al. | 2009
- 1773
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Synthesis, binding affinity and SAR of new benzolactam derivatives as dopamine D3 receptor ligandsOrtega, Raquel / Raviña, Enrique / Masaguer, Christian F. et al. | 2009
- 1779
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Synthesis and SAR of piperazinyl-N-phenylbenzamides as inhibitors of hepatitis C virus RNA replication in cell cultureConte, Immacolata / Giuliano, Claudio / Ercolani, Caterina et al. | 2009
- 1784
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Salicylate–urea-based soluble epoxide hydrolase inhibitors with high metabolic and chemical stabilitiesKasagami, Takeo / Kim, In-Hae / Tsai, Hsing-Ju et al. | 2009
- 1790
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Microbial biotransformation as a source of chemical diversity in cane toad steroid toxinsHayes, R. Andrew / Piggott, Andrew M. / Dalle, Kristian et al. | 2009
- 1793
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Relation between lipophilicity of alkyl gallates and antifungal activity against yeasts and filamentous fungiLeal, P.C. / Mascarello, A. / Derita, M. et al. | 2009
- 1797
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Discovery and optimization of piperidyl benzamide derivatives as a novel class of 11β-HSD1 inhibitorsRew, Yosup / McMinn, Dustin L. / Wang, Zhulun et al. | 2009
- 1797
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Discovery and optimization of piperidyl benzamide derivatives as a novel class of 11b-HSD1 inhibitorsRew, Y. / McMinn, D. L. / Wang, Z. et al. | 2009
- 1802
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The use of oxadiazole and triazole substituted naphthyridines as HIV-1 integrase inhibitors. Part 1: Establishing the pharmacophoreJohns, Brian A. / Weatherhead, Jason G. / Allen, Scott H. et al. | 2009
- 1807
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1,3,4-Oxadiazole substituted naphthyridines as HIV-1 integrase inhibitors. Part 2: SAR of the C5 positionJohns, Brian A. / Weatherhead, Jason G. / Allen, Scott H. et al. | 2009
- 1811
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Design, synthesis, and biological evaluation of novel 1-(1H-1,2,4-triazole-1-yl)-2-(2,4-difluorophenyl)-3-substituted benzylamino-2-propanolsChai, Xiaoyun / Zhang, Jun / Yu, Shichong et al. | 2009
- 1815
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Lithospermic acid derivatives from Lithospermum erythrorhizon increased expression of serine palmitoyltransferase in human HaCaT cellsThuong, Phuong Thien / Kang, Keon Wook / Kim, Jeong Kee et al. | 2009
- 1818
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Stereoselective synthesis of 15- and 16-substituted isosteviol derivatives and their cytotoxic activitiesWu, Ya / Dai, Gui-Fu / Yang, Jing-Hua et al. | 2008
- 1822
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Total synthesis and antihypertensive activity of (±)7,8-dihydroxy-3-methyl-isochromanone-4Liu, Jie / Ren, Hao / Xu, Jinyi et al. | 2008
- 1825
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14-O-Heterocyclic-substituted naltrexone derivatives as non-peptide mu opioid receptor selective antagonists: Design, synthesis, and biological studiesLi, Guo / Aschenbach, Lindsey C.K. / He, Hengjun et al. | 2008
- 1830
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Design, synthesis, and structure–activity relationship of novel CCR2 antagonistsKothandaraman, Shankaran / Donnely, Karla L. / Butora, Gabor et al. | 2008
- 1835
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Corrigendum to “Discovery, SAR and X-ray structure of 1H-benzimidazole-5-carboxylic acid cyclohexyl-methyl-amides as inhibitors of inducible T-cell kinase (Itk)” [Bioorg. Med. Chem. Lett. 18 (2008) 5545–5549]Moriarty, Kevin J. / Takahashi, Hidenori / Pullen, Steven S. et al. | 2008
- 1836
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Corrigendum to “Human ACAT-1 and -2 inhibitory activities of saucerneol B, manassantin A and B isolated from Saururus chinensis” [Bioorg. Med. Chem. Lett. 14 (2004) 3109–3112]Lee, Woo Song / Lee, Dae-Woo / Baek, Young-Il et al. | 2004
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Instructions to contributors| 2009
- IFC
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Editorial board| 2009