Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 5101
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Graphical contents list| 2005
- 5114
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Potent and highly selective kappa opioid receptor agonists incorporating chroman- and 2,3-dihydrobenzofuran-based constraintsChu, Guo-Hua / Gu, Minghua / Cassel, Joel A. et al. | 2005
- 5120
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Transforming bivalent ligands into retractable enzyme inhibitors through polypeptide#8211protein interactionsTolkatchev, Dmitri et al. | 2005
- 5120
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Transforming bivalent ligands into retractable enzyme inhibitors through polypeptide–protein interactionsTolkatchev, Dmitri / Vinogradova, Anna / Ni, Feng et al. | 2005
- 5124
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Estrogen receptor ligands. Part 14: Application of novel antagonist side chains to existing platformsBlizzard, Timothy A. / Morgan, Jerry D. II / Chan, Wanda et al. | 2005
- 5129
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Structural basis for the GSK-3β binding affinity and selectivity against CDK-2 of 1-(4-aminofurazan-3yl)-5-dialkylaminomethyl-1H-[1,2,3] triazole-4-carboxylic acid derivativesPande, Vineet / Ramos, Maria J. et al. | 2005
- 5129
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Structural basis for the GSK-3#946 binding affinity and selectivity against CDK-2 of 1-(4-aminofurazan-3yl)-5-dialkylaminomethyl-1H-(1,2,3) triazole-4-carboxylic acid derivativesPande, Vineet et al. | 2005
- 5136
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Carbonic anhydrase activators: X-ray crystal structure of the adduct of human isozyme II with l-histidine as a platform for the design of stronger activatorsTemperini, Claudia / Scozzafava, Andrea / Puccetti, Luca et al. | 2005
- 5142
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Highly sensitive peptide-based probes for protein tyrosine phosphatase activity utilizing a fluorogenic mimic of phosphotyrosineMitra, Sayantan / Barrios, Amy M. et al. | 2005
- 5146
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Design, synthesis, and evaluation of octahydropyranopyrrole-based inhibitors of mammalian ribonucleotide reductaseFuertes, Michael J. / Kaur, Jaskiran / Deb, Prasant et al. | 2005
- 5150
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Phosphinate, sulfonate, and sulfonamidate dipeptides as potential inhibitors of Escherichia coli aminopeptidase NYang, Ke-Wu / Golich, Frank C. / Sigdel, Tara K. et al. | 2005
- 5154
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Synthesis and structure–activity relationships of 1,2,4-triazoles as a novel class of potent tubulin polymerization inhibitorsOuyang, Xiaohu / Chen, Xiaoling / Piatnitski, Evgueni L. et al. | 2005
- 5154
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Synthesis and structure#8211activity relationships of 1,2,4-triazoles as a novel class of potent tubulin polymerization inhibitorsOuyang, Xiaohu et al. | 2005
- 5160
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Novel CCR1 antagonists with oral activity in the mouse collagen induced arthritisRevesz, Laszlo / Bollbuck, Birgit / Buhl, Thomas et al. | 2005
- 5165
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Quantitative structure–activity relationship studies of vitamin D receptor affinity for analogues of 1α,25-dihydroxyvitamin D3. 1: WHIM descriptorsGonzález, Maykel Pérez / Suárez, Pedro Lois / Fall, Yagamare et al. | 2005
- 5165
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Quantitative structure#8211activity relationship studies of vitamin D receptor affinity for analogues of 1#945,25-dihydroxyvitamin D3. 1: WHIM descriptorsGonzález, Maykel Pérez et al. | 2005
- 5170
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Nonsteroidal anti-inflammatory drugs and their analogues as inhibitors of aldo-keto reductase AKR1C3: New lead compounds for the development of anticancer agentsGobec, Stanislav / Brožič, Petra / Rižner, Tea Lanišnik et al. | 2005
- 5176
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Novel cell-penetrating #945-keto-amide calpain inhibitors as potential treatment for muscular dystrophyLescop, Cyrille et al. | 2005
- 5176
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Novel cell-penetrating α-keto-amide calpain inhibitors as potential treatment for muscular dystrophyLescop, Cyrille / Herzner, Holger / Siendt, Hervé et al. | 2005
- 5182
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Synthesis and biological evaluation of methoxylated analogs of the newer generation taxoids IDN5109 and IDN5390Barboni, Luciano / Ballini, Roberto / Giarlo, Guido et al. | 2005
- 5187
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Structure-based discovery of a new class of Hsp90 inhibitorsBarril, Xavier / Brough, Paul / Drysdale, Martin et al. | 2005
- 5192
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Carbonic anhydrase inhibitors: Inhibition of the human isozymes I, II, VA, and IX with a library of substituted difluoromethanesulfonamidesCecchi, Alessandro / Taylor, Scott D. / Liu, Yong et al. | 2005
- 5197
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3-(5-chloro-2,4-dihydroxyphenyl)-Pyrazole-4-carboxamides as inhibitors of the Hsp90 molecular chaperoneBrough, Paul A. / Barril, Xavier / Beswick, Mandy et al. | 2005
- 5202
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Heteroaryl-O-glucosides as novel sodium glucose co-transporter 2 inhibitors. Part 1Zhang, Xiaoyan / Urbanski, Maud / Patel, Mona et al. | 2005
- 5207
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In silico fragment-based discovery of indolin-2-one analogues as potent DNA gyrase inhibitorsOblak, Marko / Grdadolnik, Simona Golič / Kotnik, Miha et al. | 2005
- 5211
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Synthesis and evaluation of thiazole carboxamides as vanilloid receptor 1 (TRPV1) antagonistsXi, Ning / Bo, Yunxin / Doherty, Elizabeth M. et al. | 2005
- 5218
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A small library of trisubstituted pyrimidines as antimalarial and antitubercular agentsAgarwal, Anu / Srivastava, Kumkum / Puri, S.K. et al. | 2005
- 5222
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Synthesis and antitubercular activity of 2-hydroxy-aminoalkyl derivatives of diaryloxy methano phenanthrenesPanda, Gautam / Shagufta / Srivastava, Anil K. et al. | 2005
- 5226
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A lead compound for the development of ABA 8′-hydroxylase inhibitorsUeno, Kotomi / Yoneyama, Hidetaka / Saito, Shigeki et al. | 2005
- 5226
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A lead compound for the development of ABA 8#8242-hydroxylase inhibitorsUeno, Kotomi et al. | 2005
- 5230
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Self-complementary peptides for the formation of collagen-like triple helical supramoleculesKoide, Takaki / Homma, Daisuke L. / Asada, Shinichi et al. | 2005
- 5234
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Biaryl diamides as potent melanin concentrating hormone receptor 1 antagonistsPalani, Anandan / Shapiro, Sherry / McBriar, Mark D. et al. | 2005
- 5237
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Structure–activity relationship studies on a series of cyclohexylpiperazines bearing a phanylacetamide as ligands of the human melanocortin-4 receptorPontillo, Joseph / Tran, Joe A. / White, Nicole S. et al. | 2005
- 5237
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Structure#8211activity relationship studies on a series of cyclohexylpiperazines bearing a phanylacetamide as ligands of the human melanocortin-4 receptorPontillo, Joseph et al. | 2005
- 5241
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Discovery of a substituted 8-arylquinoline series of PDE4 inhibitors: Structure–activity relationship, optimization, and identification of a highly potent, well tolerated, PDE4 inhibitorMacdonald, Dwight / Mastracchio, Anthony / Perrier, Hélène et al. | 2005
- 5241
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Discovery of a substituted 8-arylquinoline series of PDE4 inhibitors: Structure#8211activity relationship, optimization, and identification of a highly potent, well tolerated, PDE4 inhibitorMacdonald, Dwight et al. | 2005
- 5247
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Synthesis, biological activity, and X-ray crystal structural analysis of diaryl ether inhibitors of malarial enoyl acyl carrier protein reductase. Part 1: 4′-Substituted triclosan derivativesFreundlich, Joel S. / Anderson, John W. / Sarantakis, Dimitri et al. | 2005
- 5247
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Synthesis, biological activity, and X-ray crystal structural analysis of diaryl ether inhibitors of malarial enoyl acyl carrier protein reductase. Part 1: 4#8242-Substituted triclosan derivativesFreundlich, Joel S. et al. | 2005
- 5253
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N-[(3S)-1-Benzylpyrrolidin-3-yl]-(2-thienyl)benzamides: Human dopamine D4 ligands with high affinity for the 5-HT2A receptorArora, Jalaj / Bordeleau, Michel / Dube, Laurence et al. | 2005
- 5257
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2-Cyano-4-fluoro-1-thiovalylpyrrolidine analogues as potent inhibitors of DPP-IVHaffner, Curt D. / McDougald, Darryl L. / Reister, Steven M. et al. | 2005
- 5262
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Photocurable hard and porous biomaterials from ROMP precursors cross-linked with diyl radicalsEnholm, Eric / Joshi, Aarti / Wright, Dennis L. et al. | 2005
- 5266
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Discovery of 4-heteroarylbicyclo[2.2.2]octyltriazoles as potent and selective inhibitors of 11β-HSD1: Novel therapeutic agents for the treatment of metabolic syndromeGu, Xin / Dragovic, Jasminka / Koo, Gloria C. et al. | 2005
- 5266
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Discovery of 4-heteroarylbicyclo(2.2.2)octyltriazoles as potent and selective inhibitors of 11#946-HSD1: Novel therapeutic agents for the treatment of metabolic syndromeGu, Xin et al. | 2005
- 5270
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Synthesis and ex vivo evaluation of carbon-11 labelled N-(4-methoxybenzyl)-N′-(5-nitro-1,3-thiazol-2-yl)urea ([11C]AR-A014418): A radiolabelled glycogen synthase kinase-3β specific inhibitor for PET studiesVasdev, Neil / Garcia, Armando / Stableford, Winston T. et al. | 2005
- 5270
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Synthesis and ex vivo evaluation of carbon-11 labelled N-(4-methoxybenzyl)-N#8242-(5-nitro-1,3-thiazol-2-yl)urea ((11C)AR-A014418): A radiolabelled glycogen synthase kinase-3#946 specific inhibitor for PET studiesVasdev, Neil et al. | 2005
- 5274
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Two classes of p38#945 MAP kinase inhibitors having a common diphenylether core but exhibiting divergent binding modesMichelotti, Enrique L. et al. | 2005
- 5274
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Two classes of p38α MAP kinase inhibitors having a common diphenylether core but exhibiting divergent binding modesMichelotti, Enrique L. / Moffett, Kristofer K. / Nguyen, Duyan et al. | 2005
- 5280
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Novel and expanded jadomycins incorporating non-proteogenic amino acidsJakeman, David L. / Graham, Cathy L. / Reid, Taryn R. et al. | 2005
- 5284
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Synthesis and biological evaluation of novel bisheterocycle-containing compounds as potential anti-influenza virus agentsWang, Wen-Long / Yao, De-Yong / Gu, Min et al. | 2005
- 5288
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Inhibition of Tpl2 kinase and TNF-#945 production with 1,7-naphthyridine-3-carbonitriles: Synthesis and structure#8211activity relationshipsGavrin, Lori Krim et al. | 2005
- 5288
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Inhibition of Tpl2 kinase and TNF-α production with 1,7-naphthyridine-3-carbonitriles: Synthesis and structure–activity relationshipsGavrin, Lori Krim / Green, Neal / Hu, Yonghan et al. | 2005
- 5293
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Aminopiperidine indazoles as orally efficacious melanin concentrating hormone receptor-1 antagonistsVasudevan, Anil / Souers, Andrew J. / Freeman, Jennifer C. et al. | 2005
- 5298
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Binding of amine-substituted N1-benzenesulfonylindoles at human 5-HT6 serotonin receptorsPullagurla, Manik / Siripurapu, Uma / Kolanos, Renata et al. | 2005
- 5303
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Photoregulation of DNA polymerase I (Klenow) with caged fluorescent oligodeoxynucleotidesTang, XinJing / Richards, Julia L. / Peritz, Adam E. et al. | 2005
- 5307
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Inhibitors of the serotonin transporter protein (SERT): The design and synthesis of biotinylated derivatives of 3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indoles. High-affinity serotonergic ligands for conjugation with quantum dotsTomlinson, Ian D. / Mason, John N. / Blakely, Randy D. et al. | 2005
- 5311
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Orally bioavailable highly potent HIV protease inhibitors against PI-resistant virusLu, Zhijian / Bohn, Joann / Rano, Tom et al. | 2005
- 5315
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A synthesis of 3-deoxydihydrolycoricidine: Refinement of a structurally minimum pancratistatin pharmacophoreMcNulty, James / Larichev, Vladimir / Pandey, Siyaram et al. | 2005
- 5319
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Inhibitors of phenylethanolamine N-methyltransferase devoid of α2-adrenoceptor affinityGrunewald, Gary L. / Lu, Jian / Criscione, Kevin R. et al. | 2005
- 5319
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Inhibitors of phenylethanolamine N-methyltransferase devoid of #9452-adrenoceptor affinityGrunewald, Gary L. et al. | 2005
- 5324
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Synthesis and biological evaluation of novel (l)-#945-amino acid methyl ester, heteroalkyl, and aryl substituted 1,4-naphthoquinone derivatives as antifungal and antibacterial agentsTandon, Vishnu K. et al. | 2005
- 5324
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Synthesis and biological evaluation of novel (l)-α-amino acid methyl ester, heteroalkyl, and aryl substituted 1,4-naphthoquinone derivatives as antifungal and antibacterial agentsTandon, Vishnu K. / Yadav, Dharmendra B. / Singh, Ravindra V. et al. | 2005
- 5329
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Geometric diversity through permutation of backbone configuration in cyclic peptide librariesPerlman, Zachary E. / Bock, Jonathan E. / Peterson, Jeffrey R. et al. | 2005
- 5335
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Novel 7-methoxy-6-oxazol-5-yl-2,3-dihydro-1H-quinazolin-4-ones as IMPDH inhibitorsBirch, Helen L. / Buckley, George M. / Davies, Natasha et al. | 2005
- 5340
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Rapamycin analogs with reduced systemic exposureWagner, Rolf / Mollison, Karl W. / Liu, Luping et al. | 2005
- 5344
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Selective and orally bioavailable phenylglycine tissue factor/factor VIIa inhibitorsZbinden, Katrin Groebke / Obst-Sander, Ulrike / Hilpert, Kurt et al. | 2005
- CO2
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Editorial Board| 2005
- I
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Contributors to this issue| 2005
- III
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Instructions to contributors| 2005