Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 4915
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Graphical contents list| 2008
- 4929
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Synthesis and activity of 1-(3-amino-1-phenylpropyl)indolin-2-ones: A new class of selective norepinephrine reuptake inhibitorsMcComas, Casey C. / Vu, An T. / Mahaney, Paige E. et al. | 2008
- 4932
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Structure–activity relationship study of a novel necroptosis inhibitor, necrostatin-7Zheng, Weihong / Degterev, Alexei / Hsu, Emily et al. | 2008
- 4936
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N-Alkyl-5H-pyrido[4,3-b]indol-1-amines and derivatives as novel urotensin-II receptor antagonistsWang, Yonghui / Wu, Zining / Guida, Brian F. et al. | 2008
- 4940
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New iodoreboxetine analogues for SPECT imaging of the noradrenaline transporterJobson, Nicola K. / Crawford, Andrew R. / Dewar, Deborah et al. | 2008
- 4944
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Design and synthesis of fluorescent SGLT2 inhibitorsLansdell, Mark I. / Burring, Denise J. / Hepworth, David et al. | 2008
- 4948
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Discovery of pyrazolopyrimidines as the first class of allosteric agonists for the high affinity nicotinic acid receptor GPR109AShen, Hong C. / Taggart, Andrew K.P. / Wilsie, Larissa C. et al. | 2008
- 4952
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Discovery of thieno[2,3-c]pyridines as potent COT inhibitorsGeorge, Dawn / Friedman, Michael / Allen, Hamish et al. | 2008
- 4956
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Phenylethyl cinnamides: A new series of a-glucosidase inhibitors from the leaves of Aegle marmelosPhuwapraisirisan, P. / Puksasook, T. / Jong-aramruang, J. et al. | 2008
- 4956
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Phenylethyl cinnamides: A new series of α-glucosidase inhibitors from the leaves of Aegle marmelosPhuwapraisirisan, Preecha / Puksasook, Thanchanok / Jong-aramruang, Jonkolnee et al. | 2008
- 4959
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New PPARγ ligands based on barbituric acid: Virtual screening, synthesis and receptor binding studiesSundriyal, Sandeep / Viswanad, Bhoomi / Ramarao, Poduri et al. | 2008
- 4959
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New PPARg ligands based on barbituric acid: Virtual screening, synthesis and receptor binding studiesSundriyal, S. / Viswanad, B. / Ramarao, P. et al. | 2008
- 4963
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Molecular modeling aided design of nicotinic acid receptor GPR109A agonistsDeng, Qiaolin / Frie, Jessica L. / Marley, Daria M. et al. | 2008
- 4968
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Synthesis of a 200-member library of squaric acid N-hydroxylamide amidesCharton, Julie / Déprez, Benoît P. / Déprez-Poulain, Rébecca F. et al. | 2008
- 4972
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Pharmacophore modeling and virtual screening for designing potential PLK1 inhibitorsWang, Hui-Yuan / Cao, Zhi-Xing / Li, Lin-Li et al. | 2008
- 4978
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Synthesis of N-isobutylnoroxymorphone from naltrexone by a selective cyclopropane ring opening reactionFujii, Hideaki / Osa, Yumiko / Ishihara, Marina et al. | 2008
- 4982
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Synthesis and SAR study of N-(4-hydroxy-3-(2-hydroxynaphthalene-1-yl)phenyl)-arylsulfonamides: Heat shock protein 90 (Hsp90) inhibitors with submicromolar activity in an in vitro assayGanesh, Thota / Thepchatri, Pahk / Li, Lian et al. | 2008
- 4988
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Discovery of the catechol structural moiety as a Stat3 SH2 domain inhibitor by virtual screeningHao, Wenshan / Hu, Yongbo / Niu, Chuansheng et al. | 2008
- 4993
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Design, synthesis, and evaluation of novel aryl-tetrahydropyridine PPARα/γ dual agonistsKim, Eunkyung / Park, Chan Sun / Han, Taedong et al. | 2008
- 4993
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Design, synthesis, and evaluation of novel aryl-tetrahydropyridine PPARa/g dual agonistsKim, E. / Park, C. S. / Han, T. et al. | 2008
- 4997
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Syntheses and structure–activity relationships of novel, potent, and selective trans-2-[3-oxospiro[isobenzofuran-1(3H),1′-cyclohexan]-4′-yl]benzimidazole NPY Y5 receptor antagonistsOgino, Yoshio / Ohtake, Norikazu / Nagae, Yoshikazu et al. | 2008
- 4997
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Syntheses and structure-activity relationships of novel, potent, and selective trans-2-[3-oxospiro[isobenzofuran-1(3H),1prime-cyclohexan]-4prime-yl]benzimidazole NPY Y5 receptor antagonistsOgino, Y. / Ohtake, N. / Nagae, Y. et al. | 2008
- 5002
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Hexahydro-pyrrolo- and hexahydro-1H-pyrido[1,2-b]pyridazin-2-ones as potent inhibitors of HCV NS5B polymeraseRuebsam, Frank / Sun, Zhongxiang / Ayida, Benjamin K. et al. | 2008
- 5006
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ortho-Dihydroxyisoflavone derivatives from aged Doenjang (Korean fermented soypaste) and its radical scavenging activityPark, Jun-Seong / Park, Hye Yoon / Kim, Dong Hyun et al. | 2008
- 5010
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Design, syntheses, and structure–activity relationships of novel NPY Y5 receptor antagonists: 2-{3-Oxospiro[isobenzofuran-1(3H),4′-piperidin]-1′-yl}benzimidazole derivativesOgino, Yoshio / Ohtake, Norikazu / Nagae, Yoshikazu et al. | 2008
- 5010
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Design, syntheses, and structure-activity relationships of novel NPY Y5 receptor antagonists: 2-{3-Oxospiro[isobenzofuran-1(3H),4prime-piperidin]-1prime-yl}benzimidazole derivativesOgino, Y. / Ohtake, N. / Nagae, Y. et al. | 2008
- 5015
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1,5-Dihydro-benzo[e][1,4]oxazepin-2(1H)-ones containing a 7-(5prime-cyanopyrrol-2-yl) group as nonsteroidal progesterone receptor modulatorsKern, J. C. / Terefenko, E. A. / Fensome, A. et al. | 2008
- 5015
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1,5-Dihydro-benzo[e][1,4]oxazepin-2(1H)-ones containing a 7-(5′-cyanopyrrol-2-yl) group as nonsteroidal progesterone receptor modulatorsKern, Jeffrey C. / Terefenko, Eugene A. / Fensome, Andrew et al. | 2008
- 5018
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Discovery of a novel class of PPARδ partial agonistsShearer, Barry G. / Patel, Hari S. / Billin, Andrew N. et al. | 2008
- 5018
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Discovery of a novel class of PPARd partial agonistsShearer, B. G. / Patel, H. S. / Billin, A. N. et al. | 2008
- 5023
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Structure-guided design of substituted aza-benzimidazoles as potent hypoxia inducible factor-1a prolyl hydroxylase-2 inhibitorsFrohn, M. / Viswanadhan, V. / Pickrell, A. J. et al. | 2008
- 5023
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Structure-guided design of substituted aza-benzimidazoles as potent hypoxia inducible factor-1α prolyl hydroxylase-2 inhibitorsFrohn, Mike / Viswanadhan, Vellarkad / Pickrell, Alexander J. et al. | 2008
- 5027
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1-Benzylbenzimidazoles: The discovery of a novel series of bradykinin B1 receptor antagonistsGuo, Qin / Chandrasekhar, Jayaraman / Ihle, David et al. | 2008
- 5032
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Benzimidazole-substituted (3-phenoxypropyl)amines as histamine H3 receptor ligandsAslanian, Robert / Zhu, Xiaohong / Vaccaro, Henry A. et al. | 2008
- 5037
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Discovery of novel series of benzoic acid derivatives containing biphenyl ether moiety as potent and selective human β3-adrenergic receptor agonists: Part IVNakajima, Yutaka / Imanishi, Masashi / Itou, Shinji et al. | 2008
- 5037
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Discovery of novel series of benzoic acid derivatives containing biphenyl ether moiety as potent and selective human b3-adrenergic receptor agonists: Part IVNakajima, Y. / Imanishi, M. / Itou, S. et al. | 2008
- 5041
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Synthesis and biological evaluation of 2-amino-3-(3′,4′,5′-trimethoxybenzoyl)-6-substituted-4,5,6,7-tetrahydrothieno[2,3-c]pyridine derivatives as antimitotic agents and inhibitors of tubulin polymerizationRomagnoli, Romeo / Baraldi, Pier Giovanni / Carrion, Maria Dora et al. | 2008
- 5041
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Synthesis and biological evaluation of 2-amino-3-(3prime,4prime,5prime-trimethoxybenzoyl)-6-substituted-4,5,6,7-tetrahydrothieno[2,3-c]pyridine derivatives as antimitotic agents and inhibitors of tubulin polymerizationRomagnoli, R. / Baraldi, P. G. / Carrion, M. D. et al. | 2008
- 5046
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Impacts of baicalein analogs with modification of the 6th position of A ring on the activity toward NF-κB-, AP-1-, or CREB-mediated transcriptionHuang, Sheng-Teng / Lee, Yashang / Gullen, Elizabeth A. et al. | 2008
- 5046
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Impacts of baicalein analogs with modification of the 6th position of A ring on the activity toward NF-kB-, AP-1-, or CREB-mediated transcriptionHuang, S. T. / Lee, Y. / Gullen, E. A. et al. | 2008
- 5050
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Promising core structure for nuclear receptor ligands: Design and synthesis of novel estrogen receptor ligands based on diphenylamine skeletonOhta, Kiminori / Chiba, Yuki / Ogawa, Takumi et al. | 2008
- 5054
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PNA/DNA interstrand cross-links from a modified PNA base upon photolysis or oxidative conditionsKim, Yongtae / Hong, In Seok et al. | 2008
- 5058
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Synthesis and cytotoxic activity of heterocyclic ring-substituted betulinic acid derivativesKumar, Vivek / Rani, Nidhi / Aggarwal, Pawan et al. | 2008
- 5063
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Synthesis and evaluation of cis-3,4-disubstituted piperidines as potent CC chemokine receptor 2 (CCR2) antagonistsCherney, Robert J. / Nelson, David J. / Lo, Yvonne C. et al. | 2008
- 5066
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Carbonic anhydrase inhibitors: Inhibition of the β-class enzymes from the fungal pathogens Candida albicans and Cryptococcus neoformans with simple anionsInnocenti, Alessio / Mühlschlegel, Fritz A. / Hall, Rebecca A. et al. | 2008
- 5066
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Carbonic anhydrase inhibitors: Inhibition of the b-class enzymes from the fungal pathogens Candida albicans and Cryptococcus neoformans with simple anionsInnocenti, A. / Muhlschlegel, F. A. / Hall, R. A. et al. | 2008
- 5071
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Design, synthesis and preliminary biological evaluation of new hydroxamate histone deacetylase inhibitors as potential antileukemic agentsGuandalini, L. / Cellai, C. / Laurenzana, A. et al. | 2008
- 5075
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Synthesis of 3-alkyl naphthalenes as novel estrogen receptor ligandsFang, Jing / Akwabi-Ameyaw, Adwoa / Britton, Jonathan E. et al. | 2008
- 5078
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Design, synthesis, and antibacterial activities of novel 3,6-bicyclolide oximes: Length optimization and zero carbon linker oximesTang, Datong / Gai, Yonghua / Polemeropoulos, Alexander et al. | 2008
- 5083
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Discovery and optimization of (R)-prolinol-derived agonists of the Growth Hormone Secretagogue receptor (GHSR)Zhai, Weixu / Flynn, Neil / Longhi, Daniel A. et al. | 2008
- 5087
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Synthesis and antibacterial activity of the C-7 side chain of 3-aminoquinazolinedionesHutchings, Kim M. / Tran, Tuan P. / Ellsworth, Edmund L. et al. | 2008
- 5091
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Design, synthesis, and bioactivity of putative tubulin ligands with adamantane coreZefirova, Olga N. / Nurieva, Evgeniya V. / Lemcke, Heiko et al. | 2008
- 5095
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Discovery of novel potent and selective dipeptide hepatitis C virus NS3/4A serine protease inhibitorsRaboisson, Pierre / Lin, Tse-I / Kock, Herman de et al. | 2008
- 5101
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Synthesis and evaluation of a spiro-isobenzofuranone class of histamine H3 receptor inverse agonistsJitsuoka, Makoto / Tsukahara, Daisuke / Ito, Sayaka et al. | 2008
- 5107
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Bradykinin B1 receptor antagonists: An α-hydroxy amide with an improved metabolism profileKuduk, Scott D. / Chang, Ronald K. / DiPardo, Robert M. et al. | 2008
- 5107
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Bradykinin B1 receptor antagonists: An a-hydroxy amide with an improved metabolism profileKuduk, S. D. / Chang, R. K. / DiPardo, R. M. et al. | 2008
- 5111
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Novel hypoglycemic dihydropyridones serendipitously discovered from O- versus C-alkylation in the synthesis of VMAT2 antagonistsXie, Yuli / Raffo, Anthony / Ichise, Masanori et al. | 2008
- 5115
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Discovery of amido-benzisoxazoles as potent c-Kit inhibitorsKunz, Roxanne K. / Rumfelt, Shannon / Chen, Ning et al. | 2008
- 5118
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Substituted aryl pyrimidines as potent and soluble TRPV1 antagonistsStec, Markian M. / Bo, Yunxin / Chakrabarti, Partha P. et al. | 2008
- 5123
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Synthesis and anti-CVB 3 evaluation of substituted 5-nitro-2-phenoxybenzonitrilesPürstinger, Gerhard / De Palma, Armando M. / Zimmerhofer, Günther et al. | 2008
- 5126
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Identification of ring-fused pyrazolo pyridin-2-ones as novel poly(ADP-ribose)polymerase-1 inhibitorsMoree, Wilna J. / Goldman, Phyllis / Demaggio, Anthony J. et al. | 2008
- 5130
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7-[1H-Indol-2-yl]-2,3-dihydro-isoindol-1-ones as dual Aurora-A/VEGF-R2 kinase inhibitors: Design, synthesis, and biological activityHughes, Terry V. / Emanuel, Stuart L. / O’Grady, Harold R. et al. | 2008
- 5134
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Discovery of benzoylpiperazines as a novel class of potent and selective GlyT1 inhibitorsPinard, Emmanuel / Alberati, Daniela / Borroni, Edilio et al. | 2008
- 5140
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Synthesis and biological affinity of new imidazo- and indol-arylpiperazine derivatives: Further validation of a pharmacophore model for α1-adrenoceptor antagonistsStrappaghetti, Giovannella / Mastrini, Luciano / Lucacchini, Antonio et al. | 2008
- 5140
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Synthesis and biological affinity of new imidazo- and indol-arylpiperazine derivatives: Further validation of a pharmacophore model for a1-adrenoceptor antagonistsStrappaghetti, G. / Mastrini, L. / Lucacchini, A. et al. | 2008
- 5146
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Design, synthesis, biochemical, and biological evaluation of nitrogen-containing trifluoro structural modifications of combretastatin A-4Hall, John J. / Sriram, Madhavi / Strecker, Tracy E. et al. | 2008
- 5150
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Novel and potent oxazolidinone antibacterials featuring 3-indolylglyoxamide substituentsTakhi, Mohamed / Singh, Gurpreet / Murugan, C. et al. | 2008
- 5156
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Erratum to “Structural modifications of N-arylamide oxadiazoles: Identification of N-arylpiperidine oxadiazoles as potent and selective agonists of CB2” [Bioorg. Med. Chem. Lett. 18 (2008) 4267–4274]DiMauro, Erin F. / Buchanan, John L. / Chen, Alan et al. | 2008
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Instructions to contributors| 2008
- IFC
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Editorial board| 2008