Bioorganic and Medicinal Chemistry Letters
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Table of contents
- 553
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Graphical contents list| 2004
- 569
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Publisher's Announcement—new Regional Editor for Bioorganic & Medicinal Chemistry| 2003
- 571
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Inhibition kinetics of carba- and C-fucosyl analogues of GDP-fucose against fucosyltransferase V: implication for the reaction mechanismNorris, Andrew J. / Whitelegge, Julian P. / Strouse, M.Jane et al. | 2003
- 575
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Synthesis and biological evaluation of (−)-laulimalide analoguesGallagher, Brian M. Jr. / Fang, Francis G. / Johannes, Charles W. et al. | 2003
- 581
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Synthesis and incorporation of an a-hexofuranosyl thymidine into oligodeoxynucleotides via its two exocyclic OH-groupsFilichev, Vyacheslav V. et al. | 2004
- 581
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Synthesis and incorporation of an α-hexofuranosyl thymidine into oligodeoxynucleotides via its two exocyclic OH-groupsFilichev, Vyacheslav V. / Pedersen, Erik B. et al. | 2003
- 585
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Chemoenzymatic synthesis and binding affinity of novel (R)- and (S)-3-aminomethyl-1-tetralones, potential atypical antipsychoticsCaro, Yolanda / Torrado, Marı́a / Masaguer, Christian F. et al. | 2003
- 591
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Aza-bicyclic amino acid sulfonamides as α4β1/α4β7 integrin antagonistsDyatkin, Alexey B / Hoekstra, William J / Kinney, William A et al. | 2003
- 591
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Aza-bicyclic amino acid sulfonamides as a4b1-a4b7 integrin antagonistsDyatkin, Alexey B. et al. | 2004
- 597
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Synthesis of new thiophene and benzo[b]thiophene hydrazide derivatives as human NPY Y5 antagonistsGaliano, Silvia / Erviti, Oihana / Pérez, Silvia et al. | 2003
- 601
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Rational design and synthesis of selective BACE-1 inhibitorsBrady, Stephen F. / Singh, Satendra / Crouthamel, Ming-Chih et al. | 2003
- 605
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Inhibition of estrone sulfatase (ES) by alkyl and cycloalkyl ester derivatives of 4-[(aminosulfonyl)oxy] benzoic acidPatel, Chirag K. / Owen, Caroline P. / Ahmed, Sabbir et al. | 2003
- 611
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Synthesis and biological evaluation of novel coumarin derivatives with a 7-azomethine linkageKontogiorgis, Christos A. / Hadjipavlou-Litina, Dimitra J. et al. | 2003
- 615
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Diamine derivatives with antiparasitic activitiesLabadie, Guillermo R. / Choi, Seoung-Ryoung / Avery, Mitchell A. et al. | 2003
- 621
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Synthesis and antitumor activity of 10-substituted benzylidene anthroneHu, Weixiao / Zhou, Wei et al. | 2003
- 623
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Permeation and metabolism of a series of novel lipophilic ascorbic acid derivatives, 6-O-acyl-2-O-a-d-glucopyranosyl-l-ascorbic acids with a branched-acyl chain, in a human living skin equivalent modelTai, Akihiro et al. | 2004
- 623
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Permeation and metabolism of a series of novel lipophilic ascorbic acid derivatives, 6-O-acyl-2-O-α-d-glucopyranosyl-l-ascorbic acids with a branched-acyl chain, in a human living skin equivalent modelTai, Akihiro / Goto, Satomi / Ishiguro, Yutaka et al. | 2003
- 629
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Synthesis and mitochondrial complex I inhibition of dihydroxy-cohibin A, non-THF annonaceous acetogenin analogueKonno, Hiroyuki / Hiura, Naoki / Makabe, Hidefumi et al. | 2003
- 633
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Synthesis and biological activity of a novel squalene epoxidase inhibitor, FR194738Sawada, Masae / Washizuka, Ken-ichi / Okumura, Hiroyuki et al. | 2003
- 639
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Macrocyclic piperazinones as potent dual inhibitors of farnesyltransferase and geranylgeranyltransferase-IDinsmore, Christopher J / Zartman, C.Blair / Bergman, Jeffrey M et al. | 2003
- 645
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Degradation of target protein in living cells by small-molecule proteolysis inducerZhang, Dong / Baek, Sun-Hee / Ho, Abby et al. | 2003
- 649
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Biosynthesis of agglomerin A: stereospecific incorporation of pro-R- and pro-S-hydrogens at sn-C-3 of glycerol into the branched C3 moietyMashimo, Youichi / Sekiyama, Yasuyo / Araya, Hiroshi et al. | 2003
- 653
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Synthesis and antifungal activities of phenylenedithioureasPhuong, Truong / Khac-Minh, Thai / Van Ha, Nguyen Thi et al. | 2003
- 657
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Solid-phase synthesis of a small library of 3-phenylthio-3-nicotinyl propionic acid derivatives acting as antagonists of the integrin aVb3Vianello, Paola et al. | 2004
- 657
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Solid-phase synthesis of a small library of 3-phenylthio-3-nicotinyl propionic acid derivatives acting as antagonists of the integrin αVβ3Vianello, Paola / Cozzi, Paolo / Galvani, Arturo et al. | 2003
- 663
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TMC-95A, a reversible proteasome inhibitor, induces neurite outgrowth in PC12 cellsInoue, Masayuki / Zhai, Haifeng / Sakazaki, Hayato et al. | 2003
- 667
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Manipulation of kinetic profiles in 2-aryl propionic acid cyclooxygenase inhibitorsGupta, Kushol / Kaub, Carl J. / Carey, Kristen N. et al. | 2003
- 673
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Structure–activity relationships of non-imidazole H3 receptor ligands. Part 3: 5-Substituted 3-phenyl-1,2,4-oxadiazoles as potent antagonistsGfesser, Gregory A. / Zhang, Henry / Dinges, Jurgen et al. | 2003
- 677
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Thiazoles and thiopyridines: novel series of high affinity h5HT7 ligandsThomson, Christopher G. / Beer, Margaret S. / Curtis, Neil R. et al. | 2003
- 681
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2-Hydroxy-4-isopropylbenzaldehyde, a potent partial tyrosinase inhibitorNihei, Ken-ichi / Yamagiwa, Yoshiro / Kamikawa, Tadao et al. | 2003
- 685
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Peptidyl aldehydes as slow-binding inhibitors of dual-specificity phosphatasesPark, Junguk / Fu, Hua / Pei, Dehua et al. | 2003
- 689
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A new class of potent non-imidazole H3 antagonists: 2-aminoethylbenzofuransCowart, Marlon / Pratt, John K. / Stewart, Andrew O. et al. | 2003
- 695
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Synthesis and evaluation of novel bacterial rRNA-binding benzimidazoles by mass spectrometryHe, Yun / Yang, Jun / Wu, Baogen et al. | 2003
- 701
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Inhibition of α-chymotrypsin with thiol-bearing substrate analogues in the presence of zinc ionHan, Min Su / Oh, Dong Ju / Kim, Dong H. et al. | 2003
- 701
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Inhibition of a-chymotrypsin with thiol-bearing substrate analogues in the presence of zinc ionHan, Min Su et al. | 2004
- 707
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QSAR Studies of PC-3 cell line inhibition activity of TSA and SAHA-like hydroxamic acidsWang, Di-Fei / Wiest, Olaf / Helquist, Paul et al. | 2003
- 713
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Rational design of azepane-glycoside antibiotics targeting the bacterial ribosomeBarluenga, Sofia / Simonsen, Klaus B. / Littlefield, Ethel S. et al. | 2003
- 719
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Design of small molecule ketoamide-based inhibitors of cathepsin KCatalano, John G. / Deaton, David N. / Long, Stacey T. et al. | 2003
- 723
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Enantioselective ester hydrolysis catalyzed by b-cyclodextrin conjugated with b-hairpin peptidesTsutsumi, Hiroshi et al. | 2004
- 723
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Enantioselective ester hydrolysis catalyzed by β-cyclodextrin conjugated with β-hairpin peptidesTsutsumi, Hiroshi / Ikeda, Hiroshi / Mihara, Hisakazu et al. | 2003
- 727
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3-(2-Pyrrolidin-1-ylethyl)-5-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole derivatives as high affinity human 5-HT1B/1D ligandsEgle, Ian / MacLean, Neil / Demchyshyn, Lidia et al. | 2003
- 731
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3D-QSAR studies on PU3 analogues by comparative molecular field analysisLiu, Hong-Chong / Lyu, Ping-Chiang / Leong, Max K. et al. | 2003
- 735
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Vancomycin disulfide derivatives as antibacterial agentsMu, YongQi / Nodwell, Matthew / Pace, John L. et al. | 2003
- 739
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Novel nevirapine-like inhibitors with improved activity against NNRTI-resistant HIV: 8-heteroarylthiomethyldipyridodiazepinone derivativesYoakim, C. / Bonneau, P.R. / Déziel, R. et al. | 2003
- 743
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Fluorinated dihydroquinolines as potent n-NOS inhibitorsJaroch, Stefan / Rehwinkel, Hartmut / Hölscher, Peter et al. | 2003
- 747
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Synthesis and biological results of the technetium-99m-labeled 4-nitroimidazole for imaging tumor hypoxiaChu, Taiwei / Hu, Shaowen / Wei, Bing et al. | 2003
- 751
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Benzene-di-N-octylcarbamates as conformationally constrained phospholipase A2 inhibitorsLin, Gialih / Lin, Yan-Fu / Hwang, Mei-Ting et al. | 2003
- 757
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Synthesis and antibiotic activity of the tricyclic furo[3,2-c] isochromen-2-trione unit of the pyranonaphthoquinonesBianchi, Darı́o A. / Sutich, Emma G. / Kaufman, Teodoro S. et al. | 2003
- 761
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Synthesis and biological evaluation of piperazine-based derivatives as inhibitors of plasminogen activator inhibitor-1 (PAI-1)Ye, Bin / Chou, Yuo-Ling / Karanjawala, Rushad et al. | 2003
- 767
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Synthesis of N,Nprime-disubstituted 3-aminobenzo[c] and [d]azepin-2-ones as potent and specific farnesyl transferase inhibitorsLe Diguarher, T. / Ortuno, J. C. / Shanks, D. et al. | 2004
- 767
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Synthesis of N,N′-disubstituted 3-aminobenzo[c] and [d]azepin-2-ones as potent and specific farnesyl transferase inhibitorsLe Diguarher, Thierry / Ortuno, Jean-Claude / Shanks, David et al. | 2003
- 773
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Bile acid amides derived from chiral amino alcohols: novel antimicrobials and antifungalsHazra, BrajaG. / Pore, VandanaS. / Dey, SanjeevKumar et al. | 2003
- 779
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Essential structural features of acetogenins: role of hydroxy groups adjacent to the bis-THF ringsAbe, Masato / Kenmochi, Atsushi / Ichimaru, Naoya et al. | 2003
- 783
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Omega-carboxypyridyl substituted ureas as Raf kinase inhibitorsKhire, Uday R. / Bankston, Donald / Barbosa, James et al. | 2003
- 783
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Omega-carboxypyridyl substituted ureas as Raf kinase inhibitors - SAR of the amide substituentKhire, Uday R. et al. | 2004
- 787
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N-4-Substituted-benzyl-N′-tert-butylbenzyl thioureas as vanilloid receptor ligands: investigation on the role of methanesulfonamido group in antagonistic activityPark, Hyeung-geun / Choi, Ji-yeon / Choi, Sea-hoon et al. | 2003
- 787
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N-4-Substituted-benzyl-Nprime-tert-butylbenzyl thioureas as vanilloid receptor ligands: investigation on the role of methanesulfonamido group in antagonistic activityPark, H. g. / Choi, J. y. / Choi, S. h. et al. | 2004
- 793
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Discovery of thiophene-2-carboxylic acids as potent inhibitors of HCV NS5B polymerase and HCV subgenomic RNA replication. Part 1: SulfonamidesChan, Laval / Das, Sanjoy K. / Reddy, T.Jagadeeswar et al. | 2003
- 797
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Discovery of thiophene-2-carboxylic acids as potent inhibitors of HCV NS5B polymerase and HCV subgenomic RNA replication. Part 2: Tertiary amidesChan, Laval / Pereira, Oswy / Reddy, T.Jagadeeswar et al. | 2003
- 801
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Synthesis of oligonucleotide 2′-conjugates via amide bond formation in solutionKachalova, Anna V. / Stetsenko, Dmitry A. / Gait, Michael J. et al. | 2003
- 801
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Synthesis of oligonucleotide 2prime-conjugates via amide bond formation in solutionKachalova, A. V. / Stetsenko, D. A. / Gait, M. J. et al. | 2004
- 805
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Discovery of novel aspartyl ketone dipeptides as potent and selective caspase-3 inhibitorsHan, Yongxin / Giroux, André / Grimm, Erich L. et al. | 2003
- 809
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The design and synthesis of sulfonamides as caspase-1 inhibitorsHarter, William G. / Albrect, Hans / Brady, Kenneth et al. | 2003
- 813
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3-Trifluoromethyl-4-nitro-5-arylpyrazoles are novel KATP channel agonistsPeat, Andrew J. / Townsend, Claire / Craig McKay, M. et al. | 2003
- 817
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Synthesis and SAR evaluation of 1,2,4-triazoles as A2A receptor antagonistsAlanine, Alexander / Anselm, Lilli / Steward, Lucinda et al. | 2003
- CO2
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Editorial Board| 2004
- I
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Contributors to this issue| 2004
- III
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Instuctions to Contributors| 2004