Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
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Graphical contents list| 2013
- 21
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Design of small molecule epigenetic modulatorsPachaiyappan, Boobalan / Woster, Patrick M. et al. | 2013
- 33
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Drug discovery considerations in the development of covalent inhibitorsMah, Robert / Thomas, Jason R. / Shafer, Cynthia M. et al. | 2013
- 40
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Design, synthesis and anti-Alzheimer properties of dimethylaminomethyl-substituted curcumin derivativesFang, Lei / Gou, Shaohua / Liu, Xuying et al. | 2013
- 44
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Sortase A inhibitory metabolites from the roots of Pulsatilla koreanaLee, Sooryun / Song, Inn-Hye / Lee, Jung-Ho et al. | 2013
- 49
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Synthesis and biological evaluation of @a-hydroxyalkylphosphonates as new antimicrobial agentsFaisca Phillips, A. M. / Barros, M. T. / Pacheco, M. et al. | 2014
- 49
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Synthesis and biological evaluation of α-hydroxyalkylphosphonates as new antimicrobial agentsFaísca Phillips, Ana Maria / Barros, Maria Teresa / Pacheco, Marta et al. | 2013
- 54
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Synthesis, biological evaluation and SAR of 3-benzoates of ingenol for treatment of actinic keratosis and non-melanoma skin cancerGrue-Sørensen, Gunnar / Liang, Xifu / Månsson, Kristoffer et al. | 2013
- 61
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Lactam based 7-amino suberoylamide hydroxamic acids as potent HDAC inhibitorsTaddei, Maurizio / Cini, Elena / Giannotti, Luca et al. | 2013
- 65
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Novel anthraquinone based chalcone analogues containing an imine fragment: Synthesis, cytotoxicity and anti-angiogenic activityKolundžija, Branka / Marković, Violeta / Stanojković, Tatjana et al. | 2013
- 72
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The discovery of potent, orally bioavailable pyrazolo and triazolopyrimidine CXCR2 receptor antagonistsPorter, David W. / Bradley, Michelle / Brown, Zarin et al. | 2013
- 77
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Rationally designed hybrid molecules with appreciable COX-2 inhibitory and anti-nociceptive activitiesSingh, Palwinder / Shaveta / Sharma, Surbhi et al. | 2013
- 83
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Verrulactone C with an unprecedented dispiro skeleton, a new inhibitor of Staphylococcus aureus enoyl-ACP reductase, from Penicillium verruculosum F375Kim, Nyung / Sohn, Mi-Jin / Koshino, Hiroyuki et al. | 2013
- 87
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Design and synthesis of tamoxifen derivatives as a selective estrogen receptor down-regulatorShoda, Takuji / Okuhira, Keiichiro / Kato, Masashi et al. | 2013
- 90
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Design, synthesis and antibacterial activities of 5-(pyrazin-2-yl)-4H-1,2,4-triazole-3-thiol derivatives containing Schiff base formation as FabH inhibitoryZhang, Fei / Wen, Qing / Wang, She-Feng et al. | 2013
- 96
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Syntheses of novel β-carboline derivatives and the activities against five tumor-cell linesBai, Bing / Li, Xing-Yao / Liu, Li et al. | 2013
- 96
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Syntheses of novel @b-carboline derivatives and the activities against five tumor-cell linesBai, B. / Li, X. Y. / Liu, L. et al. | 2014
- 99
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TMEDA-derived biscationic amphiphiles: An economical preparation of potent antibacterial agentsBlack, Jacob W. / Jennings, Megan C. / Azarewicz, Julianne et al. | 2013
- 103
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A tetradecapeptide somatostatin dicarba-analog: Synthesis, structural impact and biological activityMartín-Gago, Pablo / Ramón, Rosario / Aragón, Eric et al. | 2013
- 108
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Structure activity relationships of fused bicyclic and urea derivatives of spirocyclic compounds as potent CCR1 antagonistsHossain, Nafizal / Mensonides-Harsema, Marguérite / Cooper, Martin E. et al. | 2013
- 113
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Azide–alkyne cycloaddition affording enzymatically tunable bisubstrate based inhibitors of histone acetyltransferase PCAFvan Ameijde, Jeroen / Zwiebel, Addy P.R. / Ruijtenbeek, Rob et al. | 2013
- 117
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Fluorescent probes of the isoxazole–dihydropyridine scaffold: MDR-1 binding and homology modelSzabon-Watola, Monika I. / Ulatowski, Sarah V. / George, Kathleen M. et al. | 2013
- 122
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Chemical synthesis and tyrosinase inhibitory activity of rhododendrol glycosidesIwadate, Takehiro / Kashiwakura, Yutaka / Masuoka, Noriyoshi et al. | 2013
- 126
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Identification of quinones as HER2 inhibitors for the treatment of trastuzumab resistant breast cancerSridhar, Jayalakshmi / Sfondouris, Mary E. / Bratton, Melyssa R. et al. | 2013
- 132
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Synthesis and biological properties of thiazole-analogues of pyochelin, a siderophore of Pseudomonas aeruginosaNoël, Sabrina / Hoegy, Françoise / Rivault, Freddy et al. | 2013
- 136
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New titanocene derivatives with high antiproliferative activity against breast cancer cellsSaturnino, Carmela / Sirignano, Esther / Botta, Antonio et al. | 2013
- 141
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Synthesis and biological evaluation of cyclopentyl-triazolol-pyrimidine (CPTP) based P2Y12 antagonistsTu, Wangyang / Fan, Jiang / Zhang, Haitang et al. | 2013
- 147
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Synthesis and anticancer potential of benzothiazole linked phenylpyridopyrimidinones and their diones as mitochondrial apoptotic inducersKamal, Ähmed / Ashraf, Md. / Vishnu Vardhan, M.V.P.S. et al. | 2013
- 152
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Replacement of amide with bioisosteres led to a new series of potent adenosine A2A receptor antagonistsYang, Zhaohui / Li, Xuan / Ma, Haikuo et al. | 2013
- 156
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Discovery and optimization of N-(3-(1,3-dioxo-2,3-dihydro-1H-pyrrolo[3,4-c]pyridin-4-yloxy)phenyl)benzenesulfonamides as novel GPR119 agonistsYu, Ming / Wang, Yingcai / Zhu, Jiang et al. | 2013
- 161
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Synthesis and SAR of novel isoxazoles as potent c-jun N-terminal kinase (JNK) inhibitorsHe, Yuanjun / Duckett, Derek / Chen, Weimin et al. | 2013
- 165
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Synthesis and antimycobacterial activity of novel camphane-based agentsStavrakov, Georgi / Philipova, Irena / Valcheva, Violeta et al. | 2013
- 168
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Cassaine diterpene alkaloids from Erythrophleum fordii and their anti-angiogenic effectHung, Tran Manh / Cuong, To Dao / Kim, Jeong Ah et al. | 2013
- 173
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pH-rate profiles of l-arabinitol 4-dehydrogenase from Hypocrea jecorina and its application in l-xylulose productionTiwari, Manish Kumar / Singh, Raushan Kumar / Gao, Hui et al. | 2013
- 177
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The identification of AF38469: An orally bioavailable inhibitor of the VPS10P family sorting receptor SortilinSchrøder, Tenna Juul / Christensen, Søren / Lindberg, Samsa et al. | 2013
- 181
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Synthesis of licochalcone analogues with increased anti-inflammatory activityKim, Si-Jun / Kim, Cheol Gi / Yun, So-Ra et al. | 2013
- 186
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Cytotoxic activity of gypenosides and gynogenin against non-small cell lung carcinoma A549 cellsChen, Dao-Jin / Liu, Hui-Min / Xing, Shao-Fang et al. | 2013
- 192
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Synthesis and evaluation of novel azoles as potent antifungal agentsLi, Liangjing / Ding, Hao / Wang, Baogang et al. | 2013
- 195
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Linker modification reduced the renal uptake of technetium-99m-labeled Arg-Ala-Asp-conjugated alpha-melanocyte stimulating hormone peptideYang, Jianquan / Flook, Adam M. / Feng, Changjian et al. | 2013
- 199
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Modulating the interaction between CDK2 and cyclin A with a quinoline-based inhibitorDeng, Yongqi / Shipps, Gerald W. Jr. / Zhao, Lianyun et al. | 2013
- 204
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Correlation between chemotype-dependent binding conformations of HSP90α/β and isoform selectivity—Implications for the structure-based design of HSP90α/β selective inhibitors for treating neurodegenerative diseasesErnst, Justin T. / Liu, Michael / Zuccola, Harmon et al. | 2013
- 204
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Correlation between chemotype-dependent binding conformations of HSP90@a/@b and isoform selectivity-Implications for the structure-based design of HSP90@a/@b selective inhibitors for treating neurodegenerative diseasesErnst, J. T. / Liu, M. / Zuccola, H. et al. | 2014
- 209
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Synthesis of 3′-O-fluorescently mono-modified reversible terminators and their uses in sequencing-by-synthesisKim, Da-Rae / Kim, Taek-Soo / Kim, Eunsun et al. | 2013
- 214
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Oxidative cleavage of DNA by pentamethine carbocyanine dyes irradiated with long-wavelength visible lightMapp, Carla T. / Owens, Eric A. / Henary, Maged et al. | 2013
- 220
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Synthesis and biological evaluation of the pirfenidone derivatives as antifibrotic agentsMa, Zhen / Pan, Youlu / Huang, Wenhai et al. | 2013
- 224
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Discovery of hybrid Hsp90 inhibitors and their anti-neoplastic effects against gefitinib-resistant non-small cell lung cancer (NSCLC)Jeong, Chul-Ho / Park, Hee Baek / Jang, Won Jun et al. | 2013
- 228
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New anti-inflammatory cembranoid diterpenoids from the Vietnamese soft coral Lobophytum crassumThao, Nguyen Phuong / Luyen, Bui Thi Thuy / Ngan, Nguyen Thi Thanh et al. | 2013
- 233
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Rational design, synthesis and antitubercular evaluation of novel 2-(trifluoromethyl)phenothiazine-[1,2,3]triazole hybridsAddla, Dinesh / Jallapally, Anvesh / Gurram, Divya et al. | 2013
- 237
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Synthesis of a novel series of artemisinin dimers with potent anticancer activity involving Sonogashira cross-coupling reactionBuragohain, Pori / Saikia, Bishwajit / Surineni, Naresh et al. | 2013
- 240
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Sulfonamide inhibition studies of the γ-carbonic anhydrase from the oral pathogen Porphyromonas gingivalisVullo, Daniela / Del Prete, Sonia / Osman, Sameh M. et al. | 2013
- 240
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Sulfonamide inhibition studies of the @c-carbonic anhydrase from the oral pathogen Porphyromonas gingivalisVullo, D. / Del Prete, S. / Osman, S. M. et al. | 2014
- 245
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Novel pyrazole integrated 1,3,4-oxadiazoles: Synthesis, characterization and antimicrobial evaluationNingaiah, Srikantamurthy / Bhadraiah, Umesha K. / Doddaramappa, Shridevi D. et al. | 2013
- 249
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Design, synthesis and evaluation of dual pharmacology β2-adrenoceptor agonists and PDE4 inhibitorsHuang, Ling / Shan, Wenjun / Zhou, Qi et al. | 2013
- 249
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Design, synthesis and evaluation of dual pharmacology @b"2-adrenoceptor agonists and PDE4 inhibitorsHuang, L. / Shan, W. / Zhou, Q. et al. | 2014
- 254
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Concise and high-yield synthesis of T808 and T808P for radiosynthesis of [18F]-T808, a PET tau tracer for Alzheimer’s diseaseGao, Mingzhang / Wang, Min / Zheng, Qi-Huang et al. | 2013
- 258
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(E)-Alkenes as replacements of amide bonds: Development of novel and potent acyclic CGRP receptor antagonistsKim, June J. / Wood, Michael R. / Stachel, Shawn J. et al. | 2013
- 262
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Imidazole-derived agonists for the neurotensin 1 receptorHershberger, Paul M. / Hedrick, Michael P. / Peddibhotla, Satyamaheshwar et al. | 2013
- 268
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A novel indigoid anti-tuberculosis agentKlein, Larry L. / Petukhova, Valentina / Wan, Baojie et al. | 2013
- 271
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Preparation and evaluation of deconstruction analogues of 7-deoxykalafungin as AKT kinase inhibitorsKorwar, Sudha / Nguyen, Thuy / Ellis, Keith C. et al. | 2013
- 275
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Sulfonamide inhibition studies of the @d-carbonic anhydrase from the diatom Thalassiosira weissflogiiVullo, D. / Del Prete, S. / Osman, S. M. et al. | 2014
- 275
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Sulfonamide inhibition studies of the δ-carbonic anhydrase from the diatom Thalassiosira weissflogiiVullo, Daniela / Del Prete, Sonia / Osman, Sameh M. et al. | 2013
- 280
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High-throughput docking for the identification of new influenza A virus polymerase inhibitors targeting the PA–PB1 protein–protein interactionTintori, Cristina / Laurenzana, Ilaria / Fallacara, Anna Lucia et al. | 2013
- 283
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Synthesis and preliminary evaluation of a new fluorine-18 labelled triazine derivative for PET imaging of cannabinoid CB2 receptorHortala, Laurent / Arnaud, Joëlle / Roux, Pascale et al. | 2013
- 288
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Discovery and optimization of Lu AF58801, a novel, selective and brain penetrant positive allosteric modulator of alpha-7 nicotinic acetylcholine receptors: Attenuation of subchronic phencyclidine (PCP)-induced cognitive deficits in rats following oral administrationEskildsen, Jørgen / Redrobe, John P. / Sams, Anette G. et al. | 2013
- 294
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Discrimination between 5-hydroxymethylcytosine and 5-methylcytosine in DNA by selective chemical labelingHu, Jianlin / Chen, Yuqi / Xu, Xiaowei et al. | 2013
- 298
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Triazino indole–quinoline hybrid: A novel approach to antileishmanial agentsSharma, Rashmi / Pandey, Anand Kumar / Shivahare, Rahul et al. | 2013
- 302
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Synthesis, anti-HIV activity, integrase enzyme inhibition and molecular modeling of catechol, hydroquinone and quinol labdane analogsPawar, Rohan / Das, Tiyasa / Mishra, Sanjay et al. | 2013
- 308
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1,2,3-Triazole-derived naphthalimides as a novel type of potential antimicrobial agents: Synthesis, antimicrobial activity, interaction with calf thymus DNA and human serum albuminLv, Jing-Song / Peng, Xin-Mei / Kishore, Baathulaa et al. | 2013
- 314
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A near-infrared fluorescence dye for sensitive detection of hydrogen sulfide in serumWu, Xuanjun / Shi, Jiaqi / Yang, Liu et al. | 2013
- 317
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Novel di-tertiary-butyl phenylhydrazones as dual cyclooxygenase-2/5-lipoxygenase inhibitors: Synthesis, COX/LOX inhibition, molecular modeling, and insights into their cytotoxicitiesGhatak, Shibnath / Vyas, Alok / Misra, Suniti et al. | 2013
- 325
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Stereoselective total synthesis of a novel regiomer of herbarumin I and its cytotoxic and antimicrobial activitiesJangili, Paramesh / Kashanna, Jajula / Kumar, C. Ganesh et al. | 2013
- 328
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Synthesis and biological evaluation of novel N-substituted 1H-dibenzo[a,c]carbazole derivatives of dehydroabietic acid as potential antimicrobial agentsGu, Wen / Qiao, Chao / Wang, Shi-Fa et al. | 2013
- 332
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NAD-based inhibitors with anticancer potentialFelczak, Krzysztof / Vince, Robert / Pankiewicz, Krzysztof W. et al. | 2013
- 337
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Discovery of potent and efficacious cyanoguanidine-containing nicotinamide phosphoribosyltransferase (Nampt) inhibitorsZheng, Xiaozhang / Baumeister, Timm / Buckmelter, Alexandre J. et al. | 2013
- 344
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Dactyloditerpenol acetate, a new prenylbisabolane-type diterpene from Aplysia dactylomela with significant in vitro anti-neuroinflammatory activityJiménez-Romero, Carlos / Mayer, Alejandro M.S. / Rodríguez, Abimael D. et al. | 2013
- 349
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Evaluation of benzoic acid derivatives as sirtuin inhibitorsChen, Yi-Pei / Catbagan, Chad C. / Bowler, Jeannette T. et al. | 2013
- 353
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Design, synthesis and structure–activity relationships of substituted oxazole–benzamide antibacterial inhibitors of FtsZStokes, Neil R. / Baker, Nicola / Bennett, James M. et al. | 2013
- 360
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Identification through structure-based methods of a bacterial NAD+-dependent DNA ligase inhibitor that avoids known resistance mutationsMurphy-Benenato, Kerry / Wang, Hongming / McGuire, Helen M. et al. | 2013
- 367
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Preparation of 8-hydroxyquinoline derivatives as potential antibiotics against Staphylococcus aureusLam, Kim-Hung / Gambari, Roberto / Lee, Kenneth Ka-Ho et al. | 2013
- 371
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Copper ion as a delivery platform for taxanes and taxane complexesManning, Thomas J. / Phillips, Dennis / Wylie, Greg et al. | 2013
- 378
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Design and synthesis of an aminopiperidine series of γ-secretase modulatorsKobayashi, Tomonori / Iwama, Seiji / Fusano, Akira et al. | 2013
- 378
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Design and synthesis of an aminopiperidine series of @c-secretase modulatorsKobayashi, T. / Iwama, S. / Fusano, A. et al. | 2014
- 382
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Asymmetric synthesis and receptor activity of chiral simplified resiniferatoxin (sRTX) analogues as transient receptor potential vanilloid 1 (TRPV1) ligandsKim, Myeong Seop / Ki, Yooran / Ahn, Song Yeon et al. | 2013
- 386
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Simplified captopril analogues as NDM-1 inhibitorsLi, Ningning / Xu, Yintong / Xia, Qiang et al. | 2013
- 390
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Inhibition of serine and proline racemases by substrate-product analoguesHarty, Matthew / Nagar, Mitesh / Atkinson, Logan et al. | 2013
- 394
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Detection of hepatitis C virus by single-step hairpin primer RT-PCRTakei, Fumie / Tani, Hideki / Matsuura, Yoshiharu et al. | 2013
- 397
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Corrigendum to “Imidazopyridazines as potent inhibitors of Plasmodium falciparum calcium-dependent protein kinase 1 (PfCDPK1): Preparation and evaluation of pyrazole linked analogues” [Bioorg. Med. Chem. Lett. 23 (2013) 6019–6024]Large, Jonathan M. / Osborne, Simon A. / Smiljanic-Hurley, Ela et al. | 2013
- 398
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Corrigendum to “Design, synthesis and evaluation of aspirin analogues having an additional carboxylate substituent for antithrombotic activity” [Bioorg. Med. Chem. Lett. 19 (2009) 4213–4216]Alagha, Ahmed / Moman, Edelmiro / Adamo, Mauro F.A. et al. | 2013
- IFC
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Editorial board| 2013