Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 2643
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Graphical contents list| 2012
- 2664
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Isoflavones inhibit the clonogenicity of human colon cancer cellsHyun, Jiye / Shin, Soon Young / So, Kyoung Min et al. | 2012
- 2670
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Design and synthesis of potent, isoxazole-containing renin inhibitorsFournier, Pierre-André / Arbour, Mélissa / Cauchon, Elizabeth et al. | 2012
- 2675
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Synthesis and evaluation of substituted dibenzo[c,e]azepine-5-ones as P-glycoprotein-mediated multidrug resistance reversal agentsTang, Xiaobo / Gu, Xiaoke / Ren, Zhiguang et al. | 2012
- 2681
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Double-stranded oligonucleotides containing 5-aminomethyl-2′-deoxyuridine form thermostable anti-parallel triplexes with single-stranded DNA or RNAShibata, Aya / Ueno, Yoshihito / Iwata, Mari et al. | 2012
- 2681
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Double-stranded oligonucleotides containing 5-aminomethyl-2prime-deoxyuridine form thermostable anti-parallel triplexes with single-stranded DNA or RNAShibata, A. / Ueno, Y. / Iwata, M. et al. | 2012
- 2684
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Lanthanide(III) complexes of pyridine–tetraacetic acid-glycoconjugates: Synthesis and luminescence studies of mono and divalent derivativesGouin, Sébastien G. / Roger, Mélissa / Leygue, Nadine et al. | 2012
- 2689
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Design and synthesis of novel opioid ligands with an azabicyclo[2.2.2]octane skeleton and their pharmacologiesWatanabe, Yoshikazu / Kitazawa, Shota / Fujii, Hideaki et al. | 2012
- 2693
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Pyrazolopyrimidines as dual Akt/p70S6K inhibitorsRice, Kenneth D. / Kim, Moon H. / Bussenius, Joerg et al. | 2012
- 2698
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The chemical synthesis of metabolically stabilized 2-OMe-LPA analogues and preliminary studies of their inhibitory activity toward autotaxinGendaszewska-Darmach, Edyta / Laska, Edyta / Rytczak, Przemysław et al. | 2012
- 2701
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Design and synthesis of thiourea derivatives containing a benzo[5,6]cyclohepta[1,2-b]pyridine moiety as potential antitumor and anti-inflammatory agentsLiu, Wukun / Zhou, Jinpei / Zhang, Tong et al. | 2012
- 2705
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Synthesis and antiviral activity of a series of 1′-substituted 4-aza-7,9-dideazaadenosine C-nucleosidesCho, Aesop / Saunders, Oliver L. / Butler, Thomas et al. | 2012
- 2705
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Synthesis and antiviral activity of a series of 1prime-substituted 4-aza-7,9-dideazaadenosine C-nucleosidesCho, A. / Saunders, O. L. / Butler, T. et al. | 2012
- 2708
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Synthesis and in vitro anticancer and antitubercular activity of diarylpyrazole ligated dihydropyrimidines possessing lipophilic carbamoyl groupYadlapalli, Rama Krishna / Chourasia, O.P. / Vemuri, Kiranmayi et al. | 2012
- 2712
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Synthesis and biological activity of bi/tricyclic azasugars fused thiazolidin-4-one and thiazinan-4-one by microwave-assisted tandem Staudinger/aza-Wittig/cyclizationLi, Xiaoliu / Qin, Zhanbin / Yang, Tianyu et al. | 2012
- 2717
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Antitumor activity of annonaceous acetogenins in HepS and S180 xenografts bearing miceChen, Yong / Chen, Jian-wei / Xu, Sha-sha et al. | 2012
- 2720
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5-Benzylidenerhodanine and 5-benzylidene-2-4-thiazolidinedione based antibacterialsZvarec, Ondrej / Polyak, Steven W. / Tieu, William et al. | 2012
- 2723
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Sinularioside, a triacetylated glycolipid from the Indonesian soft coral Sinularia sp., is an inhibitor of NO releasePutra, Masteria Yunovilsa / Ianaro, Angela / Panza, Elisabetta et al. | 2012
- 2726
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Design, synthesis and cytotoxic activities of novel hybrid compounds between 2-phenylbenzofuran and imidazoleYang, Xiao-Dong / Wan, Wei-Chao / Deng, Xiao-Yan et al. | 2012
- 2730
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Lead optimisation of the N1 substituent of a novel series of indazole arylsulfonamides as CCR4 antagonists and identification of a candidate for clinical investigationProcopiou, Panayiotis A. / Ford, Alison J. / Graves, Rebecca H. et al. | 2012
- 2734
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Preparation and photophysical properties of a caged kynurenineMaitrani, Chandan / Heyes, Derren J. / Hay, Sam et al. | 2012
- 2738
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Discovery and evaluation of spirocyclic derivatives as antagonists of the neuropeptide Y5 receptorFichtner, Michael / Lee, Eunsun / Tomlinson, Elizabeth et al. | 2012
- 2744
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Synthesis of new bergenin derivatives as potent inhibitors of inflammatory mediators NO and TNF-aShah, M. R. / Arfan, M. / Amin, H. et al. | 2012
- 2744
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Synthesis of new bergenin derivatives as potent inhibitors of inflammatory mediators NO and TNF-αShah, Muhammad Raza / Arfan, Mohammad / Amin, Hazrat et al. | 2012
- 2748
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Synthesis and evaluation of piperidine urea derivatives as efficacious 11β-hydroxysteroid dehydrogenase type 1 inhibitors in diabetic ob/ob miceZhang, Liming / Chen, Junhua / Ning, Mengmeng et al. | 2012
- 2748
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Synthesis and evaluation of piperidine urea derivatives as efficacious 11b-hydroxysteroid dehydrogenase type 1 inhibitors in diabetic ob/ob miceZhang, L. / Chen, J. / Ning, M. et al. | 2012
- 2753
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Fluorescent nucleosides with ‘on–off’ switching function, pH-responsive fluorescent uridine derivativesSaito, Yoshio / Miyamoto, Shigenori / Suzuki, Azusa et al. | 2012
- 2757
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Synthesis of [Tyr-5-Ψ(CH2NMe)-Tyr-6]RA-VII, a reduced peptide bond analogue of RA-VII, an antitumor bicyclic hexapeptideHasuda, Tomoyo / Hitotsuyanagi, Yukio / Shinada, Mitsuyuki et al. | 2012
- 2760
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A new pancreatic lipase inhibitor from Broussonetia kanzinokiAhn, Jong Hoon / Liu, Qing / Lee, Chul et al. | 2012
- 2764
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Synthesis of highly potent novel anti-tubercular isoniazid analogues with preliminary pharmacokinetic evaluationRamani, Addepalli Venkata / Monika, Arumalla / Indira, Vadlamani Lakshmi et al. | 2012
- 2768
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Thiosemicarbazone fragment embedded within 1,2,4-triazole ring as inhibitors of Entamoeba histolyticaSiddiqui, Shadab Miyan / Salahuddin, Attar / Azam, Amir et al. | 2012
- 2772
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Design and synthesis of naphthoquinone derivatives as antiproliferative agents and 20S proteasome inhibitorsXu, Kai / Xiao, Zhiyan / Tang, Yan Bo et al. | 2012
- 2775
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Synthesis of new opioid derivatives with a propellane skeleton and their pharmacology. Part 2: Propellane derivatives with an amide side chainNagase, Hiroshi / Akiyama, Junko / Nakajima, Ryo et al. | 2012
- 2780
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Inhibition of tumor suppressor protein p53-dependent transcription by a tetramerization domain peptide via hetero-oligomerizationWada, Junya / Kamada, Rui / Imagawa, Toshiaki et al. | 2012
- 2784
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Pyrazine-based Syk kinase inhibitorsForns, Pilar / Esteve, Cristina / Taboada, Lorena et al. | 2012
- 2789
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3-(N-Arylsulfamoyl)benzamides, inhibitors of human sirtuin type 2 (SIRT2)Choi, Soo Hyuk / Quinti, Luisa / Kazantsev, Aleksey G. et al. | 2012
- 2794
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Indole-propionic acid derivatives as potent, S1P3-sparing and EAE efficacious sphingosine-1-phosphate 1 (S1P1) receptor agonistsMeng, Qinghua / Zhao, Baowei / Xu, Qiongfeng et al. | 2012
- 2798
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Development of hypoxia-sensitive Gd3+-based MRI contrast agentsIwaki, Shimpei / Hanaoka, Kenjiro / Piao, Wen et al. | 2012
- 2803
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Discovery of S-777469: An orally available CB2 agonist as an antipruritic agentOdan, Masahide / Ishizuka, Natsuki / Hiramatsu, Yoshiharu et al. | 2012
- 2807
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Substituted phenoxypropyl-(R)-2-methylpyrrolidine aminomethyl ketones as histamine-3 receptor inverse agonistsZulli, Allison L. / Aimone, Lisa D. / Mathiasen, Joanne R. et al. | 2012
- 2811
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A new class of prolylcarboxypeptidase inhibitors, Part 1: Discovery and evaluationGraham, Thomas H. / Liu, Wensheng / Verras, Andreas et al. | 2012
- 2818
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A new class of prolylcarboxypeptidase inhibitors, Part 2: The aminocyclopentanesGraham, Thomas H. / Liu, Wensheng / Verras, Andreas et al. | 2012
- 2823
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Efficient one-pot cyclization/folding of Rhesus θ-defensin-1 (RTD-1)Aboye, Teshome L. / Li, Yilong / Majumder, Subhabrata et al. | 2012
- 2827
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Bromophenols as inhibitors of protein tyrosine phosphatase 1B with antidiabetic propertiesShi, Dayong / Li, Jing / Jiang, Bo et al. | 2012
- 2833
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Deep-red fluorescent imaging probe for bacteriaWhite, Alexander G. / Gray, Brian D. / Pak, Koon Yan et al. | 2012
- 2837
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Design and synthesis of 3-(4,5,6,7-tetrahydro-3H-imidazo[4,5-c]pyridin-2-yl)-1H-quinolin-2-ones as VEGFR-2 kinase inhibitorsHan, Sun-Young / Choi, Jie Won / Yang, Jeon et al. | 2012
- 2843
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Discovery of novel and potent heterocyclic carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitorsBasu, Sujay / Prasad, Uppuleti Viplava / Barawkar, Dinesh A. et al. | 2012
- 2850
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Radioiodinated sunitinib as a potential radiotracer for imaging angiogenesis—radiosynthesis and first radiopharmacological evaluation of 5-[125I]Iodo-sunitinibKuchar, Manuela / Oliveira, Maria Cristina / Gano, Lurdes et al. | 2012
- 2856
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Medicinal chemistry approaches to avoid aldehyde oxidase metabolismPryde, David C. / Tran, Thien-Duc / Jones, Peter et al. | 2012
- 2861
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Discovery of HIV fusion inhibitors targeting gp41 using a comprehensive α-helix mimetic libraryWhitby, Landon R. / Boyle, Kristopher E. / Cai, Lifeng et al. | 2012
- 2861
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Discovery of HIV fusion inhibitors targeting gp41 using a comprehensive a-helix mimetic libraryWhitby, L. R. / Boyle, K. E. / Cai, L. et al. | 2012
- 2866
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Synthesis and SAR studies of novel heteroaryl fused tetracyclic indole-diamide compounds: Potent allosteric inhibitors of the hepatitis C virus NS5B polymeraseDing, Min / He, Feng / Hudyma, Thomas W. et al. | 2012
- 2872
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Design, synthesis, synergistic antimicrobial activity and cytotoxicity of 4-aryl substituted 3,4-dihydropyrimidinones of curcuminLal, Jaggi / Gupta, S.K. / Thavaselvam, D. et al. | 2012
- 2877
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Discovery of a novel chemotype of potent human ENaC blockers using a bioisostere approach. Part 2: a-Branched quaternary aminesHunt, T. / Atherton-Watson, H. C. / Collingwood, S. P. et al. | 2012
- 2877
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Discovery of a novel chemotype of potent human ENaC blockers using a bioisostere approach. Part 2: α-Branched quaternary aminesHunt, Thomas / Atherton-Watson, Hazel C. / Collingwood, Stephen P. et al. | 2012
- 2880
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2-Anilino-4-aryl-8H-purine derivatives as inhibitors of PDK1Blanchard, Stéphanie / Soh, Chang Kai / Lee, Chai Ping et al. | 2012
- 2885
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Prospective acetylcholinesterase inhibitory activity of indole and its analogsKhorana, Nantaka / Changwichit, Kanokwan / Ingkaninan, Kornkanok et al. | 2012
- 2889
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Consensus hologram QSAR modeling for the prediction of human intestinal absorptionModa, Tiago L. / Andricopulo, Adriano D. et al. | 2012
- 2894
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CB 1/2 dual agonists with 3-carbamoyl 2-pyridone derivatives as antipruritics: Reduction of CNS side effects by introducing polar functional groupsOdan, Masahide / Ishizuka, Natsuki / Hiramatsu, Yoshiharu et al. | 2012
- 2898
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Discovery of S-444823, a potent CB1/CB2 dual agonist as an antipruritic agentOdan, Masahide / Ishizuka, Natsuki / Hiramatsu, Yoshiharu et al. | 2012
- 2902
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Antimycobacterial activity of bisbenzylisoquinoline alkaloids from Tiliacora triandra against multidrug-resistant isolates of Mycobacterium tuberculosisSureram, Sanya / Senadeera, Sarath P.D. / Hongmanee, Poonpilas et al. | 2012
- 2906
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Design and synthesis of dihydrobenzofuran amides as orally bioavailable, centrally active γ-secretase modulatorsPettersson, Martin / Johnson, Douglas S. / Subramanyam, Chakrapani et al. | 2012
- 2906
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Design and synthesis of dihydrobenzofuran amides as orally bioavailable, centrally active g-secretase modulatorsPettersson, M. / Johnson, D. S. / Subramanyam, C. et al. | 2012
- 2912
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Calcitonin gene-related peptide (CGRP) receptor antagonists: Novel aspartates and succinatesLuo, Guanglin / Chen, Ling / Pin, Sokhom S. et al. | 2012
- 2917
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Calcitonin gene-related peptide (CGRP) receptor antagonists: Pyridine as a replacement for a core amide groupLuo, Guanglin / Chen, Ling / Civiello, Rita et al. | 2012
- 2922
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The design and synthesis of novel, phosphonate-containing transient receptor potential melastatin 8 (TRPM8) antagonistsMatthews, Jay M. / Qin, Ning / Colburn, Raymond W. et al. | 2012
- 2927
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Melanogenesis inhibitory bisabolane-type sesquiterpenoids from the roots of Angelica koreanaLee, Jin Woo / Yun, Cheong-Yong / Roh, Eunmiri et al. | 2012
- 2932
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Low brain penetrant CB1 receptor agonists for the treatment of neuropathic painAdam, Julia M. / Clark, John K. / Davies, Keneth et al. | 2012
- 2938
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Inhibition of hepatitis C virus NS5A by fluoro-olefin based γ-turn mimeticsChang, Wonsuk / Mosley, Ralph T. / Bansal, Shalini et al. | 2012
- 2938
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Inhibition of hepatitis C virus NS5A by fluoro-olefin based g-turn mimeticsChang, W. / Mosley, R. T. / Bansal, S. et al. | 2012
- 2943
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Discovery of new piperidine amide triazolobenzodiazepinones as intestinal-selective CCK1 receptor agonistsCameron, Kimberly O. / Beretta, Elena E. / Chen, Yue et al. | 2012
- 2948
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Synthesis and biological evaluation of novel small non-peptidic HIV-1 PIs: The benzothiophene ring as an effective moietyChiummiento, Lucia / Funicello, Maria / Lupattelli, Paolo et al. | 2012
- 2951
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Photo-degradation products of pramipexoleNishimura, Eiji / Kugimiya, Aya / Naoki, Hideo et al. | 2012
- 2954
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Sesquiterpene lactones from Tithonia diversifolia act as peroxisome proliferator-activated receptor agonistsLin, Hsiang-Ru et al. | 2012
- 2959
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New triazole derivatives as antifungal agents: Synthesis via click reaction, in vitro evaluation and molecular docking studiesZou, Yan / Zhao, Qingjie / Liao, Jun et al. | 2012
- 2963
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From ApoA1 upregulation to BET family bromodomain inhibition: Discovery of I-BET151Mirguet, Olivier / Lamotte, Yann / Donche, Frédéric et al. | 2012
- 2968
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Identification of a novel series of BET family bromodomain inhibitors: Binding mode and profile of I-BET151 (GSK1210151A)Seal, Jonathan / Lamotte, Yann / Donche, Frédéric et al. | 2012
- 2973
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Unambiguous structure of atractyloside and carboxyatractylosideSanchez, Jean-Frédéric / Kauffmann, Brice / Grélard, Axelle et al. | 2012
- 2976
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Phosphonium lipocations as antiparasitic agentsLong, Timothy E. / Lu, Xiao / Galizzi, Melina et al. | 2012
- 2980
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Structure–activity studies of some berberine analogs as inhibitors of Toxoplasma gondiiKrivogorsky, Bogdana / Pernat, Jennifer A. / Douglas, Kelsi A. et al. | 2012
- 2983
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Copper(I) mediated facile synthesis of potent tubulin polymerization inhibitor, 9-amino-α-noscapine from natural α-noscapineManchukonda, Naresh K. / Sridhar, Balasubramanian / Naik, Pradeep K. et al. | 2012
- 2983
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Copper(I) mediated facile synthesis of potent tubulin polymerization inhibitor, 9-amino-a-noscapine from natural a-noscapineManchukonda, N. K. / Sridhar, B. / Naik, P. K. et al. | 2012
- 2988
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Structural polymorphism of human telomere G-quadruplex induced by a pyridyl carboxamide moleculeXu, Liang / Xu, Zhouxin / Shang, Ye et al. | 2012
- 2993
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Discovery of novel P3-oxo inhibitor of hepatitis C virus NS3/4A serine proteaseDuan, Maosheng / Kazmierski, Wieslaw / Crosby, Renae et al. | 2012
- 2997
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Development of clickable active site-directed photoaffinity probes for γ-secretaseCrump, Christina J. / am Ende, Christopher W. / Eric Ballard, T. et al. | 2012
- 2997
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Development of clickable active site-directed photoaffinity probes for g-secretaseCrump, C. J. / am Ende, C. W. / Eric Ballard, T. et al. | 2012
- 3001
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Synthesis and evaluation of 1-(substituted)-3-prop-2-ynylureas as antiangiogenic agentsSanphanya, Kingkan / Wattanapitayakul, Suvara K. / Prangsaengtong, Orawin et al. | 2012
- 3006
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Identification of novel telomeric G-quadruplex-targeting chemical scaffolds through screening of three NCI librariesRahman, Khondaker M. / Tizkova, Karolina / Reszka, Anthony P. et al. | 2012
- 3011
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Footprint-based identification of viral entry inhibitors targeting HIVgp41Holden, Patrick M. / Kaur, Harmeet / Goyal, Rashi et al. | 2012
- 3017
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Pimarane diterpenes from the fungus Epicoccum sp. HS-1 associated with Apostichopus japonicusXia, Xuekui / Zhang, Jianye / Zhang, Yonggang et al. | 2012
- IFC
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Editorial board| 2012