Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 701
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The long story of camptothecin: From traditional medicine to drugsMartino, Emanuela / Della Volpe, Serena / Terribile, Elisa et al. | 2016
- 708
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Design, synthesis and evaluation of novel bifunctional tetrahydroxamate chelators for PET imaging of 89Zr-labeled antibodiesRousseau, Julie / Zhang, Zhengxing / Dias, Gemma M. et al. | 2017
- 713
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Investigation of the anti-angiogenesis effects induced by deoxypodophyllotoxin-5-FU conjugate C069 against HUVE cellsXiang, Rong / Guan, Xiao-Wen / Hui, Ling et al. | 2017
- 718
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DL-3-n-butylphthalide-Edaravone hybrids as novel dual inhibitors of amyloid-β aggregation and monoamine oxidases with high antioxidant potency for Alzheimer’s therapyQiang, Xiaoming / Li, Yan / Yang, Xia et al. | 2017
- 723
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Synthesis of cholesteryl doxorubicin and its anti-cancer activityChoi, Jong-Soo / Doh, Kyung-Oh / Kim, Bieong-Kil et al. | 2017
- 729
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Discovery and biological evaluation of some (1H-1,2,3-triazol-4-yl)methoxybenzaldehyde derivatives containing an anthraquinone moiety as potent xanthine oxidase inhibitorsZhang, Ting-jian / Li, Song-ye / Yuan, Wei-yan et al. | 2017
- 733
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Evaluation of a series of 2-napthamide derivatives as inhibitors of the drug efflux pump AcrB for the reversal of antimicrobial resistanceWang, Yinhu / Mowla, Rumana / Guo, Liwei et al. | 2017
- 740
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Synthesis of carbon-11-labeled isonicotinamides as new potential PET agents for imaging of GSK-3 enzyme in Alzheimer’s diseaseGao, Mingzhang / Wang, Min / Zheng, Qi-Huang et al. | 2017
- 744
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Design, synthesis and evaluation of antiproliferative activity of melanoma-targeted histone deacetylase inhibitorsRaji, Idris / Ahluwalia, Kabir / Oyelere, Adegboyega K. et al. | 2017
- 750
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Discovery of pyrazolopyrimidine derivatives as novel inhibitors of ataxia telangiectasia and rad3 related protein (ATR)Ramachandran, Sreekanth A. / Jadhavar, Pradeep S. / Singh, Manvendra P. et al. | 2017
- 755
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Antiparasitic lethality of sulfonamidebenzamides in kinetoplastidsHackler, Amber / Patrick, Stephen L. / Kahney, Elizabeth W. et al. | 2017
- 759
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Escape from adamantane: Scaffold optimization of novel P2X7 antagonists featuring complex polycyclesBarniol-Xicota, Marta / Kwak, Seung-Hwa / Lee, So-Deok et al. | 2017
- 764
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Synthesis, characterization, in vitro SAR and in vivo evaluation of N,N′bisnaphthylmethyl 2-alkyl substituted imidazolium salts against NSCLCDeBord, Michael A. / Southerland, Marie R. / Wagers, Patrick O. et al. | 2017
- 776
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Synthesis and biological evaluation of 2-alkoxycarbonylallyl esters as potential anticancer agentsRonayne, Conor T. / Solano, Lucas N. / Nelson, Grady L. et al. | 2017
- 781
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Indolyl-naphthyl-maleimides as potent and selective inhibitors of protein kinase C-α/βvan Eis, Maurice J. / Evenou, JeanPierre / Schuler, Walter et al. | 2017
- 787
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Anti-HSV-1, antioxidant and antifouling phenolic compounds from the deep-sea-derived fungus Aspergillus versicolor SCSIO 41502Huang, Zhonghui / Nong, Xuhua / Ren, Zhe et al. | 2017
- 792
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A novel piperazine linked β-amino alcohols bearing a benzosuberone scaffolds as anti-proliferative agentsVanguru, Sowmya / Jilla, Lavanya / Sajja, Yasodakrishna et al. | 2017
- 797
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Selenoesters and selenoanhydrides as novel multidrug resistance reversing agents: A confirmation study in a colon cancer MDR cell lineGajdács, Márió / Spengler, Gabriella / Sanmartín, Carmen et al. | 2017
- 803
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Alkaloids from the mangrove endophytic fungus Diaporthe phaseolorum SKS019Cui, Hui / Yu, Jianchen / Chen, Senhua et al. | 2017
- 808
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Development of gallic acid formazans as novel enoyl acyl carrier protein reductase inhibitors for the treatment of tuberculosisSaharan, Vanita D. / Mahajan, Supriya S. et al. | 2017
- 816
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Synthesis of Vorinostat and cholesterol conjugate to enhance the cancer cell uptake selectivityIdippily, Nethrie D. / Gan, Chunfang / Orefice, Paul et al. | 2017
- 821
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Synthesis, antimycobacterial and cytotoxic activity of α,β-unsaturated amides and 2,4-disubstituted oxazoline derivativesAvalos-Alanís, Francisco G. / Hernández-Fernández, Eugenio / Carranza-Rosales, Pilar et al. | 2017
- 826
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Discovery of peptidic miR-21 processing inhibitor by mirror image phage display: A novel method to generate RNA binding D-peptidesSakamoto, Kotaro / Otake, Kentaro / Umemoto, Tadashi et al. | 2017
- 829
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Novel 12N-substituted matrinanes as potential anti-coxsackievirus agentsLi, Ying–Hong / Tang, Sheng / Li, Yu–Huan et al. | 2017
- 834
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A new efficient method of generating photoaffinity beads for drug target identificationNishiya, Yoichi / Hamada, Tomoko / Abe, Masayuki et al. | 2017
- 841
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Synthesis and in vitro activity of dicationic indolyl diphenyl ethers as novel potent antibiotic agents against drug-resistant bacteriaChen, Xiaofang / Hu, Xinxin / Wu, Yanbin et al. | 2017
- 845
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Synthesis and biological evaluation of thiazole derivatives as novel USP7 inhibitorsChen, Chao / Song, Jiemei / Wang, Jinzheng et al. | 2017
- 850
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Benzoflavones as cholesterol esterase inhibitors: Synthesis, biological evaluation and docking studiesSingh, Harbinder / Singh, Jatinder Vir / Gupta, Manish K. et al. | 2017
- 855
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Discovery of 7-(3-(piperazin-1-yl)phenyl)pyrrolo[2,1-f][1,2,4]triazin-4-amine derivatives as highly potent and selective PI3Kδ inhibitorsQin, Lan-Ying / Ruan, Zheming / Cherney, Robert J. et al. | 2017
- 862
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Discovering novel 7-azaindole-based series as potent AXL kinase inhibitorsFeneyrolles, Clémence / Guiet, Léa / Singer, Mathilde et al. | 2017
- 867
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Design, synthesis and biological evaluation of novel 3-substituted 4-anilino-coumarin derivatives as antitumor agentsLuo, Guoshun / Muyaba, Moses / Lyu, Weiting et al. | 2017
- 875
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Nardonaphthalenones A and B from the roots and rhizomes of Nardostachys chinensis Batal.Deng, Xu / Wu, Yi-Jing / Chen, Ying-Peng et al. | 2017
- 880
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Anticomplement triterpenoids from the roots of Ilex asprellaWen, Quan / Lu, Yan / Chao, Zhi et al. | 2017
- 887
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Synthesis and structure–activity relationship studies of phenolic hydroxyl derivatives based on quinoxalinone as aldose reductase inhibitors with antioxidant activityHao, Xin / Han, Zhongfei / Li, Yang et al. | 2017
- 893
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A novel monoterpenoid indole alkaloid with anticancer activity from Melodinus khasianusZhou, Jie / Feng, Jin-Hong / Fang, Lei et al. | 2017
- 897
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New synthetic route to ethynyl-dUTP: A means to avoid formation of acetyl and chloro vinyl base-modified triphosphates that could poison SELEX experimentsRöthlisberger, Pascal / Levi-Acobas, Fabienne / Hollenstein, Marcel et al. | 2017
- 901
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Antifungal activity of substituted auronesSutton, Caleb L. / Taylor, Zachary E. / Farone, Mary B. et al. | 2017
- 904
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Synthesis and antiviral evaluation of novel heteroarylpyrimidines analogs as HBV capsid effectorsBoucle, Sebastien / Lu, Xiao / Bassit, Leda et al. | 2017
- 911
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Mesoionic pyrido[1,2-a]pyrimidinones: Discovery of dicloromezotiaz as a lepidoptera insecticide acting on nicotinic acetylcholine receptors1,2Zhang, Wenming / Holyoke, Caleb W. Jr. / Barry, James et al. | 2017
- 918
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Study of antileishmanial activity of 2-aminobenzoyl amino acid hydrazides and their quinazoline derivativesKhattab, Sherine Nabil / Haiba, Nesreen Saied / Asal, Ahmed Mosaad et al. | 2017
- 922
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Quinolidene based monocarbonyl curcumin analogues as promising antimycobacterial agents: Synthesis and molecular docking studySubhedar, Dnyaneshwar D. / Shaikh, Mubarak H. / Nawale, Laxman et al. | 2017
- 929
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Discovery of furan carboxylate derivatives as novel inhibitors of ATP-citrate lyase via virtual high-throughput screeningJernigan, Finith E. / Hanai, Jun-ichi / Sukhatme, Vikas P. et al. | 2017
- 936
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Shape-based virtual screening, synthesis and evaluation of novel pyrrolone derivatives as antiviral agents against HCVBassetto, Marcella / Leyssen, Pieter / Neyts, Johan et al. | 2016
- 941
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In vivo evaluation of IGF1R/IR PET ligand [18F]BMS-754807 in rodentsPrabhakaran, Jaya / Dewey, Stephen L. / McClure, Richard et al. | 2016
- 944
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Discovery of new MurA inhibitors using induced-fit simulation and dockingRožman, Kaja / Lešnik, Samo / Brus, Boris et al. | 2016
- 950
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Design, synthesis, and bioactivities of novel oxadiazole-substituted pyrazole oximesDai, Hong / Chen, Jia / Li, Gang et al. | 2016
- 954
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DNA-duplex linker for AFM-SELEX of DNA aptamer against human serum albuminTakenaka, Musashi / Okumura, Yuzo / Amino, Tomokazu et al. | 2016
- 958
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Design, synthesis and biological activity evaluation of novel 2,6-difluorobenzamide derivatives through FtsZ inhibitionBi, Fangchao / Guo, Liwei / Wang, Yinhu et al. | 2016
- 963
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Design, synthesis and biological evaluation of six dinuclear platinum(II) complexesYu, Congtao / Gao, Chuanzhu / Bai, Linkui et al. | 2016
- 967
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Discovery of medium ring thiophosphorus based heterocycles as antiproliferative agentsFeng, Wei / Novera, Wisna / Peh, Kaye et al. | 2016
- 973
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Natural potential neuroinflammatory inhibitors from Alhagi sparsifolia Shap.Zhou, Di / Wei, Hongyan / Jiang, Zhe et al. | 2016
- 979
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Synthesis and cell imaging applications of fluorescent mono/di/tri-heterocyclyl-2,6-dicyanoanilinesPisal, Mahesh M. / Annadate, Ritesh A. / Athalye, Meghana C. et al. | 2016
- 989
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Inhibition of invasion by N-trans-feruloyloctopamine via AKT, p38MAPK and EMT related signals in hepatocellular carcinoma cellsBai, Zhong-Tian / Wu, Zheng-Rong / Xi, Li-Li et al. | 2016
- 994
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Design, synthesis and biological evaluation of regioisomers of 666-15 as inhibitors of CREB-mediated gene transcriptionXie, Fuchun / Li, Bingbing X. / Xiao, Xiangshu et al. | 2016
- 999
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A tetramic acid derivative with protein tyrosine phosphatase 1B inhibitory activity and a new nortriterpene glycoside from the Indonesian marine sponge Petrosia sp.Maarisit, Wilmar / Yamazaki, Hiroyuki / Kanno, Syu-ichi et al. | 2016
- 1003
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Chitosan cross-linked with poly(ethylene glycol)dialdehyde via reductive amination as effective controlled release carriers for oral protein drug deliveryJing, Zi-Wei / Ma, Zhi-Wei / Li, Chen et al. | 2016
- 1007
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Discovery of FZU-03,010 as a self-assembling anticancer amphiphile for acute myeloid leukemiaChen, Yingyu / Li, Cailong / Zheng, Yunquan et al. | 2016
- 1012
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Synthesis, evaluation and quantitative structure–activity relationship (QSAR) analysis of Wogonin derivatives as cytotoxic agentsBian, Jinlei / Li, Tinghan / Weng, Tianwei et al. | 2016
- 1017
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Novel 2,4-dichlorophenoxy acetic acid substituted thiazolidin-4-ones as anti-inflammatory agents: Design, synthesis and biological screeningAli, Yakub / Alam, Mohammad Sarwar / Hamid, Hinna et al. | 2016
- 1026
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Microbial hydroxylation and glycosylation of pentacyclic triterpenes as inhibitors on tissue factor procoagulant activityWang, Wei-Wei / Xu, Shao-Hua / Zhao, Ya-Zheng et al. | 2016
- 1031
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Identification of a selective inhibitor of transforming growth factor β-activated kinase 1 by biosensor-based screening of focused librariesMiura, Takaaki / Matsuo, Atsushi / Muraoka, Terushige et al. | 2016
- 1037
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Synthesis and evaluation of 5-(1H-indol-3-yl)-N-aryl-1,3,4-oxadiazol-2-amines as Bcl-2 inhibitory anticancer agentsHamdy, Rania / Ziedan, Noha I. / Ali, Samia et al. | 2016
- 1041
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Synthesis and antioxidant activity of a procyanidin B3 analogueMizuno, Mirei / Nakanishi, Ikuo / Matsubayashi, Satoko et al. | 2016
- 1045
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Sulfonamide-based non-alkyne LpxC inhibitors as Gram-negative antibacterial agentsKawai, Tetsuya / Kazuhiko, Iwase / Takaya, Noriko et al. | 2016
- 1050
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Benzenesulphonamide inhibitors of the cytolytic protein perforinSpicer, Julie A. / Miller, Christian K. / O'Connor, Patrick D. et al. | 2016
- 1055
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Virtual screening and experimental validation identify novel modulators of nuclear receptor RXRα from Drugbank databaseXu, Dan / Cai, Lijun / Guo, Shangjie et al. | 2016
- 1062
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Discovery of MK-1832, a Kv1.5 inhibitor with improved selectivity and pharmacokineticsWolkenberg, Scott E. / Nolt, M. Brad / Bilodeau, Mark T. et al. | 2016
- 1070
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Bifunctional bisphosphonate derivatives and platinum complexes with high affinity for bone hydroxyapatiteSun, Yanyan / Chen, Lei / Wu, Xiwen et al. | 2016
- 1076
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Sulfamic and succinic acid derivatives of 25-OH-PPD and their activities to MCF-7, A-549, HCT-116, and BGC-823 cell linesZhou, Wu-Xi / Cao, Jia-Qing / Wang, Xu-De et al. | 2016
- 1081
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Combined treatment with zingerone and its novel derivative synergistically inhibits TGF-β1 induced epithelial-mesenchymal transition, migration and invasion of human hepatocellular carcinoma cellsKim, Young-Joo / Jeon, Youngsic / Kim, Taejung et al. | 2016
- 1089
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Functionalized triazines as potent HCV entry inhibitorsMull, Eric S. / Sun, Li-Qiang / Zhao, Qian et al. | 2016
- 1094
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Investigation of piperazine benzamides as human β3 adrenergic receptor agonists for the treatment of overactive bladderHarper, Bart H. / Wang, Liping / Zhu, Cheng et al. | 2016
- 1099
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Structure-based optimization of 1H-imidazole-2-carboxamides as Axl kinase inhibitors utilizing a Mer mutant surrogateKeung, Walter / Boloor, Amogh / Brown, Jason et al. | 2016
- 1105
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Discovery of core-structurally novel PTP1B inhibitors with specific selectivity containing oxindole-fused spirotetrahydrofurochroman by one-pot reactionDong, Suzhen / Lei, Yubing / Jia, Shikun et al. | 2016
- 1109
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The design and synthesis of novel spirocyclic heterocyclic sulfone ROMK inhibitors as diureticsChobanian, Harry R. / Guo, Yan / Pio, Barbara et al. | 2016
- IFC
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Editorial board| 2017