Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 6925
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Graphical contents list| 2011
- 6941
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Structure-based design of isoindoline-1,3-diones and 2,3-dihydrophthalazine-1,4-diones as novel B-Raf inhibitorsWang, Xiaolun / Salaski, Edward J. / Berger, Dan M. et al. | 2011
- 6945
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Improved radiosynthesis of the apoptosis marker 18F-ICMT11 including biological evaluationGlaser, Matthias / Goggi, Julian / Smith, Graham et al. | 2011
- 6950
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Design and synthesis of pyridin-2-ylmethylaminopiperidin-1-ylbutyl amide CCR5 antagonists that are potent inhibitors of M-tropic (R5) HIV-1 replicationSkerlj, Renato / Bridger, Gary / Zhou, Yuanxi et al. | 2011
- 6955
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Synthesis and SAR of a novel metabotropic glutamate receptor 4 (mGlu4) antagonist: Unexpected ‘molecular switch’ from a closely related mGlu4 positive allosteric modulatorUtley, Thomas / Haddenham, Dustin / Salovich, James M. et al. | 2011
- 6960
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Alkaloids from Chelidonium majus and their inhibitory effects on LPS-induced NO production in RAW264.7 cellsPark, Ji Eun / Cuong, To Dao / Hung, Tran Manh et al. | 2011
- 6964
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Synthesis and docking study of 2-phenylaminopyrimidine Abl tyrosine kinase inhibitorsLü, Shuang / Luo, Qun / Hao, Xiang et al. | 2011
- 6969
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Identification of nonplanar small molecule for G-quadruplex grooves: Molecular docking and molecular dynamic studyLi, Jinlian / Jin, Xiaoqiang / Hu, LiHong et al. | 2011
- 6973
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Antibacterial and antitubercular activity of fosmidomycin, FR900098, and their lipophilic analogsUh, Eugene / Jackson, Emily R. / San Jose, Géraldine et al. | 2011
- 6977
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Discovery of new aminopyrimidine-based phosphoinositide 3-kinase beta (PI3Kb) inhibitors with selectivity over PI3KaKim, J. / Hong, S. et al. | 2011
- 6977
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Discovery of new aminopyrimidine-based phosphoinositide 3-kinase beta (PI3Kβ) inhibitors with selectivity over PI3KαKim, Jinhee / Hong, Seunghee / Hong, Sungwoo et al. | 2011
- 6982
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III. Identification of novel CXCR3 chemokine receptor antagonists with a pyrazinyl–piperazinyl–piperidine scaffoldKim, Seong Heon / Anilkumar, Gopinadhan N. / Zawacki, Lisa Guise et al. | 2011
- 6987
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[18F]Azadibenzocyclooctyne ([18F]ADIBO): A biocompatible radioactive labeling synthon for peptides using catalyst free [3+2] cycloadditionArumugam, Selvanathan / Chin, Joshua / Schirrmacher, Ralf et al. | 2011
- 6992
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Fluoride-18 radiolabeling of peptides bearing an aminooxy functional group to a prosthetic ligand via an oxime bondCarberry, Patrick / Carpenter, Alan P. / Kung, Hank F. et al. | 2011
- 6996
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Anti-staphylococcal activity and b-lactam resistance attenuating capacity of structural analogues of (-)-epicatechin gallateAnderson, J. C. / McCarthy, R. A. / Paulin, S. et al. | 2011
- 6996
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Anti-staphylococcal activity and β-lactam resistance attenuating capacity of structural analogues of (−)-epicatechin gallateAnderson, James C. / McCarthy, Robert A. / Paulin, Sarah et al. | 2011
- 7001
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Discovery of a novel series of melanin-concentrating hormone receptor 1 antagonists for the treatment of obesityMihalic, Jeffrey T. / Chen, Xiaoqi / Fan, Pingchen et al. | 2011
- 7006
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Novel tricyclic inhibitors of IKK2: Discovery and SAR leading to the identification of 2-methoxy-N-((6-(1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-7-yl)pyridin-2-yl)methyl)acetamide (BMS-066)Watterson, Scott H. / Langevine, Charles M. / Van Kirk, Katy et al. | 2011
- 7013
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Spacer length effects on in vitro imaging and surface accessibility of fluorescent inhibitors of prostate specific membrane antigenLiu, Tiancheng / Nedrow-Byers, Jessie R. / Hopkins, Mark R. et al. | 2011
- 7017
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Radiosynthesis of three [11C]ureido-substituted benzenesulfonamides as PET probes for carbonic anhydrase IX in tumorsAsakawa, Chiharu / Ogawa, Masanao / Kumata, Katsushi et al. | 2011
- 7021
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Stabilization of DNA duplex by 2-substituted adenine as a minor groove modifierTanaka, Makiko / Kozakai, Ryota / Saito, Yoshio et al. | 2011
- 7025
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Novel antileukemic agents derived from tamibarotene and nitric oxide donorsBian, Haiyong / Feng, Jinhong / Li, Minyong et al. | 2011
- 7030
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Substrate profiling of IGF-1R and InsR: Identification of a potent pentamer substrateChapelat, Julien / Berst, Frédéric / Marzinzik, Andreas L. et al. | 2011
- 7034
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Synthesis of novel 3-carboxamide-benzocoumarin derivatives as orally active antithrombotic agentsSashidhara, Koneni V. / Kumar, Abdhesh / Kumar, Manoj et al. | 2011
- 7041
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Ungeremine effectively targets mammalian as well as bacterial type I and type II topoisomerasesCasu, Laura / Cottiglia, Filippo / Leonti, Marco et al. | 2011
- 7045
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TACN-containing cationic lipids with ester bond: Preparation and application in gene deliveryZhang, Qin-Fang / Yang, Wei-Han / Yi, Wen-Jing et al. | 2011
- 7050
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Discovery of small molecules that enhance astrocyte differentiation in rat fetal neural stem cellsChang, Dong Jo / Jeong, Mi Young / Song, Jiho et al. | 2011
- 7054
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Synthesis and cytotoxic evaluation of novel paraconic acid analogsLe Floch, Camille / Le Gall, Erwan / Léonel, Eric et al. | 2011
- 7059
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Anisotropy studies of tRNA-T box antiterminator RNA complex in the presence of 1,4-disubstituted 1,2,3-triazolesZhou, S. / Acquaah-Harrison, G. / Bergmeier, S.C. et al. | 2011
- 7064
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Novel inhibitors of Mycobacterium tuberculosis dTDP-6-deoxy-l-lyxo-4-hexulose reductase (RmlD) identified by virtual screeningWang, Yi / Hess, Tamara Noelle / Jones, Victoria et al. | 2011
- 7068
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A small molecule that preferentially binds the closed conformation of Hsp90Alexander, Leslie D. / Partridge, James R. / Agard, David A. et al. | 2011
- 7072
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Synthesis and SAR of 2-Phenoxypyridines as novel c-Jun N-terminal kinase inhibitorsSong, Xinyi / Chen, Weimin / Lin, Li et al. | 2011
- 7076
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Synthesis and evaluation of pyridone-phenoxypropyl-R-2-methylpyrrolidine analogues as histamine H3 receptor antagonistsBecknell, Nadine C. / Lyons, Jacquelyn A. / Aimone, Lisa D. et al. | 2011
- 7081
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Enzymatic synthesis of d-sorbose and d-psicose with aldolase RhaD: Effect of acceptor configuration on enzyme stereoselectivityLi, Zijie / Cai, Li / Qi, Qingsheng et al. | 2011
- 7085
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The synthesis of xanthones, xanthenediones, and spirobenzofurans: Their antibacterial and antifungal activityOmolo, Justin J. / Johnson, Myron M. / van Vuuren, Sandy F. et al. | 2011
- 7089
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Thiophene inhibitors of PDE4: Crystal structures show a second binding mode at the catalytic domain of PDE4D2Nankervis, Jacob L. / Feil, Susanne C. / Hancock, Nancy C. et al. | 2011
- 7094
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Synthesis and antiviral activity of 2′-deoxy-2′-fluoro-2′-C-methyl-7-deazapurine nucleosides, their phosphoramidate prodrugs and 5′-triphosphatesShi, Junxing / Zhou, Longhu / Zhang, Hongwang et al. | 2011
- 7094
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Synthesis and antiviral activity of 2prime-deoxy-2prime-fluoro-2prime-C-methyl-7-deazapurine nucleosides, their phosphoramidate prodrugs and 5prime-triphosphatesShi, J. / Zhou, L. / Zhang, H. et al. | 2011
- 7099
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Usabamycins A–C: New anthramycin-type analogues from a marine-derived actinomyceteSato, Seizo / Iwata, Fumie / Yamada, Shoichi et al. | 2011
- 7102
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Biological evaluation of glucose and deoxyglucose derivatives radiolabeled with [99mTc(CO)3(H2O)3]+ core as potential melanoma imaging agentsDapueto, Rosina / Castelli, Romina / Fernández, Marcelo et al. | 2011
- 7107
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Discovery and optimization of indoles and 7-azaindoles as Rho kinase (ROCK) inhibitors (part-I)Chowdhury, Sarwat / Sessions, E. Hampton / Pocas, Jennifer R. et al. | 2011
- 7113
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Discovery and optimization of indole and 7-azaindoles as Rho kinase (ROCK) inhibitors (Part-II)Sessions, E. Hampton / Chowdhury, Sarwat / Yin, Yan et al. | 2011
- 7119
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Facile synthesis of new 4-aza-podophyllotoxin analogs via microwave-assisted multi-component reactions and evaluation of their cytotoxic activityShi, Feng / Zeng, Xiao-Ning / Zhang, Ge et al. | 2011
- 7124
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Discovery of N-Aryl-2-acylindole human glucagon receptor antagonistsSinz, Christopher / Bittner, Amy / Brady, Ed et al. | 2011
- 7131
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Discovery of cyclic guanidines as potent, orally active, human glucagon receptor antagonistsSinz, Christopher / Chang, Jiang / Lins, Ashley Rouse et al. | 2011
- 7137
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The de-guanidinylated derivative of peramivir remains a potent inhibitor of influenza neuraminidaseBromba, Caleb M. / Mason, Jeremy W. / Brant, Michael G. et al. | 2011
- 7142
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Synthesis and antimicrobial activity of brominated resorcinol dimersBouthenet, Elise / Oh, Ki-Bong / Park, Seungil et al. | 2011
- 7146
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Synthesis and biological activity of acetyl-protected hydroxybenzyl diethyl phosphates (EHBP) as potential chemotherapeutic agentsKodela, Ravinder / Chattopadhyay, Mitali / Nath, Niharika et al. | 2011
- 7151
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Synthesis and biological evaluation of salicylate-based compounds as a novel class of methionine aminopeptidase inhibitorsWang, Wen-Long / Chai, Sergio C. / Ye, Qi-Zhuang et al. | 2011
- 7155
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Discovery of a novel class of non-ATP site DFG-out state p38 inhibitors utilizing computationally assisted virtual fragment-based drug design (vFBDD)Moffett, Kristofer / Konteatis, Zenon / Nguyen, Duyan et al. | 2011
- 7166
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Synthesis of GSK3b mimetic inhibitors of Akt featuring a novel extended dipeptide surrogateRanatunga, S. / Del Valle, J. R. et al. | 2011
- 7166
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Synthesis of GSK3β mimetic inhibitors of Akt featuring a novel extended dipeptide surrogateRanatunga, Sujeewa / Del Valle, Juan R. et al. | 2011
- 7170
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Synthesis and biological evaluation of arylated novobiocin analogs as Hsp90 inhibitorsKusuma, Bhaskar Reddy / Duerfeldt, Adam S. / Blagg, Brian S.J. et al. | 2011
- 7175
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Isolation and identification of diadenosine 5prime,5-P1,P4-tetraphosphate binding proteins using magnetic bio-panningGuo, W. / Azhar, M. A. / Xu, Y. et al. | 2011
- 7175
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Isolation and identification of diadenosine 5′,5‴-P 1,P 4-tetraphosphate binding proteins using magnetic bio-panningGuo, Wei / Azhar, M. Ameruddin / Xu, Yuhong et al. | 2011
- 7180
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Identification of novel, exosite-binding matrix metalloproteinase-13 inhibitor scaffoldsRoth, Joshua / Minond, Dmitriy / Darout, Etzer et al. | 2011
- 7185
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Design and synthesis of triazolopyridazines substituted with methylisoquinolinone as selective c-Met kinase inhibitorsRyu, Jae Wook / Han, Sun-Young / Yun, Jeong In et al. | 2011
- 7189
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Transformation of quercitols into 4-methylenecyclohex-5-ene-1,2,3-triol derivatives, precursors for the chemical chaperones N-octyl-4-epi-b-valienamine (NOEV) and N-octyl-b-valienamine (NOV)Kuno, S. / Takahashi, A. / Ogawa, S. et al. | 2011
- 7189
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Transformation of quercitols into 4-methylenecyclohex-5-ene-1,2,3-triol derivatives, precursors for the chemical chaperones N-octyl-4-epi-β-valienamine (NOEV) and N-octyl-β-valienamine (NOV)Kuno, Shinichi / Takahashi, Atsushi / Ogawa, Seiichiro et al. | 2011
- 7193
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Molecular design, synthesis and bioactivity of glycosyl hydrazine and hydrazone derivatives: Notable effects of the sugar moietyCui, Zining / Yang, Xinling / Shi, Yanxia et al. | 2011
- 7197
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Identification of small-molecule inhibitors of Trypansoma cruzi replicationGermain, Andrew R. / Carmody, Leigh C. / Dockendorff, Chris et al. | 2011
- 7201
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Crassocolides N–P, three cembranoids from the Formosan soft coral Sarcophyton crassocauleWang, Guey-Horng / Huang, Ho-Cheng / Su, Jui-Hsin et al. | 2011
- 7205
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Discovery and optimization of 2-phenyloxazole derivatives as diacylglycerol acyltransferase-1 inhibitorsYun, Weiya / Ahmad, Mushtaq / Chen, Yingsi et al. | 2011
- 7210
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Synthesis and biological evaluation of novel pyrimidine derivatives as sub-micromolar affinity ligands of GalR2Sagi, Vasudeva Naidu / Liu, Tianyu / Lu, Xiaoying et al. | 2011
- 7216
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Synthesis and testing of trifluoromethyl-containing phosphonate–peptide conjugates as inhibitors of serine hydrolasesSokolova, Nadezhda V. / Nenajdenko, Valentine G. / Sokolov, Vladimir B. et al. | 2011
- 7219
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3D-QSAR and molecular docking studies of 2-pyrimidinecarbonitrile derivatives as inhibitors against falcipain-3Potshangbam, Angamba Meetei / Tanneeru, Karunakar / Reddy, Bandi Madhusudhan et al. | 2011
- 7224
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Synthesis and activity study of phosphonamidate dipeptides as potential inhibitors of VanXYang, Ke-Wu / Cheng, Xu / Zhao, Chuan et al. | 2011
- 7228
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Corrigendum to “Discovery of 3-aryl-5-acylpiperazinyl-pyrazoles as antagonists to the NK3 receptor” [Bioorg. Med. Chem. Lett. 21 (2011) 1991–1996]Hoveyda, Hamid R. / Roy, Marie-Odile / Blanc, Sebastien et al. | 2011
- 7229
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Corrigendum to “Oxidative stimuli-responsive nanoprodrug of camptothecin kills glioblastoma cells” [Bioorg. Med. Chem. Lett. 20 (2010) 5262]Lee, Bong-Seop / Nalla, Aruna K. / Stock, Ilana R. et al. | 2011
- IFC
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Editorial board| 2011