Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 4395
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Graphical contents list| 2007
- 4411
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Aminopyrrolidineamide inhibitors of site-1 proteaseHay, Bruce A. / Abrams, Barbara / Zumbrunn, Allice Y. et al. | 2007
- 4415
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Rational design of 7-arylquinolines as non-competitive metabotropic glutamate receptor subtype 5 antagonistsMilbank, Jared B.J. / Knauer, Christopher S. / Augelli-Szafran, Corinne E. et al. | 2007
- 4419
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SAR and X-ray structures of enantiopure 1,2-cis-(1R,2S)-cyclopentyldiamine and cyclohexyldiamine derivatives as inhibitors of coagulation Factor XaQiao, Jennifer X. / Chang, Chong-Hwan / Cheney, Daniel L. et al. | 2007
- 4428
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Synthesis, cytotoxicity, and antiviral activities of new neolignans related to honokiol and magnololAmblard, Franck / Govindarajan, Baskaran / Lefkove, Benjamin et al. | 2007
- 4432
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N-(5-Chloro-2-(hydroxymethyl)-N-alkyl-arylsulfonamides as g-secretase inhibitorsParker, M. F. / Barten, D. M. / Bergstrom, C. P. et al. | 2007
- 4432
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N-(5-Chloro-2-(hydroxymethyl)-N-alkyl-arylsulfonamides as γ-secretase inhibitorsParker, Michael F. / Barten, Donna M. / Bergstrom, Carl P. et al. | 2007
- 4437
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Thiotetrazole alkynylacetanilides as potent and bioavailable non-nucleoside inhibitors of the HIV-1 wild type and K103N/Y181C double mutant reverse transcriptasesGagnon, Alexandre / Amad, Ma’an H. / Bonneau, Pierre R. et al. | 2007
- 4442
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2-Aryl-N-acyl indole derivatives as liver X receptor (LXR) agonistsKher, Sunil / Lake, Kirk / Sircar, Ila et al. | 2007
- 4447
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Convergent synthesis and in vivo inhibitory effect on fat accumulation of (−)-ternatin, a highly N-methylated cyclic peptideShimokawa, Kenichiro / Yamada, Kaoru / Kita, Masaki et al. | 2007
- 4450
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Identification and optimization of novel 1,3,4-oxadiazole EP1 receptor antagonistsHall, Adrian / Brown, Susan H. / Chowdhury, Anita et al. | 2007
- 4456
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Design, synthesis, and molecular modeling studies of 5′-deoxy-5′-ureidoadenosine: 5′-ureido group as multiple hydrogen bonding donor in the active site of S-adenosylhomocysteine hydrolaseWang, Ting / Lee, Hyun Joo / Tosh, Dilip K. et al. | 2007
- 4456
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Design, synthesis, and molecular modeling studies of 5prime-deoxy-5prime-ureidoadenosine: 5prime-ureido group as multiple hydrogen bonding donor in the active site of S-adenosylhomocysteine hydrolaseWang, T. / Lee, H. J. / Tosh, D. K. et al. | 2007
- 4460
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Gypsophin: A novel α-glucosidase inhibitory cyclic peptide from the roots of Gypsophila oldhamianaLuo, Jian-Guang / Wang, Xiao-Bing / Ma, Li et al. | 2007
- 4460
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Gypsophin: A novel a-glucosidase inhibitory cyclic peptide from the roots of Gypsophila oldhamianaLuo, J. G. / Wang, X. B. / Ma, L. et al. | 2007
- 4464
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Identification of a novel series of benzimidazoles as potent and selective antagonists of the human melanocortin-4 receptorPoitout, Lydie / Brault, Valérie / Sackur, Carole et al. | 2007
- 4471
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Synthesis and bioevaluation of N-(arylalkyl)-homospermidine conjugatesXie, Songqiang / Cheng, Pengfei / Liu, Guangchao et al. | 2007
- 4476
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Synthesis and biological evaluation of N-acetyl-β-aryl-1,2-didehydroethylamines as new HIV-1 RT inhibitors in vitroCheng, Pi / Jiang, Zhi-Yong / Wang, Rui-Rui et al. | 2007
- 4476
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Synthesis and biological evaluation of N-acetyl-b-aryl-1,2-didehydroethylamines as new HIV-1 RT inhibitors in vitroCheng, P. / Jiang, Z. Y. / Wang, R. R. et al. | 2007
- 4481
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Design, synthesis, and discovery of stilbene derivatives based on lithospermic acid B as potent protein tyrosine phosphatase 1B inhibitorsJung, Mankil / Lee, Yongnam / Park, Moonsoo et al. | 2007
- 4487
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Synthesis and SAR of tetrahydropyrrolo[1,2-b][1,2,5]thiadiazol-2(3H)-one 1,1-dioxide analogues as highly potent selective androgen receptor modulatorsManfredi, Mark C. / Bi, Yingzhi / Nirschl, Alexandra A. et al. | 2007
- 4491
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Induction of GRP78 by valproic acid is dependent upon histone deacetylase inhibitionShi, Yuanyuan / Gerritsma, David / Bowes, Anna J. et al. | 2007
- 4495
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Synthesis and matrix metalloproteinase (MMP)-12 inhibitory activity of ageladine A and its analogsAndo, Naoki / Terashima, Shiro et al. | 2007
- 4500
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Proinsecticide candidates N-(5-methyl-2-oxo-1,3-dioxol-4-yl)methyl derivatives of imidacloprid and 1-chlorothiazolylmethyl-2-nitroimino-imidazolidineOhno, Ikuya / Hirata, Koichi / Ishida, Chiharu et al. | 2007
- 4504
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Synthesis and pharmacological evaluation of condensed heterocyclic 6-substituted-1,2,4-triazolo[3,4-b]-1,3,4-thiadiazole derivatives of naproxenAmir, Mohammad / Kumar, Harish / Javed, Sadique A. et al. | 2007
- 4509
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Himbacine derived thrombin receptor (PAR-1) antagonists: SAR of the pyridine ringXia, Yan / Chackalamannil, Samuel / Clasby, Martin et al. | 2007
- 4514
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Synthesis and reactivity of azobenzene-based bispropargyl sulfones: Interesting comparison between cyclic and acyclic systemsMitra, Debarati / Kar, Moumita / Pal, Rhitankar et al. | 2007
- 4518
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Novel prodrug approach to photodynamic therapy: Fmoc solid-phase synthesis of a cell permeable peptide incorporating 5-aminolaevulinic acidDixon, Mark J. / Bourré, Ludovic / MacRobert, Alexander J. et al. | 2007
- 4523
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Synthesis and antibacterial activity of novel fluoroquinolones containing substituted piperidinesDang, Zhao / Yang, Yushe / Ji, Ruyun et al. | 2007
- 4527
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Synthesis of symmetrical C- and pseudo-symmetrical O-linked disaccharide analogs for arabinosyltransferase inhibitory activity in Mycobacterium tuberculosisPathak, Ashish K. / Pathak, Vibha / Riordan, James R. et al. | 2007
- 4531
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Design and synthesis of novel, conformationally restricted HMG-CoA reductase inhibitorsPfefferkorn, Jeffrey A. / Choi, Chulho / Song, Yuntao et al. | 2007
- 4538
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Design and synthesis of hepatoselective, pyrrole-based HMG-CoA reductase inhibitorsPfefferkorn, Jeffrey A. / Song, Yuntao / Sun, Kuai-Lin et al. | 2007
- 4545
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Cytostatic activity of novel 4prime-aminochalcone-based imidesJha, A. / Mukherjee, C. / Rolle, A. J. et al. | 2007
- 4545
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Cytostatic activity of novel 4′-aminochalcone-based imidesJha, Amitabh / Mukherjee, Chandrani / Rolle, Alfred J. et al. | 2007
- 4551
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In-silico fragment-based identification of novel angiogenesis inhibitorsDakshanamurthy, Sivanesan / Kim, Min / Brown, Milton L. et al. | 2007
- 4557
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Design, synthesis, and evaluation of 3,4-disubstituted pyrazole analogues as anti-tumor CDK inhibitorsLin, Ronghui / Chiu, George / Yu, Yang et al. | 2007
- 4562
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Benzo[b]thiophene-based histone deacetylase inhibitorsWitter, David J. / Belvedere, Sandro / Chen, Liqiang et al. | 2007
- 4568
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Design, synthesis, and biological evaluation of pyrazinones containing novel P1 needles as inhibitors of TF/VIIaTrujillo, John I. / Huang, Horng-Chih / Neumann, William L. et al. | 2007
- 4575
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Inhibitors of anthrax lethal factorGaddis, Brandon D. / Avramova, Larisa V. / Chmielewski, Jean et al. | 2007
- 4579
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Discovery of 3-aminopiperidines as potent, selective, and orally bioavailable dipeptidyl peptidase IV inhibitorsCox, Jason M. / Harper, Bart / Mastracchio, Anthony et al. | 2007
- 4584
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Design, synthesis, and preliminary biological evaluation of a novel triazole analogue of ceramideKim, Sanghee / Cho, Minjae / Lee, Taeho et al. | 2007
- 4588
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Synthesis of 4-phenoxybenzamide adenine dinucleotide as NAD analogue with inhibitory activity against enoyl-ACP reductase (InhA) of Mycobacterium tuberculosisBonnac, Laurent / Gao, Guang-Yao / Chen, Liqiang et al. | 2007
- 4592
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Respiratory syncytial virus fusion inhibitors. Part 5: Optimization of benzimidazole substitution patterns towards derivatives with improved activityWang, Xiangdong Alan / Cianci, Christopher W. / Yu, Kuo-Long et al. | 2007
- 4599
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N-(6,7-Dichloro-2,3-dioxo-1,2,3,4-tetrahydroquinoxalin-5-yl)-N-alkylsulfonamides as peripherally restricted N-methyl-d-aspartate receptor antagonists for the treatment of painDeur, Christopher / Agrawal, Arun K. / Baum, Heidi et al. | 2007
- 4604
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A computational docking study for prediction of binding mode of diospyrin and derivatives: Inhibitors of human and leishmanial DNA topoisomerase-IChhabra, Sandeep et al. | 2007
- 4613
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Design and synthesis of 6-methyl-2-oxo-1,2,3,4-tetrahydro-pyrimidine-5-carboxylic acid derivatives as PPARg activatorsKumar, R. / Mittal, A. / Ramachandran, U. et al. | 2007
- 4613
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Design and synthesis of 6-methyl-2-oxo-1,2,3,4-tetrahydro-pyrimidine-5-carboxylic acid derivatives as PPARγ activatorsKumar, Rakesh / Mittal, Amit / Ramachandran, Uma et al. | 2007
- 4619
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Design of novel histone deacetylase inhibitorsSiliphaivanh, Phieng / Harrington, Paul / Witter, David J. et al. | 2007
- 4625
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Design of a partial PPARd agonistPettersson, I. / Ebdrup, S. / Havranek, M. et al. | 2007
- 4625
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Design of a partial PPARδ agonistPettersson, Ingrid / Ebdrup, Søren / Havranek, Miroslav et al. | 2007
- 4630
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Discovery of a novel class of benzazepinone Nav1.7 blockers: Potential treatments for neuropathic painHoyt, Scott B. / London, Clare / Gorin, David et al. | 2007
- 4635
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Synthesis and in vitro activity of 2-thiazolylhydrazone derivatives compared with the activity of clotrimazole against clinical isolates of Candida spp.Chimenti, Franco / Bizzarri, Bruna / Maccioni, Elias et al. | 2007
- 4641
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Heterocyclic α-helix mimetics for targeting protein–protein interactionsBiros, Shannon M. / Moisan, Lionel / Mann, Enrique et al. | 2007
- 4641
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Heterocyclic a-helix mimetics for targeting protein-protein interactionsBiros, S. M. / Moisan, L. / Mann, E. et al. | 2007
- 4646
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Human serum albumin binding assay based on displacement of a non selective fluorescent inhibitorThorarensen, Atli / Sarver, Ronald W. / Tian, Fang et al. | 2007
- 4650
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Selective oxidation of sulfides to sulfoxides catalyzed by ruthenium (III) meso-tetraphenylporphyrin chloride in the presence of molecular oxygenZhou, Xian-Tai / Ji, Hong-Bing / Cheng, Zhao et al. | 2007
- 4654
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Adenosine phosphonate inhibitors of lipid II: Alanyl tRNA ligase MurM from Streptococcus pneumoniaeCressina, Elena / Lloyd, Adrian J. / De Pascale, Gianfranco et al. | 2007
- 4657
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Novel tetrahydro-b-carboline-1-carboxylic acids as inhibitors of mitogen activated protein kinase-activated protein kinase 2 (MK-2)Trujillo, J. I. / Meyers, M. J. / Anderson, D. R. et al. | 2007
- 4657
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Novel tetrahydro-β-carboline-1-carboxylic acids as inhibitors of mitogen activated protein kinase-activated protein kinase 2 (MK-2)Trujillo, John I. / Meyers, Marvin J. / Anderson, David R. et al. | 2007
- 4664
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The discovery of carboline analogs as potent MAPKAP-K2 inhibitorsWu, Jiang-Ping / Wang, Ji / Abeywardane, Asitha et al. | 2007
- 4670
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Synthesis and evaluation of potent and selective β3 adrenergic receptor agonists containing heterobiaryl carboxylic acidsShearer, Barry G. / Chao, Esther Y. / Uehling, David E. et al. | 2007
- 4670
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Synthesis and evaluation of potent and selective b3 adrenergic receptor agonists containing heterobiaryl carboxylic acidsShearer, B. G. / Chao, E. Y. / Uehling, D. E. et al. | 2007
- 4678
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Synthesis and structure–activity relationship of a novel, non-hydroxamate series of TNF-α converting enzyme inhibitorsGilmore, John L. / King, Bryan W. / Asakawa, Naoyuki et al. | 2007
- 4678
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Synthesis and structure-activity relationship of a novel, non-hydroxamate series of TNF-a converting enzyme inhibitorsGilmore, J. L. / King, B. W. / Asakawa, N. et al. | 2007
- 4683
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Cycloalkanediamine derivatives as novel blood coagulation factor Xa inhibitorsNagata, Tsutomu / Yoshino, Toshiharu / Haginoya, Noriyasu et al. | 2007
- 4689
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Design and synthesis of highly potent and selective human peroxisome proliferator-activated receptor a agonistsYamazaki, Y. / Abe, K. / Toma, T. et al. | 2007
- 4689
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Design and synthesis of highly potent and selective human peroxisome proliferator-activated receptor α agonistsYamazaki, Yukiyoshi / Abe, Kazutoyo / Toma, Tsutomu et al. | 2007
- 4694
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Synthesis and SAR of novel conformationally-restricted oxazolidinones possessing Gram-positive and fastidious Gram-negative antibacterial activity. Part 1: Substituted pyrazolesBoyer, Frederick E. / Vara Prasad, J.V.N. / Choy, Allison L. et al. | 2007
- 4699
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Synthesis and SAR of novel conformationally restricted oxazolidinones possessing Gram-positive and fastidious Gram-negative antibacterial activity. Part 2: Amino substitutions on heterocyclic D-ring systemChoy, Allison L. / Vara Prasad, J.V.N. / Boyer, Frederick E. et al. | 2007
- 4703
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Synthesis, in vitro and in vivo cytotoxicity of 6,7-diaryl-2,3,8,8a-tetrahydroindolizin-5(1H)-onesKimball, F. Scott / Tunoori, Ashok Rao / Victory, Samuel F. et al. | 2007
- 4708
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Design, synthesis, and structure–activity relationship studies of new phenolic DNA gyrase inhibitorsLübbers, Thomas / Angehrn, Peter / Gmünder, Hans et al. | 2006
- I
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Instructions to contributors| 2007
- IFC
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Editorial board| 2007