Bioorganic and Medicinal Chemistry Letters
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Table of contents
- 2993
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Graphical contents list| 2004
- 3013
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Porphyrin–DNA cross-linking agent hybrids: chemical synthesis and biological studiesHe, Hanping / Tian, Tian / Wang, Ping et al. | 2004
- 3017
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Discovering selective agonists of endothelial target for acetylcholine (ETA) via diversity-guided pharmacophore simplification and simulationYang, Rifang / Zhao, Rusheng / Chen, Dongmei et al. | 2004
- 3027
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A novel mixed-ligand antimycobacterial dimeric copper complex of ciprofloxacin and phenanthrolineSaha, Dilip Kumar / Sandbhor, Uday / Shirisha, K. et al. | 2004
- 3033
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A new lead compound for abscisic acid biosynthesis inhibitors targeting 9-cis-epoxycarotenoid dioxygenaseHan, Sun-young / Kitahata, Nobutaka / Saito, Tamio et al. | 2004
- 3037
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Identification and optimization of novel partial agonists of Neuromedin B receptor using parallel synthesisShuttleworth, Stephen J. / Lizarzaburu, Mike E. / Chai, Anne et al. | 2004
- 3043
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A novel series of potent and selective small molecule inhibitors of the complement component C1sSubasinghe, Nalin L. / Ali, Farah / Illig, Carl R. et al. | 2004
- 3049
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Synthesis and pharmacological evaluation of piperidinoalkanoyl-1,2,3,4-tetrahydroisoquinoline derivatives as novel specific bradycardic agentsKubota, Hideki / Watanabe, Toshihiro / Kakefuda, Akio et al. | 2004
- 3053
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N-Isoquinolin-5-yl-N′-aralkyl-urea and -amide antagonists of human vanilloid receptor 1Jetter, Michele C. / Youngman, Mark A. / McNally, James J. et al. | 2004
- 3053
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N-Isoquinolin-5-yl-Nprime-aralkyl-urea and -amide antagonists of human vanilloid receptor 1Jetter, M. C. / Youngman, M. A. / McNally, J. J. et al. | 2004
- 3057
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Synthesis of 1,7-annulated indoles and their applications in the studies of cyclin dependent kinase inhibitorsZhu, Guoxin / Conner, Scott E. / Zhou, Xun et al. | 2004
- 3063
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Interaction with the S1b-pocket of urokinase: 8-heterocycle substituted and 6,8-disubstituted 2-naphthamidine urokinase inhibitorsWendt, Michael D. et al. | 2004
- 3063
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Interaction with the S1β-pocket of urokinase: 8-heterocycle substituted and 6,8-disubstituted 2-naphthamidine urokinase inhibitorsWendt, Michael D. / Geyer, Andrew / McClellan, William J. et al. | 2004
- 3069
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The synthesis and antimicrobial evaluation of a new series of isoxazolinyl oxazolidinonesWeidner-Wells, Michele A. / Werblood, Harvey M. / Goldschmidt, Raul et al. | 2004
- 3073
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Bridgehead-methyl analog of SC-53116 as a 5-HT4 agonistBecker, Daniel P. / Flynn, Daniel L. / Villamil, Clara I. et al. | 2004
- 3077
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A TOPS-MODE approach to predict adenosine kinase inhibitionGonzález, Maykel Pérez / Moldes, Maria del Carmen Terán et al. | 2004
- 3081
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Image contrast agents activated by prostate specific antigen (PSA)Jones, Graham B. / Xie, Longfei / El-Shafey, Ahmed et al. | 2004
- 3085
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Molecular modeling studies on the active binding site of the blood–brain barrier choline transporterGeldenhuys, Werner J. / Lockman, Paul R. / McAfee, James H. et al. | 2004
- 3093
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Structural differences between paroxetine and femoxetine responsible for differential inhibition of Staphylococcus aureus efflux pumpsWei, Peng / Kaatz, Glenn W. / Kerns, Robert J. et al. | 2004
- 3099
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SAR study of a subtype selective allosteric potentiator of metabotropic glutamate 2 receptor, N-(4-phenoxyphenyl)-N-(3-pyridinylmethyl)ethanesulfonamideBarda, David A. / Wang, Zhao-Qing / Britton, Thomas C. et al. | 2004
- 3103
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Conformationally restricted analogs of deoxynegamycinRaju, B. / Anandan, Sampathkumar / Gu, Shihai et al. | 2004
- 3109
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Human ACAT-1 and -2 inhibitory activities of saucerneol B, manassantin A and B isolated from Saururus chinensisLee, Woo Song / Lee, Dae-Woo / Baek, Young-Il et al. | 2004
- 3113
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Synthesis and activity of phosphinic tripeptide inhibitors of cathepsin CMucha, Artur / Pawełczak, Małgorzata / Hurek, Józef et al. | 2004
- 3117
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Lingshuiol, a novel polyhydroxyl compound with strongly cytotoxic activity from the marine dinoflagellate Amphidinium spHuang, Xiao-Chun / Zhao, Di / Guo, Yue-Wei et al. | 2004
- 3121
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Novel nonpeptidic inhibitors of HIV-1 protease obtained via a new multicomponent chemistry strategyYehia, Nasser A.M. / Antuch, Walfrido / Beck, Barbara et al. | 2004
- 3127
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Synthesis and biological evaluation of novel b-carboline derivatives as Tat-TAR interaction inhibitorsYu, Xiaolin et al. | 2004
- 3127
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Synthesis and biological evaluation of novel β-carboline derivatives as Tat–TAR interaction inhibitorsYu, Xiaolin / Lin, Wei / Li, Jingyun et al. | 2004
- 3131
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Development of an isotope-coded activity-based probe for the quantitative profiling of cysteine proteasesvan Swieten, Paul F. / Maehr, Rene / van den Nieuwendijk, Adrianus M.C.H. et al. | 2004
- 3135
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2-Alkylsulfanyl estrogen derivatives: synthesis of a novel class of multi-targeted anti-tumour agentsLeese, Mathew P. / Newman, Simon P. / Purohit, Atul et al. | 2004
- 3139
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Oxazolidinone: search for highly potent antibacterialLohray, Braj Bhushan / Lohray, Vidya Bhushan / Srivastava, Brijesh Kumar et al. | 2004
- 3143
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Synthesis and evaluation of nonpeptide substituted spirobenzazepines as potent vasopressin antagonistsXiang, Min Amy / Chen, Robert H. / Demarest, Keith T. et al. | 2004
- 3147
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An efficient sequence for the preparation of small secondary amine hydrochloride salts for focused library generation without need for distillation or chromatographic purificationDubowchik, Gene M. / Michne, Jodi A. / Zuev, Dmitry et al. | 2004
- 3151
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Exploring the possible binding sites at the interface of triosephosphate isomerase dimer as a potential target for anti-tripanosomal drug designEspinoza-Fonseca, L.Michel / Trujillo-Ferrara, José G. et al. | 2004
- 3155
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In vitro SAR of (5-(2H)-isoxazolonyl) ureas, potent inhibitors of hormone-sensitive lipaseLowe, Derek B. / Magnuson, Steven / Qi, Ning et al. | 2004
- 3161
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A new 2-carbamoyl pteridine that inhibits mycobacterial FtsZReynolds, R.C. / Srivastava, S. / Ross, L.J. et al. | 2004
- 3165
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Structure-based design, synthesis, and antimicrobial activity of purine derived SAH/MTA nucleosidase inhibitorsTedder, Martina E. / Nie, Zhe / Margosiak, Stephen et al. | 2004
- 3169
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Synthesis of 3-O-acyl/3-benzylidene/3-hydrazone/3-hydrazine/17-carboxyacryloyl ester derivatives of betulinic acid as anti-angiogenic agentsMukherjee, Rama / Jaggi, Manu / Rajendran, Praveen et al. | 2004
- 3173
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5-Alkyl-2-[(aryl and alkyloxylcarbonylmethyl)thio]-6-(1-naphthylmethyl) pyrimidin-4(3H)-ones as an unique HIV reverse transcriptase inhibitors of S-DABO seriesHe, Yanping / Chen, Fener / Sun, Guangfu et al. | 2004
- 3177
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Potential hypotensive agents: synthesis and hypotensive activity of oxime ethers derived from 1-naphthoxepines and related compoundsTandon, Vishnu K. / Kumar, Manoj / Awasthi, Anoop K. et al. | 2004
- 3181
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Design and synthesis of β-amino-α-hydroxy amide derivatives as inhibitors of MetAP2 and HUVEC growthSendzik, Martin / Janc, James W. / Cabuslay, Ronnel et al. | 2004
- 3181
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Design and synthesis of b-amino-a-hydroxy amide derivatives as inhibitors of MetAP2 and HUVEC growthSendzik, Martin et al. | 2004
- 3185
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High-throughput identification of fucosyltransferase inhibitors using carbohydrate microarraysBryan, Marian C. / Lee, Lac V. / Wong, Chi-Huey et al. | 2004
- 3189
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Synthesis and structure–activity relationships of 3-substituted 1,4-dihydro-4-oxo-1-(2-thiazolyl)-1,8-naphthyridines as novel antitumor agentsTsuzuki, Yasunori / Tomita, Kyoji / Sato, Yuji et al. | 2004
- 3195
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Benzimidazoles as new potent and selective DP antagonists for the treatment of allergic rhinitisBeaulieu, Christian / Wang, Zhaoyin / Denis, Danielle et al. | 2004
- 3201
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First total synthesis of structurally unique flavonoids and their strong anti-inflammatory effectNakatsuka, Takashi / Tomimori, Yoshiaki / Fukuda, Yoshiaki et al. | 2004
- 3205
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Development of l-3-aminotyrosine suitably protected for the synthesis of a novel nonphosphorylated hexapeptide with low-nanomolar Grb2-SH2 domain-binding affinitySong, Yan-Li / Roller, Peter P. / Long, Ya-Qiu et al. | 2004
- 3209
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New highly active taxoids from 9b-dihydrobaccatin-9,10-acetals. Part 5Takeda, Yasuyuki et al. | 2004
- 3209
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New highly active taxoids from 9β-dihydrobaccatin-9,10-acetals. Part 5Takeda, Yasuyuki / Uoto, Kouichi / Iwahana, Michio et al. | 2004
- 3217
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1,7-Annulated indolocarbazoles as cyclin-dependent kinase inhibitorsAl-awar, Rima S. / Ray, James E. / Hecker, Kyle A. et al. | 2004
- 3221
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Critical structural motif for the catalytic inhibition of human topoisomerase II by UK-1 and analogsWang, Ben B. / Maghami, Nima / Goodlin, Vanessa L. et al. | 2004
- 3227
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Selective urokinase-type plasminogen activator (uPA) inhibitors. Part 3: 1-IsoquinolinylguanidinesBarber, Christopher G. / Dickinson, Roger P. / Fish, Paul V. et al. | 2004
- 3231
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Synthesis and CB1 receptor activities of novel arachidonyl alcohol derivativesParkkari, Teija / Savinainen, Juha R. / Rauhala, Anu L. et al. | 2004
- 3235
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Potent and selective, sulfamide-based human b3-adrenergic receptor agonistsDow, Robert L. et al. | 2004
- 3235
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Potent and selective, sulfamide-based human β3-adrenergic receptor agonistsDow, Robert L. / Paight, Ernest S. / Schneider, Steven R. et al. | 2004
- 3241
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3,3prime-Oxybis(dimethoxytrityl chloride) (O-DMTCl): synthesis and applications of a novel bifunctional protecting groupOka, N. / Sanghvi, Y. S. / Theodorakis, E. A. et al. | 2004
- 3241
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3,3′-Oxybis(dimethoxytrityl chloride) (O-DMTCl): synthesis and applications of a novel bifunctional protecting groupOka, Natsuhisa / Sanghvi, Yogesh S. / Theodorakis, Emmanuel A. et al. | 2004
- 3245
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3-(7-Azaindolyl)-4-arylmaleimides as potent, selective inhibitors of glycogen synthase kinase-3Zhang, Han-Cheng / Ye, Hong / Conway, Bruce R. et al. | 2004
- 3251
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Novel thrombin inhibitors incorporating weakly basic heterobicyclic P1-arginine mimetics: optimization via modification of P1 and P3 moietiesKranjc, Andreja / Peterlin-Mašič, Lucija / Ilaš, Janez et al. | 2004
- 3257
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The monoethyl ester of meconic acid is an active site inhibitor of HCV NS5B RNA-dependent RNA polymerasePace, Paola / Nizi, Emanuela / Pacini, Barbara et al. | 2004
- 3263
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A novel 18b-glycyrrhetinic acid analogue as a potent and selective inhibitor of 11b-hydroxysteroid dehydrogenase 2Vicker, Nigel et al. | 2004
- 3263
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A novel 18β-glycyrrhetinic acid analogue as a potent and selective inhibitor of 11β-hydroxysteroid dehydrogenase 2Vicker, Nigel / Su, Xiangdong / Lawrence, Harshani et al. | 2004
- 3269
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2,3-Dihydro-1,3-dioxo-1H-isoindole-5-carboxylic acid derivatives: a novel class of small molecule heparanase inhibitorsCourtney, Stephen M. / Hay, Philip A. / Buck, Richard T. et al. | 2004
- 3275
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Long chain amines and long chain ammonium salts as novel inhibitors of dynamin GTPase activityHill, Timothy A. / Odell, Luke R. / Quan, Annie et al. | 2004
- 3279
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Simple and an efficient method for the synthesis of 1-(2-dimethylamino-1-(4-methoxy-phenyl)-ethyl)-cyclohexanol hydrochloride: ((plus-minus)) venlafaxine racemic mixturesBasappa et al. | 2004
- 3279
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Simple and an efficient method for the synthesis of 1-[2-dimethylamino-1-(4-methoxy-phenyl)-ethyl]-cyclohexanol hydrochloride: (±) venlafaxine racemic mixturesBasappa / Kavitha, C.V. / Rangappa, K.S. et al. | 2004
- 3283
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Carbonic anhydrase inhibitors: the first QSAR study on inhibition of tumor-associated isoenzyme IX with aromatic and heterocyclic sulfonamidesJaiswal, Mona / Khadikar, Padmakar V. / Scozzafava, Andrea et al. | 2004
- 3291
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Design and synthesis of dysidiolide analogs from vitamin D3: novel class of Cdc25A inhibitorsShimazawa, Rumiko / Suzuki, Toshiyuki / Dodo, Kosuke et al. | 2004
- 3295
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The effect of 6-substituted-4′,4″-difluorobenztropines on monoamine transporters and the muscarinic M1 receptorGrundt, Peter / Kopajtic, Theresa A. / Katz, Jonathan L. et al. | 2004
- 3295
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The effect of 6-substituted-4prime,4Prime-difluorobenztropines on monoamine transporters and the muscarinic M1 receptorGrundt, P. / Kopajtic, T. A. / Katz, J. L. et al. | 2004
- 3299
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Novel inhibitors of bacterial protein synthesis: structure–activity relationships for 1,8-naphthyridine derivatives incorporating position 3 and 4 variantsClark, Richard F. / Wang, Sanyi / Ma, Zhenkun et al. | 2004
- 3303
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New substituted triaza-benzo[cd]azulen-9-ones as promising phosphodiesterase-4 inhibitorsDevillers, Ingrid / Pevet, Isabelle / Jacobelli, Henry et al. | 2004
- 3307
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Comparison of inhibitory activity of isomeric triazolopyridine derivatives towards adenosine receptor subtypes or do similar structures reveal similar bioactivities?Guba, Wolfgang / Nettekoven, Matthias / Püllmann, Bernd et al. | 2004
- 3313
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Thiol-based SAHA analogues as potent histone deacetylase inhibitorsSuzuki, Takayoshi / Kouketsu, Akiyasu / Matsuura, Azusa et al. | 2004
- 3319
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The first synthesis of glucosylgalactosyl hydroxylysine (Glu-Gal-Hyl) an important biological indicator of collagen turnoverAllevi, Pietro / Anastasia, Mario / Paroni, Rita et al. | 2004
- 3323
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Synthesis of analogues of a potent antitumor saponin OSW-1Morzycki, Jacek W. / Wojtkielewicz, Agnieszka / Wołczyński, Sławomir et al. | 2004
- 3327
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Carbonic anhydrase inhibitors. Inhibition of the zinc and cobalt γ-class enzyme from the archaeon Methanosarcina thermophila with anionsInnocenti, Alessio / Zimmerman, Sabrina / Ferry, James G. et al. | 2004
- 3327
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Carbonic anhydrase inhibitors. Inhibition of the zinc and cobalt g-class enzyme from the archaeon Methanosarcina thermophila with anionsInnocenti, Alessio et al. | 2004
- 3333
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Nucleosides and nucleotides. Part 226: Alternate-strand triple-helix formation by 3′-3′-linked oligodeoxynucleotides composed of asymmetrical sequencesHoshika, Shuichi / Ueno, Yoshihito / Kamiya, Hiroyuki et al. | 2004
- 3333
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Nucleosides and nucleotides. Part 226: Alternate-strand triple-helix formation by 3prime-3prime-linked oligodeoxynucleotides composed of asymmetrical sequencesHoshika, S. / Ueno, Y. / Kamiya, H. et al. | 2004
- 3337
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Preparation of alkylation agents for bulged DNA microenvironmentsFouad, Farid S. / Xi, Zhen / Goldberg, Irving H. et al. | 2004
- 3341
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Anti-AIDS agents. Part 58: Synthesis and anti-HIV activity of 1-thia-di-O-(−)-camphanoyl-(+)-cis-khellactone (1-thia-DCK) analoguesXia, Peng / Yin, Zhi-Jian / Chen, Ying et al. | 2004
- 3345
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N2-Benzyl-N1-(1-(1-naphthyl)ethyl)-3-phenylpropane-1,2-diamines and conformationally restrained indole analogues: development of calindol as a new calcimimetic acting at the calcium sensing receptorKessler, Albane / Faure, Hélène / Petrel, Christophe et al. | 2004
- 3351
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Potent S1P receptor agonists replicate the pharmacologic actions of the novel immune modulator FTY720Hale, Jeffrey J. / Neway, William / Mills, Sander G. et al. | 2004
- 3357
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A new approach to the synthesis of optically active alkylated adenine derivativesZakirova, N.F. / Shipitsyn, A.V. / Belanov, E.F. et al. | 2003
- 3361
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Corrigendum to "Hydroxytriamides as potent g-secretase inhibitors"Prasad, C. V. / Wallace, O. B. / Noonan, J. W. et al. | 2004
- 3361
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Corrigendum to “Hydroxytriamides as potent γ-secretase inhibitors”Prasad, C.V.C. / Wallace, Owen B. / Noonan, Jeffrey W. et al. | 2004
- 3361
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Corrigendum to "Hydroxytriamides as potent g-secretase inhibitors" - (Bioorg. Med. Chem. Lett. 14 (2004) 1917)Prasad, C.V.C. et al. | 2004
- 3363
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Corrigendum to “Bridged bicyclic vasopressin receptor antagonists with V2-selective or dual V1a/V2 activity”Dyatkin, Alexey B. / Hoekstra, William J. / Hlasta, Dennis J. et al. | 2002
- 3363
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Corrigendum to "Bridged bicyclic vasopressin receptor antagonists with V2-selective or dual V1a-V2 activity" - (Bioorg. Med. Chem. Lett. 12 (2002) 3081)Dyatkin, Alexey B. et al. | 2004
- CO2
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Editorial board| 2004
- I
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Contributors to this issue| 2004
- V
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Instructions to contributors| 2004