Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 567
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Graphical contents list| 2007
- 583
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Synthesis and biological activation of an ethylene glycol-linked amino acid conjugate of cyclic cidofovirEriksson, Ulrika / Hilfinger, John M. / Kim, Jae-Seung et al. | 2006
- 587
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Design and synthesis of conformationally constrained tri-substituted ureas as potent antagonists of the human glucagon receptorLiang, Rui / Abrardo, Lauren / Brady, Edward J. et al. | 2006
- 593
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Synthesis and antimalarial activity of new 1,12-bis(N,Nprime-acetamidinyl)dodecane derivativesOuattara, M. / Wein, S. / Calas, M. et al. | 2007
- 593
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Synthesis and antimalarial activity of new 1,12-bis(N,N′-acetamidinyl)dodecane derivativesOuattara, Mahama / Wein, Sharon / Calas, Michèle et al. | 2006
- 597
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Highly constrained bicyclic VLA-4 antagonistsChang, Linda L. / Truong, Quang / Doss, George A. et al. | 2006
- 602
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Discovery of [7-(2,6-dichlorophenyl)-5-methylbenzo [1,2,4]triazin-3-yl]-[4-(2-pyrrolidin-1-ylethoxy)phenyl]amine—a potent, orally active Src kinase inhibitor with anti-tumor activity in preclinical assaysNoronha, Glenn / Barrett, Kathy / Boccia, Antonio et al. | 2006
- 609
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An efficient synthesis of quinoxaline derivatives from 4-chloro-4-deoxy-a-d-galactose and their cytotoxic activitiesYan, L. / Liu, F. W. / Dai, G. F. et al. | 2007
- 609
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An efficient synthesis of quinoxaline derivatives from 4-chloro-4-deoxy-α-d-galactose and their cytotoxic activitiesYan, Lin / Liu, Feng-Wu / Dai, Gui-Fu et al. | 2006
- 613
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Remarkable immunostimulation effects of hybrid liposomes on human peripheral blood mononuclear cells in vitroKomizu, Yuji / Tomonaga, Yuka / Goto, Koichi et al. | 2006
- 617
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Synthesis of 2prime-paclitaxel methyl 2-glucopyranosyl succinate for specific targeted delivery to cancer cellsLiu, D. Z. / Sinchaikul, S. / Reddy, P. V. et al. | 2007
- 617
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Synthesis of 2′-paclitaxel methyl 2-glucopyranosyl succinate for specific targeted delivery to cancer cellsLiu, Der-Zen / Sinchaikul, Supachok / Reddy, Peddiahgari Vasu Govardhana et al. | 2006
- 621
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Molecular iodine catalyzed synthesis of aryl-14H-dibenzo[a, j]xanthenes under solvent-free conditionPasha, Mohamed A. / Jayashankara, Vaderapura P. et al. | 2006
- 624
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Identification of the benzodiazepines as a new class of antileishmanial agentClark, Rachel L. / Carter, Katharine C. / Mullen, Alexander B. et al. | 2006
- 628
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Carbonic anhydrase activators: l-Adrenaline plugs the active site entrance of isozyme II, activating better isoforms I, IV, VA, VII, and XIVTemperini, Claudia / Innocenti, Alessio / Scozzafava, Andrea et al. | 2006
- 636
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Natural dibenzoxazepinones from leaves of Carex distachya: Structural elucidation and radical scavenging activityFiorentino, Antonio / D’Abrosca, Brigida / Pacifico, Severina et al. | 2006
- 640
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Synthesis of pyochelin–norfloxacin conjugatesRivault, Freddy / Liébert, Clémence / Burger, Alain et al. | 2006
- 645
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Synthesis and biological study of medicinally important Mannich bases derived from 4-(dimethylamino)-1,4,4a,5,5a,6,11,12a-octahydro-3,6,10,12,12a pentahydroxy naphthacene carboxamideJoshi, Sheela / Manikpuri, Anju Das / Tiwari, Prapti et al. | 2006
- 649
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Design of cell-permeable, fluorescent activity-based probes for the lysosomal cysteine protease asparaginyl endopeptidase (AEP)/legumainSexton, Kelly B. / Witte, Martin D. / Blum, Galia et al. | 2006
- 654
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Solid-phase synthesis of Stat3 inhibitors incorporating O-carbamoylserine and O-carbamoylthreonine as glutamine mimicsMandal, Pijus K. / Heard, Patricia A. / Ren, Zhiyong et al. | 2006
- 657
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Novel pyrazolopiperazinone- and pyrrolopiperazinone-based MCH-R1 antagonistsMeyers, Kenneth M. / Méndez-Andino, José / Colson, Anny-Odile et al. | 2006
- 662
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Synthesis and SAR of novel 2-arylthiazolidinones as selective analgesic N-type calcium channel blockersKnutsen, Lars J.S. / Hobbs, Christopher J. / Earnshaw, Christopher G. et al. | 2006
- 668
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Discovery of a new class of 4-anilinopyrimidines as potent c-Jun N-terminal kinase inhibitors: Synthesis and SAR studiesLiu, Mei / Wang, Sanyi / Clampit, Jill E. et al. | 2006
- 673
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Constrained analogs of CB-1 antagonists: 1,5,6,7-Tetrahydro-4H-pyrrolo[3,2-c]pyridine-4-one derivativesSmith, Roger A. / Fathi, Zahra / Brown, Su-Ellen et al. | 2006
- 679
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Core exploration in optimization of chemokine receptor CCR4 antagonistsPurandare, Ashok V. / Wan, Honghe / Somerville, John E. et al. | 2006
- 683
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Synthesis and biological activities of novel dexibuprofen tetraacetylriboflavin conjugatesBanekovich, Christian / Ott, Ingo / Koch, Thao et al. | 2006
- 688
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Structural basis for the inhibition of Aurora A kinase by a novel class of high affinity disubstituted pyrimidine inhibitorsTari, Leslie W. / Hoffman, Isaac D. / Bensen, Daniel C. et al. | 2006
- 692
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Influence of an additional 2-amino substituent of the 1-aminoethyl pharmacophore group on the potency of rimantadine against influenza virus ATataridis, Dimitrios / Fytas, George / Kolocouris, Antonios et al. | 2006
- 697
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Identification and structure–activity relationships of 1-aryl-3-piperidin-4-yl-urea derivatives as CXCR3 receptor antagonistsAllen, Daniel R. / Bolt, Amanda / Chapman, Gayle A. et al. | 2006
- 702
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Dual serotonin transporter/histamine H3 ligands: Optimization of the H3 pharmacophoreKeith, John M. / Gomez, Leslie A. / Letavic, Michael A. et al. | 2006
- 707
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Design, synthesis, and evaluation of efflux substrate–metal chelator conjugates as potential antimicrobial agentsZhang, Yanling / Eric Ballard, C. / Zheng, Shi-Long et al. | 2006
- 712
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Structure–activity relationship in the 3-iodo-4-phenoxypyridinone (IOPY) series: The nature of the C-3 substituent on anti-HIV activityBenjahad, Abdellah / Oumouch, Said / Guillemont, Jerôme et al. | 2006
- 717
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Thiosialoside clusters using carbosilane dendrimer core scaffolds as a new class of influenza neuraminidase inhibitorsSakamoto, Jun-Ichi / Koyama, Tetsuo / Miyamoto, Daisei et al. | 2006
- 722
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Pharmacophore identification of KSP inhibitorsLiu, Fei / You, Qi-Dong / Chen, Ya-Dong et al. | 2006
- 727
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Spirodiketopiperazine-based CCR5 antagonists: Lead optimization from biologically active metaboliteNishizawa, Rena / Nishiyama, Toshihiko / Hisaichi, Katsuya et al. | 2006
- 732
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1,5-Biaryl pyrrole derivatives as EP1 receptor antagonists: Structure–activity relationships of 4- and 5-substituted benzoic acid derivativesHall, Adrian / Brown, Susan H. / Chessell, Iain P. et al. | 2006
- 736
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Benzothiazole benzimidazole (S)-isothiazolidinone derivatives as protein tyrosine phosphatase-1B inhibitorsSparks, Richard B. / Polam, Padmaja / Zhu, Wenyu et al. | 2006
- 741
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Synthesis of a technetium-99m labeled tricyclic ganciclovir analog for non-invasive reporter gene expression imagingZhang, Yi / Lin, Jing / Pan, Dongfeng et al. | 2006
- 745
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Analogues of the dopamine D2 receptor antagonist L741,626: Binding, function, and SARGrundt, Peter / Jane Husband, Sarah Little / Luedtke, Robert R. et al. | 2006
- 750
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Discovery of adamantane ethers as inhibitors of 11β-HSD-1: Synthesis and biological evaluationPatel, Jyoti R. / Shuai, Qi / Dinges, Jurgen et al. | 2006
- 750
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Discovery of adamantane ethers as inhibitors of 11b-HSD-1: Synthesis and biological evaluationPatel, J. R. / Shuai, Q. / Dinges, J. et al. | 2007
- 756
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Design and synthesis of phenethyl benzo[1,4]oxazine-3-ones as potent inhibitors of PI3KinaseγLanni, Thomas B. Jr. / Greene, Keri L. / Kolz, Christine N. et al. | 2006
- 756
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Design and synthesis of phenethyl benzo[1,4]oxazine-3-ones as potent inhibitors of PI3KinasegLanni, T. B. / Greene, K. L. / Kolz, C. N. et al. | 2007
- 761
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Molecular dynamics simulation of the P2Y14 receptor. Ligand docking and identification of a putative binding site of the distal hexose moietyIvanov, Andrei A. / Fricks, Ingrid / Kendall Harden, T. et al. | 2006
- 767
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Dopamine-selective potentiometric responses by new ditopic sensory elements based on a hexahomotrioxacalix[3]areneSaijo, Ryosuke / Tsunekawa, Saori / Murakami, Hiroyuki et al. | 2006
- 772
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Anti-influenza virus activity of biflavonoidsMiki, Kazuhiko / Nagai, Takayuki / Suzuki, Kazushige et al. | 2006
- 776
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Chemico-enzymatic synthesis of a new fluorescent-labeled DNA by PCR with a thymidine nucleotide analogue bearing an acridone derivativeShoji, Atsushi / Hasegawa, Tomoya / Kuwahara, Masayasu et al. | 2006
- 780
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Synthesis and antiproliferative activity of (2R,3R)-disubstituted tetrahydropyrans. Part 2: Effect of side chain homologationCarrillo, Romen / León, Leticia G. / Martı´n, Tomás et al. | 2006
- 784
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Synthesis and SAR of potent and selective androgen receptor antagonists: 5,6-Dichloro-benzimidazole derivativesNg, Raymond A. / Guan, Jihua / Alford, Vernon C. Jr. et al. | 2006
- 789
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PDE5 inhibitors: An original access to novel potent arylated analogues of tadalafilBeghyn, Terence / Hounsou, Candide / Deprez, Benoit P. et al. | 2006
- 793
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Discovery of galectin ligands in fully randomized combinatorial one-bead-one-compound (glyco)peptide librariesAndré, Sabine / Maljaars, C. Elizabeth P. / Halkes, Koen M. et al. | 2006
- 799
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Chalcone based aryloxypropanolamines as potential antihyperglycemic agentsShukla, Poonam / Singh, Amar Bahadur / Srivastava, Arvind Kumar et al. | 2006
- 803
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Synthesis and DNA-binding ability of C2R-fluoro substituted DC-81 and its dimersKamal, Ahmed / Rajasekhar Reddy, D. / Murali Mohan Reddy, P.S. et al. | 2006
- 807
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Diaryl substituted pyrazoles as potent CCR2 receptor antagonistsPinkerton, Anthony B. / Huang, Dehua / Cube, Rowena V. et al. | 2006
- 814
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Aminomethyl tetrahydronaphthalene biphenyl carboxamide MCH-R1 antagonists—Increasing selectivity over hERGMeyers, Kenneth M. / Kim, Nicholas / Méndez-Andino, José L. et al. | 2006
- 819
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Aminomethyl tetrahydronaphthalene ketopiperazine MCH-R1 antagonists—Increasing selectivity over hERGMeyers, Kenneth M. / Méndez-Andino, José L. / Colson, Anny-Odile et al. | 2006
- 823
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Evaluating scoring functions for docking and designing b-secretase inhibitorsKatharine Holloway, M. / McGaughey, G. B. / Coburn, C. A. et al. | 2007
- 823
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Evaluating scoring functions for docking and designing β-secretase inhibitorsKatharine Holloway, M. / McGaughey, Georgia B. / Coburn, Craig A. et al. | 2006
- 828
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SAR studies of 3-arylpropionic acids as potent and selective agonists of sphingosine-1-phosphate receptor-1 (S1P1) with enhanced pharmacokinetic propertiesYan, Lin / Huo, Pei / Hale, Jeffrey J. et al. | 2006
- 832
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MCH-R1 antagonists based on an arginine scaffold: SAR studies on the amino-terminusMéndez-Andino, José / Colson, Anny-Odile / Denton, Daniel et al. | 2006
- 836
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Solid phase-assisted synthesis and screening of a small library of N-(4-hydroxyphenyl)retinamide (4-HPR) analogsMershon, Serena M. / Anding, Allyson L. / Chapman, Jason S. et al. | 2006
- 841
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Synthesis of thiazolone-based sulfonamides as inhibitors of HCV NS5B polymeraseDing, Yili / Smith, Kenneth L. / Varaprasad, Chamakura V.N.S. et al. | 2006
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Editorial board| 2007
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Instructions to contributors| 2007