Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 4369
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Graphical contents list| 2011
- 4385
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Simple but powerful: Phenanthroline-based small molecules for cellular imaging and cancer screeningSergeeva, Natalia N. / Donnier-Marechal, Marion / Vaz, Gisela M. et al. | 2011
- 4389
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New C-23 modified of silybin and 2,3-dehydrosilybin: Synthesis and preliminary evaluation of antioxidant propertiesZarrelli, Armando / Sgambato, Alessandro / Petito, Valentina et al. | 2011
- 4393
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Construction of a 19F-lectin biosensor for glycoprotein imaging by using affinity-guided DMAP chemistrySun, Yedi / Takaoka, Yousuke / Tsukiji, Shinya et al. | 2011
- 4397
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Nothospondin, a new AP-1 inhibitory quassinoid from the Cameroonian plant Nothospondias staudtiiDiyabalanage, Thushara / Ratnayake, Ranjala / Wilson, Jennifer A. et al. | 2011
- 4400
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Flavans from Iris tenuifolia and their effects on β-amyloid aggregation and neural stem cells proliferation in vitroCui, Yan-Mei / Wang, Hui / Liu, Quan-Ru et al. | 2011
- 4400
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Flavans from Iris tenuifolia and their effects on b-amyloid aggregation and neural stem cells proliferation in vitroCui, Y. M. / Wang, H. / Liu, Q. R. et al. | 2011
- 4404
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Synthesis, molecular modeling and bio-evaluation of cycloalkyl fused 2-aminopyrimidines as antitubercular and antidiabetic agentsSingh, Nimisha / Pandey, Sarvesh Kumar / Anand, Namrata et al. | 2011
- 4409
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Azepanone-based inhibitors of human cathepsin S: Optimization of selectivity via the P2 substituentKerns, Jeffrey K. / Nie, Hong / Bondinell, William et al. | 2011
- 4416
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Antiproliferative activity and QSAR studies of a series of new 4-aminomethylidene derivatives of some pyrazol-5-onesMarković, Violeta / Erić, Slavica / Stanojković, Tatjana et al. | 2011
- 4422
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Identification of MK-5710 ((8aS)-8a-methyl-1,3-dioxo-2-[(1S,2R)-2-phenylcyclopropyl]-N-(1-phenyl-1H-pyrazol-5-yl)hexahydroimid azo[1,5-a]pyrazine-7(1H)-carboxamide), a potent smoothened antagonist for use in Hedgehog pathway dependent malignancies, Part 1Malancona, Savina / Altamura, Sergio / Filocamo, Gessica et al. | 2011
- 4429
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Identification of MK-5710 ((8aS)-8a-methyl-1,3-dioxo-2-[(1S,2R)-2-phenylcyclo- propyl]-N-(1-phenyl-1H-pyrazol-5-yl)hexahydro-imidazo[1,5-a]pyrazine-7(1H)-carboxamide), a potent smoothened antagonist for use in Hedgehog pathway dependent malignancies, Part 2Kinzel, Olaf / Alfieri, Anna / Altamura, Sergio et al. | 2011
- 4436
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Development of potent B-RafV600E inhibitors containing an arylsulfonamide headgroupStellwagen, John C. / Adjabeng, George M. / Arnone, Marc R. et al. | 2011
- 4441
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New isoprenylated flavonoids and adipogenesis-promoting constituents from Morus notabilisHu, Xiao / Ji, Jun / Wang, Meng et al. | 2011
- 4447
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N-β-Glycosyl sulfamides are selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XIIRodríguez, Oscar M. / Maresca, Alfonso / Témpera, Carlos A. et al. | 2011
- 4447
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N-b-Glycosyl sulfamides are selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XIIRodriguez, O. M. / Maresca, A. / Tempera, C. A. et al. | 2011
- 4451
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Design, synthesis and antimycobacterial evaluation of novel 3-substituted-N-aryl-6,7-dimethoxy-3a,4-dihydro-3H-indeno[1,2-c]pyrazole-2-carboxamide analoguesAhsan, Mohamed Jawed / Samy, Jeyabalan Govinda / Dutt, Kunduri Rajeswar et al. | 2011
- 4454
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Synthesis and antihistamine evaluations of novel loratadine analoguesWang, Yue / Wang, Juan / Lin, Yan et al. | 2011
- 4457
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Structure–activity study on a series of α-glutamic acid scaffold based compounds as new ADAMTS inhibitorsPeng, Lijie / Duan, Lei / Liu, Xiaofeng et al. | 2011
- 4457
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Structure-activity study on a series of a-glutamic acid scaffold based compounds as new ADAMTS inhibitorsPeng, L. / Duan, L. / Liu, X. et al. | 2011
- 4462
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Cytotoxicity of aporphines in human colon cancer cell lines HCT-116 and Caco-2: An SAR studyPonnala, Shashikanth / Chaudhary, Sandeep / González-Sarrias, Antonio et al. | 2011
- 4465
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C-Aryl glucosides substituted at the 4prime-position as potent and selective renal sodium-dependent glucose co-transporter 2 (SGLT2) inhibitors for the treatment of type 2 diabetesXu, B. / Feng, Y. / Cheng, H. et al. | 2011
- 4465
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C-Aryl glucosides substituted at the 4′-position as potent and selective renal sodium-dependent glucose co-transporter 2 (SGLT2) inhibitors for the treatment of type 2 diabetesXu, Baihua / Feng, Yan / Cheng, Huawei et al. | 2011
- 4471
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Synthesis, in vitro evaluation and molecular docking studies of new triazole derivatives as antifungal agentsJiang, Yongwei / Zhang, Jun / Cao, Yongbing et al. | 2011
- 4476
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Hydrophobic tag-assisted liquid-phase synthesis of a growth hormone-inhibiting peptide somatostatinKitada, Shingo / Fujita, Shuji / Okada, Yohei et al. | 2011
- 4480
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Synthesis and anti-inflammatory activity of novel biscoumarin–chalcone hybridsSashidhara, Koneni V. / Kumar, Manoj / Modukuri, Ram K. et al. | 2011
- 4485
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Limonoids from seeds of Thai Xylocarpus moluccensisRavangpai, Warin / Sommit, Damrong / Teerawatananond, Thapong et al. | 2011
- 4490
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Pharmacophore modeling and virtual screening to identify potential RET kinase inhibitorsShih, Kuei-Chung / Shiau, Chung-Wai / Chen, Ting-Shou et al. | 2011
- 4498
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New salicylamide and sulfonamide derivatives of quinoxaline 1,4-di-N-oxide with antileishmanial and antimalarial activitiesBarea, Carlos / Pabón, Adriana / Castillo, Denis et al. | 2011
- 4503
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Facile conversion of RNA aptamers to modular fluorescent sensors with tunable detection wavelengthsNakano, Shun / Nakata, Eiji / Morii, Takashi et al. | 2011
- 4507
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Synthesis and SAR of new pyrazolo[4,3-h]quinazoline-3-carboxamide derivatives as potent and selective MPS1 kinase inhibitorsCaldarelli, Marina / Angiolini, Mauro / Disingrini, Teresa et al. | 2011
- 4512
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Synthesis and biological activities of 4-N-(anilinyl-n-[oxazolyl])-7-chloroquinolines (n=3prime or 4prime) against Plasmodium falciparum in in vitro modelsGordey, E. E. / Yadav, P. N. / Merrin, M. P. et al. | 2011
- 4512
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Synthesis and biological activities of 4-N-(anilinyl-n-[oxazolyl])-7-chloroquinolines (n =3′ or 4′) against Plasmodium falciparum in in vitro modelsGordey, Erin E. / Yadav, Paras N. / Merrin, Marcus P. et al. | 2011
- 4516
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A facile synthesis of 1,5-disubstituted-2-aminoimidazoles: Antibiotic activity of a first generation libraryHarris, Tyler L. / Worthington, Roberta J. / Melander, Christian et al. | 2011
- 4520
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Synthesis of aurones and their inhibitory effects on nitric oxide and PGE2 productions in LPS-induced RAW 264.7 cellsShin, Seo Young / Shin, Min Cheol / Shin, Ji-Sun et al. | 2011
- 4524
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Structure–activity studies of RNA-binding oxazolidinone derivativesMaciagiewicz, Iwona / Zhou, Shu / Bergmeier, Stephen C. et al. | 2011
- 4528
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Identification of benzofuran-4,5-diones as novel and selective non-hydroxamic acid, non-peptidomimetic based inhibitors of human peptide deformylaseAntczak, Christophe / Shum, David / Bassit, Bhramdeo et al. | 2011
- 4533
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Benzimidazolone as potent chymase inhibitor: Modulation of reactive metabolite formation in the hydrophobic (P1) regionLo, Ho Yin / Nemoto, Peter A. / Kim, Jin Mi et al. | 2011
- 4540
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Nobiletin metabolites: Synthesis and inhibitory activity against matrix metalloproteinase-9 productionOshitari, Tetsuta / Okuyama, Yuji / Miyata, Yoshiki et al. | 2011
- 4545
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Benzisothiazolones as modulators of macrophage migration inhibitory factorJorgensen, William L. / Trofimov, Alexander / Du, Xin et al. | 2011
- 4550
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Discovery of imidazo[1,2-b]pyridazines as IKKβ inhibitors. Part 3: Exploration of effective compounds in arthritis modelsShimizu, Hiroki / Yamasaki, Tomonori / Yoneda, Yoshiyuki et al. | 2011
- 4550
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Discovery of imidazo[1,2-b]pyridazines as IKKb inhibitors. Part 3: Exploration of effective compounds in arthritis modelsShimizu, H. / Yamasaki, T. / Yoneda, Y. et al. | 2011
- 4556
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Discovery of bacterial NAD+-dependent DNA ligase inhibitors: Optimization of antibacterial activityStokes, Suzanne S. / Huynh, Hoan / Gowravaram, Madhusudhan et al. | 2011
- 4561
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Antiplasmodial and cytotoxicity evaluation of 3-functionalized 2-azetidinone derivativesSingh, Pardeep / Sachdeva, Shaveta / Raj, Raghu et al. | 2011
- 4564
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Photosynthesis—Inhibiting efficiency of 4-chloro-2-(chlorophenylcarbamoyl)phenyl alkylcarbamatesImramovsky, Ales / Pesko, Matus / Ferriz, Juana Monreal et al. | 2011
- 4568
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Antiproliferative activity of dmoPTA–Ru(II) complexes against human solid tumor cellsRíos-Luci, Carla / León, Leticia G. / Mena-Cruz, Adrián et al. | 2011
- 4572
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Synthesis and antiproliferative activity of novel a- and b-dialkoxyphosphoryl isothiocyanatesPsurski, M. / Blazewska, K. / Gajda, A. et al. | 2011
- 4572
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Synthesis and antiproliferative activity of novel α- and β-dialkoxyphosphoryl isothiocyanatesPsurski, Mateusz / Błażewska, Katarzyna / Gajda, Anna et al. | 2011
- 4577
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Rigidized 1-aryl sulfonyl tryptamines: Synthesis and pharmacological evaluation as 5-HT6 receptor ligandsNirogi, Ramakrishna / Dwarampudi, Adireddy / Kambhampati, Ramasastry et al. | 2011
- 4581
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Cytotoxic diterpenoid quinonemethides from the roots of Pygmacopremna herbaceaSatish, K. / Vishnuvardhan, M.V.P.S. / Lakshma Nayak, V. et al. | 2011
- 4585
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Synthesis and evaluation of 1-cyclopropyl-2-thioalkyl-8-methoxy fluoroquinolonesMarks, Kevin R. / Malik, Muhammad / Mustaev, Arkady et al. | 2011
- 4589
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A convenient method to prepare emulsified polyacrylate nanoparticles from for drug delivery applicationsGaray-Jimenez, Julio C. / Turos, Edward et al. | 2011
- 4592
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Synthesis of an aryloxy oxo pyrimidinone library that displays ALK-selective inhibitionSlavish, P. Jake / Price, Jeanine E. / Jiang, Qin et al. | 2011
- 4597
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The tandem chain extension aldol reaction used for synthesis of ketomethylene tripeptidomimetics targeting hPEPT1Thorn, Karina / Nielsen, Carsten Uhd / Jakobsen, Palle et al. | 2011
- 4602
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Discovery of a stable macrocyclic o-aminobenzamide Hsp90 inhibitor which significantly decreases tumor volume in a mouse xenograft modelZapf, Christoph W. / Bloom, Jonathan D. / Li, Zhong et al. | 2011
- 4608
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Discovery and synthesis of a new class of opioid ligand having a 3-azabicyclo[3.1.0]hexane core. An example of a ‘magic methyl’ giving a 35-fold improvement in bindingLunn, Graham / Banks, Bernard J. / Crook, Robert et al. | 2011
- 4612
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Design-driven LO: The discovery of new ultra long acting dibasic β2-adrenoceptor agonistsConnolly, Stephen / Alcaraz, Lilian / Bailey, Andrew et al. | 2011
- 4612
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Design-driven LO: The discovery of new ultra long acting dibasic b2-adrenoceptor agonistsConnolly, S. / Alcaraz, L. / Bailey, A. et al. | 2011
- 4617
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Osteogenic constituents from Pterospermum acerifolium Willd. flowersDixit, Preety / Khan, Mohd Parvez / Swarnkar, Gaurav et al. | 2011
- 4622
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Optimisation of pharmacokinetic properties to afford an orally bioavailable and selective V1A receptor antagonistArbuckle, William / Baker, James / Barn, David et al. | 2011
- 4629
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Synthesis of d-labeled and unlabeled benzoyloxysuccinimides and application to quantitative analysis of peptides and a protein by isotope differential mass spectrometryZabet-Moghaddam, Masoud / Shaikh, Aarif L. / Jones, Lauren B. et al. | 2011
- 4633
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Discovery of pyrrolo[2,1-f][1,2,4]triazine C6-ketones as potent, orally active p38α MAP kinase inhibitorsDyckman, Alaric J. / Li, Tianle / Pitt, Sidney et al. | 2011
- 4633
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Discovery of pyrrolo[2,1-f][1,2,4]triazine C6-ketones as potent, orally active p38a MAP kinase inhibitorsDyckman, A. J. / Li, T. / Pitt, S. et al. | 2011
- 4638
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Internalization of a C17α-alkynylestradiol-porphyrin conjugate into estrogen receptor positive MCF-7 breast cancer cellsSadler, Sara / Persons, Kelly S. / Jones, Graham B. et al. | 2011
- 4638
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Internalization of a C17a-alkynylestradiol-porphyrin conjugate into estrogen receptor positive MCF-7 breast cancer cellsSadler, S. / Persons, K. S. / Jones, G. B. et al. | 2011
- 4642
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Phenylpropenamide derivatives: Anti-hepatitis B virus activity of the Z isomer, SAR and the search for novel analogsWang, Peiyuan / Naduthambi, Devan / Mosley, Ralph T. et al. | 2011
- 4648
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The novel 3,4-dihydropyrimidin-2(1H)-one urea derivatives of N-aryl urea: Synthesis, anti-inflammatory, antibacterial and antifungal activity evaluationTale, Rajesh H. / Rodge, Atish H. / Hatnapure, Girish D. et al. | 2011
- 4652
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Discovery of potent, soluble and orally active TRPV1 antagonists. Structure–activity relationships of a series of isoxazolesRatcliffe, Paul / Abernethy, Lynn / Ansari, Nasrin et al. | 2011
- 4658
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Corrigendum to "Selective a-glucosidase substrates and inhibitors containing short aromatic peptidyl moieties" [Bioorg. Med. Chem. Lett. 21 (2011) 2441-2444]Park, S. / Hyu, S. / Do, S. i. et al. | 2011
- 4658
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Corrigendum to “Selective α-glucosidase substrates and inhibitors containing short aromatic peptidyl moieties” [Bioorg. Med. Chem. Lett. 21 (2011) 2441–2444]Park, Sangeun / Hyu, Soonsil / Do, Su-il et al. | 2011
- IFC
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Editorial board| 2011