Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 4031
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Graphical contents list| 2015
- 4047
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Recent progress on MAP kinase pathway inhibitorsUehling, David E. / Harris, Philip A. et al. | 2015
- 4057
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Recent progress in the development of small-molecule glucagon receptor antagonistsSammons, Matthew F. / Lee, Esther C.Y. et al. | 2015
- 4065
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Synthesis and herbicidal activities of benzothiazole N,O-acetalsJi, Zhiqin / Zhou, Fengxing / Wei, Shaopeng et al. | 2015
- 4069
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Discovery of novel nonpeptide allosteric inhibitors interrupting the interaction of CDK2/cyclin A3 by virtual screening and bioassaysHu, Yutong / Li, Shuai / Liu, Fang et al. | 2015
- 4074
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Efficient cleavage of DNA oligonucleotides by a non-FokI-type zinc finger nuclease containing one His4-type finger domain derived from the first finger domain of Sp1Negi, Shigeru / Yoshioka, Michiko / Mima, Hiroko et al. | 2015
- 4074
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Efficient cleavage of DNA oligonucleotides by a non-FokI-type zinc finger nuclease containing one His₄-type finger domain derived from the first finger domain of Sp1Kano, Koji et al. | 2015
- 4078
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Syntheses of new chlorin derivatives containing maleimide functional group and their photodynamic activity evaluationGuo, Xiuhan / Wang, Liu / Wang, Shisheng et al. | 2015
- 4082
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Dicarabrol, a new dimeric sesquiterpene from Carpesium abrotanoides L.Wang, Jun-Feng / He, Wei-Jun / Zhang, Xiao-Xiao et al. | 2015
- 4085
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Integrated kinetic studies and computational analysis on naphthyl chalcones as mushroom tyrosinase inhibitorsRadhakrishnan, Sini / Shimmon, Ronald / Conn, Costa et al. | 2015
- 4092
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Synthesis, structure–activity relationship and biological evaluation of novel nitrogen mustard sophoridinic acid derivatives as potential anticancer agentsLi, Dong-Dong / Dai, Lin-Lin / Zhang, Na et al. | 2015
- 4097
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Catechols and 3-hydroxypyridones as inhibitors of the DNA repair complex ERCC1-XPFChapman, Timothy M. / Gillen, Kevin J. / Wallace, Claire et al. | 2015
- 4104
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N-Hydroxyimides and hydroxypyrimidinones as inhibitors of the DNA repair complex ERCC1–XPFChapman, Timothy M. / Wallace, Claire / Gillen, Kevin J. et al. | 2015
- 4109
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Identification of N-sulfonyl-tetrahydroquinolines as RORc inverse agonistsFauber, Benjamin P. / Gobbi, Alberto / Savy, Pascal et al. | 2015
- 4114
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Tris(3-hydroxypropyl)phosphine (THPP): A mild, air-stable reagent for the rapid, reductive cleavage of small-molecule disulfidesMcNulty, James / Krishnamoorthy, Venkatesan / Amoroso, Dino et al. | 2015
- 4118
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Identification of triazolo[4,5-b]pyrazine derivatives as hepatocyte growth factor receptor inhibitors through structure–activity relationships and molecular docking simulationsDong, Minghui / Ren, Yujie / Gao, Xiaodong et al. | 2015
- 4127
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Solid-phase synthesis of 5′-triantennary N-acetylgalactosamine conjugated antisense oligonucleotides using phosphoramidite chemistryPrakash, Thazha P. / Brad Wan, W. / Low, Audrey et al. | 2015
- 4131
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Differential influence of 7 cations on 16 non-competitive NMDA receptor blockersBerger, Michael L. / Rebernik, Patrick et al. | 2015
- 4136
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The imidazo[1,2-a]pyridine ring system as a scaffold for potent dual phosphoinositide-3-kinase (PI3K)/mammalian target of rapamycin (mTOR) inhibitorsStec, Markian M. / Andrews, Kristin L. / Bo, Yunxin et al. | 2015
- 4143
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A novel series of indazole-/indole-based glucagon receptor antagonistsLin, Songnian / Zhang, Fengqi / Jiang, Guoqiang et al. | 2015
- 4148
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Design, synthesis and biological evaluation of multifunctional ligands targeting opioid and bradykinin 2 receptorsDeekonda, Srinivas / Rankin, David / Davis, Peg et al. | 2015
- 4153
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Predicting hydration propensities of biologically relevant α-ketoamidesWedler, Henry B. / Palazzo, Teresa A. / Pemberton, Ryan P. et al. | 2015
- 4158
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Design and synthesis of N-[6-(Substituted Aminoethylideneamino)-2-Hydroxyindan-1-yl]arylamides as selective and potent muscarinic M1 agonistsLiu, Bin / Croy, Carrie H. / Hitchcock, Stephen A. et al. | 2015
- 4158
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Design and synthesis of N-[6-(Substituted Aminoethylideneamino)-2-Hydroxyindan-1-yl]arylamides as selective and potent muscarinic M₁ agonistsLiu, Bin et al. | 2015
- 4164
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Expanding the structural diversity of Bcr-Abl inhibitors: Hybrid molecules based on GNF-2 and ImatinibPan, Xiaoyan / Dong, Jinyun / Shao, Ruili et al. | 2015
- 4169
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One-pot synthesis of new triazole—Imidazo[2,1-b][1,3,4]thiadiazole hybrids via click chemistry and evaluation of their antitubercular activityRamprasad, Jurupula / Nayak, Nagabhushana / Dalimba, Udayakumar et al. | 2015
- 4174
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Design and synthesis of carborane-containing estrogen receptor-beta (ERβ)-selective ligandsOhta, Kiminori / Ogawa, Takumi / Oda, Akifumi et al. | 2015
- 4179
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A simple and efficient dispersion correction to the Hartree–Fock theory (2): Incorporation of a geometrical correction for the basis set superposition errorYoshida, Tatsusada / Hayashi, Takahisa / Mashima, Akira et al. | 2015
- 4185
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Design and synthesis of 11α-substituted bile acid derivatives as potential anti-tuberculosis agentsPore, Vandana S. / Divse, Jaisingh M. / Charolkar, Chaitanya R. et al. | 2015
- 4191
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Induction of apoptosis by genipin inhibits cell proliferation in AGS human gastric cancer cells via Egr1/p21 signaling pathwayKo, Hyeonseok / Kim, Jee Min / Kim, Sun-Joong et al. | 2015
- 4197
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Nanoparticle-encapsulated P2X7 receptor antagonist in a pH-sensitive polymer as a potential local drug delivery system to acidic inflammatory environmentsLee, Sun-Mi / Cho, Joong-Heui / Lee, So-Deok et al. | 2015
- 4197
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Nanoparticle-encapsulated P2X₇ receptor antagonist in a pH-sensitive polymer as a potential local drug delivery system to acidic inflammatory environmentsCho, Joong-Heui et al. | 2015
- 4203
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7-(Pyrazol-4-yl)-3H-imidazo[4,5-b]pyridine-based derivatives for kinase inhibition: Co-crystallisation studies with Aurora-A reveal distinct differences in the orientation of the pyrazole N1-substituentBavetsias, Vassilios / Pérez-Fuertes, Yolanda / McIntyre, Patrick J. et al. | 2015
- 4210
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Biological evaluation of angular disubstituted naphthoimidazoles as anti-inflammatory agentsCuadrado-Berrocal, Irene / Guedes, Gema / Estevez-Braun, Ana et al. | 2015
- 4214
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A novel sesquiterpene and three new phenolic compounds from the rhizomes of Acorus tatarinowii SchottLiang, Shuang / Ying, Shu-Song / Wu, Hong-Hua et al. | 2015
- 4219
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Discovery, synthesis and biochemical profiling of purine-2,6-dione derivatives as inhibitors of the human poly(A)-selective ribonuclease Caf1Jadhav, Gopal P. / Kaur, Ishwinder / Maryati, Maryati et al. | 2015
- 4225
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2-(3′-Indolyl)-N-arylthiazole-4-carboxamides: Synthesis and evaluation of antibacterial and anticancer activitiesTantak, Mukund P. / Wang, Jing / Singh, Rajnish Prakash et al. | 2015
- 4232
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Synthesis of BF3 catalyzed Mannich derivatives with excellent ee from phenylpropanolamine, study of their antimicrobial activity and molecular dockingChennakesava Rao, K. / Easwaramoorthi, K. / Arun, Y. et al. | 2015
- 4232
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Synthesis of BF₃ catalyzed Mannich derivatives with excellent ee from phenylpropanolamine, study of their antimicrobial activity and molecular dockingBalachandran, C et al. | 2015
- 4239
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One-pot synthesis of podophyllotoxin-thiourea congeners by employing NH₂SO₃H/NaI: Anticancer activity, DNA topoisomerase-II inhibition, and apoptosis inducing agentsShankaraiah, Nagula et al. | 2015
- 4239
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One-pot synthesis of podophyllotoxin–thiourea congeners by employing NH2SO3H/NaI: Anticancer activity, DNA topoisomerase-II inhibition, and apoptosis inducing agentsShankaraiah, Nagula / Kumar, Niggula Praveen / Amula, Suresh Babu et al. | 2015
- 4245
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Discovery of novel 5,6,7,8-tetrahydro[1,2,4]triazolo[4,3-a]pyridine derivatives as γ-secretase modulatorsTakai, Takafumi / Hoashi, Yasutaka / Tomata, Yoshihide et al. | 2015
- 4250
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Novel 11β-HSD1 inhibitors: C-1 versus C-2 substitution and effect of the introduction of an oxygen atom in the adamantane scaffoldLeiva, Rosana / Seira, Constantí / McBride, Andrew et al. | 2015
- 4254
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Technetium glucose complexes as potential cancer imaging agentsDapueto, Rosina / Aguiar, Rodrigo B. / Moreno, María et al. | 2015
- 4260
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Optimization of a small molecule probe that restores e-cadherin expressionBrogan, John T. / Stoops, Sydney L. / Brady, Suzanne et al. | 2015
- 4265
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Design and synthesis of carbazole carboxamides as promising inhibitors of Bruton’s tyrosine kinase (BTK) and Janus kinase 2 (JAK2)Liu, Qingjie / Batt, Douglas G. / Lippy, Jonathan S. et al. | 2015
- 4270
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Factors influencing the cytotoxicity of α-methylene-γ-hydroxy esters against pancreatic cancerRamachandran, P. Veeraraghavan / Helppi, Matthew A. / Lehmkuhler, Arlie L. et al. | 2015
- 4274
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Thiophene-expanded guanosine analogues of GemcitabineChen, Zhe / Ku, Therese C. / Seley-Radtke, Katherine L. et al. | 2015
- 4277
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2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFRL858R/T790MChan, Shingpan / Han, Kun / Qu, Rong et al. | 2015
- 4277
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2,4-Diarylamino-pyrimidines as kinase inhibitors co-targeting IGF1R and EGFR(L⁸⁵⁸R/T⁷⁹⁰M)Cheng, Huimin et al. | 2015
- 4282
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Synthesis and biological evaluation of new symmetric curcumin derivativesSribalan, Rajendran / Kirubavathi, Maruthan / Banuppriya, Govindharaj et al. | 2015
- 4287
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Probing a 3,4′-bis-guanidinium diaryl derivative as an allosteric inhibitor of the Ras pathwayDiez-Cecilia, Elena / Carson, Robert / Kelly, Brendan et al. | 2015
- 4293
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Chemical structure and biological activity of a quorum sensing pheromone from Bacillus subtilis subsp. nattoOkada, Masahiro / Nakamura, Yuta / Hayashi, Shunsuke et al. | 2015
- 4297
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Expanding the chemical space of human serine racemase inhibitorsDellafiora, Luca / Marchetti, Marialaura / Spyrakis, Francesca et al. | 2015
- 4304
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Vascular barrier protective effects of 3-N- or 3-O-cinnamoyl carbazole derivativesKu, Sae-Kwang / Lee, Jee-Hyun / O, Yuseok et al. | 2015
- 4308
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Design of novel dispirooxindolopyrrolidine and dispirooxindolopyrrolothiazole derivatives as potential antitubercular agentsMhiri, Chourouk / Boudriga, Sarra / Askri, Moheddine et al. | 2015
- 4314
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Re-engineering nalidixic acid’s chemical scaffold: A step towards the development of novel anti-tubercular and anti-bacterial leads for resistant pathogensPeraman, Ramalingam / Varma, Raghu Veer / Reddy, Y. Padmanabha et al. | 2015
- 4320
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Discovery of 1-hydroxypyridine-2-thiones as selective histone deacetylase inhibitors and their potential application for treating leukemiaMuthyala, Ramaiah / Shin, Woo Shik / Xie, Jiashu et al. | 2015
- 4325
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Isolation and structure of vanitaracin A, a novel anti-hepatitis B virus compound from Talaromyces sp.Matsunaga, Hiroki / Kamisuki, Shinji / Kaneko, Manabu et al. | 2015
- 4329
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Chemo-enzymatic synthesis of imidazolium-tagged sialyllactosamine probesSittel, Imke / Galan, M. Carmen et al. | 2015
- 4333
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Pandalisines A and B, novel indolizidine alkaloids from the leaves of Pandanus utilisCheng, Yuan-Bin / Tsai, Yi-Hong / Lo, I-Wen et al. | 2015
- 4337
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Discovery of selective N-[3-(1-methyl-piperidine-4-carbonyl)-phenyl]-benzamide-based 5-HT1F receptor agonists: Evolution from bicyclic to monocyclic coresZhang, Deyi / Blanco, Maria-Jesus / Ying, Bai-Ping et al. | 2015
- 4337
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Discovery of selective N-[3-(1-methyl-piperidine-4-carbonyl)-phenyl]-benzamide-based 5-HT₁ F receptor agonists: Evolution from bicyclic to monocyclic coresBlanco, Maria-Jesus et al. | 2015
- 4342
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Synthesis of oxygenated oleanolic and ursolic acid derivatives with anti-inflammatory propertiesNelson, Andrew T. / Camelio, Andrew M. / Claussen, Karin R. et al. | 2015
- IFC
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Editorial board| 2015