Bioorganic and Medicinal Chemistry Letters
The tables of contents are generated automatically and are based on the data records of the individual contributions available in the index of the TIB portal. The display of the Tables of Contents may therefore be incomplete.
Table of contents
- 1451
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Graphical contents list| 2006
- 1468
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6H-Benzo[c]chromen-6-one derivatives as selective ERβ agonistsSun, Wanying / Cama, Lovji D. / Birzin, Elizabeth T. et al. | 2005
- 1468
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6H-Benzo[c]chromen-6-one derivatives as selective ERb agonistsSun, Wanying et al. | 2006
- 1473
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Design of novel synthetic MTS conjugates of bile acids for site-directed sulfhydryl labeling of cysteine residues in bile acid binding and transporting proteinsRay, Abhijit / Banerjee, Antara / Chang, Cheng et al. | 2005
- 1477
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Imidazo[1,2-b][1,2,4]triazines as a2-a3 subtype selective GABAA agonists for the treatment of anxietyJennings, Andrew S.R. et al. | 2006
- 1477
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Imidazo[1,2-b][1,2,4]triazines as α2/α3 subtype selective GABAA agonists for the treatment of anxietyJennings, Andrew S.R. / Lewis, Richard T. / Russell, Michael G.N. et al. | 2005
- 1481
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6H,13H-Pyrazino[1,2-a;4,5-a′]diindole analogs: Probing the pharmacophore for allosteric ligands of muscarinic M2 receptorsZlotos, Darius P. / Tränkle, Christian / Abdelrahman, Aliaa et al. | 2005
- 1486
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Arylaminoethyl amides as noncovalent inhibitors of cathepsin S. Part 2: Optimization of P1 and N-arylAlper, Phillip B. / Liu, Hong / Chatterjee, Arnab K. et al. | 2005
- 1491
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Anti-HBV nucleotide prodrug analogs: Synthesis, bioreversibility, and cytotoxicity studiesPadmanabhan, Seetharamaiyer / Coughlin, John E. / Zhang, Guangrong et al. | 2005
- 1495
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Synthesis and screening of bicyclic carbohydrate-based compounds: A novel type of antiviralsHoof, Steven Van / Ruttens, Bart / Hubrecht, Idzi et al. | 2005
- 1499
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Cyclodextrin-grafted polysaccharides as supramolecular carrier systems for naproxenRamírez, Héctor L. / Valdivia, Aymara / Cao, Roberto et al. | 2005
- 1502
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4-Aminophenoxyacetic acids as a novel class of reversible cathepsin K inhibitorsShinozuka, Tsuyoshi / Shimada, Kousei / Matsui, Satoshi et al. | 2005
- 1506
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Synthesis and biological investigation of new 4″-malonyl tethered derivatives of erythromycin and clarithromycinSherman, Daniel / Xiong, Liqun / Mankin, Alexander S. et al. | 2005
- 1510
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Inhibition of jack bean urease by organobismuth compoundsMurafuji, Toshihiro / Azuma, Takako / Miyoshi, Youhei et al. | 2005
- 1514
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Schiff base conjugates of p-aminosalicylic acid as antimycobacterial agentsPatole, Jayendra / Shingnapurkar, Dipti / Padhye, Subhash et al. | 2005
- 1518
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8-Fluoroimidazo[1,2-a]pyridine: Synthesis, physicochemical properties and evaluation as a bioisosteric replacement for imidazo[1,2-a]pyrimidine in an allosteric modulator ligand of the GABAA receptorHumphries, Alexander C. / Gancia, Emanuela / Gilligan, Myra T. et al. | 2005
- 1523
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Cyclodextrin retinylidene: A biomimetic kinetic trap model for rhodopsinKpegba, Kafui / Murtha, Matthew / Nesnas, Nasri et al. | 2005
- 1527
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Guanidinylated 2,5-dideoxystreptamine derivatives as anthrax lethal factor inhibitorsJiao, Guan-Sheng / Cregar, Lynne / Goldman, Mark E. et al. | 2005
- 1532
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Identification of a novel series of tetrahydrodibenzazocines as inhibitors of 17b-hydroxysteroid dehydrogenase type 3Fink, Brian E. et al. | 2006
- 1532
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Identification of a novel series of tetrahydrodibenzazocines as inhibitors of 17β-hydroxysteroid dehydrogenase type 3Fink, Brian E. / Gavai, Ashvinikumar V. / Tokarski, John S. et al. | 2005
- 1537
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Synthesis, X-ray crystallographic analysis, and antitumor activity of N-(benzothiazole-2-yl)-1-(fluorophenyl)-O,O-dialkyl-a-aminopho- sphonatesJin, Linhong et al. | 2006
- 1537
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Synthesis, X-ray crystallographic analysis, and antitumor activity of N-(benzothiazole-2-yl)-1-(fluorophenyl)-O,O-dialkyl-α-aminophosphonatesJin, Linhong / Song, Baoan / Zhang, Guoping et al. | 2005
- 1544
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Discovery and synthesis of a novel series of quinoline-based thrombin receptor (PAR-1) antagonistsClasby, Martin C. / Chackalamannil, Samuel / Czarniecki, Michael et al. | 2005
- 1549
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Discovery and SAR study of novel dihydroquinoline containing glucocorticoid receptor ligandsTakahashi, Hidenori / Bekkali, Younes / Capolino, Alison J. et al. | 2005
- 1553
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Structure–activity relationship studies on niphimycin, a guanidylpolyol macrolide antibiotic. Part 1: The role of the N-methyl-N″-alkylguanidinium moietyUsuki, Yoshinosuke / Matsumoto, Keiji / Inoue, Takatsugu et al. | 2005
- 1557
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Novel 4-N-substituted aryl pent-2-ene-1,4-dione derivatives of piperazinyloxazolidinones as antibacterialsLohray, Braj Bhushan / Lohray, Vidya Bhushan / Srivastava, Brijesh Kumar et al. | 2005
- 1562
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Synthesis and evaluation of novel 8-oxo-8H-cyclopenta[a]acenaphthylene-7-carbonitriles as long-wavelength fluorescent markers for hypoxic cells in solid tumorLiu, Yan / Xu, Yufang / Qian, Xuhong et al. | 2005
- 1567
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Nuphar alkaloids with immediately apoptosis-inducing activity from Nuphar pumilum and their structural requirements for the activityMatsuda, Hisashi / Yoshida, Kazutoshi / Miyagawa, Katsutoshi et al. | 2005
- 1574
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1,2,3,4-Tetrahydroisoquinolinyl sulfamic acids as phosphatase PTP1B inhibitorsKlopfenstein, Sean R. / Evdokimov, Artem G. / Colson, Anny-Odile et al. | 2005
- 1579
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Arylphthalazines. Part 2: 1-(Isoquinolin-5-yl)-4-arylamino phthalazines as potent inhibitors of VEGF receptors I and IIDuncton, Matthew A.J. / Piatnitski, Evgueni L. / Katoch-Rouse, Reeti et al. | 2005
- 1582
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Imidazo[1,2-a]pyrazin-8-ones, imidazo[1,2-d][1,2,4]triazin-8-ones and imidazo[2,1-f][1,2,4]triazin-8-ones as a2-a3 subtype selective GABAA agonists for the treatment of anxietyGoodacre, Simon C. et al. | 2006
- 1582
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Imidazo[1,2-a]pyrazin-8-ones, imidazo[1,2-d][1,2,4]triazin-8-ones and imidazo[2,1-f][1,2,4]triazin-8-ones as α2/α3 subtype selective GABAA agonists for the treatment of anxietyGoodacre, Simon C. / Hallett, David J. / Carling, Robert W. et al. | 2005
- 1586
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Novel dual inhibitors of calpain and lipid peroxidation with enhanced cellular activityAuvin, Serge / Pignol, Bernadette / Navet, Edith et al. | 2005
- 1590
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The water-soluble fullerene derivative ‘Radical Sponge®’ exerts cytoprotective action against UVA irradiation but not visible-light-catalyzed cytotoxicity in human skin keratinocytesXiao, Li / Takada, Hiroya / Gan, Xue hui et al. | 2005
- 1596
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Factor VIIa inhibitors: Gaining selectivity within the trypsin familyShrader, William D. / Kolesnikov, Aleksandr / Burgess-Henry, Jana et al. | 2005
- 1601
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Synthesis and evaluation of an N-acylated photoactivatable analogue of glutathione as probe for glutathione-utilizing enzymesBernardi, Dan / Battaglia, Eric / Kirsch, Gilbert et al. | 2005
- 1605
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Acetylenic TACE inhibitors. Part 3: Thiomorpholine sulfonamide hydroxamatesLevin, J.I. / Chen, J.M. / Laakso, L.M. et al. | 2005
- 1610
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Brequinar derivatives and species-specific drug design for dihydroorotate dehydrogenaseHurt, Darrell E. / Sutton, Amanda E. / Clardy, Jon et al. | 2005
- 1616
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Structural modifications of the cannabinoid side chain towards C3-aryl and 1′,1′-cycloalkyl-1′-cyano cannabinoidsPapahatjis, Demetris P. / Nahmias, Victoria R. / Andreou, Thanos et al. | 2005
- 1621
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Depeptidization efforts on α-ketoamide inhibitors of HCV NS3-4A serine protease: Effect on HCV replicon activityBogen, Stéphane L. / Ruan, Sumei / Liu, Rong et al. | 2005
- 1621
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Depeptidization efforts on a-ketoamide inhibitors of HCV NS3-4A serine protease: Effect on HCV replicon activityBogen, Stéphane L. et al. | 2006
- 1621
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Depeptidization efforts on Formula Not Shown α-ketoamide inhibitors of HCV NS3-4A serine protease: Effect on HCV replicon activityBogen, S. p. / Ruan, S. / Liu, R. et al. | 2006
- 1628
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Novel inhibitors of hepatitis C NS3–NS4A serine protease derived from 2-aza-bicyclo[2.2.1]heptane-3-carboxylic acidVenkatraman, Srikanth / Njoroge, F. George / Wu, Wanli et al. | 2005
- 1633
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Inhibitors of epidermal growth factor receptor tyrosine kinase: Novel C-5 substituted anilinoquinazolines designed to target the ribose pocketBallard, Peter / Bradbury, Robert H. / Harris, Craig S. et al. | 2005
- 1638
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Discovery and optimization of a novel series of liver X receptor-a agonistsLi, Leping et al. | 2006
- 1638
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Discovery and optimization of a novel series of liver X receptor-α agonistsLi, Leping / Liu, Jiwen / Zhu, Liusheng et al. | 2005
- 1643
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Tricyclic azepine derivatives: Pyrimido[4,5-b]-1,4-benzoxazepines as a novel class of epidermal growth factor receptor kinase inhibitorsSmith, Leon II / Piatnitski, Evgueni L. / Kiselyov, Alexander S. et al. | 2005
- 1647
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DNA triplex stabilization by a δ-carboline derivative tethered to third strand oligonucleotidesTodorović, Nina / Phuong, Nguyen Thi Bich / Langer, Peter et al. | 2005
- 1651
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New photoantimicrobial films composed of porphyrinated lipophilic cellulose estersKrouit, Mohammed / Granet, Robert / Branland, Pierre et al. | 2005
- 1656
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Synthesis and biological activity of (+)-hedychilactone A and its analogs from (+)-sclareolideOh, Sangtae / Jeong, In Howa / Shin, Woon-Seob et al. | 2005
- 1660
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Biological studies of photoinducible phenol quaternary ammonium derivativesSong, Yang / Wang, Ping / Wu, Juanjuan et al. | 2005
- 1665
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Convenient methods for the synthesis of P1-farnesyl-P2-indicator diphosphatesFeld, Birte K. / Weiss, Gregory A. et al. | 2005
- 1668
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Aryl O- and S-galactosides and lactosides as specific inhibitors of human galectins-1 and -3: Role of electrostatic potential at O-3Giguère, Denis / Sato, Sachiko / St-Pierre, Christian et al. | 2005
- 1673
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Design and synthesis of potent and subtype-selective PPARa agonistsDesai, Ranjit C. et al. | 2006
- 1673
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Design and synthesis of potent and subtype-selective PPARα agonistsDesai, Ranjit C. / Metzger, Edward / Santini, Conrad et al. | 2005
- 1679
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Discovery of trans-3,4′-bispyridinylethylenes as potent and novel inhibitors of protein kinase B (PKB/Akt) for the treatment of cancer: Synthesis and biological evaluationLi, Qun / Li, Tongmei / Zhu, Gui-Dong et al. | 2005
- 1686
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Anticancer activity of a series of platinum complexes integrating demethylcantharidin with isomers of 1,2-diaminocyclohexaneYu, Chun-Wing / Li, Kay K.W. / Pang, Siu-Kwong et al. | 2005
- 1692
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Synthesis of the first sulfur-35-labeled hERG radioligandRaab, Conrad E. / Butcher, John W. / Connolly, Thomas M. et al. | 2005
- 1696
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Indole-glucosides as novel sodium glucose co-transporter 2 (SGLT2) inhibitors. Part 2Zhang, Xiaoyan / Urbanski, Maud / Patel, Mona et al. | 2005
- 1702
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Synthesis and insecticidal activity of fluorinated 2-(2,6-dichloro-4-trifluoromethylphenyl)-2,4,5,6-tetrahydrocyclopentapyrazolesMeegalla, Sanath K. / Doller, Dario / Liu, Ruiping et al. | 2005
- 1707
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Natural and synthetic G-quadruplex interactive berberine derivativesFranceschin, Marco / Rossetti, Luigi / D’Ambrosio, Anna et al. | 2005
- 1712
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Synthesis and antiviral activity of 2′-deoxy-2′-fluoro-2′-C-methyl purine nucleosides as inhibitors of hepatitis C virus RNA replicationClark, Jeremy L. / Mason, J. Christian / Hollecker, Laurent et al. | 2005
- 1716
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CDK2/cyclinA inhibitors: Targeting the cyclinA recruitment site with small molecules derived from peptide leadsCastanedo, Georgette / Clark, Kevin / Wang, Shumei et al. | 2005
- 1721
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Synthesis of Tic-d-Phe Ψ[CH2–CH2] isostere and its use in the development of melanocortin receptor agonistsTian, Xinrong / Chen, Xuemei / Gan, Lixian et al. | 2005
- 1726
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2-((1H-Azol-1-yl)methyl)-N-arylbenzamides: Novel dual inhibitors of VEGFR-1/2 kinasesKiselyov, Alexander S. / Semenova, Marina / Semenov, Victor V. et al. | 2005
- 1731
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Seco-prolinenitrile inhibitors of dipeptidyl peptidase IV define minimal pharmacophore requirements at P1Magnin, David R. / Taunk, Prakash C. / Robertson, James G. et al. | 2005
- 1735
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Novel, potent P2–P3 pyrrolidine derivatives of ketoamide-based cathepsin K inhibitorsBarrett, David G. / Catalano, John G. / Deaton, David N. et al. | 2005
- 1740
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Design and modular parallel synthesis of a MCR derived α-helix mimetic protein–protein interaction inhibitor scaffoldAntuch, Walfrido / Menon, Sanjay / Chen, Quin-Zene et al. | 2005
- 1740
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Design and modular parallel synthesis of a MCR derived a-helix mimetic protein–protein interaction inhibitor scaffoldAntuch, Walfrido et al. | 2006
- 1744
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The reversed binding of β-phenethylamine inhibitors of DPP-IV: X-ray structures and properties of novel fragment and elaborated inhibitorsNordhoff, Sonja / Cerezo-Gálvez, Silvia / Feurer, Achim et al. | 2005
- 1744
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The reversed binding of b-phenethylamine inhibitors of DPP-IV: X-ray structures and properties of novel fragment and elaborated inhibitorsNordhoff, Sonja et al. | 2006
- 1749
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Synthesis and SAR of substituted tetrahydrocarbazole derivatives as new NPY-1 antagonistsDi Fabio, Romano / Giovannini, Riccardo / Bertani, Barbara et al. | 2005
- 1753
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Synthesis of 3-benzyl-2-substituted quinoxalines as novel monoamine oxidase A inhibitorsHassan, Seham Y. / Khattab, Sherine N. / Bekhit, Adnan A. et al. | 2005
- 1757
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Erratum to “Efficient cleavage of RNA, enhanced cellular uptake, and controlled intracellular localization of conjugate DNAzymes” [Bioorg. Med. Chem. Lett. 15 (2005) 167–170]Kubo, Takanori / Takamori, Kengo / Kanno, Ken-ichi et al. | 2004
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Editorial Board| 2006
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Instructions to contributors| 2006