Bioorganic and Medicinal Chemistry Letters
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Table of contents
- 305
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Graphical Abstracts| 2002
- 321
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Myxovirescin analogues via macrocyclic ring–closing metathesisContent, Stéphane / Dutton, Christopher J / Roberts, Lee et al. | 2002
- 327
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Chemoenzymatic synthesis of high-mannose type HIV-1 gp120 glycopeptidesSingh, Suddham / Ni, Jiahong / Wang, Lai-Xi et al. | 2002
- 331
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Solid-phase synthesis of cyclic RGD-furanoid sugar amino acid peptides as integrin inhibitorsvan Well, Renate M. / Overkleeft, Herman S. / van der Marel, Gijsbert A. et al. | 2002
- 335
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2,5-Bis-(2-hydroxybenzoylamino)pentanoic acid, a salicylic acid-metabolite isolated from chicken: characterization and independent synthesisHillaert, Ulrik / Baert, Kris / Rozenski, Jef et al. | 2002
- 339
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Stereochemical studies on phosphopantothenoylcysteine decarboxylase from Escherichia coliStrauss, Erick / Begley, Tadhg P et al. | 2002
- 343
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Synthesis and GABAA receptor activity of a 6,19-Oxido analogue of pregnanoloneVeleiro, Adriana S / Rosenstein, Ruth E / Jaliffa, Carolina O et al. | 2002
- 347
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Imidazopyrimidines, potent inhibitors of p38 MAP kinaseRupert, Kenneth C / Henry, James R / Dodd, John H et al. | 2002
- 351
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[3H]-Methoxymethyl-MTEP and [3H]-Methoxy-PEPy: potent and selective radioligands for the metabotropic glutamate subtype 5 (mGlu5) receptorCosford, Nicholas D.P / Roppe, Jeffrey / Tehrani, Lida et al. | 2002
- 355
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Synthesis and In vitro efficacy of acid-Sensitive poly(ethylene glycol) paclitaxel conjugatesRodrigues, Paula C.A / Scheuermann, Karin / Stockmar, Cornelia et al. | 2002
- 361
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Structure–Activity relationships of novel anti-Malarial agents: Part 5. N-(4-acylamino-3-benzoylphenyl)-[5-(4-nitrophenyl)-2-furyl]acrylic acid amidesWiesner, Jochen / Kettler, Katja / Sakowski, Jacek et al. | 2002
- 365
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Nociceptin/Orphanin FQ(1–13)NH2 analogues modified in the Phe1-Gly2 peptide bondGuerrini, Remo / Rizzi, Daniela / Zucchini, Marina et al. | 2002
- 369
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Nonbenzamidine tetrazole derivatives as factor Xa inhibitorsQuan, Mimi L / Ellis, Christopher D / He, Ming Y et al. | 2002
- 375
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Synthesis and In vivo anti-inflammatory activity of long-chain 2-amino-alcoholsMagrioti, Victoria / Hadjipavlou-Litina, Dimitra / Constantinou-Kokotou, Violetta et al. | 2002
- 379
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Discovery of a novel series of 6-azauracil-based thyroid hormone receptor ligands: potent, TRβ subtype-selective thyromimeticsDow, Robert L. / Schneider, Steven R. / Paight, Ernest S. et al. | 2002
- 379
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Discovery of a novel series of 6-azauracil-based thyroid hormone receptor ligands: potent, TRb subtype-selective thyromimeticsDow, Robert L. et al. | 2003
- 383
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Evaluation of vinylsulfamides as sulfhydryl selective alkylation reagents in protein modificationLi, Min / Wu, Robert S. / Tsai, Jane S.C. et al. | 2002
- 387
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Synthesis and evaluation of d-Lactams (Piperazones) as elastase inhibitorsSeibel, Jürgen et al. | 2003
- 387
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Synthesis and evaluation of δ-Lactams (Piperazones) as elastase inhibitorsSeibel, Jürgen / Brown, David / Amour, Augustin et al. | 2002
- 391
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Synthesis of labelled PNA oligomers by a post-synthetic modification approachde la Torre, Beatriz G / Eritja, Ramon et al. | 2002
- 395
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Synthesis of antioxidant propyl gallate using tannase from Aspergillus niger van Teighem in nonaqueous mediaSharma, Shweta / Gupta, Munishwar N et al. | 2002
- 399
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Novel thieno oxazine analogues as antihyperglycemic and lipid modulating agentsDas, Saibal Kumar / Reddy, K.Anantha / Abbineni, Chandrasekhar et al. | 2002
- 405
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SLV310, a novel, potential antipsychotic, combining potent dopamine D2 receptor antagonism with serotonin reuptake inhibitionvan Hes, Rolf / Smid, Pieter / Stroomer, Cees N.J et al. | 2002
- 409
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Zinc(II)-mediated inhibition of a ribonuclease by an N-hydroxyurea nucleotideHiggin, Joshua J / Yakovlev, Gennady I / Mitkevich, Vladimir A et al. | 2002
- 413
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2,3-Diarylbenzopyran derivatives as a novel class of selective cyclooxygenase-2 inhibitorsHyup Joo, Yung / Kwan Kim, Jin / Kang, Seon-Hwa et al. | 2002
- 419
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QSAR Study on solubility of alkanes in water and Their partition coefficients in different solvent systems using PI indexKhadikar, Padmakar V. / Mandloi, Dheeraj / Bajaj, Amrit V. et al. | 2002
- 423
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A series of 2(Z)-2-Benzylidene-6,7-dihydroxybenzofuran-3[2H]-ones as inhibitors of chorismate synthaseThomas, Michael G / Lawson, Chris / Allanson, Nigel M et al. | 2002
- 427
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1,3,4 trisubstituted pyrrolidine CCR5 receptor antagonists bearing 4-aminoheterocycle substituted piperidine side chainsWilloughby, Christopher A / Rosauer, Keith G / Hale, Jeffery J et al. | 2002
- 433
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Novel antifungal b-amino acids: synthesis and activity against Candida albicansMittendorf, Joachim et al. | 2003
- 433
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Novel antifungal β-amino acids: synthesis and activity against Candida albicansMittendorf, Joachim / Kunisch, Franz / Matzke, Michael et al. | 2002
- 437
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Discovery of orally bioavailable NK1 receptor antagonistsGenicot, C. / Christophe, B. / Collart, P. et al. | 2002
- 443
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Characterization of the mechanism of anticonvulsant activity for a selected set of putative AMPA receptor antagonistsGrasso, Silvana / Micale, Nicola / Zappalà, Maria et al. | 2002
- 447
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Modelling of carbonic anhydrase inhibitory activity of sulfonamides using molecular negentropyAgrawal, Vijay K / Khadikar, Padmakar V et al. | 2002
- 455
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Synthesis and antitumor activity of novel C-8 ester derivatives of leinamycinKanda, Yutaka / Ashizawa, Tadashi / Kawashima, Kenji et al. | 2002
- 459
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Synthesis and preliminary cytotoxicity of nitrogen mustard derivatives of distamycin AWang, Yuqiang / Wright, Susan C / Larrick, James W et al. | 2002
- 463
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Synthesis and biological evaluation of novel 1b-methylcarbapenems with isothiazoloethenyl side chainsKang, Yong Koo et al. | 2003
- 463
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Synthesis and biological evaluation of novel 1β-methylcarbapenems with isothiazoloethenyl side chainsKang, Yong Koo / Lee, Kyung Seok / Yoo, Kyung Ho et al. | 2002
- 467
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p38 Inhibitors: piperidine- and 4-aminopiperidine-substituted naphthyridinones, quinolinones, and dihydroquinazolinonesHunt, Julianne A / Kallashi, Florida / Ruzek, Rowena D et al. | 2002
- 471
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Antitumour benzothiazoles. Part 20:Hutchinson, I. / Bradshaw, T. D. / Matthews, C. S. et al. | 2003
- 471
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Antitumour benzothiazoles. Part 20: 3'-Cyano and 3'-Alkynyl-Substituted 2-(4'-Aminophenyl)benzothiazoles as new potent and selective analoguesHutchinson, Ian et al. | 2003
- 471
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Antitumour benzothiazoles. Part 20:† For Part 19 of the series, see ref 1. 3′-Cyano and 3′-Alkynyl-Substituted 2-(4′-Aminophenyl)benzothiazoles as new potent and selective analoguesHutchinson, Ian / Bradshaw, Tracey D / Matthews, Charles S et al. | 2002
- 475
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Synthesis and SAR of α-Acylaminoketone ligands for control of gene expressionTice, Colin M / Hormann, Robert E / Thompson, Christine S et al. | 2002
- 475
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Synthesis and SAR of a-Acylaminoketone ligands for control of gene expressionTice, Colin M. et al. | 2003
- 479
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2-Phenylspiroindenes: a novel class of selective estrogen receptor modulators (SERMs)Blizzard, Timothy A / Morgan, II, Jerry D / Mosley, Ralph T et al. | 2002
- 485
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Inhibition of mast cell leukotriene release by thiourea derivativesVenkatachalam, Taracad K / Qazi, Sanjive / Samuel, Peter et al. | 2002
- 489
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Discovery, SAR, synthesis, pharmacokinetic and biochemical characterization of A-192411: A novel fungicidal lipopeptide-(I)Wang, Weibo / Li, Qun / Hasvold, Lisa et al. | 2002
- 495
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In vivo characterization of A-192411: a novel fungicidal lipopeptide (II)Meulbroek, Jonathan A / Nilius, Angela M / Li, Qun et al. | 2002
- 499
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1,4-Diazepane-2-ones as novel inhibitors of LFA-1Wattanasin, Sompong / Albert, Rainer / Ehrhardt, Claus et al. | 2002
- 503
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Thiophene-based vitronectin receptor antagonistsBubenik, Monica / Meerovitch, Karen / Bergeron, Frédéric et al. | 2002
- 507
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Structure–Activity relationships of substituted benzothiophene-anthranilamide factor Xa inhibitorsChou, Yuo-Ling / Davey, David D / Eagen, Keith A et al. | 2002
- 513
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Pharmacophore-Based discovery of substituted pyridines as novel dopamine transporter inhibitorsEnyedy, Istvan J / Sakamuri, Sukumar / Zaman, Wahiduz A et al. | 2002
- 519
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Sordaricin antifungal agentsQuesnelle, Claude A / Gill, Patrice / Dodier, Marco et al. | 2002
- 525
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5-Azidoepibatidine: an exceptionally potent photoaffinity ligand for neuronal a4b2 and a7 nicotinic acetylcholine receptorsZhang, Nanjing et al. | 2003
- 525
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5-Azidoepibatidine: an exceptionally potent photoaffinity ligand for neuronal α4β2 and α7 nicotinic acetylcholine receptorsZhang, Nanjing / Tomizawa, Motohiro / Casida, John E et al. | 2002
- 529
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Synthesis, opioid receptor binding, and functional activity of 5′-substituted 17-cyclopropylmethylpyrido[2′,3′:6,7]morphinansAnanthan, Subramaniam / Kezar, III, Hollis S / Saini, Surendra K et al. | 2002
- 529
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Synthesis, opioid receptor binding, and functional activity of 5prime-substituted 17-cyclopropylmethylpyrido[2prime,3prime:6,7]morphinansAnanthan, S. / Kezar, III, H. S. / Saini, S. K. et al. | 2003
- 533
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Both 5-arylidene-2-thioxodihydropyrimidine-4,6(1H,5H)-diones and 3-thioxo-2,3-dihydro-1H-imidazo(1,5-a)indol-1-ones are light-Dependent tumor necrosis factor-a antagonistsVoss, Matthew E. et al. | 2003
- 533
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Both 5-arylidene-2-thioxodihydropyrimidine-4,6(1H,5H)-diones and 3-thioxo-2,3-dihydro-1H-imidazo[1,5-a]indol-1-ones are light-Dependent tumor necrosis factor-α antagonistsVoss, Matthew E / Carter, Percy H / Tebben, Andrew J et al. | 2002
- 539
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Cephalosporin prodrugs of paclitaxel for immunologically specific activation by L-49-sFv-b-Lactamase fusion proteinVrudhula, Vivekananda M. et al. | 2003
- 539
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Cephalosporin prodrugs of paclitaxel for immunologically specific activation by L-49-sFv-β-Lactamase fusion proteinVrudhula, Vivekananda M. / Kerr, David E. / Siemers, Nathan O. et al. | 2002
- 543
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Novel inhibitors of IMPDHWatterson, Scott H. / Carlsen, Marianne / Murali Dhar, T.G. et al. | 2002
- 543
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Novel inhibitors of IMPDH - a highly potent and selective quinolone-based seriesWatterson, Scott H. et al. | 2003
- 547
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Quinolone-Based IMPDH inhibitors: introduction of basic residues on ring D and SAR of the corresponding mono, di and benzofused analoguesDhar, T.G.Murali / Watterson, Scott H. / Chen, Ping et al. | 2002
- 553
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Synthesis and dopamine transporter affinity of chiral 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(2-hydroxypropyl)piperazines as potential cocaine abuse therapeutic agentsHsin, Ling-Wei / Prisinzano, Thomas / Wilkerson, Chavon R et al. | 2002
- 557
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A facile synthesis of C2-symmetric 17b-estradiol dimersRabouin, Daniel et al. | 2003
- 557
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A facile synthesis of C2-symmetric 17β-estradiol dimersRabouin, Daniel / Perron, Valérie / N'Zemba, Blaise et al. | 2002
- 561
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Design, synthesis and structure–Activity relationships of benzoxazinone-Based factor Xa inhibitorsHuang, Wenrong / Zhang, Penglie / Zuckett, Jingmei F et al. | 2002
- 567
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Piperazine-based CCR5 antagonists as HIV-1 inhibitors. III: synthesis, antiviral and pharmacokinetic profiles of symmetrical heteroaryl carboxamidesMcCombie, Stuart W. / Tagat, Jayaram R. / Vice, Susan F. et al. | 2002
- 573
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Condensed aromatic peptide family of microbial metabolites, inhibitors of CD28–CD80 interactionsHegde, Vinod R / Puar, Mohindar S / Dai, Ping et al. | 2002
- 577
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Selective phenolic acylation of 10-hydroxycamptothecin using poly (ethylene glycol) carboxylic acidGreenwald, Richard B. / Choe, Yun H. / Wu, Dechun et al. | 2002
- 581
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Organic phenyl arsonic acid compounds with potent antileukemic activityLiu, Xing-Ping / Narla, Rama Krishna / Uckun, Fatih M et al. | 2002
- 585
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Erratum to "Design and Synthesis of a b-Amino Phosphotyrosyl Mimetic Suitably Protected for Peptide Synthesis"(Bioorg. Med. Chem. Lett. 12 (2002) 3399)Lee, Kyeoung et al. | 2003
- 585
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Erratum to “Design and Synthesis of a β-Amino Phosphotyrosyl Mimetic Suitably Protected for Peptide Synthesis”[Bioorg. Med. Chem. Lett. 12 (2002) 3399]Lee, Kyeoung / Zhang, Manchao / Yang, Dajun et al. | 2002
- CO2
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Editorial Board| 2002
- I
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Instructions to Contributors| 2002
- iii
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Contents List| 2002
- vii
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Contributors to this issue| 2002